PCT/2000/51 - World Intellectual Property Organization

51/2000
19098 PCT Gazette - Section I - Gazette du PCT 21 Dec/déc 2000
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 241/18, 241/20, 405/12, A61K
31/497, A61P 25/00
(11) WO 00/76984 (13) A2
(21) PCT/SE00/01017
(22) 19 May/mai 2000 (19.05.2000)
(25) en (26) en
(30) 9901884-8 21 May/mai 1999
(21.05.1999)
SE
(30) 60/137,527 3 Jun/juin 1999 US
(03.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) NOVEL COMPOUNDS, THEIR USE
AND PREPARATION
NOUVEAUX COMPOSES, ET UTILI-
SATION ET PREPARATION DE CES
DERNIERS
(71) PHARMACIA & UPJOHN AB [SE/SE];
S-112 87 Stockholm (SE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) NILSSON, Björn [SE/SE]; Djäknegatan
15:650, S-754 23 Uppsala (SE). TEJBRANT,
Jan [SE/SE]; Bäckaskiftsvägen 13, S-122
42 Enskede (SE). PELCMAN, Benjamin
[SE/SE]; Döbelnsgatan 93, S-113 52 Stockholm
(SE). RINGBERG, Erik [SE/SE];
Gröna gatan 23F, S-753 26 Uppsala (SE).
THOR, Markus [SE/SE]; Gredelbyvägen
14C, S-741 40 Knivsta (SE). NILSSON,
Jonas [SE/SE]; Gnejsvägen 1B, S-752 43
Uppsala (SE). JÖNSSON, Mattias [SE/SE];
August Södermans väg 71, S-756 49 Uppsala
(SE).
(74) WIDÉN, Björn et al. / etc.; Pharmacia &
Upjohn AB, S-112 87 Stockholm (SE).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CR CU CZ DE DK DM EE ES FI
GB GD GE GH GM HR HU ID IL IN IS JP
KE KG KP KR KZ LC LK LR LS LT LU LV
MA MD MG MK MN MW MX NO NZ PL
PT RO RU SD SE SG SI SK SL TJ TM TR
TT TZ UA UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 273/00, 413/12, 417/12, 413/14,
A61K 31/395, A61P 33/00
(11) WO 00/76985
(21) PCT/EP00/04935
(13) A1
(22) 30 May/mai 2000 (30.05.2000)
(25) de (26) de
(30) 199 26 620.4 11 Jun/juin 1999
(11.06.1999)
DE
(43) 21 Dec/déc 2000 (21.12.2000)
(54) CYCLO-IMINO DEPSIPEPTIDES AND
THEIR UTILIZATION IN CONTROL-
LING ENDOPARASITES
CYCLO-IMINODEPSIPEPTIDES ET
LEUR UTILISATION POUR LUTTER
CONTRE LES ENDOPARASITES
(71) BAYER AKTIENGESELLSCHAFT
[DE/DE]; D-51368 Leverkusen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) JESCHKE, Peter [DE/DE]; Kalmüntener
Str. 44a, D-51467 Bergisch Gladbach
(DE). HARDER, Achim [DE/DE]; Europaring
54, D-51109 Köln (DE). VON
SAMSON-HIMMELSTJERNA, Georg
[DE/DE]; Neuenkamper Str. 21, D-42657
Solingen (DE). BONSE, Gerhard [DE/DE];
Gerstenkamp 1, D-51061 Köln (DE).
(74) BAYER AKTIENGESELLSCHAFT;
D-51368 Leverkusen (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID IL
IN IS JP KE KG KP KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
MZ NO NZ PL PT RO RU SD SE SG SI SK
SL TJ TM TR TT TZ UA UG US UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 277/04
(11) WO 00/76986 (13) A1
(21) PCT/EP00/03213
(22) 11 Apr/avr 2000 (11.04.2000)
(25) de (26) de
(30) 199 26 233.0 10 Jun/juin 1999
(10.06.1999)
DE
(43) 21 Dec/déc 2000 (21.12.2000)
(54) METHOD FOR THE PRODUCTION OF
THIAZOLIDIN
PROCEDE DE PREPARATION DE
THIAZOLIDINE
(71) PROBIODRUG GESELLSCHAFT
FÜR ARZNEIMITTELFORSCHUNG
MBH [DE/DE]; Weinbergweg 22, 06120
Halle/Saale (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) DEMUTH, Hans-Ulrich [DE/DE];
Hegelstrasse 14, 06114 Halle/Saale (DE).
KRUBER, Susanne [DE/DE]; Reilstrasse 9,
06114 Halle (DE).
(74) FORSTMEYER, Dietmar et al. / etc.;
Boeters & Bauer, Bereiteranger 15, 81541
München (DE).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CR CU CZ DE DK DM EE ES FI
GB GD GE GH GM HR HU ID IL IN IS JP
KE KG KP KR KZ LC LK LR LS LT LU LV
MA MD MG MK MN MW MX NO NZ PL
PT RO RU SD SE SG SI SK SL TJ TM TR
TT TZ UA UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW SD SL SZ TZ UG
ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF
BJ CF CG CI CM GA GN GW ML MR NE
SN TD TG).
(51) 7 C07D 277/20, 277/36, 417/06, A61K
31/426, 31/427, A61P 25/28
(11) WO 00/76987 (13) A1
(21) PCT/US00/15069
(22) 31 May/mai 2000 (31.05.2000)
(25) en (26) en
(30) 60/138,544 10 Jun/juin 1999 US
(10.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) RHODANINE DERIVATIVES FOR USE
IN A METHOD OF INHIBITING AMY-
LOID PROTEIN AGGREGATION AND
IMAGING AMYLOID DEPOSITS
DERIVES DE RHODANINE UTILISES
DANS UN PROCEDE D’INHIBITION
DE L’AGREGATION DE PROTEINES
AMYLOIDES ET DE FORMATION
D’IMAGES DE DEPOTS AMYLOIDES
(71) WARNER-LAMBERT COMPANY
[US/US]; 201 Tabor Road, Morris Plains,
NJ 07950 (US). YAMANOUCHI PHAR-
MACEUTICAL COMPANY [JP/JP];
17-1, Hasune 3-chome, Itabashi Ku, Tokyo
174-8612 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) AUGELLI-SZAFRAN, Corinne, Elizabeth
[US/US]; 2812 Aspen Ridge Drive,
Ann Arbor, MI 48103 (US). GLASE, Shelly,
Ann [US/US]; 4468 Hillside Court, Ann
Arbor, MI 48105 (US). WALKER, Lary,
Craswell [US/US]; 4890 North Ridgeside
Circle, Ann Arbor, MI 48105 (US).
YASUNAGA, Tomoyuki [JP/JP]; 13-18,
Minami 3-chome, Ushiku, Ibaraki 300-1222
(JP).
(74) RYAN, M., Andrea; Warner-Lambert Company,
201 Tabor Road, Morris Plains, NJ
07950 (US) et al. / etc.
(81) AE AG AL AU BA BB BG BR CA CN CR
CU CZ DM DZ EE GD GE HR HU ID IL IN
IS JP KP KR LC LK LR LT LV MA MG MK
MN MX MZ NO NZ PL RO SG SI SK SL TR
TT UA US UZ VN YU ZA.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 277/36, 417/06, 417/10, 417/14,
A61K 31/426, 31/427, 51/04, A61P 25/28
// A61K 123:00
(11) WO 00/76988
(21) PCT/US00/15072
(13) A1
(22) 31 May/mai 2000 (31.05.2000)
(25) en (26) en
(30) 60/138,545 10 Jun/juin 1999
(10.06.1999)
US
(43) 21 Dec/déc 2000 (21.12.2000)
(54) RHODANINE DERIVATIVES AND
THEIR USE IN INHIBITING AND
IMAGING AMYLOIDS