PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO

01/2002
122 PCT Gazette - Section I - Gazette du PCT 3 Jan/jan 2002
(43) 3 Jan/jan 2002 (03.01.2002)
(54) ARYL FUSED SUBSTITUTED 4-OXY-
PYRIDINES
4-OXY-PYRIDINES SUBSTITUEES A
FUSION ARYLE
(71) NEUROGEN CORPORATION [US/US];
35 Northeast Industrial Road, Branford, CT
06405 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) CAI, Guolin [US/US]; 2382 White
Chapel Place, Thousand Oaks, CA 91362
(US). ALBAUGH, Pamela [US/US]; 10475
Trebah Circle, Carmel, IN 46032 (US).
YUAN, Jun [US/US]; 40 Spruce Hill Drive,
Guilford, CT 06437 (US).
(74) SARUSSI, Steven, J.; McDonnell Boehnen
Hulbert & Berghoff, Suite 3200, 300 South
Wacker Drive, Chicago, IL 60606 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EE ES FI GB GD GE GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC
LK LR LS LT LU LV MA MD MG MK MN
MW MX MZ NO NZ PL PT RO RU SD SE
SG SI SK SL TJ TM TR TT TZ UA UG US
UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 215/22, A61K 31/47, A61P 35/00,
C07D 401/12
(11) WO 02/00624 (13) A2
(21) PCT/US01/10849
(22) 12 Jun/juin 2001 (12.06.2001)
(25) en (26) en
(30) 60/213,380 23 Jun/juin 2000 US
(23.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) METHODS AND COMPOUNDS FOR
INHIBITING MRP1
PROCEDES ET COMPOSES D’INHIBI-
TION DU MRP1
(71) ELI LILLY AND COMPANY [US/US];
Lilly Corporate Center, DC 1104, Indianapolis,
IN 46285 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BONJOUKLIAN, Rosanne [US/US];
318 Dominion Drive, Zionsville, IN 46077
(US). YORK, Jeremy, Schulenburg
[US/US]; 8866 Doral East Drive, Apartment
F, Indianapolis, IN 46250 (US).
(74) LEE, Kirby, W. et al. / etc.; Lilly Corporate
Center, DC1104, Indianapolis, IN 46285
(US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT TZ UA UG
US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 215/28
(11) WO 02/00625 (13) A2
(21) PCT/EP01/07258
(22) 26 Jun/juin 2001 (26.06.2001)
(25) en (26) en
(30) 1274/00 28 Jun/juin 2000 CH
(28.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) PROCESS FOR THE PREPARATION OF
QUINOLINE DERIVATIVES
PROCEDE DE PREPARATION DE DE-
RIVES DE QUINOLINE
(71) SYNGENTA PARTICIPATIONS AG
[CH/CH]; Schwarzwaldallee 215, CH-4058
Basel (CH).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) SCHEUZGER, Karl [CH/CH]; St.
Gallerring 189, CH-4054 Basel (CH).
(74) BASTIAN, Werner; c/o Syngenta Participations
AG, Intellectual Property, P.O. Box,
CH-4002 Basel (CH).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT TZ UA UG
US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 223/16, A61K 31/55, A61P 13/00,
C07D 401/06, 243/12, 495/04
(11) WO 02/00626 (13) A1
(21) PCT/GB01/02737
(22) 21 Jun/juin 2001 (21.06.2001)
(25) en (26) en
(30) 0015601.8 26 Jun/juin 2000 GB
(26.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) FUSED AZEPINE DERIVATIVES
AND THEIR USE AS ANTIDIURETIC
AGENTS
DERIVES D’AZEPINE FUSIONNES ET
LEURS UTILISATIONS COMME ANTI-
DIURETIQUES
(71) FERRING B.V. [NL/NL]; Polaris Avenue
144, NL-2132 JX Hoofddorp (NL).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ASHWORTH, Doreen, Mary
[GB/GB]; 10 The Glades, Locks Heath,
Southampton, Hampshire SO31 6UY (GB).
PITT, Gary, Robert, William [GB/GB];
18 Kingfishers, Shipton-Bellinger, Tidworth,
Hampshire SP9 7US (GB). HUDSON, Peter
[GB/GB]; 12 Tottehale Close, North Baddesley,
Southampton, Hampshire SO52 9NQ
(GB). YEA, Christopher, Martyn [GB/GB];
11 Gaston Gardens, Romsey, Hampshire
SO51 7RZ (GB). FRANKLIN, Richard,
Jeremy [GB/GB]; 208 Finchampstead Road,
Wokingham, Berkshire RG40 3HB (GB).
SEMPLE, Graeme [GB/SE]; AstraZeneca
R & D Molndal, S-431 83 Molndal (SE).
(74) GEERING, Keith, Edwin; Reddie & Grose,
16 Theobalds Road, London WC1X 8PL
(GB).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EE ES FI GB GD GE GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC
LK LR LS LT LU LV MA MD MG MK MN
MW MX MZ NO NZ PL PT RO RU SD SE
SG SI SK SL TJ TM TR TT TZ UA UG US
UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 231/12, A61K 31/415
(11) WO 02/00627 (13) A1
(21) PCT/TR01/00025
(22) 26 Jun/juin 2001 (26.06.2001)
(25) en (26) en
(30) 2000/01872 26 Jun/juin 2000 TR
(26.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) A CRYSTALLINE FORM OF CELE-
COXIB
FORME CRISTALLINE DE CELE-
COXIB
(71) FAKO ILACLARI A.S. [TR/TR];
Buyukdere Caddesi No: 205, 4. Levent,
80650 Istanbul (TR).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) GUNDUZ, A., Halit [TR/TR]; FAKO
ILACLARI A.S., Buyukdere Caddesi
No:205, 4. Levent, 80650 Istanbul (TR).
GOKTEPE, Mehmet [TR/TR]; FAKO
ILACLARI A.S., Buyukdere Caddesi
No:205, 4. Levent, 80650 Istanbul (TR). BA-
HAR, Mehmet [TR/TR]; FAKO ILACLARI
A.S., Buyukdere Caddesi No:205, 4. Levent,
80650 Istanbul (TR).
(74) AKSOY DANISMANLIK GIDA TEK-
STIL ITHALAT IHRACAT TICARET
LTD. STI.; 1. Cadde 5/6, Bahcelievler,
06500 Ankara (TR).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).