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PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

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<strong>42</strong>/<strong>2000</strong><br />

15246 <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 19 Oct/oct <strong>2000</strong><br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

(54) BICYCLIC HETEROAROMATIC<br />

COMPOUNDS USEFUL AS LH AGO-<br />

NISTS<br />

COMPOSES HETEROAROMATIQUES<br />

BICYCLIQUES UTILES EN TANT<br />

QU’AGONISTES DE L’HORMONE<br />

LUTEINISANTE (LH)<br />

(71) AKZO NOBEL N.V. [NL/NL]; Velperweg<br />

76, NL–6824 BM Arnhem (NL).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) GERRITSMA, Gerrildina, Geziena<br />

[NL/NL]; Vezelstraat 20, NL–5345 XD Oss<br />

(NL). VAN STRATEN, Nicole, Corine,<br />

Renée [NL/NL]; De Bongerd 132, NL–5345<br />

JW Oss (NL). ADANG, Anton, Egbert,<br />

Peter [NL/NL]; Le Sage ten Broeklaan 77,<br />

NL–5615 CR Eindhoven (NL).<br />

(74) HERMANS, F., G., M.; P.O. Box 20,<br />

NL–5340 BH Oss (NL).<br />

(81) AL AU BA BB BG BR CA CN CU CZ EE<br />

GE HR HU ID IL IN IS JP KP KR LC LK<br />

LR LT LV MG MK MN MX NO NZ PL RO<br />

RU SG SI SK SL TR TT UA US UZ VN YU<br />

ZA; AP (GH GM KE LS MW SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 C07D 495/14, A61K 31/55, A61P 5/00 //<br />

(C07D 495/14, 333:00, 243:00, 221:00)<br />

(11) WO 00/61587 (13) A1<br />

(21) <strong>PCT</strong>/FR00/00881<br />

(22) 7 Apr/avr <strong>2000</strong> (07.04.<strong>2000</strong>)<br />

(25) fr (26) fr<br />

(30) 99/04440 9 Apr/avr 1999<br />

(09.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

FR<br />

(54) PYRIDO–THIENO–DIAZEPINES, ME-<br />

THOD FOR THE PRODUCTION<br />

THEREOF AND PHARMACEUTICAL<br />

COMPOSITIONS CONTAINING SAID<br />

PYRIDO–THIENO–DIAZEPINES<br />

PYRIDO–THIENO–DIAZEPINES,<br />

LEUR PROCEDE DE PREPARATION<br />

ET LES COMPOSITIONS PHARMA-<br />

CEUTIQUES LES CONTENANT<br />

(71) SOCIETE DE CONSEILS DE RE-<br />

CHERCHES ET D’APPLICATIONS<br />

SCIENTIFIQUES (S.C.R.A.S.) [FR/FR];<br />

51/53, rue du Docteur Blanche, F–75016<br />

Paris (FR).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) LIBERATORE, Anne–Marie [FR/FR];<br />

10, rue de la Croix Picard, Saint Benoist,<br />

F–78610 Auffargis (FR). BIGG, Dennis<br />

[FR/FR]; 12, rue des Bénédictines, F–91190<br />

Gif–sur–Yvette (FR).<br />

(74) BOURGOUIN, André; Beaufour Ipsen –<br />

S.C.A.F., Direction de la Propriété Industrielle,<br />

<strong>42</strong>, rue du Docteur Blanche, F–75016<br />

Paris (FR).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID<br />

IL IN IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MA MD MG MK MN MW<br />

MX NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ<br />

VN YU ZA ZW; AP (GH GM KE LS MW<br />

SD SL SZ TZ UG ZW); EA (AM AZ BY<br />

KG KZ MD RU TJ TM); EP (AT BE CH<br />

CY DE DK ES FI FR GB GR IE IT LU MC<br />

NL PT SE); OA (BF BJ CF CG CI CM GA<br />

GN GW ML MR NE SN TD TG).<br />

(51) 7 C07F 7/18, C07C 177/00<br />

(11) WO 00/61588 (13) A1<br />

(21) <strong>PCT</strong>/GB00/01375<br />

(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 9908326.3 12 Apr/avr 1999<br />

(12.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

GB<br />

(54) NOVEL INTERMEDIATE FOR THE<br />

SYNTHESIS OF PROSTAGLANDINS<br />

NOUVEAU PRODUIT INTERME-<br />

DIAIRE POUR LA SYNTHESE DES<br />

PROSTAGLANDINES<br />

(71) CHIROTECH TECHNOLOGY LIMI-<br />

TED [GB/GB]; Cambridge Science Park,<br />

Milton Road, Cambridge CB4 0WG (GB).<br />

(72) JACKSON, Philip, Mark; Chirotech<br />

Technology Limited, Cambridge Science<br />

Park, Milton Road, Cambridge CB4 0WG<br />

(GB). LENNON, Ian, Campbell; Chirotech<br />

Technology Limited, Cambridge Science<br />

Park, Milton Road, Cambridge CB4 0WG<br />

(GB).<br />

(74) GILL JENNINGS & EVERY; Broadgate<br />

House, 7 Eldon Street, London EC2M 7LH<br />

(GB).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID<br />

IL IN IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MA MD MG MK MN MW<br />

MX NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG UZ VN<br />

YU ZA ZW; AP (GH GM KE LS MW SD<br />

SL SZ TZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY<br />

DE DK ES FI FR GB GR IE IT LU MC NL<br />

PT SE); OA (BF BJ CF CG CI CM GA GN<br />

GW ML MR NE SN TD TG).<br />

(51) 7 C07F 9/653, 15/00, C07B 53/00, C07D<br />

263/06<br />

(11) WO 00/61589 (13) A1<br />

(21) <strong>PCT</strong>/GB00/00758<br />

(22) 3 Mar/mar <strong>2000</strong> (03.03.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 9907895.8 8 Apr/avr 1999<br />

(08.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

GB<br />

(54) NOVEL LIGANDS FOR CHIRAL CA-<br />

TALYSIS<br />

NOUVEAUX LIGANDS POUR CATA-<br />

LYSE CHIRALE<br />

(71) THE TEXAS A & M UNIVERSITY SYS-<br />

TEM [US/US]; 310 Wisenbaker, College<br />

Station, TX 77843–3369 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) BURGESS, Kevin [GB/US]; 764 S Rosemary,<br />

Bryan, TX 77802 (US).<br />

(74) WISHART, Ian, Carmichael; Johnson<br />

Matthey Technology Centre, Blounts Court,<br />

Sonning Common, Reading RG4 9NH (GB).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CU CZ DE DK EE ES FI GB<br />

GD GE GH GM HR HU ID IL IN IS JP KE<br />

KG KP KR KZ LC LK LR LS LT LU LV<br />

MD MG MK MN MW MX NO NZ PL PT<br />

RO RU SD SE SG SI SK SL TJ TM TR TT<br />

UA UG US UZ VN YU ZA ZW; AP (GH<br />

GM KE LS MW SD SL SZ TZ UG ZW);<br />

EA (AM AZ BY KG KZ MD RU TJ TM);<br />

EP (AT BE CH CY DE DK ES FI FR GB<br />

GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(51) 7 C07F 15/00 // A61K 31/28, A61P 35/00<br />

(11) WO 00/61590 (13) A1<br />

(21) <strong>PCT</strong>/CA00/00385<br />

(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/128,939 13 Apr/avr 1999<br />

(13.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

US<br />

(54) PROCESS FOR PREPARING AMINE<br />

PLATINUM COMPLEXES<br />

PROCEDE DE PREPARATION DE<br />

COMPLEXES DE PLATINE<br />

(71) ANORMED, INC. [CA/CA]; <strong>No</strong>. 200,<br />

20353–64th Avenue, Langley, British Columbia<br />

V2Y 1N5 (CA).<br />

(72) WONG, Ernest, S., Y.; Unit 50,<br />

8844–208th Street, Langley, British Columbia<br />

V1M 3X7 (CA). GIANDOMENICO,<br />

Christen, M.; 778 Elm Avenue, Blaine, WA<br />

98230 (US).<br />

(74) ROBINSON, J., Christopher et al. / etc.;<br />

Fetherstonhaugh & Co., Box 11560, Suite<br />

2200, 650 West Georgia Street, Vancouver,<br />

British Columbia V6B 4N8 (CA).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID<br />

IL IN IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MA MD MG MK MN MW<br />

MX NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG UZ VN<br />

YU ZA ZW; AP (GH GM KE LS MW SD<br />

SL SZ TZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY<br />

DE DK ES FI FR GB GR IE IT LU MC NL<br />

PT SE); OA (BF BJ CF CG CI CM GA GN<br />

GW ML MR NE SN TD TG).

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