section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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44/2002<br />
21728 PCT Gazette - Section I - Gazette du PCT 31 Oct/oct 2002<br />
(22) 4 Apr/avr 2002 (04.04.2002)<br />
(25) en (26) en<br />
(30) 0108999.4 10 Apr/avr 2001<br />
(10.04.2001)<br />
(30) 0127426.5 15 Nov/nov 2001<br />
(15.11.2001)<br />
GB<br />
GB<br />
(43) 31 Oct/oct 2002 (31.10.2002)<br />
(54) PYRAZOLE DERIVATIVES FOR<br />
TREATING HIV<br />
DERIVES DE PYRAZOLE POUR LE<br />
TRAITEMENT DE VIH<br />
(71) PFIZER LIMITED [GB/GB]; Ramsgate<br />
Road, Sandwich, Kent CT13 9NJ (GB).<br />
(only for / seulement pour GB)<br />
(71) PFIZER INC. [US/US]; 235 East 42nd<br />
Street, New York, NY 10017 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf GB)<br />
(72, 75) JONES, Lyn, Howard [GB/GB]; Pfizer<br />
Global Research and Development, Ramsgate<br />
Road, Sandwich, Kent CT13 9NJ (GB).<br />
MOW BRAY, Charles, Eric [GR/GB];<br />
Pfizer Global Research and Development,<br />
Ramsgate Road, Sandwich, Kent CT13 9NJ<br />
(GB). PRICE, Davis, Anthony [GB/GB];<br />
Pfizer Global Research and Development,<br />
Ramsgate Road, Sandwich, Kent CT13 9NJ<br />
(GB). SELBY, Matthew, Duncan [GB/GB];<br />
Pfizer Global Research and Development,<br />
Ramsgate Road, Sandwich, Kent CT13 9NJ<br />
(GB). STUPPLE, Paul, Anthony [GB/GB];<br />
Pfizer Global Research and Development,<br />
Ramsgate Road, Sandwich, Kent CT13 9NJ<br />
(GB).<br />
(74) LANE, Graham, Mark et al. / etc.; Pfizer<br />
Limited, Ramsgate Road, Sandwich, Kent<br />
CT13 9NJ (GB).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ OM PH PL PT RO<br />
RU SD SE SG SI SK SL TJ TM TN TR TT<br />
TZ UA UG US UZ VN YU ZA ZM ZW.<br />
(84)AP(GHGMKELSMWMZSDSLSZTZ<br />
UG ZM ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE TR);<br />
OA(BFBJCFCGCICMGAGNGQGW<br />
ML MR NE SN TD TG).<br />
(51) 7 C07D 233/26, A61K 31/4164, A61P 43/00,<br />
C07D 405/12, 409/12<br />
(11) WO 02/085861<br />
(21) PCT/US02/12647<br />
(13) A1<br />
(22) 19 Apr/avr 2002 (19.04.2002)<br />
(25) en (26) en<br />
(30) 09/838,551 19 Apr/avr 2001<br />
(19.04.2001)<br />
US<br />
(43) 31 Oct/oct 2002 (31.10.2002)<br />
(54) IMIDAZOLIDINE COMPOUNDS AND<br />
THEIR USE AS CXCR3 ANTAGONISTS<br />
COMPOSES D’IMIDAZOLIDINE ET<br />
LEUR UTILISATION COMME ANTA-<br />
GONISTES DE CXCR3<br />
(63) US 09/838,551 (CON)<br />
19 Apr/avr 2001 (19.04.2001)<br />
(71) MILLENNIUM PHARMACEUTICALS,<br />
INC. [US/US]; 75 Sidney Street, Cambridge,<br />
MA 02139 (US). KYOWA HAKKO KO-<br />
GYO., LTD. [JP/JP]; 1-6-1 Ohtemachi,<br />
Chiyoda-ku, Tokyo 100-8185 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(71) OHSHIMA, Etsuo [JP/JP]; 2-223, Edogawadai-Nishi,<br />
Nagareyama-shi, Chiba (JP).<br />
(only for / seulement pour US)<br />
(72, 75) SONE, Hiroki [JP/JP]; 1188 Shimotogari,<br />
Nagizumi-cho, Sunto-gun, Shizuoka<br />
(JP). KOTERA, Osamu [JP/JP]; 1064-11,<br />
Shimotogari, Nagaizumi-cho, Sunto-gun,<br />
Shizuoka (JP). KOMATSU, Rie [JP/JP];<br />
393-2, Nameri, Nagaizumi-cho, Sunto-gun,<br />
Shizuoka (JP). LAROSA, Gregory, J.<br />
[US/US]; 16 Alameda Road, W. Roxbury,<br />
MA 02132 (US). LULY,Jay,R.[US/US]; 24<br />
Damien Road, Wellesley, MA 02181 (US).<br />
(74) CARROLL, Alice, O. et al. / etc.; Hamilton,<br />
Brook, Smith & Reynolds, P.C., 530 Virginia<br />
Road, P.O. Box 9133, Concord, MA 01742-<br />
9133 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ OM PH PL PT RO<br />
RU SD SE SG SI SK SL TJ TM TN TR TT<br />
TZ UA UG US UZ VN YU ZA ZM ZW.<br />
(84)AP(GHGMKELSMWMZSDSLSZTZ<br />
UG ZM ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE TR);<br />
OA(BFBJCFCGCICMGAGNGQGW<br />
ML MR NE SN TD TG).<br />
Published / Publiée : (c)<br />
(51) 7 C07D 233/26, A61K 31/4164, A61P 29/00<br />
(11) WO 02/085862<br />
(21) PCT/US02/12650<br />
(13) A1<br />
(22) 19 Apr/avr 2002 (19.04.2002)<br />
(25) en (26) en<br />
(30) 09/838,657 19 Apr/avr 2001<br />
(19.04.2001)<br />
US<br />
(43) 31 Oct/oct 2002 (31.10.2002)<br />
(54) IMIDAZOLIDINE DERIVATIVES AS<br />
CHEMOKINE RECEPTOR MODULA-<br />
TORS<br />
DERIVES D’IMIDAZOLIDINE EN<br />
TANT QUE MODULATEURS DE RE-<br />
CEPTEUR DE CHIMIOKINE<br />
(63) US 09/838,657 (CON)<br />
19 Apr/avr 2001 (19.04.2001)<br />
(71) MILLENNIUM PHARMACEUTICALS,<br />
INC. [US/US]; 75 Sidney Street, Cambridge,<br />
MA 02139 (US). KYOWA HAKKO KO-<br />
GYO CO., LTD. [JP/JP]; 1-6-1, Ohtemachi,<br />
Chiyoda-ku, Tokyo 100-8185 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) OHSHIMA, Etsuo [JP/JP]; 2-223, Edogawadai-Nishi,<br />
Nagareyama-shi, Chiba (JP).<br />
SONE, Hiroki [JP/JP]; 1188 Shimotogari,<br />
Nagaizumi-cho, Sunto-gun, Shizuoka<br />
(JP). KOTERA, Osamu [JP/JP]; 1064-11,<br />
Shimotogari, Nagaizumi-cho, Sunto-gun,<br />
Shizuoka (JP). KOMATSU, Rie [JP/JP];<br />
393-2, Nameri, Nagaizumi-cho, Sunto-gun,<br />
Shizuoka (JP). LAROSA, Gregory, J.<br />
[US/US]; 16 Alameda Road, W. Roxbury,<br />
MA 02132 (US). LULY,Jay,R.[US/US]; 24<br />
Damien Road, Wellesley, MA 02181 (US).<br />
(74) CARROLL, Alice, O. et al. / etc.; Hamilton,<br />
Brook, Smith & Reynolds, P.C., 530 Virginia<br />
Road, P.O. Box 9133, Concord, MA 01742-<br />
9133 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ OM PH PL PT RO<br />
RU SD SE SG SI SK SL TJ TM TN TR TT<br />
TZ UA UG US UZ VN YU ZA ZM ZW.<br />
(84)AP(GHGMKELSMWMZSDSLSZTZ<br />
UG ZM ZW); EA (AM AZ BY KG KZ MD<br />
RUTJTM);EP(ATBECHCYDEDKES<br />
FI FR GB GR IE IT LU MC NL PT SE TR);<br />
OA(BFBJCFCGCICMGAGNGQGW<br />
ML MR NE SN TD TG).<br />
(51) 7 C07D 233/54, 405/12, A61K 31/415 //<br />
(C07D 405/12, 307:00, 233:00)<br />
(11) WO 02/085863 (13) A1<br />
(21) PCT/FR02/01411<br />
(22) 24 Apr/avr 2002 (24.04.2002)<br />
(25) fr (26) fr<br />
(30) 01/05497 24 Apr/avr 2001<br />
(24.04.2001)<br />
FR<br />
(43) 31 Oct/oct 2002 (31.10.2002)<br />
(54) NOVEL COMPOUNDS OF THE FAM-<br />
ILY OF 3-ALKYL-(4,5 DIPHENYL-IM-<br />
IDAZOL-1-YL) AND THEIR USE AS<br />
SOOTHING AGENTS<br />
COMPOSES DE LA FAMILLE DES<br />
3-ALKYL-(4, 5 DIPHENYL-IMIDA-<br />
ZOL-1-YL) ET LEUR UTILISATION<br />
COMME APAISANTS<br />
(71) L’OREAL [FR/FR]; 14, rue Royal, F-75008<br />
Paris (FR).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) GALEY, Jean-Baptiste [FR/FR]; 12,<br />
rue Ch.-Dordain, F-93600 Aulnay-sous-Bois<br />
(FR). DALKO, Maria [FR/FR]; 16, Résidence<br />
du Château de Courcelles, F-91190<br />
Gif sur Yvette (FR). MAHE, Yann [FR/FR];<br />
36, avenue de l’Epargne, F-91390 Morsang-sur-Orge<br />
(FR). DUMATS, Jacqueline<br />
[FR/FR]; 13, rue Ambroise Croizat, F-93420<br />
Villepinte (FR).<br />
(74) L’OREAL; Myriam ALLAB-DPI, 6, rue<br />
Bertrand Sincholle, F-92585 Clichy Cedex<br />
(FR).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ OM PH PL PT RO<br />
RU SD SE SG SI SK SL TJ TM TN TR TT<br />
TZ UA UG US UZ VN YU ZA ZM ZW.<br />
(84)AP(GHGMKELSMWMZSDSLSZTZ<br />
UG ZM ZW); EA (AM AZ BY KG KZ MD<br />
RUTJTM);EP(ATBECHCYDEDKES<br />
FI FR GB GR IE IT LU MC NL PT SE TR);<br />
OA(BFBJCFCGCICMGAGNGQGW<br />
ML MR NE SN TD TG).
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