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PCT/2000/51 - World Intellectual Property Organization

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<strong>51</strong>/<strong>2000</strong><br />

21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19091<br />

Frontiers Science Park South, Third Avenue,<br />

Harlow, Essex CM19 5AW (GB).<br />

ENGBERTS, Jan, Bernard, Frederick,<br />

Nicolaas [NL/NL]; University of Groningen,<br />

Nijenborgh 4, NL-9747 Groningen (NL).<br />

FIELDEN, Matthew, Leigh [AU/NL]; University<br />

of Groningen, Nijenborgh 4, NL-9747<br />

Groningen (NL). KREMER, Andreas<br />

[DE/GB]; SmithKline Beecham Pharmaceuticals,<br />

New Frontiers Science Park South,<br />

Third Avenue, Harlow, Essex CM19 5AW<br />

(GB).<br />

(74) GIDDINGS, Peter, John; SmithKline<br />

Beecham, Two New Horizons Court, Brentford,<br />

Middlesex TW8 9EP (GB).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07C 215/52, A61K 31/135, A61P 25/24<br />

(11) WO 00/76955 (13) A1<br />

(21) <strong>PCT</strong>/US00/16388<br />

(22) 14 Jun/juin <strong>2000</strong> (14.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/333,594 15 Jun/juin 1999 US<br />

(15.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) ENANTIOMERS OF O-DESMETHYL<br />

VENLAFAXINE<br />

ENANTIOMERES DE O-DESMETHYL<br />

VENLAFAXINE<br />

(71) AMERICAN HOME PRODUCTS COR-<br />

PORATION [US/US]; Five Giralda Farms,<br />

Madison, NJ 07940-0874 (US).<br />

(72) YARDLEY, John, Patrick; 154 Hughes<br />

Road, King of Prussia, PA 19406 (US). AS-<br />

SELIN, Andre, Alfred; 64 Ackerman Drive,<br />

Mahwah, NJ 07430 (US).<br />

(74) ECK, Steven, R.; American Home Products<br />

Corporation, Patent Law Dept. - 2B, One<br />

Campus Drive, Parsippany, NJ 07054 (US) et<br />

al. / etc.<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07C 217/00<br />

(11) WO 00/76956 (13) A2<br />

(21) <strong>PCT</strong>/US00/16439<br />

(22) 14 Jun/juin <strong>2000</strong> (14.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/333,207 15 Jun/juin 1999 US<br />

(15.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) ENANTIOMERS OF N-DESMETHYL<br />

VENLAFAXINE<br />

ENANTIOMERES DE N-DESMETHYL<br />

VENLAFAXINE<br />

(71) AMERICAN HOME PRODUCTS COR-<br />

PORATION [US/US]; Five Giralda Farms,<br />

Madison, NJ 07940-0874 (US).<br />

(72) YARDLEY, John, Patrick; 154 Hughes<br />

Road, King of Prussia, PA 19406 (US). AS-<br />

SELIN, Andre, Alfred; 64 Ackerman Drive,<br />

Mahwah, NJ 07430 (US).<br />

(74) ECK, Steven, R.; American Home Products<br />

Corporation, Patent Law Dept. - 2B, One<br />

Campus Drive, Parsippany, NJ 07054 (US) et<br />

al. / etc.<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07C 217/10, 233/69, C07D 215/14,<br />

307/79, 317/54, 319/18, 277/64, 333/54,<br />

333/62, 333/70, 409/04, 311/04, 235/06,<br />

241/42, A61K 31/47, 31/343, 31/36, 31/357,<br />

31/428, 31/381, 31/4436, 31/352, 31/4184,<br />

31/498, 31/135, A61P 25/28, 25/16, 25/14,<br />

11/16<br />

(11) WO 00/76957<br />

(21) <strong>PCT</strong>/JP00/03748<br />

(13) A1<br />

(22) 9 Jun/juin <strong>2000</strong> (09.06.<strong>2000</strong>)<br />

(25) ja (26) ja<br />

(30) 11/165879 11 Jun/juin 1999<br />

(11.06.1999)<br />

JP<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) N-ALKOXYALKYL-N,N-DIALKY-<br />

LAMINE DERIVATIVES OR SALTS<br />

THEREOF, AND REMEDIES FOR<br />

NERVE DEGENERATION DISEASES<br />

CONTAINING THE SAME<br />

DERIVES DE N-ALKOXYALKYL,<br />

N-DIALKYLAMINE OU LEURS SELS<br />

ET REMEDES CONTRE LES MALA-<br />

DIES A DEGENERESCENCE NER-<br />

VEUSE, QUI LES CONTIENNENT<br />

(71) TOYAMA CHEMICAL CO., LTD.<br />

[JP/JP]; 2-5, Nishishinjuku 3-chome, Shinjuku-ku,<br />

Tokyo 160-0023 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) ONO, Satoshi [JP/JP]; 2-5, Nakajima<br />

3-chome, Toyama-shi, Toyama 930-0801<br />

(JP). SAITOH, Akihito [JP/JP]; 6-12,<br />

Toyoshiro-cho, Toyama-shi, Toyama<br />

931-8324 (JP). IWAKAMI, Noboru [JP/JP];<br />

3-20, Sengoku-machi, Takaoka-shi, Toyama<br />

933-0847 (JP). NAKAGAWA, Masaya<br />

[JP/JP]; 67, Nakaaoide, Kamiichi-machi,<br />

Nakaniikawa-gun, Toyama 930-0386 (JP).<br />

YAMAGUCHI, Sumie [JP/JP]; 6-27, Shimookui<br />

1-chome, Toyama-shi, Toyama<br />

930-0817 (JP).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07C 229/08, A61K 31/197, C07C 229/30,<br />

229/22, 229/34, 229/32, 229/20, A61P 25/00,<br />

1/00<br />

(11) WO 00/76958 (13) A2<br />

(21) <strong>PCT</strong>/US00/15070<br />

(22) 31 May/mai <strong>2000</strong> (31.05.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,485 10 Jun/juin 1999 US<br />

(10.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) MONO- AND DISUBSTITUTED<br />

3-PROPYL GAMMA-AMINOBUTYRIC<br />

ACIDS<br />

ACIDES 3-PROPYLE GAMMA-AMI-<br />

NOBUTYRIQUES MONOSUBSTITUES<br />

ET DISUBSTITUES<br />

(71) WARNER-LAMBERT COMPANY<br />

[US/US]; 201 Tabor Road, Morris Plains,<br />

NJ 07950 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) BELLIOTTI, Thomas, Richard<br />

[US/US]; 6125 Lodi Lane, Saline, MI 48176<br />

(US). BRYANS, Justin, Stephen [GB/GB];<br />

Dean Cottage, 3 W. Wickham Road, Balsham<br />

CB1 6DZ (GB). EKHATO, Ihoezo,<br />

Victor [NG/US]; 1005 Edgemill Way, Steeplechase<br />

on Radley Run, West Chester, PA<br />

19382 (US). OSUMA, Augustine, Tobi<br />

[US/US]; 1174 Paddock Place #202, Ann Arbor,<br />

MI 48108 (US). SCHELKUN, Robert,<br />

Michael [US/US]; 221 E. Braman Avenue,<br />

Milan, MI 48160 (US). SCHWARZ, Roy,<br />

Douville [US/US]; 9340 Lake Crest Drive,<br />

Whitmore Lake, MI 48189 (US). THORPE,<br />

Andrew, John [GB/US]; 570 Landings<br />

Boulevard, Ann Arbor, MI 48103 (US).<br />

WISE, Lawrence, David [US/US]; 1241<br />

Barrister, Ann Arbor, MI 48105 (US). WUS-<br />

TROW, David, Juergen [US/US]; <strong>51</strong>01 John<br />

Holmes Road, Ann Arbor, MI 48103 (US).<br />

YUEN, Po-Wai [US/US]; 2178 Maple Creek<br />

Circle, Ann Arbor, MI 48108 (US).<br />

(74) RYAN, M., Andrea; Warner-Lambert Company,<br />

201 Tabor Road, Morris Plains, NJ<br />

07950 (US) et al. / etc.<br />

(81) AE AG AL AU BA BB BG BR CA CN CR<br />

CU CZ DM DZ EE GD GE HR HU ID IL IN<br />

IS JP KP KR LC LK LR LT LV MA MG MK<br />

MN MX MZ NO NZ PL RO SG SI SK SL TR<br />

TT UA US UZ VN YU ZA.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU

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