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Bulletin 2010/45 - European Patent Office

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(C07D) I.1(2)<br />

(30) 28.03.2005 JP 2005090831<br />

15.06.2005 JP 2005174738<br />

15.07.2005 JP 2005206808<br />

09.08.2005 JP 2005230666<br />

(54) • Alkyl-3-[2-(benzo[b]thiophen-5-yl)ethoxy]-propanoate<br />

als Intermediate in der<br />

Herstellung von Azetidin-3-ol Derivativen<br />

• Alkyl-3-[2-(benzo[b]thiophen-5-yl)ethoxy]-propanoates<br />

as intermediates in<br />

the production of Azetidin-3-ol derivatives<br />

• Alkyl-3-[2-(benzo[b]thiophèn-5-yl)éthoxy]-propanoates<br />

en tant qu'intermediaires<br />

dans la production de dérivés<br />

d'azétidin-3-ol<br />

(71) TOYAMA CHEMICAL CO., LTD., 2-5, 3chome,<br />

Nishishinjuku, Shinjuku-ku, Tokyo<br />

160-0023, JP<br />

(72) Saitoh, Akihito, Toyama-shi,Toyama, JP<br />

Suzuki, Yoshiaki, Toyama-shi,Toyama, JP<br />

Yonezawa, Kenji, Toyama-shi,Toyama, JP<br />

Kawamura, Mitsuhide, Toyama-shi,Toyama,<br />

JP<br />

Kusanagi, Takahiko, Toyama-shi,Toyama, JP<br />

Nakai, Takashi, Toyama-shi,Toyama, JP<br />

(74) Blodig, Wolfgang, Wächtershäuser & Hartz<br />

<strong>Patent</strong>anwaltspartnerschaft Weinstraße 8,<br />

80333 München, DE<br />

(62) 06730075.6 / 1 864 978<br />

C07D 333/64 → (51) C07D 333/54<br />

C07D 401/04 → (51) C07D 295/12<br />

C07D 401/10 → (51) C07D 239/94<br />

(51) C07D 401/12 (11) 2 248 810 A1<br />

C07D 211/58 C07D 213/74<br />

C07D 213/75 C07D 213/81<br />

(25) Ja (26) En<br />

(21) 09713617.0 (22) 13.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) JP 2009/052401 13.02.2009<br />

(87) WO 2009/10<strong>45</strong>20 2009/35 27.08.2009<br />

(30) 18.02.2008 JP 2008036161<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

PHENOXYPYRIDIN-DERIVATS<br />

• METHOD FOR PRODUCING PHENOXY-<br />

PYRIDINE DERIVATIVE<br />

• PROCÉDÉ DE FABRICATION D'UN DÉRIVÉ<br />

DE PHÉNOXYPYRIDINE<br />

(71) Eisai R&D Management Co., Ltd., 6-10,<br />

Koishikawa 4-chome Bunkyo-ku, Tokyo 112-<br />

8088, JP<br />

(72) NAGAI, Mitsuo, Tsukuba-shi Ibaraki 300-<br />

2635, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

C07D 401/12 → (51) C07D 239/94<br />

C07D 401/14 → (51) C07D 239/94<br />

C07D 403/04 → (51) C07D 239/94<br />

C07D 403/10 → (51) C07D 239/94<br />

C07D 403/12 → (51) C07D 239/94<br />

C07D 405/10 → (51) C07D 239/94<br />

(51) C07D 405/12 (11) 2 248 811 A1<br />

A61K 31/4178 A61P 3/06<br />

A61P 3/10 A61P 9/10<br />

A61P 25/28 A61P 29/00<br />

A61P 37/00 C07D 405/14<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

C07D 409/14 C07D 413/12<br />

C07D 417/12<br />

(25) Ja (26) En<br />

(21) 09715052.8 (22) 27.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) JP 2009/000872 27.02.2009<br />

(87) WO 2009/107387 2009/36 03.09.2009<br />

(30) 29.02.2008 US 32651<br />

(54) • 2-OXOCHROMEN-DERIVAT<br />

• 2-OXOCHROMENE DERIVATIVE<br />

• DÉRIVÉ DE 2-OXOCHROMÈNE<br />

(71) Kowa Company, Ltd., 6-29, Nishiki 3-chome,<br />

Naka-ku Nagoya-shi, Aichi-ken 460-8625, JP<br />

(72) OKUDA, Ayumu, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

MATSUDA, Takayuki, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

MIURA, Toru, Higashimurayama-shi Tokyo<br />

189-0022, JP<br />

OZAWA, Hidefumi, Tokyo 103-8433, JP<br />

TOSAKA, Ayako, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

YAMAZAKI, Koichi, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

YAMAGUCHI, Yuki, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

KUROBUCHI, Sayaka, deceased, JP<br />

WATANABE, Yuuichirou, Higashimurayamashi<br />

Tokyo 189-0022, JP<br />

SHIBUYA, Kimiyuki, Higashimurayama-shi<br />

Tokyo 189-0022, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

C07D 405/12 → (51) A01N 43/40<br />

C07D 405/14 → (51) C07D 239/94<br />

C07D 405/14 → (51) C07D 405/12<br />

(51) C07D 409/12 (11) 2 248 812 A2<br />

A61K 31/192 A61P 3/10<br />

(25) En (26) En<br />

(21) 10172951.5 (22) 26.06.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 27.06.2006 JP 2006177099<br />

(54) • Kondensierte cyclische Verbindungen als<br />

GPR40 Modulatoren<br />

• Fused cyclic compounds as GPR40 receptor<br />

modulators<br />

• Composés cycliques condensés comme<br />

modulateurs du recepteur GPR40<br />

(71) Takeda Pharmaceutical Company Limited, 1-<br />

1, Doshomachi 4-chome Chuo-ku, Osakashi,<br />

Osaka 541-00<strong>45</strong>, JP<br />

(72) Yasuma, Tsuneo, Osaka 532-8686, JP<br />

Negoro, Nobuyuki, Osaka 532-8686, JP<br />

Yamashita, Masayuki, Osaka 532-8686, JP<br />

Itou, Masahiro, Osaka 532-8686, JP<br />

(74) von Kreisler Selting Werner, Deichmannhaus<br />

am Dom Bahnhofsvorplatz 1, 50667 Köln,<br />

DE<br />

(62) 07767983.5 / 2 041 123<br />

C07D 409/12 → (51) A01N 43/40<br />

C07D 409/14 → (51) C07D 405/12<br />

C07D 413/12 → (51) C07D 405/12<br />

C07D 417/12 → (51) A01N 43/40<br />

236<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>45</strong>/<strong>2010</strong>) 10.11.<strong>2010</strong><br />

C07D 417/12 → (51) C07D 405/12<br />

(51) C07D 473/10 (11) 2 248 813 A1<br />

A61K 31/522 A61P 9/08<br />

A61P 9/12 A61P 25/26<br />

(25) Ja (26) En<br />

(21) 09708909.8 (22) 06.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) JP 2009/052117 06.02.2009<br />

(87) WO 2009/099221 2009/33 13.08.2009<br />

(30) 07.02.2008 JP 2008027944<br />

(54) • VERFAHREN UND VORRICHTUNG ZUR<br />

HERSTELLUNG EINER ZUSAMMENSET-<br />

ZUNG MIT HOHEM THEOBROMINGEHALT<br />

• PRODUCTION METHOD AND PRODUC-<br />

TION DEVICE FOR COMPOSITION HAVING<br />

HIGH CONTENT OF THEOBROMINE<br />

• PROCÉDÉ DE PRODUCTION ET DISPOSI-<br />

TIF DE PRODUCTION POUR UNE COM-<br />

POSITION PRÉSENTANT UNE TENEUR<br />

ÉLEVÉE EN THÉOBROMINE<br />

(71) Meiji Seika Kaisha, Ltd., 4-16, Kyobashi 2chome,<br />

Chuo-ku Tokyo 104-8002, JP<br />

(72) Satoshi HANAMURA, Saitama-ken 350-<br />

0289, JP<br />

Ken CHIKAUCHI, Saitama-Ken 350-0289, JP<br />

Shigeru KANAZAWA, Saitama-ken 350-0289,<br />

JP<br />

Jinichiro KOGA, Saitama-ken 350-0289, JP<br />

Minoru KANEGAE, Saitama-ken, JP<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

(51) C07D 487/04 (11) 2 248 814 A2<br />

A61P 25/26 A61P 25/18<br />

A61P 9/10 A61P 25/08<br />

A61P 25/28 A61P 3/08<br />

A61P 25/16 A61K 31/519<br />

A61P 3/04<br />

(25) Ru (26) En<br />

(21) 09703618.0 (22) 23.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) IB 2009/050275 23.01.2009<br />

(87) WO 2009/093210 2009/31 30.07.2009<br />

(88) 08.10.2009<br />

(30) 24.01.2008 RU 2008102154<br />

17.09.2008 RU 2008137217<br />

(54) • SUBSTITUIERTE CYCLOALKAN[E UND D]<br />

PYRAZOLO[1,5-A]PYRIMIDINE/ANTAGO-<br />

NISTEN VON SEROTONIN-5-HT6-REZEPT-<br />

OREN UND VERFAHREN ZU DEREN<br />

HERSTELLUNG UND DEREN VERWEN-<br />

DUNG<br />

• SUBSTITUTED CYCLOALCANO[e AND d]<br />

PYRAZOLO [1,5-a] PYRIMIDINES/<br />

ANTAGONISTS OF SEROTONIN 5-HT6<br />

RECEPTORS AND METHODS FOR PRO-<br />

DUCTION AND THE USE THEREOF<br />

• CYCLO-ALCANOÝE ET D¨PYRAZOLOÝ1,5-<br />

A¨PYRIMIDINES SUBSTITUÉES FONC-<br />

TIONNANT COMME DES ANTAGONISTES<br />

DES RÉCEPTEURS 5-HT6 DE SÉROTO-<br />

NINE, PROCÉDÉS DE FABRICATION ET<br />

D'UTILISATION<br />

(71) Alla Chem, LLC., 318 N. Carson Street, Suite<br />

208, Carson City, NV 89701, US<br />

Ivashchenko, Andrey Alexandrovich,<br />

Abramtsevskaya 4 Korp. 2, kv. 27, Moscow<br />

127576, RU<br />

(72) IVASHCHENKO, Andrey Alexandrovich,<br />

Moscow 127576, RU

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