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Bulletin 2010/45 - European Patent Office

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(C07D) I.1(1)<br />

A61K 31/5025<br />

(25) En (26) En<br />

(21) 09716067.5 (22) 16.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) EP 2009/051761 16.02.2009<br />

(87) WO 2009/1064<strong>45</strong> 2009/36 03.09.2009<br />

(30) 25.02.2008 US 31035<br />

22.01.2009 US 146528<br />

(54) • PYRROLOPYRAZINKINASEINHIBITOREN<br />

• PYRROLOPYRAZINE KINASE INHIBITORS<br />

• INHIBITEURS DE KINASE PYRROLOPY-<br />

RAZINE<br />

(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) DU BOIS, Daisy, Joe, Palo Alto California<br />

94304, US<br />

ELWORTHY, Todd, Richard, Los Altos California<br />

94022, US<br />

HENDRICKS, Robert, Than, San Carlos<br />

California 94070, US<br />

HERMANN, Johannes, Cornelius, San Francisco<br />

California 94107, US<br />

KONDRU, Rama, K., Sunnyvale California<br />

94086, US<br />

LOU, Yan, San Jose California 95130, US<br />

OWENS, Timothy, D., Mountain View California<br />

94040, US<br />

PARK, Jaehyeon, Sunnyvale California<br />

94087, US<br />

SMITH, David, Bernard, San Mateo California<br />

94403, US<br />

SOTH, Michael, Milpitas California 95035, US<br />

YEE, Calvin, Wesley, Daly City California<br />

94015, US<br />

(74) Heiroth, Ulrike Hildegard, F. Hoffmann-La<br />

Roche AG <strong>Patent</strong> Department, Grenzacherstrasse<br />

124, CH-4070 Basel, CH<br />

(51) C07D 487/04 (11) 2 247 596 A2*<br />

A61K 31/519 A61P 35/00<br />

(25) En (26) En<br />

(21) 09761144.6 (22) 12.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) IN 2009/000037 12.01.2009<br />

(87) WO 2009/098715 2009/33 13.08.2009<br />

(88) 15.10.2009<br />

(30) 11.01.2008 IN CH01092008<br />

(54) • NEUARTIGE PYRAZOL-[3,4-D-]PYRIMI-<br />

DIN-DERIVATE ALS WIRKSTOFFE GEGEN<br />

KREBS<br />

• NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE<br />

DERIVATIVES AS ANTI -CANCER AGENTS<br />

• NOUVEAUX DERIVES DE PYRAZOLO [3,4<br />

-D] PYRIMIDINE EN TANT QU'AGENTS<br />

ANTICANCEREUX<br />

(71) Natco Pharma Limited, Natco House, Road<br />

No. 2, Banjara Hills, Hyderabad 500 033,<br />

Andhra Pradesh, IN<br />

(72) KONAKANCHI, Durga, Prasad, Hyderabad<br />

500 033, Andhra Pradesh, IN<br />

Subba Rao, Hyderabad 500 033, Andhra<br />

Pradesh, IN<br />

ANANTHANENI, Lakshmi, Hyderabad 500<br />

033, Andhra Pradesh, IN<br />

PILLI, Ramakrishna, Hyderabad 500 033,<br />

Andhra Pradesh, IN<br />

PULLA REDDY, Muddasani, Hyderabad 500<br />

033, Andhra Pradesh, IN<br />

ADIBHATLA KALI SATYA, Bhujanga Rao,<br />

Hyderabad 500 033, Andhra Pradesh, IN<br />

VENKAIAH CHOWDARY, Nannapaneni,<br />

Hyderabad 500 033, IN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) Srinivasan, Ravi Chandran, J.A. Kemp & Co.<br />

14 South Square Gray's Inn, London WC1R<br />

5JJ, GB<br />

(51) C07D 491/04 (11) 2 247 597 A1*<br />

A61P 3/00 A61P 29/00<br />

A61P 37/00 A61K 31/436<br />

C07D 491/147<br />

(25) En (26) En<br />

(21) 09708143.4 (22) 05.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/033134 05.02.2009<br />

(87) WO 2009/100171 2009/33 13.08.2009<br />

(30) 07.02.2008 US 26816<br />

(54) • KONDENSIERTE HETEROARYLE ALS<br />

MODULATOREN DER AKTIVITÄT DES<br />

GLUCOCORTICOIDREZEPTORS, VON AP-1<br />

UND/ODER NF-KB UND DEREN VERWEN-<br />

DUNG<br />

• FUSED HETEROARYL MODULATORS OF<br />

GLUCOCORTICOID RECEPTOR, AP-1,<br />

AND/OR NF-KB ACTIVITY AND USE<br />

THEREOF<br />

• MODULATEURS HÉTÉROARYLE CONDEN-<br />

SÉS, DE L'ACTIVITÉ AP-1 ET/OU NF- B DU<br />

RÉCEPTEUR DES GLUCOCORTICOÏDES ET<br />

LEUR UTILISATION<br />

(71) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton, NJ<br />

05843-4000, US<br />

(72) DUAN, Jingwu, Princeton, New Jersey<br />

08543, US<br />

WEINSTEIN, David, S., Princeton, New<br />

Jersey 08543, US<br />

JIANG, Bin, Princeton, New Jersey 08543,<br />

US<br />

(74) Beacham, Annabel Rose, Dehns St Bride's<br />

House 10 Salisbury Square, London EC4Y<br />

8JD, GB<br />

C07D 491/147→ (51) C07D 491/04<br />

C07D 493/04 → (51) C07D 403/12<br />

C07D 495/04 → (51) C07D 403/12<br />

(51) C07D 498/04 (11) 2 247 598 A1*<br />

C07D 519/00 A61K 31/33<br />

A61P 25/00<br />

(25) En (26) En<br />

(21) 09706447.1 (22) 27.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) IB 2009/000293 27.01.2009<br />

(87) WO 2009/095787 2009/32 06.08.2009<br />

(30) 29.01.2008 EP 08290077<br />

(54) • SUBSTITUIERTE HETEROARYLAMIDOXA-<br />

ZEPINOPYRIMIDONDERIVATE<br />

• SUBSTITUTED HETEROARYLAMIDE OXA-<br />

ZEPINOPYRIMIDONE DERIVATIVES<br />

• DÉRIVÉS D'HÉTÉROARYLAMIDE OXAZÉ-<br />

PINOPYRIMIDONE SUBSTITUÉS<br />

(71) Sanofi-Aventis, 174 Avenue de France,<br />

75013 Paris, FR<br />

Mitsubishi Tanabe Pharma Corporation, 2-6-<br />

18, Kitahama Chuo-ku Osaka-shi, Osaka<br />

541-8505, JP<br />

(72) FAYOL, Aude, F-75013 Paris, FR<br />

LOCHEAD, Alistair, F-75013 Paris, FR<br />

SAADY, Mourad, F-75013 Paris, FR<br />

VACHE, Julien, F-75013 Paris, FR<br />

YAICHE, Philippe, F-75013 Paris, FR<br />

75<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>45</strong>/<strong>2010</strong>) 10.11.<strong>2010</strong><br />

(74) Dépré, Marie-Line, et al, Sanofi-Aventis<br />

Département Brevets 174, avenue de France,<br />

F-75013 Paris, FR<br />

(51) C07D 498/04 (11) 2 247 599 A1*<br />

A61K 31/33 A61P 25/00<br />

(25) En (26) En<br />

(21) 09706539.5 (22) 27.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) IB 2009/000298 27.01.2009<br />

(87) WO 2009/095788 2009/32 06.08.2009<br />

(30) 29.01.2008 EP 08290075<br />

(54) • SUBSTITUIERTE ARYLAMIDOXAZEPINO-<br />

PYRIMIDONDERIVATE<br />

• SUBSTITUTED ARYLAMIDE OXAZEPINO-<br />

PYRIMIDONE DERIVATIVES<br />

• DÉRIVÉS D'ARYLAMIDE OXAZÉPINOPY-<br />

RIMIDONE SUBSTITUÉS<br />

(71) Sanofi-Aventis, 174 Avenue de France,<br />

75013 Paris, FR<br />

Mitsubishi Tanabe Pharma Corporation, 2-6-<br />

18, Kitahama Chuo-ku Osaka-shi, Osaka<br />

541-8505, JP<br />

(72) FAYOL, Aude, F-75013 Paris, FR<br />

LOCHEAD, Alistair, F-75013 Paris, FR<br />

SAADY, Mourad, F-75013 Paris, FR<br />

VACHE, Julien, F-75013 Paris, FR<br />

YAICHE, Philippe, F-75013 Paris, FR<br />

(74) Dépré, Marie-Line, et al, Sanofi-Aventis<br />

Département Brevets 174, avenue de France,<br />

F-75013 Paris, FR<br />

(51) C07D 498/04 (11) 2 247 600 A2*<br />

(25) En (26) En<br />

(21) 09708325.7 (22) 15.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/031163 15.01.2009<br />

(87) WO 2009/099736 2009/33 13.08.2009<br />

(88) 08.10.2009<br />

(30) 06.02.2008 US 26690<br />

(54) • BENZOXAZOLCARBONSÄUREAMIDE ALS<br />

INHIBITOREN VON POLY(ADP-RIBOSE)<br />

POLYMERASE (PARP)<br />

• BENZOXAZOLE CARBOXAMIDE INHIBI-<br />

TORS OF POLY(ADP-RIBOSE)POLYMER-<br />

ASE (PARP)<br />

• INHIBITEURS À BASE DE COMPOSÉS<br />

BENZOXAZOLE-CARBOXAMIDE DE L<br />

ACTIVITÉ POLY(ADP-RIBOSE)POLYMÉ-<br />

RASE (PARP)<br />

(71) Lead Therapeutics, Inc., 999 Bayhill Drive,<br />

Suite 130, San Bruno, CA 94066, US<br />

(72) CHU, Daniel, Santa Clara California 95051,<br />

US<br />

WANG, Bing, San Jose Arizona 95138, US<br />

(74) Ritter, Thomas Kurt, Jones Day<br />

Prinzregentenstraße 11, 80538 München, DE<br />

C07D 498/04 → (51) C07D 471/04<br />

(51) C07D 513/04 (11) 2 247 601 A1*<br />

A61K 31/519 A61P 31/18<br />

(25) En (26) En<br />

(21) 09771847.2 (22) 02.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) AU 2009/000856 02.07.2009<br />

(87) WO <strong>2010</strong>/000030 <strong>2010</strong>/01 07.01.<strong>2010</strong>

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