PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
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01/<strong>2002</strong><br />
42 <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 3 Jan/jan <strong>2002</strong><br />
(30) 60/223,212 4 Aug/août 2000 US<br />
(04.08.2000)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) RAPIDLY EXPANDING COMPOSI-<br />
TION FOR GASTRIC RETENTION<br />
AND CONTROLLED RELEASE<br />
OF THERAPEUTIC AGENTS, AND<br />
DOSAGE FORMS INCLUDING THE<br />
COMPOSITION<br />
COMPOSITION A EXPANSION RA-<br />
PIDE POUR RETENTION GAS-<br />
TRIQUE ET LIBERATION REGULEE<br />
D’AGENTS THERAPEUTIQUES, ET<br />
FORMES POSOLOGIQUES RENFER-<br />
MANT CETTE COMPOSITION<br />
(71) TEVA PHARMACEUTICAL INDUS-<br />
TRIES LTD. [IL/IL]; 5 Basel Street, P.O.<br />
Box 3190, 49131 Petah Tiqva (IL).<br />
(for all designated States except / pour tous<br />
les États désignés sauf BB US)<br />
(71) TEVA PHARMACEUTICALS USA, INC.<br />
[US/US]; 1090 Horsham Road, P.O. Box<br />
1090, <strong>No</strong>rth Wales, PA 19454-1090 (US).<br />
(only for / seulement pour BB)<br />
(72, 75) FLESHNER-BARAK, Moshe [IL/IL];<br />
Hefetz Mordechai 15, Petach Tikva (IL).<br />
LERNER, E., Itzhak [IL/IL]; Wolfson 32,<br />
Petach Tikva (IL). ROSENBERGER, Vered<br />
[IL/IL]; Ms. Landau 3, Givat, Masuah,<br />
Jerusalem (IL). DAHAN, Mazal [IL/IL];<br />
Moshe Sharet Street 8/10, 96920 Jerusalem<br />
(IL). IMAKOV, Yisrael [IL/IL]; Ha Narkiss<br />
20, Carmei Yosef (IL).<br />
(74) BRAINARD, Charles, R. et al. / etc.;<br />
Kenyon & Kenyon, One Broadway, New<br />
York, NY 10004 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ PL PT RO RU SD<br />
SE SG SI SK SL TJ TM TR TT TZ UA UG<br />
US UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 A61K 31/35, A61P 17/00, 17/16<br />
(11) WO 02/00214 (13) A1<br />
(21) <strong>PCT</strong>/DE01/02285<br />
(22) 20 Jun/juin 2001 (20.06.2001)<br />
(25) de (26) de<br />
(30) 100 31 457.0 28 Jun/juin 2000 DE<br />
(28.06.2000)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) FLAVONE/FLAVANONE DERIVA-<br />
TIVES FOR THE SYSTEMIC TREAT-<br />
MENT AND PROPHYLAXIS OF UV-IN-<br />
DUCED DERMATOSES<br />
DERIVES DE FLAVONE/FLAVANONE<br />
POUR LE TRAITEMENT SYSTEMA-<br />
TIQUE ET LA PROPHYLAXIE DE<br />
DERMATOSES ASSOCIEES AUX UV<br />
(71, 72) KRUTMANN, Jean [DE/DE]; Rathausplatz<br />
19, 41844 Wegberg (DE). STEGE, Helger<br />
[DE/DE]; Marie-Juchacz-Weg 41, 79111<br />
Freiburg (DE).<br />
(74) MILLER RECHTSANWÄLTE;<br />
Kaiser-Joseph-Strasse 260, Postfach 03<br />
10, 79003 Freiburg (DE).<br />
(81) AE AG AL AU BA BB BG BR BZ CA CN<br />
CO CR CU CZ DM DZ EE GD GE HR HU<br />
ID IL IN IS JP KP KR LC LK LR LT LV MA<br />
MG MK MN MX NO NZ PL RO SG SI SK<br />
SL TT UA US UZ VN YU ZA.<br />
Published / Publiée :(c)<br />
Declaration / Déclaration :<br />
(u) for / pour US only / seulement<br />
(51) 7 A61K 31/395, 31/55, 31/44, 31/40<br />
(11) WO 02/00215 (13) A1<br />
(21) <strong>PCT</strong>/US01/19958<br />
(22) 22 Jun/juin 2001 (22.06.2001)<br />
(25) en (26) en<br />
(30) 60/304,189 23 Jun/juin 2000 US<br />
(23.06.2000)<br />
(30) 60/264,695 30 Jan/jan 2001 US<br />
(30.01.2001)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) SUBTYPE SELECTIVE MELATONER-<br />
GICS<br />
MELATONERGIQUES A SELECTI-<br />
VITE DE SOUS-TYPES<br />
(71) COGNETIX, INC. [US/US]; 421 Wakara<br />
Way, Suite 201, Salt Lake City, UT 84108<br />
(US).<br />
(72) JONES, Robert, M.; 44 West Broadway<br />
#2103 South, Salt Lake City, UT 84101-3223<br />
(US).<br />
(74) IHNEN, Jeffrey, L. et al. / etc.; Rothwell,<br />
Figg, Ernst & Manbeck, P.C., 555 13th Street,<br />
N.W., Suite 701-E, Washington, DC 20004<br />
(US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ PL PT RO RU SD<br />
SE SG SI SK SL TJ TM TR TT TZ UA UG<br />
UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 A61K 31/40, A61P 9/00, C07D 209/82<br />
(11) WO 02/00216<br />
(21) <strong>PCT</strong>/US01/20760<br />
(13) A1<br />
(22) 28 Jun/juin 2001 (28.06.2001)<br />
(25) en (26) en<br />
(30) 60/214,356 28 Jun/juin 2000<br />
(28.06.2000)<br />
US<br />
(30) 60/246,358 7 <strong>No</strong>v/nov 2000<br />
(07.11.2000)<br />
US<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) CARVEDILOL<br />
CARVEDILOL<br />
(71) TEVA PHARMACEUTICAL INDUS-<br />
TRIES LTD. [IL/IL]; Basel Street 5, P.O.<br />
Box 3190, 49131 Petah Tiqva (IL).<br />
(for all designated States except / pour tous<br />
les États désignés sauf BB US)<br />
(71) TEVA PHARMACEUTICALS USA, INC.<br />
[US/US]; 1090 Horsham Road, P.O. Box<br />
1090, <strong>No</strong>rth Wales, PA 19454-1090 (US).<br />
(only for / seulement pour BB)<br />
(72, 75) HILDESHEIM, Jean [IL/IL]; Rothchild<br />
30, Mazkeret Batya (IL). FINOGUEEV,<br />
Sergey [IL/IL]; P.O. Box 3029, 90100<br />
Quiriat Arbaa 213/8 (IL). ARONHIME,<br />
Judith [IL/IL]; Hava Lutzky 9/7, Rechovot<br />
(IL). DOLITZKY, Ben-Zion [IL/IL];<br />
Lochamei Hagettaot 32, Petach Tikva (IL).<br />
BEN-VALID, Shoshana [IL/IL]; Havered<br />
Street 369/12, Sderot (IL). KOR, Ilan<br />
[IL/IL]; Ha’Tavor 131, P.O. Box 1583,<br />
Shoham (IL).<br />
(74) BRAINARD, Charles, R. et al. / etc.;<br />
Kenyon & Kenyon, One Broadway, New<br />
York, NY 10004 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ PL PT RO RU SD<br />
SE SG SI SK SL TJ TM TR TT TZ UA UG<br />
US UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 A61K 31/405, A61P 43/00, 25/00 // C07D<br />
209/34<br />
(11) WO 02/00217<br />
(21) <strong>PCT</strong>/DK01/00412<br />
(13) A1<br />
(22) 14 Jun/juin 2001 (14.06.2001)<br />
(25) en (26) en<br />
(30) PA 2000 01022 29 Jun/juin 2000<br />
(29.06.2000)<br />
DK<br />
(30) PA 2001 00394 8 Mar/mar 2001<br />
(08.03.2001)<br />
DK<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) USE OF 3-SUBSTITUTED OXINDOLE<br />
DERIVATIVES AS KCNQ POTASSIUM<br />
CHANNEL MODULATORS<br />
UTILISATION DE DERIVES D’OXIN-<br />
DOLE 3-SUBSTITUE COMME MODU-<br />
LATEURS DU CANAL POTASSIQUE<br />
KCNQ<br />
(71) NEUROSEARCH A/S [DK/DK]; 93 Pederstrupvej,<br />
DK-2750 Ballerup (DK).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) JENSEN, Bo, Skaaning [DK/DK];<br />
c/o NeuroSearch A/S, 93 Pederstrupvej,<br />
DK-2750 Ballerup (DK). SCHRØDER,<br />
Rikke, L. [DK/DK]; Julius Valentiners vej<br />
13, st. th, DK-2000 Frederiksberg (DK).<br />
STRØBÆK, Dorte [DK/DK]; c/o NeuroSearch<br />
A/S, 93 Pederstrupvej, DK-2750<br />
Ballerup (DK). OLESEN, Søren, Peter<br />
[DK/DK]; c/o NeuroSearch A/S, 93 Pederstrupvej,<br />
DK-2750 Ballerup (DK).