Bulletin 2010/45 - European Patent Office
Bulletin 2010/45 - European Patent Office
Bulletin 2010/45 - European Patent Office
Create successful ePaper yourself
Turn your PDF publications into a flip-book with our unique Google optimized e-Paper software.
(C07D) II.1(1)<br />
(30) 04.03.2005 US 658791 P<br />
(54) • Verfahren zur Verminderung von Alpha,<br />
Beta-ungesättigten Ketonen in Opioidzusammensetzungen<br />
• Method of reducing alpha, beta- unsaturated<br />
ketones in opioid compositions<br />
• Procédé de réduction de cétones insaturées<br />
alpha et bêta dans des compositions<br />
d'opioides<br />
(73) EURO-CELTIQUE S.A., 2, avenue Charles de<br />
Gaulle, 1653 Luxembourg, LU<br />
(72) Kupper, Robert Joe, East Greenwich, RI<br />
02818, US<br />
(74) Vos, Derk, Maiwald <strong>Patent</strong>anwalts GmbH<br />
Elisenhof Elisenstraße 3, 80335 München,<br />
DE<br />
(62) 06707309.8 / 1 861 405<br />
C07D 487/08 → (51) C07D <strong>45</strong>1/04<br />
C07D 491/04 → (51) C07D 401/12<br />
(51) C07D 491/048 (11) 2 146 997 B1<br />
A61K 31/4355 A61P 3/04<br />
A61P 25/18 A61P 25/22<br />
A61P 25/28<br />
(25) En (26) En<br />
(21) 08742647.4 (22) 07.04.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
(43) 27.01.<strong>2010</strong><br />
(86) US 2008/00<strong>45</strong>33 07.04.2008<br />
(87) WO 2008/127585 2008/43 23.10.2008<br />
(30) 11.04.2007 US 922851 P<br />
(54) • SUBSTITUIERTE FURO[2,3-B]PYRIDIN-<br />
DERIVATE ALS CANNABINOID-1-REZEPT-<br />
ORMODULATOREN<br />
• SUBSTITUTED FURO[2,3-B]PYRIDINE<br />
DERIVATIVES AS CANNABINOID-1<br />
RECEPTOR MODULATORS<br />
• DÉRIVÉS FURO[2,3-B]PYRIDINE SUBSTI-<br />
TUÉS UTILES EN TANT QUE MODULA-<br />
TEURS DU RÉCEPTEUR DES<br />
CANNABINOÏDES 1<br />
(73) Merck Sharp & Dohme Corp., 126 East<br />
Lincoln Avenue, Rahway, NJ 07065, US<br />
(72) CLEMENTS, Matthew, J., Rahway, New<br />
Jersey 07065-0907, US<br />
DEBENHAM, John, S., Rahway, New Jersey<br />
07065-0907, US<br />
HALE, Jeffrey, J., Rahway, New Jersey<br />
07065-0907, US<br />
MADSEN-DUGGAN, Christina, B., Rahway,<br />
New Jersey 07065-0907, US<br />
WALSH, Thomas, F., Rahway, New Jersey<br />
07065-0907, US<br />
PERESYPKIN, Andrey, V., Rahway, New<br />
Jersey 07065-0907, US<br />
HELMY, Roy, Rahway, New Jersey 07065-<br />
0907, US<br />
(74) Buchan, Gavin MacNicol, et al, Merck & Co.,<br />
Inc. <strong>European</strong> <strong>Patent</strong> Department Hertford<br />
Road, Hoddesdon, Hertfordshire EN11 9BU,<br />
GB<br />
(51) C07D 491/22 (11) 1 995 249 B1<br />
A61K 31/47<strong>45</strong> A61P 35/00<br />
(25) Zh (26) En<br />
(21) 07702109.5 (22) 17.01.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
(43) 26.11.2008<br />
(86) CN 2007/000177 17.01.2007<br />
(87) WO 2007/104214 2007/38 20.09.2007<br />
(30) 10.03.2006 CN 20061002<strong>45</strong>90<br />
(54) • CAMPTOTHECINDERIVATE UND IHRE<br />
VERWENDUNG<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
• CAMPTOTHECIN DERIVATIVES AND<br />
THEIR USE<br />
• DÉRIVÉS DE LA CAMPTOTHÉCINE ET<br />
LEURS UTILISATIONS<br />
(73) Shanghai Institute of Materia Medica, Chinese<br />
Academy of Sciences, 555 Zu Chong<br />
Zhi Road Zhangjlang Hi-Tech Park Pudong<br />
New District, Shanghai <strong>2010</strong>23, CN<br />
(72) LU, Wei, Shanghai 201203, CN<br />
DING, Jian, Shanghai 201203, CN<br />
GAO, Heyong, Shanghai 201203, CN<br />
LIN, Liping, Shanghai 201203, CN<br />
CHEN, Yi, Shanghai 201203, CN<br />
(74) Solf, Alexander, <strong>Patent</strong>anwälte Dr. Solf &<br />
Zapf Candidplatz 15, 81543 München, DE<br />
(51) C07D 495/04 (11) 1 618 113 B1<br />
A61K 31/4365 A61P 7/02<br />
(25) En (26) En<br />
(21) 04768414.7 (22) 09.09.2004<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />
TR<br />
(43) 25.01.2006<br />
(86) GB 2004/003867 09.09.2004<br />
(87) WO 2005/026174 2005/12 24.03.2005<br />
(30) 11.09.2003 GB 0321256<br />
(54) • NEUE KRISTALLINE POLYMORPHE VON<br />
CLOPIDOGREL<br />
• NOVEL CRYSTALLINE POLYMORPHS OF<br />
CLOPIDOGREL<br />
• POLYMORPHES CRISTALLINS DU CLOPI-<br />
DOGREL<br />
(73) Generics (UK) Limited, Albany Gate, Darkes<br />
Lane, Potters Bar, Hertfordshire EN6 1AG,<br />
GB<br />
(72) ARUL, Ramakrishnan Merck Dev. Centre<br />
Private Ltd., Maharashtra 410 208, IN<br />
RAWAT, Ajay Singh Merck Dev. Centre<br />
Private Ltd., Maharashtra 410 208, IN<br />
GADAKAR,Maheshkumar Merck Dev. Centre<br />
Private Ltd., Maharashtra 410 208, IN<br />
RAO, Rajesh Merck Development Centre<br />
Private Ltd., Maharashtra 410 208, IN<br />
PISE, Abhinay Merck Development Centre<br />
Private Ltd, Maharashtra410 208, IN<br />
GRAY, Jason Generics (UK) Limited, Hertfordshire<br />
EN6 1AG, GB<br />
(74) Elend, Almut Susanne, et al, Venner Shipley<br />
LLP Byron House Cambridge Business Park<br />
Cowley Road, Cambridge CB4 0WZ, GB<br />
(60) 06124847.2 / 1 837 337<br />
06124851.4 / 1 772 <strong>45</strong>6<br />
09159491.1 / 2 149 578<br />
(51) C07D 498/04 (11) 1 987 040 B1<br />
(25) En (26) En<br />
(21) 07705876.6 (22) 14.02.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
(43) 05.11.2008<br />
(86) IB 2007/050482 14.02.2007<br />
(87) WO 2007/093963 2007/34 23.08.2007<br />
(30) 15.02.2006 PCT/IB2006/050505<br />
(54) • ANTIBIOTISCHE ETHANOL- ODER 1,2-<br />
ETHANDIOL-CYCLOHEXYL-DERIVATE<br />
• ETHANOL OR 1,2-ETHANEDIOL CYCLO-<br />
HEXYL ANTIBIOTIC DERIVATIVES<br />
• DÉRIVÉS D'ÉTHANOL OU DE 1,2-ÉTHA-<br />
NEDIOL DE TYPE CYCLOHEXYLE À ACTI-<br />
VITÉ ANTIBIOTIQUE<br />
(73) Actelion Pharmaceuticals Ltd., Gewerbestrasse<br />
16, 4123 Allschwil, CH<br />
(72) HUBSCHWERLEN, Christian, F-68480 Durmenach,<br />
FR<br />
SURIVET, Jean-Philippe, F-68680 Kembs, FR<br />
ZUMBRUNN ACKLIN, Cornelia, CH-4058<br />
Basel, CH<br />
567<br />
<strong>Patent</strong>e<br />
<strong>Patent</strong>s<br />
Brevets (<strong>45</strong>/<strong>2010</strong>) 10.11.<strong>2010</strong><br />
(74) Ruhlmann, Eric, et al, Actelion Pharmaceuticals<br />
Ltd Gewerbestrasse 16, 4123 Allschwil,<br />
CH<br />
(51) C07D 513/04 (11) 1 869 056 B1<br />
A61K 31/519 A61P 11/06<br />
A61P 25/00 A61P 9/10<br />
(25) En (26) En<br />
(21) 06717078.7 (22) 03.04.2006<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
AL BA HR MK YU<br />
(43) 26.12.2007<br />
(86) SE 2006/000399 03.04.2006<br />
(87) WO 2006/107258 2006/41 12.10.2006<br />
(30) 06.04.2005 SE 0500767<br />
(54) • NEUE 5-SUBSTITUIERTE 7-AMINO-[1,3]<br />
THIAZOLO[4,5-D]PYRIMIDIN-2(3H)-<br />
ONDERIVATE<br />
• NOVEL 5-SUBSTITUTED 7-AMINO-<br />
Ý1,3¨THIAZOLOÝ4,5-D¨PYRIMIDINE<br />
DERIVATIVES<br />
• NOUVEAUX DÉRIVÉS DE 7-AMINO-<br />
Ý1,3¨THIAZOLOÝ4,5-D¨PYRIMIDINE 5<br />
SUBSTITUÉ<br />
(73) AstraZeneca AB, 151 85 Södertälje, SE<br />
(72) NORDVALL, Gunnar, S-151 85 Södertälje,<br />
SE<br />
RAY, Colin, S-151 85 Södertälje, SE<br />
REIN, Tobias, S-151 85 Södertälje, SE<br />
SOHN, Daniel, S-151 85 Södertälje, SE<br />
C07F 7/18 → (51) C08F 4/60<br />
(51) C07F 7/30 (11) 1 990 3<strong>45</strong> B1<br />
C23C 16/28<br />
(25) En (26) En<br />
(21) 08163178.0 (22) 01.04.2004<br />
(84) DE FR GB<br />
(43) 12.11.2008<br />
(30) 22.10.2003 US 513476 P<br />
05.04.2003 US 460791 P<br />
(54) • Zur Verwendung in Dampfphasenabscheidungsprozessen<br />
geeignete, metallorganische<br />
Germanium-Verbindungen<br />
• Organometallic germanium compounds<br />
suitable for use in vapor deposition<br />
processes<br />
• Composés organométalliques du germanium<br />
utilisables dans des procédés de<br />
dépôt en phase vapeur<br />
(73) Rohm and Haas Electronic Materials LLC,<br />
<strong>45</strong>5 Forest Street, Marlborough, MA 01752,<br />
US<br />
(72) Shenai-Khatkhate, Deodatta Vinayak, Danvers,<br />
MA 01923, US<br />
Power, Michael Brendan, Newburyport, MA<br />
01950, US<br />
(74) Buckley, Guy Julian, <strong>Patent</strong> Outsourcing<br />
Limited 1 King Street Bakewell, Derbyshire<br />
DE<strong>45</strong> 1DZ, GB<br />
(62) 04251948.8 / 1 464 724<br />
(51) C07F 9/06 (11) 1 756 125 B1<br />
C05G 3/08<br />
(25) De (26) De<br />
(21) 05707288.6 (22) 09.02.2005<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />
SI SK TR<br />
(43) 28.02.2007<br />
(86) EP 2005/001300 09.02.2005<br />
(87) WO 2005/118602 2005/50 15.12.2005<br />
(30) 28.05.2004 DE 102004026143