PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO
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01/<strong>2002</strong><br />
3 Jan/jan <strong>2002</strong> <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 135<br />
STEROÏDES 20-FLUORO-17(20)-VINY-<br />
LIQUES CONVENANT COMME INHI-<br />
BITEURS CE LA C17-20-LYASE ET DE<br />
LA 5-ALPHA REDUCTASE<br />
(71) AVENTIS PHARMACEUTICALS INC.<br />
[US/US]; Patent Dept., Route 202-206, P.O.<br />
Box 6800, Bridgewater, NJ 08807-0800 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) PEET, <strong>No</strong>rton, P. [US/US]; 50 Blue<br />
Ridge Road, <strong>No</strong>rth Andover, MA 01845<br />
(US). WEINTRAUB, Philip, M. [US/US];<br />
33 Casale Drive South, Warren, NJ 07059<br />
(US). BURKHART, Joseph, P. [US/US];<br />
701 Andrews Boulevard, Plainfield, IN 46168<br />
(US). GATES, Cynthia, A. [US/US]; 177<br />
Pemberton Street, <strong>No</strong>. 11, Cambridge, MA<br />
02140 (US).<br />
(74) MARTIN, Lawrence, L. et al. / etc.; Aventis<br />
Pharmaceuticals Inc., Route 202-206, P.O.<br />
Box 6800, Bridgewater, NJ 08807-0800 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ VN<br />
YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07J 53/00, A61K 31/565, A61P 5/30,<br />
5/36<br />
(11) WO 02/00682 (13) A1<br />
(21) <strong>PCT</strong>/EP01/04868<br />
(22) 1 May/mai 2001 (01.05.2001)<br />
(25) en (26) en<br />
(30) 00201986.7 6 Jun/juin 2000 EP<br />
(06.06.2000)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) 16, 17-CARBOCYCLIC CONDENSED<br />
STEROID COMPOUNDS HAVING SE-<br />
LECTIVE ESTROGENIC ACTIVITY<br />
COMPOSES STEROIDES CONDENSES<br />
16, 17-CARBOCYCLIQUES A ACTI-<br />
VITE OESTROGENIQUE SELECTIVE<br />
(71) AKZO NOBEL N.V. [NL/NL]; Velperweg<br />
76, NL-6824 BM Arnhem (NL).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) LOOZEN, Hubert, Jan, Jozef<br />
[NL/NL]; Meerhoek 602, NL-5403 AC<br />
Uden (NL).<br />
(74) KRAAK, Hajo; P.O. Box 20, NL-5340 BH<br />
Oss (NL).<br />
(81) AE AG AL AU BA BB BG BR BZ CA CN<br />
CO CR CU CZ DM DZ EE GD GE HR HU<br />
ID IL IN IS JP KP KR LC LK LR LT LV MA<br />
MG MK MN MX MZ NO NZ PL RO RU SG<br />
SI SK SL TR TT UA US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07K<br />
(11) WO 02/00683 (13) A2<br />
(21) <strong>PCT</strong>/US01/19969<br />
(22) 25 Jun/juin 2001 (25.06.2001)<br />
(25) en (26) en<br />
(30) 60/213,826 23 Jun/juin 2000 US<br />
(23.06.2000)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) NOVEL CHAIN-BREAKING ANTIOXI-<br />
DANTS<br />
NOUVEAUX ANTIOXYDANTS A RUP-<br />
TURE DE CHAINE<br />
(71) VANDERBILT UNIVERSITY [US/US];<br />
305 Kirkland Hall, Nashville, TN 37240<br />
(US).<br />
(72) PRATT, Derek, A.; 2114 Sharondale Drive,<br />
Nashville, TN 37215 (US). DILABIO, Gino,<br />
A.; 91 Pearson Street, Apartment 8, Aylmer,<br />
Québec J9H 6G1 (CA). VALGIMIGLA,<br />
Luca; Via Campo di Marte 51, I-47100 Forli<br />
(IT).<br />
(74) SHOUSE, Emily, A.; Waddey & Patterson,<br />
Suite 2020, 414 Union Street, Bank of America<br />
Plaza, Nashville, TN 37219 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07K 1/00<br />
(11) WO 02/00684<br />
(21) <strong>PCT</strong>/RU01/00256<br />
(13) A2<br />
(22) 26 Jun/juin 2001 (26.06.2001)<br />
(25) en (26) en<br />
(30) 2000116791 29 Jun/juin 2000<br />
(29.06.2000)<br />
RU<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) METHOD OF OBTAINING PEPTIDES<br />
WITH TISSUE-SPECIFIC ACTIVITY<br />
AND PHARMACEUTICAL COMPOSI-<br />
TIONS ON THEIR BASIS<br />
PROCEDE DE FABRICATION DE PEP-<br />
TIDES A ACTIVITE SPECIFIQUE AUX<br />
TISSUS ET COMPOSITIONS PHAR-<br />
MACEUTIQUES A BASE DE CEUX-CI<br />
(71) SANKT-PETERBURGSKAYA OB-<br />
SCHESTVENNAYA OGRANIZAT-<br />
SIYA "INSTITUT BIOREGULYAT-<br />
SII I GERONTOLOGII CZO RAMN"<br />
[RU/RU]; pr.<br />
197110 (RU).<br />
Dinamo, 3, St.Petersburg,<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) KHAVINSON, Vladimir Khatskelevich<br />
[RU/RU]; ul. Savushkina, 26-2-7,<br />
St.Petersburg, 197374 (RU).<br />
(74) SANKT-PETERBURGSKAYA OB-<br />
SCHESTVENNAYA OGRANIZAT-<br />
SIYA "INSTITUT BIOREGULYATSII<br />
I GERONTOLOGII CZO RAMN"; pr.<br />
Dinamo, 3, St.Petersburg, 197110 (RU).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA<br />
CH CN CU CZ DE DK EE ES FI GB GD GE<br />
GH GM HR HU ID IL IS JP KE KG KP KR<br />
KZ LC LK LR LS LT LU LV MD MG MK<br />
MN MW MX NO NZ PL PT RO RU SD SE<br />
SG SI SK SL TJ TM TR TT UA UG US UZ<br />
VN YU ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07K 1/00, 16/00, A61K 39/395, 45/00<br />
(11) WO 02/00685 (13) A1<br />
(21) <strong>PCT</strong>/US01/20597<br />
(22) 28 Jun/juin 2001 (28.06.2001)<br />
(25) en (26) en<br />
(30) 60/214,865 28 Jun/juin 2000 US<br />
(28.06.2000)<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) LOCALIZED DELIVERY TO A TAR-<br />
GET SURFACE<br />
ADMINISTRATION LOCALISEE SUR<br />
UNE SURFACE CIBLE<br />
(71) UNIVERSITY OF PITTSBURGH OF<br />
THE COMMONWEALTH SYSTEM OF<br />
HIGHER EDUCATION [US/US]; 200<br />
Gardner Steel Conference Center, Pittsburg,<br />
PA 15260 (US).<br />
(72) WAGNER, William, R.; 5930 Howe Street<br />
#301, Pittsburgh, PA 15232 (US). VIL-<br />
LANUEVA, Flordeliza, S.; 7146 Roycrest<br />
Place, Pittsburgh, PA 15208 (US). DEGLAU,<br />
Timothy, E.; 2215 Eagles Nest Lane, Monroeville,<br />
PA 15146 (US).<br />
(74) ANDERSON, Debra, Z.; Eckert Seamans<br />
Cherin & Mellott, LLC, 600 Grant Street -<br />
44th Floor, Pittsburgh, PA 15219 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CO CR CU CZ DE DK<br />
DM DZ EC EE ES FI GB GD GE GH GM<br />
HR HU ID IL IN IS JP KE KG KP KR KZ<br />
LC LK LR LS LT LU LV MA MD MG MK<br />
MN MW MX MZ NO NZ PL PT RO RU SD<br />
SE SG SI SK SL TJ TM TR TT TZ UA UG<br />
UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07K 5/00<br />
(11) WO 02/00686<br />
(21) <strong>PCT</strong>/US01/20045<br />
(13) A2<br />
(22) 21 Jun/juin 2001 (21.06.2001)<br />
(25) en (26) en<br />
(30) 60/213,364 23 Jun/juin 2000<br />
(23.06.2000)<br />
US<br />
(43) 3 Jan/jan <strong>2002</strong> (03.01.<strong>2002</strong>)<br />
(54) BIOELASTOMER<br />
AND BIOSENSORS<br />
NANOMACHINES