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PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO

PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO

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01/<strong>2002</strong><br />

118 <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 3 Jan/jan <strong>2002</strong><br />

417/12, A61K 31/433, 31/4535, C07D<br />

333/40, 317/58<br />

(11) WO 02/00606 (13) A1<br />

(21) <strong>PCT</strong>/JP01/05541<br />

(22) 28 Jun/juin 2001 (28.06.2001)<br />

(25) ja (26) ja<br />

(30) 2000-200118 28 Jun/juin 2000 JP<br />

(28.06.2000)<br />

(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />

(54) BIPHENYL COMPOUND<br />

COMPOSE BIPHENYLE<br />

(71) TAKEDA CHEMICAL INDUSTRIES,<br />

LTD. [JP/JP]; 1-1, Doshomachi 4-chome,<br />

Chuo-ku, Osaka-shi, Osaka 541-0045 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) TARUI, Naoki [JP/JP]; 6-1, Mitsugarasu<br />

1-chome, Nara-shi, Nara 631-0061<br />

(JP). SANTO, Takashi [JP/JP]; 2-14-401,<br />

Motoyamaminamimachi 9-chome, Higashinada-ku,<br />

Kobe-shi, Hyogo 658-0015<br />

(JP). WATANABE, Hiroyuki [JP/JP];<br />

26-3-907, Kojidai 2-chome, Nishi-ku,<br />

Kobe-shi, Hyogo 651-2273 (JP). ASO,<br />

Kazuyoshi [JP/JP]; 10-5-307, Kamihamuro<br />

1-chome, Takatsuki-shi, Osaka<br />

569-1044 (JP). MIWA, Tetsuo [JP/JP];<br />

9-31-404, Fukaeminamimachi 1-chome, Higashinada-ku,<br />

Kobe-shi, Hyogo 658-0022<br />

(JP). TAKEKAWA, Shiro [JP/JP]; B-305,<br />

5-3, Umezono 2-chome, Tsukuba-shi, Ibaraki<br />

305-0045 (JP).<br />

(74) AOYAMA, Tamotsu et al. / etc.; AOYAMA<br />

& PARTNERS, IMP Building, 3-7, Shiromi<br />

1-chome, Chuo-ku, Osaka-shi, Osaka<br />

540-0001 (JP).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS JP KE KG KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07C 235/34, 235/60, 321/20, 321/28,<br />

327/44, A01N 37/18, 37/34, 43/08, 43/10,<br />

43/12, 43/30, 43/32, 43/40, 43/52, 43/54,<br />

43/56, 43/60, 43/78, 47/22, C07D 319/18,<br />

333/24, 333/28, 307/54, 307/56, 213/54,<br />

213/61, 239/28, 241/12, 277/30, 231/12,<br />

277/64, 333/54, 333/60, 307/79, 235/16,<br />

285/14<br />

(11) WO 02/00607<br />

(21) <strong>PCT</strong>/JP01/05037<br />

(13) A1<br />

(22) 13 Jun/juin 2001 (13.06.2001)<br />

(25) ja (26) ja<br />

(30) 2000-195649 29 Jun/juin 2000<br />

(29.06.2000)<br />

JP<br />

(30) 2000-378666 13 Dec/déc 2000<br />

(13.12.2000)<br />

JP<br />

(30) 2001-096096 29 Mar/mar 2001<br />

(29.03.2001)<br />

JP<br />

(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />

(54) AMIDE COMPOUNDS AND USE<br />

THEREOF<br />

COMPOSES D’AMIDES ET UTILISA-<br />

TION ASSOCIEE<br />

(71) SUMITOMO CHEMICAL COMPANY,<br />

LIMITED [JP/JP]; 5-33, Kitahama 4-chome,<br />

Chuo-ku, Osaka-shi, Osaka 541-8550 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) SAKAGUCHI, Hiroshi [JP/JP]; 2-11-8-<br />

407, Sonehigashi-machi, Toyonaka-shi, Osaka<br />

561-0802 (JP).<br />

(74) JINNO, Naoyoshi et al. / etc.; c/o Sumitomo<br />

Chemical Intellectual Property Service, Limited,<br />

5-33, Kitahama 4-chome, Chuo-ku, Osaka-shi,<br />

Osaka 541-8550 (JP).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS KE KG KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 C07C 255/46, 49/697, 45/67<br />

(11) WO 02/00608 (13) A2<br />

(21) <strong>PCT</strong>/EP01/06578<br />

(22) 11 Jun/juin 2001 (11.06.2001)<br />

(25) en (26) en<br />

(30) 60/210,768 12 Jun/juin 2000 US<br />

(12.06.2000)<br />

(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />

(54) A PROCESS FOR THE PREPA-<br />

RATION OF 2,2-DIMETHYL-5-(4-<br />

CHLOROBENZYL) CYCLOPEN-<br />

TANONE AND AN INTERMEDIATE<br />

USEFUL THEREFOR<br />

PROCEDE DE PREPARATION D’UN<br />

2,2-DIMETHYL-5-(4-CHLOROBEN-<br />

ZYL) CYCLOPENTANONE ET PRO-<br />

DUITS INTERMEDIAIRES UTILISES<br />

POUR CELUI-CI<br />

(71) BASF AKTIENGESELLSCHAFT<br />

[DE/DE]; 67056 Ludwigshafen (DE).<br />

(72) WONG, George, S., K.; 61 Hawthorne<br />

Place, Summit, NJ 07901 (US).<br />

(74) BASF AKTIENGESELLSCHAFT; 67056<br />

Ludwigshafen (DE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS JP KE KG KP KR KZ<br />

LC LK LR LS LT LU LV MA MD MG MK<br />

MN MW MX MZ NO NZ PL PT RO RU SD<br />

SE SG SI SK SL TJ TM TR TT TZ UA UG<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 C07C 265/10, 233/32, 271/24, 239/14,<br />

225/20, 217/74, 69/757, 61/00, A61K<br />

31/192, 31/16, A61P 29/00, 11/00<br />

(11) WO 02/00609 (13) A2<br />

(21) <strong>PCT</strong>/IT01/00311<br />

(22) 15 Jun/juin 2001 (15.06.2001)<br />

(25) en (26) en<br />

(30) RM2000A000342 23 Jun/juin 2000 IT<br />

(23.06.2000)<br />

(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />

(54) 2,6,7-SUBSTITUTED TETRALINES<br />

USEFUL FOR THE PREPARATION OF<br />

MEDICAMENTS WITH PHOSPHODI-<br />

ESTERASE IV INHIBITORY ACTIVITY<br />

TETRALINES 2,6,7-SUBSTITUEES<br />

CONVENANT A L’ELABORATION DE<br />

MEDICAMENTS INHIBITEURS DE LA<br />

PHOSPHODIESTERASE IV<br />

(71) SIGMA-TAU INDUSTRIE FARMACEU-<br />

TICHE RIUNITE S.P.A. [IT/IT]; Viale<br />

Skakespeare, 47, I-00144 Rome (IT).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FANTO’, Nicola [IT/IT]; Via Giulio<br />

Cesare, 3, I-00040 Pomezia (IT). TINTI,<br />

Maria, Ornella [IT/IT]; Via Ernesto Basile,<br />

81, I-00182 Rome (IT).<br />

(74) SPADARO, Marco; c/o Sigma-Tau Industrie<br />

Farmaceutiche Riunite S.p.A., Via Pontina,<br />

Km. 30,400, I-00040 Pomezia (IT).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS JP KE KG KP KR KZ<br />

LC LK LR LS LT LU LV MA MD MG MK<br />

MN MW MX MZ NO NZ PL PT RO RU SD<br />

SE SG SI SK SL TJ TM TR TT TZ UA UG<br />

US UZ VN YU ZA ZW.<br />

Declarations / Déclarations :<br />

(s) for the following designations / pour les<br />

désignations suivantes : AE AG AL AM AT AU<br />

AZ BA BB BG BR BY BZ CA CH CN CO CR CU<br />

CZ DE DK DM DZ EC EE ES FI GB GD GE GH<br />

GM HR HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI SK SL<br />

TJ TM TR TT TZ UA UG UZ VN YU ZA ZW AP<br />

(GH GM KE LS MW MZ SD SL SZ TZ UG ZW)<br />

EA (AM AZ BY KG KZ MD RU TJ TM) EP (AT<br />

BE CH CY DE DK ES FI FR GB GR IE IT LU<br />

MC NL PT SE TR) OA (BF BJ CF CG CI CM GA<br />

GN GW ML MR NE SN TD TG)<br />

(t) for the following designation / pour la<br />

désignation suivante : US<br />

(u) for / pour US only / seulement<br />

(51) 7 C07C 271/10, C08F 220/24, 290/12, B01F<br />

17/00, G03G 9/13, C08F 8/30<br />

(11) WO 02/00610<br />

(21) <strong>PCT</strong>/US00/32385<br />

(13) A1<br />

(22) 28 <strong>No</strong>v/nov 2000 (28.11.2000)<br />

(25) en (26) en<br />

(30) 09/605,211 28 Jun/juin 2000<br />

(28.06.2000)<br />

US<br />

(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />

(54) FLUOROALKYLOXY DISPERSANT<br />

DISPERSANT FLUOROALKYLOXY<br />

(71) 3M INNOVATIVE PROPERTIES COM-<br />

PANY [US/US]; 3M Center, P.O. Box 33427,<br />

Saint Paul, MN 55133-3427 (US).

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