PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
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<strong>51</strong>/<strong>2000</strong><br />
21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19011<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065-0907 (US). MACCOSS, Malcolm<br />
[GB/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MILLS, Sander, G.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/445, C07D 211/06, 215/12,<br />
215/14, 401/08<br />
(11) WO 00/76<strong>51</strong>4 (13) A1<br />
(21) <strong>PCT</strong>/US00/15769<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,761 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS DE CYCLOPENTYLE<br />
DE L’ACTIVITE DU RECEPTEUR DE<br />
CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). HILFIKER, Kerry, A. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065-0907 (US). LOEBACH, Jennifer, L.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MACCOSS, Malcolm<br />
[GB/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MILLS, Sander, G.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). SHEN, Dong-Ming<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). OATES, Bryan<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/47, 31/495, 31/38, 31/17<br />
(11) WO 00/76<strong>51</strong>5 (13) A1<br />
(21) <strong>PCT</strong>/US00/16<strong>51</strong>0<br />
(22) 15 Jun/juin <strong>2000</strong> (15.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,673 16 Jun/juin 1999 US<br />
(16.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) IL-8 RECEPTOR ANTAGONISTS<br />
ANTAGONISTES DU RECEPTEUR IL-8<br />
(71) SMITHKLINE BEECHAM CORPO-<br />
RATION [US/US]; One Franklin Plaza,<br />
Philadelphia, PA 19103 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WIDDOWSON, Katherine, L.<br />
[CA/US]; 1047 Old Valley Forge Road,<br />
King of Prussia, PA 19406 (US). BENSON,<br />
Gregory, Martin [GB/GB]; New Frontiers<br />
Science Park South, Harlow, Essex CM19<br />
5AW (GB).<br />
(74) SIMON, Soma, G. et al. / etc.; SmithKline<br />
Beecham Corporation, Corporate <strong>Intellectual</strong><br />
<strong>Property</strong>, UW2220, 709 Swedeland<br />
Road, P.O. Box 1539, King of Prussia, PA<br />
19406-0939 (US).<br />
(81) AE AL AU BA BB BG BR CA CN CZ DZ<br />
EE GE GH GM HR HU ID IL IN IS JP KP<br />
KR LC LK LR LT LV MA MG MK MN MX<br />
NO NZ PL RO SG SI SK SL TR TT TZ UA<br />
US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/47, 31/495, 31/38, 47/28, 31/17<br />
(11) WO 00/76<strong>51</strong>6<br />
(21) <strong>PCT</strong>/US00/16813<br />
(13) A1<br />
(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,674 16 Jun/juin 1999<br />
(16.06.1999)<br />
US<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) IL-8 RECEPTOR ANTAGONISTS<br />
ANTAGONISTES DE RECEPTEURS DE<br />
IL-8<br />
(71) SMITHKLINE BEECHAM CORPO-<br />
RATION [US/US]; One Franklin Plaza,<br />
Philadelphia, PA 19103 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BRYAN, Deborah, L. [US/US]; 341<br />
MacKenzie Drive, West Chester, PA 19380<br />
(US). GLEASON, John, G. [CA/US];<br />
8 Heron Hill Drive, Downingtown, PA<br />
19335 (US). WIDDOWSON, Katherine, L.<br />
[CA/US]; 1047 Old Valley Forge Road, King<br />
of Prussia, PA 19406 (US). BENSON, Gregory,<br />
M. [GB/GB]; Nazeing, Essex (GB).<br />
(74) SIMON, Soma, G. et al. / etc.; SmithKline<br />
Beecham Corporation, Corporate <strong>Intellectual</strong><br />
<strong>Property</strong>, UW2220, 709 Swedeland<br />
Road, P.O. Box 1539, King of Prussia, PA<br />
19406-0939 (US).<br />
(81) AE AL AU BA BB BG BR CA CN CZ DZ<br />
EE GE GH GM HR HU ID IL IN IS JP KP<br />
KR LC LK LR LT LV MA MG MK MN MX<br />
NO NZ PL RO SG SI SK SL TR TT TZ UA<br />
US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/47, 31/495, 31/38, 31/17<br />
(11) WO 00/76<strong>51</strong>7 (13) A1<br />
(21) <strong>PCT</strong>/US00/16814<br />
(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,677 16 Jun/juin 1999 US<br />
(16.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) IL-8 RECEPTOR ANTAGONISTS<br />
ANTAGONISTES DES RECEPTEURS<br />
DE IL-8<br />
(71) SMITHKLINE BEECHAM CORPO-<br />
RATION [US/US]; One Franklin Plaza,<br />
Philadelphia, PA 19103 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BRYAN, Deborah, L. [US/US]; 341<br />
MacKenzie Drive, West Chester, PA 19380<br />
(US). GLEASON, John, G. [CA/US];<br />
8 Heron Hill Drive, Downingtown, PA<br />
19335 (US). WIDDOWSON, Katherine, L.<br />
[CA/US]; 1047 Old Valley Forge Road, King<br />
of Prussia, PA 19406 (US). BENSON, Gregory,<br />
M. [GB/GB]; Nazeing, Essex (GB).<br />
(74) SIMON, Soma, G. et al. / etc.; SmithKline<br />
Beecham Corporation, Corporate <strong>Intellectual</strong><br />
<strong>Property</strong>, UW2220, 709 Swedeland<br />
Road, P.O. Box 1539, King of Prussia, PA<br />
19406-0939 (US).<br />
(81) AE AL AU BA BB BG BR CA CN CZ DZ<br />
EE GE GH GM HR HU ID IL IN IS JP KP<br />
KR LC LK LR LT LV MA MG MK MN MX<br />
NO NZ PL RO SG SI SK SL TR TT TZ UA<br />
US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/4745, 31/437, C07D 471/02<br />
(11) WO 00/76<strong>51</strong>8 (13) A1<br />
(21) <strong>PCT</strong>/US00/15656<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,365 10 Jun/juin 1999<br />
(10.06.1999)<br />
(30) 09/589,236 7 Jun/juin <strong>2000</strong><br />
(07.06.<strong>2000</strong>)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
US<br />
US<br />
(54) UREA SUBSTITUTED IMIDAZO-<br />
QUINOLINES