PCT/2000/51 - World Intellectual Property Organization

51/2000
19102 PCT Gazette - Section I - Gazette du PCT 21 Dec/déc 2000
1007 Market Street, Wilmington, DE 19898
(US).
(81) AU BR CA CN CZ EE HU IL IN JP KR LT
LV MX NO NZ PL RO SG SI SK TR UA VN
ZA.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE).
Published / Publiée :(c)
(51) 7 C07D 471/16, A61K 31/554, 31/4985,
31/5517, A61P 25/00, C07D 487/16 //
(C07D 471/16, 241:00, 221:00, 209:00)
(C07D 471/16, 243:00, 221:00, 209:00)
(C07D 487/16, 241:00, 223:00, 209:00)
(11) WO 00/77002 (13) A1
(21) PCT/US00/16498
(22) 15 Jun/juin 2000 (15.06.2000)
(25) en (26) en
(30) 60/139,321 15 Jun/juin 1999 US
(15.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) SUBSTITUTED HETEROCYCLE
FUSED GAMMA-CARBOLINES
GAMMA-CARBOLINES FUSIONNEES
A HETEROCYCLE SUBSTITUE
(71) DU PONT PHARMACEUTICALS
COMPANY [US/US]; 974 Centre Road,
WR-1ST18, Wilmington, DE 19807 (US).
(72) ROBICHAUD, Albert, J.; 120 Stonegate
Drive, Landenberg, PA 19350 (US). LEE,
Taekyu; 110 Berry Drive, Wilmington,
DE 19808 (US). DENG, Wei; 1314 Copley
Drive, Wilmington, DE 19803 (US).
MITCHELL, Ian, S.; Apartment #601, 201
South 25th Street, Philadelphia, PA 19103
(US). YANG, Michael, Guang; 15 South
Hampshire Court, Wilmington, DE 19807
(US). HAYDAR, Simon; 49 Brendan Lane,
Niskayuna, NY 12309 (US). CHEN, Wenting;
252 Apple Drive, Exton, PA 19341
(US). MC CLUNG, Christopher, D.; 2129
Biddle Street, Wilmington, DE 19805 (US).
CALVELLO, Emilie, J., B.; 18 North
Roberts Road, Bryn Mawr, PA 19010 (US).
ZAWROTNY, David, M.; 225 Laurence
Drive, Moorestown, NJ 08057 (US).
(74) LARSEN, Scott, K.; Du Pont Pharmaceuticals
Company, Legal Patent Records Center,
1007 Market Street, Wilmington, DE 19898
(US).
(81) AU BR CA CN CZ EE HU IL IN JP KR LT
LV MX NO NZ PL RO SG SI SK TR UA VN
ZA.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE).
Published / Publiée :(c)
(51) 7 C07D 487/04, A61K 31/5025, A61P 31/04,
1/04
(11) WO 00/77003
(21) PCT/JP00/03895
(13) A1
(22) 15 Jun/juin 2000 (15.06.2000)
(25) ja (26) ja
(30) 11/167679 15 Jun/juin 1999
(15.06.1999)
JP
(43) 21 Dec/déc 2000 (21.12.2000)
(54) OPTICALLY ACTIVE PYRROLOPYRI-
DAZINE COMPOUNDS
COMPOSES DE PYRROLOPYRIDA-
ZINE OPTIQUEMENT ACTIFS
(71) SANKYO COMPANY, LIMITED [JP/JP];
5-1, Nihonbashi Honcho 3-chome, Chuo-ku,
Tokyo 103-8426 (JP). UBE INDUSTRIES,
LTD. [JP/JP]; 12-32, Nishi Honmachi
1-chome, Ube-shi, Yamaguchi 755-0052
(JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) HAGIHARA, Masahiko [JP/JP]; Ube
Research Laboratory, Ube Industries Ltd.,
1978-5, Oaza Kogushi, Ube-shi, Yamaguchi
755-0067 (JP). SHIBAKAWA, Nobuhiko
[JP/JP]; Ube Research Laboratory, Ube Industries
Ltd., 1978-5, Oaza Kogushi, Ube-shi,
Yamaguchi 755-0067 (JP). MATSUNOBU,
Keiji [JP/JP]; Ube Research Laboratory,
Ube Industries Ltd., 1978-5, Oaza Kogushi,
Ube-shi, Yamaguchi 755-0067 (JP). FUJI-
WARA, Hiroshi [JP/JP]; Ube Research Laboratory,
Ube Industries Ltd., 1978-5, Oaza
Kogushi, Ube-shi, Yamaguchi 755-0067 (JP).
ITO, Keiichi [JP/JP]; Sankyo Company,
Limited, 2-58, Hiromachi 1-chome, Shinagawa-ku,
Tokyo 140-8710 (JP).
(74) NAKAMURA, Minoru et al. / etc.; Room
646, Shin-Tokyo Bldg, 3-1, Marunouchi
3-chome, Chiyoda-ku, Tokyo 100-8355 (JP).
(81) AU BR CA CN CZ HU ID IL IN KR MX NO
NZ PL RU TR US ZA.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE).
(51) 7 C07D 487/04, 471/02, A61K 31/437,
31/4353, 31/55
(11) WO 00/77004 (13) A1
(21) PCT/US00/16683
(22) 14 Jun/juin 2000 (14.06.2000)
(25) en (26) en
(30) 60/138,135 14 Jun/juin 1999 US
(14.06.1999)
(30) 09/332,318 14 Jun/juin 1999 US
(14.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) 1-AZATRICYCLIC-4-BENZYLPIPER-
AZINES
1-AZATRICYCLICO-4-BENZYLPIPE-
RAZINES
(71) NEUROGEN CORPORATION [US/US];
35 Northeast Industrial Road, Branford, CT
06405 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ZHANG, Sophie [CN/US]; Apartment
11-74, 140 Mill Street, East Haven, CT 06512
(US). HODGETTS, Kevin [US/US]; Valley
Court #10, 1171 Main Street, Branford,
CT 06405 (US). RACHWAL, Stanislaw
[PL/US]; 133 Montoya Drive, Branford,
CT 06405 (US). ROSEWATER, Daniel
[US/US]; 69 Church Street #2, Branford,
CT 06405 (US). THURKAUF, Andrew
[US/US]; 16 Fox Den Road, Danbury, CT
06811 (US).
(74) SARUSSI, Steven, J.; McDonnell Boehnen
Hulbert & Berghoff, Suite 3200, 300 South
Wacker Drive, Chicago, IL 60606 (US).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CR CU CZ DE DK DM DZ EE
ES FI GB GD GE GH GM HR HU ID IL IN
IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MA MD MG MK MN MW MX NO
NZ PL PT RO RU SD SE SG SI SK SL TJ TM
TR TT TZ UA UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07D 491/052, C08G 73/06, G02B 5/23,
G03C 1/73, C07D 221/18, C08K 5/3415 //
(C07D 491/052, 311:00, 221:00)
(11) WO 00/77005 (13) A1
(21) PCT/EP00/05162
(22) 5 Jun/juin 2000 (05.06.2000)
(25) en (26) en
(30) 99/07356 10 Jun/juin 1999 FR
(10.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) NAPHTHOPYRANS ANNELATED
IN C5-C6 WITH A LACTAM-TYPE C6
RING AND COMPOSITIONS AND
(CO)POLYMER CONTAINING THEM
NAPHTOPYRANES ANNELES EN
C5-C6 ET PORTEURS EN C6 D’UN
NOYAU DU TYPE LACTAME, ET
COMPOSITIONS ET (CO)POLYMERES
RENFERMANT LESDITS COMPOSES
(71) CORNING S.A. [FR/FR]; 7 bis, avenue de
Valvins, F-77920 Samois-sur-Seine (FR).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BREYNE, Olivier [FR/FR]; 5, rue Rosset,
F-69004 Lyon (FR).
(74) LE ROUX, Martine et al. / etc.; Cabinet
Beau De Loménie, 158, rue de l’Université,
F-75340 Paris Cedex 07 (FR).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID IL
IN IS JP KE KG KP KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
MZ NO NZ PL PT RO RU SD SE SG SI SK
SL TJ TM TR TT TZ UA UG US UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(a)
(51) 7 C07D 491/052
(11) WO 00/77006
(21) PCT/IB00/00760
(13) A1
(22) 7 Jun/juin 2000 (07.06.2000)
(25) en (26) en
(30) 865/DEL/99 11 Jun/juin 1999
(11.06.1999)
IN
(30) 09/412,455 4 Oct/oct 1999
(04.10.1999)
US
(43) 21 Dec/déc 2000 (21.12.2000)
(54) PROCESS FOR THE PREPARATION
OF 1,8-DISUBSTITUTED-1,3,4,9-