PCT/2002/1 : PCT Gazette, Weekly Issue No. 1, 2002 - WIPO

01/2002
3 Jan/jan 2002 PCT Gazette - Section I - Gazette du PCT 127
(Utility model / modèle d’utilité) ESFIFI
(Utility model / modèle d’utilité)GBGDGE
GH GM HR HU ID IL IN IS JP KE KG KP
KR KZ LC LK LR LS LT LU LV MA MD
MG MK MN MW MX MZ NO NZ PL PT
RO RU SD SE SG SI SK SK (Utility model
/ modèle d’utilité) SLTJTMTRTTTZUA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 403/06, 413/14, A61K 31/404
(11) WO 02/00646 (13) A1
(21) PCT/US01/20458
(22) 27 Jun/juin 2001 (27.06.2001)
(25) en (26) en
(30) 60/214,280 27 Jun/juin 2000 US
(27.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) FATTY ACID SYNTHASE INHIBITORS
INHIBITEURS DE SYNTHASE
D’ACIDE GRAS
(71) SMITHKLINE BEECHAM CORPO-
RATION [GB/GB]; One Franklin Plaza,
Philadelphia, PA 19103 (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) DAINES, Robert, A. [US/US]; 709
Swedeland Road, King of Prussia, PA (US).
PENDRAK, Israil [US/US]; 709 Swedeland
Road, King of Prussia, PA (US).
(74) SIMON, Soma, G. et al. / etc.; SmithKline
Beecham Corporation, Corporate Intellectual
Property, UW2220, 709 Swedeland
Road, P.O. Box 1539, King of Prussia, PA
19406-0939 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT TZ UA UG
US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 403/10, 417/10, 403/14, 417/14,
401/10, 413/10, 413/14, A61K 31/41, 31/44,
A61P 7/02
(11) WO 02/00647
(21) PCT/US01/20112
(13) A1
(22) 22 Jun/juin 2001 (22.06.2001)
(25) en (26) en
(30) 60/214,033 23 Jun/juin 2000
(23.06.2000)
US
(43) 3 Jan/jan 2002 (03.01.2002)
(54) HETEROARYL-PHENYL SUBSTI-
TUTED FACTOR XA INHIBITORS
INHIBITEURS DU FACTEUR XA A
SUBSTITUTION HETEROARYL-PHE-
NYLE
(71) DUPONT PHARMACEUTICALS COM-
PANY [US/US]; Chestnut Run Plaza, 974
Centre Road, Wilmington, DE 19805 (US).
(72) PINTO, Donald, J.P.; 425 Brentford Road,
Kennett Square, PA 19348 (US). QUAN,
Mimi, L.; 113 Venus Drive, Newark, DE
19711 (US). WOERNER, Francis, J.; 241
Cornwell Drive, Bear, DE 19701 (US).
(74) ROPER, David, J.; Dupont Pharmaceuticals
Company, Legal Patent Records Center, 1007
Market Street, Wilmington, DE 19898 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 403/12, 401/14, 409/14, 401/12,
405/12, 233/60, 405/14, A61K 31/497,
31/4439, 31/444, 31/4164, A61P 43/00,
29/00, 19/02, 19/10
(11) WO 02/00648
(21) PCT/JP01/04836
(13) A1
(22) 8 Jun/juin 2001 (08.06.2001)
(25) ja (26) ja
(30) 2000-194024 28 Jun/juin 2000
(28.06.2000)
JP
(43) 3 Jan/jan 2002 (03.01.2002)
(54) IMIDAZOLE DERIVATIVES OR SALTS
THEREOF AND DRUGS CONTAINING
THE DERIVATIVES OR THE SALTS
DERIVES IMIDAZOLE OU SELS DE
CES DERNIERS, ET MEDICAMENTS
CONTENANT LES DERIVES OU LES
SELS
(71) SSP CO., LTD. [JP/JP]; 2-12-4, NIHON-
BASHIHAMACHO, CHUO-KU, Tokyo 103-
8481 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) KONNO, Fujiko [JP/JP]; 395-202,
HIYOSHIKURA, TOMISATO-MACHI,
INBA-GUN, Chiba 286-0202 (JP). NA-
GAO, Yoshihiro [JP/JP]; 1147-18, IGO-
DAI, NARITA-SHI, Chiba 286-0035
(JP). ISOMAE, Kazuo [JP/JP]; 2-10-18,
HIRAGAGAKUENDAI, INBA-MURA,
INBA-GUN, Chiba 270-1606 (JP). OHT-
SUKA, Mari [JP/JP]; 4-7-15-704, YATSU,
NARASHINO-SHI, Chiba 275-0026
(JP). TAKAHASHI, Yoshiyuki [JP/JP];
3-5-12-106, HASHIGADAI, NARITA-SHI,
Chiba 286-0037 (JP). ISHII, Fumio [JP/JP];
3-15-106, SHIHEIMACHI, AOBA-KU,
SENDAI-SHI, Miyagi 981-0944 (JP).
HIROTA, Hiroyuki [JP/JP]; 5-8-6-406,
KARABE, NARITA-SHI, Chiba 286-0036
(JP). TAKEDA, Sunao [JP/JP]; 4-25-7-302,
KARABE, NARITA-SHI, Chiba 286-0036
(JP). KAWAMOTO, Noriyuki [JP/JP];
5-8-2-302, KARABE, NARITA-SHI, Chiba
286-0036 (JP). HONDA, Haruyoshi [JP/JP];
1049-8, NEKONA, TOMISATO-MACHI,
INBA-GUN, Chiba 286-0205 (JP). SATO,
Susumu [JP/JP]; 6-15-5, TAMATSUKURI,
NARITA-SHI, Chiba 286-0011 (JP).
(74) ARUGA, Mitsuyuki et al. / etc.; KYODO
BLDG., 3-6, NIHONBASHININGYOCHO
1-CHOME, CHUO-KU, Tokyo 103-0013
(JP).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 403/12, 409/12, 413/12, A61K
31/505, A61P 35/00
(11) WO 02/00649 (13) A1
(21) PCT/SE01/01450
(22) 21 Jun/juin 2001 (21.06.2001)
(25) en (26) en
(30) 00401842.0 28 Jun/juin 2000 EP
(28.06.2000)
(43) 3 Jan/jan 2002 (03.01.2002)
(54) SUBSTITUTED QUINAZOLINE
DERIVATIVES AND THEIR USE AS
INHIBITORS
DERIVES DE LA QUINAZOLINE SUB-
STITUES ET LEUR UTILISATION
COMME INHIBITEURS
(71) ASTRAZENECA AB [SE/SE]; S-151 85
Södertälje (SE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MORTLOCK, Andrew [GB/GB]; AstraZeneca
R & D Alderley, Alderley Park,
Macclesfield, Cheshire SK10 4TG (GB).
JUNG, Frederic [FR/FR]; AstraZeneca
Pharma, Parc Industriel Pompelle, Chemin
de Vrilly, BP 1050, F-51689 Reims Cedex 2
(FR).
(74) GLOBAL INTELLECTUAL PROPERTY
ASTRAZENCA AB; Global Intellectual
Property, S-151 85 Södertälje (SE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT TZ UA UG
US UZ VN YU ZA ZW.
Published / Publiée :(c)
Declaration / Déclaration :
(u) for / pour US only / seulement
(51) 7 C07D 403/14, A61K 31/395, A61P 31/00,
35/00, C07D 209/42, 207/34, 409/14, 401/14
(11) WO 02/00650 (13) A2
(21) PCT/US01/20334