PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
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<strong>51</strong>/<strong>2000</strong><br />
21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19091<br />
Frontiers Science Park South, Third Avenue,<br />
Harlow, Essex CM19 5AW (GB).<br />
ENGBERTS, Jan, Bernard, Frederick,<br />
Nicolaas [NL/NL]; University of Groningen,<br />
Nijenborgh 4, NL-9747 Groningen (NL).<br />
FIELDEN, Matthew, Leigh [AU/NL]; University<br />
of Groningen, Nijenborgh 4, NL-9747<br />
Groningen (NL). KREMER, Andreas<br />
[DE/GB]; SmithKline Beecham Pharmaceuticals,<br />
New Frontiers Science Park South,<br />
Third Avenue, Harlow, Essex CM19 5AW<br />
(GB).<br />
(74) GIDDINGS, Peter, John; SmithKline<br />
Beecham, Two New Horizons Court, Brentford,<br />
Middlesex TW8 9EP (GB).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG US UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07C 215/52, A61K 31/135, A61P 25/24<br />
(11) WO 00/76955 (13) A1<br />
(21) <strong>PCT</strong>/US00/16388<br />
(22) 14 Jun/juin <strong>2000</strong> (14.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 09/333,594 15 Jun/juin 1999 US<br />
(15.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) ENANTIOMERS OF O-DESMETHYL<br />
VENLAFAXINE<br />
ENANTIOMERES DE O-DESMETHYL<br />
VENLAFAXINE<br />
(71) AMERICAN HOME PRODUCTS COR-<br />
PORATION [US/US]; Five Giralda Farms,<br />
Madison, NJ 07940-0874 (US).<br />
(72) YARDLEY, John, Patrick; 154 Hughes<br />
Road, King of Prussia, PA 19406 (US). AS-<br />
SELIN, Andre, Alfred; 64 Ackerman Drive,<br />
Mahwah, NJ 07430 (US).<br />
(74) ECK, Steven, R.; American Home Products<br />
Corporation, Patent Law Dept. - 2B, One<br />
Campus Drive, Parsippany, NJ 07054 (US) et<br />
al. / etc.<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07C 217/00<br />
(11) WO 00/76956 (13) A2<br />
(21) <strong>PCT</strong>/US00/16439<br />
(22) 14 Jun/juin <strong>2000</strong> (14.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 09/333,207 15 Jun/juin 1999 US<br />
(15.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) ENANTIOMERS OF N-DESMETHYL<br />
VENLAFAXINE<br />
ENANTIOMERES DE N-DESMETHYL<br />
VENLAFAXINE<br />
(71) AMERICAN HOME PRODUCTS COR-<br />
PORATION [US/US]; Five Giralda Farms,<br />
Madison, NJ 07940-0874 (US).<br />
(72) YARDLEY, John, Patrick; 154 Hughes<br />
Road, King of Prussia, PA 19406 (US). AS-<br />
SELIN, Andre, Alfred; 64 Ackerman Drive,<br />
Mahwah, NJ 07430 (US).<br />
(74) ECK, Steven, R.; American Home Products<br />
Corporation, Patent Law Dept. - 2B, One<br />
Campus Drive, Parsippany, NJ 07054 (US) et<br />
al. / etc.<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07C 217/10, 233/69, C07D 215/14,<br />
307/79, 317/54, 319/18, 277/64, 333/54,<br />
333/62, 333/70, 409/04, 311/04, 235/06,<br />
241/42, A61K 31/47, 31/343, 31/36, 31/357,<br />
31/428, 31/381, 31/4436, 31/352, 31/4184,<br />
31/498, 31/135, A61P 25/28, 25/16, 25/14,<br />
11/16<br />
(11) WO 00/76957<br />
(21) <strong>PCT</strong>/JP00/03748<br />
(13) A1<br />
(22) 9 Jun/juin <strong>2000</strong> (09.06.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/165879 11 Jun/juin 1999<br />
(11.06.1999)<br />
JP<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) N-ALKOXYALKYL-N,N-DIALKY-<br />
LAMINE DERIVATIVES OR SALTS<br />
THEREOF, AND REMEDIES FOR<br />
NERVE DEGENERATION DISEASES<br />
CONTAINING THE SAME<br />
DERIVES DE N-ALKOXYALKYL,<br />
N-DIALKYLAMINE OU LEURS SELS<br />
ET REMEDES CONTRE LES MALA-<br />
DIES A DEGENERESCENCE NER-<br />
VEUSE, QUI LES CONTIENNENT<br />
(71) TOYAMA CHEMICAL CO., LTD.<br />
[JP/JP]; 2-5, Nishishinjuku 3-chome, Shinjuku-ku,<br />
Tokyo 160-0023 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) ONO, Satoshi [JP/JP]; 2-5, Nakajima<br />
3-chome, Toyama-shi, Toyama 930-0801<br />
(JP). SAITOH, Akihito [JP/JP]; 6-12,<br />
Toyoshiro-cho, Toyama-shi, Toyama<br />
931-8324 (JP). IWAKAMI, Noboru [JP/JP];<br />
3-20, Sengoku-machi, Takaoka-shi, Toyama<br />
933-0847 (JP). NAKAGAWA, Masaya<br />
[JP/JP]; 67, Nakaaoide, Kamiichi-machi,<br />
Nakaniikawa-gun, Toyama 930-0386 (JP).<br />
YAMAGUCHI, Sumie [JP/JP]; 6-27, Shimookui<br />
1-chome, Toyama-shi, Toyama<br />
930-0817 (JP).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG US UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07C 229/08, A61K 31/197, C07C 229/30,<br />
229/22, 229/34, 229/32, 229/20, A61P 25/00,<br />
1/00<br />
(11) WO 00/76958 (13) A2<br />
(21) <strong>PCT</strong>/US00/15070<br />
(22) 31 May/mai <strong>2000</strong> (31.05.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,485 10 Jun/juin 1999 US<br />
(10.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) MONO- AND DISUBSTITUTED<br />
3-PROPYL GAMMA-AMINOBUTYRIC<br />
ACIDS<br />
ACIDES 3-PROPYLE GAMMA-AMI-<br />
NOBUTYRIQUES MONOSUBSTITUES<br />
ET DISUBSTITUES<br />
(71) WARNER-LAMBERT COMPANY<br />
[US/US]; 201 Tabor Road, Morris Plains,<br />
NJ 07950 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BELLIOTTI, Thomas, Richard<br />
[US/US]; 6125 Lodi Lane, Saline, MI 48176<br />
(US). BRYANS, Justin, Stephen [GB/GB];<br />
Dean Cottage, 3 W. Wickham Road, Balsham<br />
CB1 6DZ (GB). EKHATO, Ihoezo,<br />
Victor [NG/US]; 1005 Edgemill Way, Steeplechase<br />
on Radley Run, West Chester, PA<br />
19382 (US). OSUMA, Augustine, Tobi<br />
[US/US]; 1174 Paddock Place #202, Ann Arbor,<br />
MI 48108 (US). SCHELKUN, Robert,<br />
Michael [US/US]; 221 E. Braman Avenue,<br />
Milan, MI 48160 (US). SCHWARZ, Roy,<br />
Douville [US/US]; 9340 Lake Crest Drive,<br />
Whitmore Lake, MI 48189 (US). THORPE,<br />
Andrew, John [GB/US]; 570 Landings<br />
Boulevard, Ann Arbor, MI 48103 (US).<br />
WISE, Lawrence, David [US/US]; 1241<br />
Barrister, Ann Arbor, MI 48105 (US). WUS-<br />
TROW, David, Juergen [US/US]; <strong>51</strong>01 John<br />
Holmes Road, Ann Arbor, MI 48103 (US).<br />
YUEN, Po-Wai [US/US]; 2178 Maple Creek<br />
Circle, Ann Arbor, MI 48108 (US).<br />
(74) RYAN, M., Andrea; Warner-Lambert Company,<br />
201 Tabor Road, Morris Plains, NJ<br />
07950 (US) et al. / etc.<br />
(81) AE AG AL AU BA BB BG BR CA CN CR<br />
CU CZ DM DZ EE GD GE HR HU ID IL IN<br />
IS JP KP KR LC LK LR LT LV MA MG MK<br />
MN MX MZ NO NZ PL RO SG SI SK SL TR<br />
TT UA US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU