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PCT/2000/51 - World Intellectual Property Organization

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<strong>51</strong>/<strong>2000</strong><br />

19106 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 21 Dec/déc <strong>2000</strong><br />

NOUVEAUX COMPOSES DERIVES DE<br />

NUCLEOSIDES, LEURS PROCEDES<br />

DE PREPARATION ET LES COMPO-<br />

SITIONS PHARMACEUTIQUES EN<br />

RENFERMANT<br />

(71) LABORATOIRES LAPHAL S.A.<br />

[FR/FR]; Avenue de Provence, F-13190<br />

Allauch (FR).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) VLIEGHE, Patrick [FR/FR]; Résidence<br />

Prado-Plaza, Bâtiment A, 30, rue des<br />

Mousses, F-13008 Marseille (FR). KRAUS,<br />

Jean-Louis [FR/FR]; 24, boulevard des Platanes,<br />

F-13008 Marseille (FR). CLERC,<br />

Thierry [FR/FR]; 286, Chemin du Roucas<br />

Blanc, F-13007 Marseille (FR). SALLES,<br />

Jean-Pierre [FR/FR]; Chemin de Vergon,<br />

F-13<strong>51</strong>0 Eguilles (FR).<br />

(74) BURTIN, Jean-François; Cabinet GEFIB,<br />

85, rue Anatole France, F-92300 Levallois<br />

Perret (FR).<br />

(81) AL AU BR CA CN CZ HU IL JP KR LT LV<br />

MK MX NO NZ PL RO RU SI US VN.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA (BF<br />

BJ CF CG CI CM GA GN GW ML MR NE<br />

SN TD TG).<br />

(<strong>51</strong>) 7 C07H 21/00, C07K 5/00<br />

(11) WO 00/77021 (13) A1<br />

(21) <strong>PCT</strong>/US00/1<strong>51</strong>35<br />

(22) 1 Jun/juin <strong>2000</strong> (01.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,632 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) 48 HUMAN SECRETED PROTEINS<br />

48 PROTEINES HUMAINES SECRE-<br />

TEES<br />

(71) HUMAN GENOME SCIENCES, INC.<br />

[US/US]; 9410 Key West Avenue, Rockville,<br />

MD 20850 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(71, 72) ROSEN, Craig, A. [US/US]; 22400<br />

Rolling Hill Road, Laytonsville, MD 20882<br />

(US).<br />

(72, 75) RUBEN, Steven, M. [US/US]; 18528<br />

Heritage Hills Drive, Laytonsville, MD<br />

20882 (US). KOMATSOULIS, George,<br />

A. [US/US]; 9<strong>51</strong>8 Garwood Street, Silver<br />

Spring, MD 20901 (US).<br />

(74) HOOVER, Kenley, K. et al. / etc.; Human<br />

Genome Sciences, Inc., 9410 Key West Avenue,<br />

Rockville, MD 20850 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

Published / Publiée :(c)<br />

(<strong>51</strong>) 7 C07H 21/00, C07K 2/00, C12P 19/34,<br />

C12N 15/12<br />

(11) WO 00/77022 (13) A1<br />

(21) <strong>PCT</strong>/US00/1<strong>51</strong>36<br />

(22) 1 Jun/juin <strong>2000</strong> (01.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,629 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) 50 HUMAN SECRETED PROTEINS<br />

50 PROTEINES HUMAINES SECRE-<br />

TEES<br />

(71) HUMAN GENOME SCIENCES, INC.<br />

[US/US]; 9410 Key West Avenue, Rockville,<br />

MD 20850 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) ROSEN, Craig, A. [US/US]; 22400<br />

Rolling Hill Road, Laytonsville, MD 20882<br />

(US). RUBEN, Steven, M. [US/US]; 18528<br />

Heritage Hill Drive, Olney, MD 20832 (US).<br />

KOMATSOULIS, George, A. [US/US];<br />

9<strong>51</strong>8 Garwood Street, Silver Spring, MD<br />

20901 (US).<br />

(74) HOOVER, Kenley, K. et al. / etc.; Human<br />

Genome Sciences, Inc., 9410 Key West Avenue,<br />

Rockville, MD 20850 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07H 21/02, 21/04, C12N 15/00, 15/09,<br />

15/63, 15/70, 15/74, 15/63, 15/85, 15/87,<br />

A61K 38/00, C07K 2/00, 4/00, 5/00, 7/00,<br />

14/00, 16/00, 17/00, 1/00<br />

(11) WO 00/77023 (13) A1<br />

(21) <strong>PCT</strong>/US00/14964<br />

(22) 1 Jun/juin <strong>2000</strong> (01.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,627 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) 48 HUMAN SECRETED PROTEINS<br />

48 PROTEINES SECRETEES HU-<br />

MAINES<br />

(71) HUMAN GENOME SCIENCES, INC.<br />

[US/US]; 9410 Key West Avenue, Rockville,<br />

MD 20850 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) ROSEN, Craig, A. [US/US]; 22400<br />

Rolling Hill Road, Laytonsville, MD 20882<br />

(US). RUBEN, Steven, M. [US/US]; 18528<br />

Heritage Hills Drive, Laytonsville, MD<br />

20882 (US). KOMATSOULIS, George,<br />

A. [US/US]; 9<strong>51</strong>8 Garwood Street, Silver<br />

Spring, MD 20901 (US).<br />

(74) HOOVER, Kenley, K. et al. / etc.; Human<br />

Genome Sciences, Inc., 9410 Key West Avenue,<br />

Rockville, MD 20850 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07H 21/02, 21/04, A01K 67/00<br />

(11) WO 00/77024 (13) A1<br />

(21) <strong>PCT</strong>/US00/16412<br />

(22) 14 Jun/juin <strong>2000</strong> (14.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/333,229 14 Jun/juin 1999 US<br />

(14.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) CAMELLO GENE FAMILY AND USES<br />

THEREOF<br />

FAMILLE DE GENES CAMELLO ET<br />

L’UTILISATION DESDITS GENES<br />

(71) NEW YORK BLOOD CENTER, INC.<br />

[US/US]; 310 East 67th Street, New York,<br />

NY 10021 (US).<br />

(72) BELYAVSKY, Alexander V.; 504 East 63rd<br />

Street, #10L, New York, NY 10021 (US).<br />

POPSUEVA, Anna, E.; Antti Korpintie<br />

4A8, FIN-00600 Helsinki (FI). LUCHIN-<br />

SKAYA, Natalia N.; 56-2 Vavilova Street,<br />

#212, Moscow, 117296 (RU).<br />

(74) GEORGE, Kenneth, P. et al. / etc.; Amster,<br />

Rothstein & Ebenstein, 90 Park Avenue, New<br />

York, NY 10016 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07J 73/00, 75/00<br />

(11) WO 00/77025<br />

(21) <strong>PCT</strong>/HU00/00048<br />

(13) A1<br />

(22) 26 May/mai <strong>2000</strong> (26.05.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) P 9901938 10 Jun/juin 1999<br />

(10.06.1999)<br />

HU<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) NEW PROCESS FOR THE SYNTHESIS<br />

OF 17β-HYDROXY-17α-METHYL-2-<br />

OXA-5α-ANDROSTANE-3-ONE

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