PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
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<strong>42</strong>/<strong>2000</strong><br />
15246 <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 19 Oct/oct <strong>2000</strong><br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
(54) BICYCLIC HETEROAROMATIC<br />
COMPOUNDS USEFUL AS LH AGO-<br />
NISTS<br />
COMPOSES HETEROAROMATIQUES<br />
BICYCLIQUES UTILES EN TANT<br />
QU’AGONISTES DE L’HORMONE<br />
LUTEINISANTE (LH)<br />
(71) AKZO NOBEL N.V. [NL/NL]; Velperweg<br />
76, NL–6824 BM Arnhem (NL).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) GERRITSMA, Gerrildina, Geziena<br />
[NL/NL]; Vezelstraat 20, NL–5345 XD Oss<br />
(NL). VAN STRATEN, Nicole, Corine,<br />
Renée [NL/NL]; De Bongerd 132, NL–5345<br />
JW Oss (NL). ADANG, Anton, Egbert,<br />
Peter [NL/NL]; Le Sage ten Broeklaan 77,<br />
NL–5615 CR Eindhoven (NL).<br />
(74) HERMANS, F., G., M.; P.O. Box 20,<br />
NL–5340 BH Oss (NL).<br />
(81) AL AU BA BB BG BR CA CN CU CZ EE<br />
GE HR HU ID IL IN IS JP KP KR LC LK<br />
LR LT LV MG MK MN MX NO NZ PL RO<br />
RU SG SI SK SL TR TT UA US UZ VN YU<br />
ZA; AP (GH GM KE LS MW SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07D 495/14, A61K 31/55, A61P 5/00 //<br />
(C07D 495/14, 333:00, 243:00, 221:00)<br />
(11) WO 00/61587 (13) A1<br />
(21) <strong>PCT</strong>/FR00/00881<br />
(22) 7 Apr/avr <strong>2000</strong> (07.04.<strong>2000</strong>)<br />
(25) fr (26) fr<br />
(30) 99/04440 9 Apr/avr 1999<br />
(09.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
FR<br />
(54) PYRIDO–THIENO–DIAZEPINES, ME-<br />
THOD FOR THE PRODUCTION<br />
THEREOF AND PHARMACEUTICAL<br />
COMPOSITIONS CONTAINING SAID<br />
PYRIDO–THIENO–DIAZEPINES<br />
PYRIDO–THIENO–DIAZEPINES,<br />
LEUR PROCEDE DE PREPARATION<br />
ET LES COMPOSITIONS PHARMA-<br />
CEUTIQUES LES CONTENANT<br />
(71) SOCIETE DE CONSEILS DE RE-<br />
CHERCHES ET D’APPLICATIONS<br />
SCIENTIFIQUES (S.C.R.A.S.) [FR/FR];<br />
51/53, rue du Docteur Blanche, F–75016<br />
Paris (FR).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) LIBERATORE, Anne–Marie [FR/FR];<br />
10, rue de la Croix Picard, Saint Benoist,<br />
F–78610 Auffargis (FR). BIGG, Dennis<br />
[FR/FR]; 12, rue des Bénédictines, F–91190<br />
Gif–sur–Yvette (FR).<br />
(74) BOURGOUIN, André; Beaufour Ipsen –<br />
S.C.A.F., Direction de la Propriété Industrielle,<br />
<strong>42</strong>, rue du Docteur Blanche, F–75016<br />
Paris (FR).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ<br />
VN YU ZA ZW; AP (GH GM KE LS MW<br />
SD SL SZ TZ UG ZW); EA (AM AZ BY<br />
KG KZ MD RU TJ TM); EP (AT BE CH<br />
CY DE DK ES FI FR GB GR IE IT LU MC<br />
NL PT SE); OA (BF BJ CF CG CI CM GA<br />
GN GW ML MR NE SN TD TG).<br />
(51) 7 C07F 7/18, C07C 177/00<br />
(11) WO 00/61588 (13) A1<br />
(21) <strong>PCT</strong>/GB00/01375<br />
(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 9908326.3 12 Apr/avr 1999<br />
(12.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
GB<br />
(54) NOVEL INTERMEDIATE FOR THE<br />
SYNTHESIS OF PROSTAGLANDINS<br />
NOUVEAU PRODUIT INTERME-<br />
DIAIRE POUR LA SYNTHESE DES<br />
PROSTAGLANDINES<br />
(71) CHIROTECH TECHNOLOGY LIMI-<br />
TED [GB/GB]; Cambridge Science Park,<br />
Milton Road, Cambridge CB4 0WG (GB).<br />
(72) JACKSON, Philip, Mark; Chirotech<br />
Technology Limited, Cambridge Science<br />
Park, Milton Road, Cambridge CB4 0WG<br />
(GB). LENNON, Ian, Campbell; Chirotech<br />
Technology Limited, Cambridge Science<br />
Park, Milton Road, Cambridge CB4 0WG<br />
(GB).<br />
(74) GILL JENNINGS & EVERY; Broadgate<br />
House, 7 Eldon Street, London EC2M 7LH<br />
(GB).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG UZ VN<br />
YU ZA ZW; AP (GH GM KE LS MW SD<br />
SL SZ TZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE); OA (BF BJ CF CG CI CM GA GN<br />
GW ML MR NE SN TD TG).<br />
(51) 7 C07F 9/653, 15/00, C07B 53/00, C07D<br />
263/06<br />
(11) WO 00/61589 (13) A1<br />
(21) <strong>PCT</strong>/GB00/00758<br />
(22) 3 Mar/mar <strong>2000</strong> (03.03.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 9907895.8 8 Apr/avr 1999<br />
(08.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
GB<br />
(54) NOVEL LIGANDS FOR CHIRAL CA-<br />
TALYSIS<br />
NOUVEAUX LIGANDS POUR CATA-<br />
LYSE CHIRALE<br />
(71) THE TEXAS A & M UNIVERSITY SYS-<br />
TEM [US/US]; 310 Wisenbaker, College<br />
Station, TX 77843–3369 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BURGESS, Kevin [GB/US]; 764 S Rosemary,<br />
Bryan, TX 77802 (US).<br />
(74) WISHART, Ian, Carmichael; Johnson<br />
Matthey Technology Centre, Blounts Court,<br />
Sonning Common, Reading RG4 9NH (GB).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CU CZ DE DK EE ES FI GB<br />
GD GE GH GM HR HU ID IL IN IS JP KE<br />
KG KP KR KZ LC LK LR LS LT LU LV<br />
MD MG MK MN MW MX NO NZ PL PT<br />
RO RU SD SE SG SI SK SL TJ TM TR TT<br />
UA UG US UZ VN YU ZA ZW; AP (GH<br />
GM KE LS MW SD SL SZ TZ UG ZW);<br />
EA (AM AZ BY KG KZ MD RU TJ TM);<br />
EP (AT BE CH CY DE DK ES FI FR GB<br />
GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(51) 7 C07F 15/00 // A61K 31/28, A61P 35/00<br />
(11) WO 00/61590 (13) A1<br />
(21) <strong>PCT</strong>/CA00/00385<br />
(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/128,939 13 Apr/avr 1999<br />
(13.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
US<br />
(54) PROCESS FOR PREPARING AMINE<br />
PLATINUM COMPLEXES<br />
PROCEDE DE PREPARATION DE<br />
COMPLEXES DE PLATINE<br />
(71) ANORMED, INC. [CA/CA]; <strong>No</strong>. 200,<br />
20353–64th Avenue, Langley, British Columbia<br />
V2Y 1N5 (CA).<br />
(72) WONG, Ernest, S., Y.; Unit 50,<br />
8844–208th Street, Langley, British Columbia<br />
V1M 3X7 (CA). GIANDOMENICO,<br />
Christen, M.; 778 Elm Avenue, Blaine, WA<br />
98230 (US).<br />
(74) ROBINSON, J., Christopher et al. / etc.;<br />
Fetherstonhaugh & Co., Box 11560, Suite<br />
2200, 650 West Georgia Street, Vancouver,<br />
British Columbia V6B 4N8 (CA).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG UZ VN<br />
YU ZA ZW; AP (GH GM KE LS MW SD<br />
SL SZ TZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE); OA (BF BJ CF CG CI CM GA GN<br />
GW ML MR NE SN TD TG).