section 1 - World Intellectual Property Organization

44/2002
31 Oct/oct 2002 PCT Gazette - Section I - Gazette du PCT 21733
(51) 7 C07D 311/56, A61K 31/37
(11) WO 02/085882 (13) A1
(21) PCT/US02/13163
(22) 24 Apr/avr 2002 (24.04.2002)
(25) en (26) en
(30) 60/286,079 24 Apr/avr 2001 US
(24.04.2001)
(43) 31 Oct/oct 2002 (31.10.2002)
(54) COUMARIN DERIVATIVES TO BE
USED AS ANTICOAGULANTS
DERIVES DE COUMARINE POUVANT
ETRE UTILISES COMME ANTICOA-
GULANTS
(71) ARXY THERAPEUTICS [US/US]; Suite
F, 2255 Martin Avenue, Santa Clara, CA
95050 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) DRUZGALA, Pascal [FR/US]; 1512
Mission Boulevard, Santa Rosa, CA 95409
(US). ZHANG, Xiaoming [US/US]; 2290
Cervantes Way, Campbell, CA 95008 (US).
PFISTER, Jurg, R. [US/US]; 1500 Oak
Avenue, Los Altos, CA 94024 (US).
(74) SALIWANCHIK, David, R.; Saliwanchik,
Lloyd & Saliwanchik, 2421 N.W. 41st Street,
Suite A-1, Gainesville, FL 32606 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ OM PH PL PT RO
RU SD SE SG SI SK SL TJ TM TN TR TT
TZ UA UG US UZ VN YU ZA ZM ZW.
(84)AP(GHGMKELSMWMZSDSLSZTZ
UG ZM ZW); EA (AM AZ BY KG KZ MD
RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE TR);
OA(BFBJCFCGCICMGAGNGQGW
ML MR NE SN TD TG).
Published / Publiée : (c)
(51) 7 C07D 313/12, A61K 31/335, C07C 259/06,
C07D 209/88, A61P 35/00
(11) WO 02/085883
(21) PCT/EP02/04349
(13) A1
(22) 19 Apr/avr 2002 (19.04.2002)
(25) en (26) en
(30) 01109428.1 23 Apr/avr 2001
(23.04.2001)
EP
(43) 31 Oct/oct 2002 (31.10.2002)
(54) TRICYCLIC ALKYLHYDROXAM-
ATES, THEIR PREPARATION AND
THEIR USE AS CELL PROLIFERA-
TION INHIBITORS
ALKYLHYDROXAMATES TRICY-
CLIQUES, PROCEDES DE PREPARA-
TION ET D’UTILISATION DE CES
DERNIERS EN TANT QU’INHIBI-
TEURS DE LA PROLIFERATION CEL-
LULAIRE
(71) F. HOFFMANN-LA ROCHE AG
[CH/CH]; 124 Grenzacherstrasse, CH-4070
Basle (CH).
(72) GROSSMANN, Adelbert; Heimgartenstrasse
1, 82436 Eglfing (DE). VON DER
SAAL, Wolfgang; Wachenbergstrasse 9,
69469 Weinheim (DE). SATTELKAU,
Tim; Renzstrasse 1, 68161 Mannheim (DE).
TIBES, Ulrich; Am Sandberg 102, D-60599
Frankfurt (DE).
(74) SCHREINER, Siegfried; Roche Diagnostics
GmbH, Patent Department (TR-E), P.O.
Box 11 52, 82372 Penzberg (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ OM PH PL PT RO
RU SD SE SG SI SK SL TJ TM TN TR TT
TZ UA UG UZ VN YU ZA ZM ZW.
(84)AP(GHGMKELSMWMZSDSLSZTZ
UG ZM ZW); EA (AM AZ BY KG KZ MD
RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE TR);
OA(BFBJCFCGCICMGAGNGQGW
ML MR NE SN TD TG).
(51) 7 C07D 327/10
(11) WO 02/085884 (13) A1
(21) PCT/IN01/00092
(22) 24 Apr/avr 2001 (24.04.2001)
(25) en (26) en
(43) 31 Oct/oct 2002 (31.10.2002)
(54) A PROCESS FOR THE STERE-
OSELECTIVE PREPARATION OF
INSECTICIDE 6,7,8,9,10-10-HEX-
AHALO-1,5,5A,6,9,9A-HEXAHY-
DRO-6,9-METHANO-2,4,3-BENZO-
DIOXATHIEPIN-3-OXIDE
PROCESSUS DE PREPARA-
TION STEREOSELECTIVE D’IN-
SECTICIDE 6,7,8,9,10-10-HEXA-
HALO-1,5,5A,6,9,9A-HEXAHY-
DRO-6,9-METHANO-2,4,3-BENZO-
DIOXATHIEPIN-3-OXYDE
(71) EXCEL INDUSTRIES LIMITED [IN/IN];
184/87, Swami Vivekanand Road, Jogeshwari,
Mumbai 400102, Maharashtra (IN).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) SHROFF, Ashwin, Champraj [IN/IN];
Excel Industries Limited, 184/87, Swami
Vivekanand Road, Jogeshwari, Mumbai
400102, Maharashtra (IN). PUROHIT, Abhijit,
Premvallabh [IN/IN]; Excel Industries
Limited, 184/87, Swami Vivekanand Road,
Jogeshwari, Mumbai 400102, Maharashtra
(IN). VADORARIA, Sanjay, Dhirajlal
[IN/IN]; Excel Industries Limited, 184/87,
Swami Vivekanand Road, Jogeshwari, Mumbai
400102, Maharashtra (IN).
(74) DEPENNING, Robert, G. et al. / etc.; Depenning
& Depenning, Alaknanda, 16 Nepean
Sea Road, Mumbai 400 036, Maharashtra
(IN).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EE ES FI GB GD GE GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC
LK LR LS LT LU LV MA MD MG MK MN
MW MX MZ NO NZ PL PT RO RU SD SE
SG SI SK SL TJ TM TR TT TZ UA UG US
UZ VN YU ZA ZW.
(84)AP(GHGMKELSMWMZSDSLSZTZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BFBJCFCGCICMGAGNGWMLMR
NE SN TD TG).
(51) 7 C07D 401/04, 401/14, 407/04, 403/04,
413/14, 237/32, 405/04, A61K 31/502, A61P
11/06
(11) WO 02/085885
(21) PCT/EP02/04494
(13) A1
(22) 24 Apr/avr 2002 (24.04.2002)
(25) en (26) en
(30) 01110227.4 25 Apr/avr 2001
(25.04.2001)
EP
(43) 31 Oct/oct 2002 (31.10.2002)
(54) PIPERAZINO-DERIVATIVES
THEIR USE AS PDE4 INHIBITOR
AND
DERIVES PIPERAZINES ET LEUR
UTILISATION EN TANT QU’INHIBI-
TEURS DE PDE4
(71) ALTANA PHARMA AG [DE/DE];
Byk-Gulden-Strasse
(DE).
2, 78467 Konstanz
(for all designated States except / pour tous
les États désignés sauf US)
(72) HATZELMANN, Armin; Alter Wall 3,
78467 Konstanz (DE). BUNDSCHUH,
Daniela; Rheingutstrasse 17, 78462 Konstanz
(DE). BARSIG, Johannes; Bleichenweg 11,
78467 Konstanz (DE). KLEY, Hans-Peter;
Im Weinberg 3b, 78476 Allensbach (DE).
(72, 75) GRUNDLER, Gerhard [DE/DE];
Meersburger Str. 4, 78464 Konstanz (DE).
SCHMIDT, Beate [DE/DE]; Allensbacher
Str. 5, 78476 Allensbach (DE). STERK,
Geert, Jan [NL/NL]; Stadhouderslaan 38,
NL-3583 JJ Utrecht (NL).
(74) ALTANA PHARMA AG; Byk-Gulden-
Strasse 2, 78467 Konstanz (DE).
(81) AE AL AU BA BG BR CA CN CO CU CZ
DZ EC EE GE HR HU ID IL IN IS JP KR LT
LV MA MK MX NO NZ PH PL RO SG SI
SK TN UA US VN YU ZA ZW.
(84) EA (AM AZ BY KG KZ MD RU TJ TM); EP
(ATBECHCYDEDKESFIFRGBGRIE
IT LU MC NL PT SE TR).
(51) 7 C07D 401/04, 413/04, A61P 31/04, A61K
31/47
(11) WO 02/085886
(21) PCT/IN02/00111
(13) A2
(22) 24 Apr/avr 2002 (24.04.2002)
(25) en (26) en
(30) 60/286,291 25 Apr/avr 2001
(25.04.2001)
US
(30) 60/287,104 27 Apr/avr 2001
(27.04.2001)
US
(30) 60/341,365 13 Dec/déc 2001
(13.12.2001)
US
(43) 31 Oct/oct 2002 (31.10.2002)
(54) NEW GENERATION TRIPLE-TARGET-
ING, CHIRAL, BROAD-SPECTRUM
ANTIMICROBIAL 7-SUBSTITUTED
PIPERIDINO-QUINOLONE CAR-
BOXYLIC ACID DERIVATIVES, THEIR
PREPARATION, COMPOSITIONS AND
USE AS MEDICAMENTS
NOUVELLE GENERATION DE DE-
RIVES CHIRAUX D’ACIDE PIPERI-
DINO-QUINOLONE CARBOXYLIQUE