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PCT/2000/51 - World Intellectual Property Organization

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<strong>51</strong>/<strong>2000</strong><br />

21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19095<br />

Road, Heaton Moor, Stockport SK4 4LD<br />

(GB). CAMP, Nicholas, Paul [GB/GB]; Flat<br />

2, Sliver Court, Fosseway, Nailsea, Avon<br />

BS48 2BX (GB). JONES, Stuart, Donald<br />

[GB/GB]; 17 Oakwood Drive, Prestbury,<br />

Cheshire SK10 4HG (GB). MORGAN,<br />

Phillip, John [GB/GB]; 11 Woodland Avenue,<br />

Congleton, Cheshire CW12 1LN (GB).<br />

RICHARDS, Simon, James [GB/GB];<br />

39 Vicarage Road, Blackrod, Bolton BL6<br />

5DA (GB). WYLIE, William, Alexander<br />

[GB/GB]; Flat 4, 39 Station Road, Reddish,<br />

Stockport SK5 6LT (GB). MASTERS, John,<br />

Joseph [US/US]; 12047 Flint Stone Court,<br />

Fishers, IN 46038 (US). WILEY, Michael,<br />

Robert [US/US]; 7725 Langwood Drive,<br />

Indianapolis, IN 46268 (US).<br />

(74) HAY, Martin, A.; Martin A. Hay & Co., 13<br />

Queen Victoria Street, Macclesfield, Cheshire<br />

SK11 6LP (GB).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07D 211/14, 271/12, 239/42, 231/12,<br />

277/30, 263/32, A61K 31/4409, A61P 37/00,<br />

31/18<br />

(11) WO 00/76972 (13) A1<br />

(21) <strong>PCT</strong>/US00/15736<br />

(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,886 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(30) 09/330,810 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) N-CYCLOPENTYL MODULATORS OF<br />

CHEMOKINE RECEPTOR ACTIVITY<br />

MODULATEURS N-CYCLOPENTY-<br />

LIQUES DE L’ACTIVITE DU RECEP-<br />

TEUR DE LA CHIMIOKINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). HILFIKER, Kerry, A. [US/US];<br />

126 East Lincoln Avenue, Rahway, NJ<br />

07065-0907 (US). MACCOSS, Malcolm<br />

[GB/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). CHAPMAN, Kevin, T.<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). LOEBACH, Jennifer,<br />

L. [US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). MILLS, Sander,<br />

G. [US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). GUTHIKONDA,<br />

Ravi, N. [US/US]; 126 East Lincoln Avenue,<br />

Rahway, NJ 07065-0907 (US). SHAH,<br />

Shrenik, K. [US/US]; 126 East Lincoln Avenue,<br />

Rahway, NJ 07065-0907 (US). KIM,<br />

Dooseop [KR/US]; 126 East Lincoln Avenue,<br />

Rahway, NJ 07065-0907 (US). SHEN,<br />

Dong-Ming [US/US]; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

OATES, Bryan [US/US]; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

(74) MERCK & CO., INC.; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KR KZ LC LK LR LS LT<br />

LU LV MA MD MG MK MN MW MX MZ<br />

NO NZ PL PT RO RU SD SE SG SI SK SL<br />

TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

Published / Publiée :(c)<br />

(<strong>51</strong>) 7 C07D 211/54, 211/56, 401/06, 403/06,<br />

409/06, 413/06, A61K 31/4453, C07F<br />

31/4453<br />

(11) WO 00/76973 (13) A1<br />

(21) <strong>PCT</strong>/US00/15724<br />

(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/139,078 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) N-CYCLOPENTYL MODULATORS OF<br />

CHEMOKINE RECEPTOR ACTIVITY<br />

MODULATEURS N-CYCLOPENTY-<br />

LIQUES DE L’ACTIVITE DU RECEP-<br />

TEUR DE LA CHIMIOKINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). CHAPMAN, Kevin, T. [US/US];<br />

126 East Lincoln Avenue, Rahway, NJ<br />

07065-0907 (US). LOEBACH, Jennifer, L.<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). MACCOSS, Malcolm<br />

[GB/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). MILLS, Sander, G.<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). OATES, Bryan<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US).<br />

(74) MERCK & CO., INC.; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KR KZ LC LK LR LS LT<br />

LU LV MA MD MG MK MN MW MX MZ<br />

NO NZ PL PT RO RU SD SE SG SI SK SL<br />

TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07D 211/60, 207/16, 241/24, A61K<br />

31/40, 31/4523, 31/496, A61P 43/00<br />

(11) WO 00/76974 (13) A2<br />

(21) <strong>PCT</strong>/US00/16188<br />

(22) 13 Jun/juin <strong>2000</strong> (13.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,972 14 Jun/juin 1999 US<br />

(14.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) OLIGOMERS AND POLYMERS OF<br />

CYCLIC IMINO CARBOXYLIC ACIDS<br />

OLIGOMERES ET POLYMERES<br />

D’ACIDES IMINO CARBOXYLIQUES<br />

CYCLIQUES<br />

(71) WISCONSIN ALUMNI RESEARCH<br />

FOUNDATION [US/US]; 614 Walnut<br />

Street, Madison, WI 53707-7365 (US).<br />

(72) GELLMAN, Samuel, H.; 222 Glacier<br />

Drive, Madison, WI 53705 (US). HUCK,<br />

Bayard, R.; 304 Princeton Avenue, #6,<br />

Madison, WI 53705 (US). RICHARDS,<br />

Michele, R.; 155 Lakewood Gardens Lane,<br />

Madison, WI 53704 (US).<br />

(74) LEONE, Joseph, T. et al. / etc.; DeWitt Ross<br />

& Stevens S.C., 8000 Excelsior Drive, Madison,<br />

WI 53717-1914 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07D 213/22 // 213/84, 401/04<br />

(11) WO 00/76975<br />

(21) <strong>PCT</strong>/JP00/03831<br />

(13) A1<br />

(22) 13 Jun/juin <strong>2000</strong> (13.06.<strong>2000</strong>)<br />

(25) ja (26) ja<br />

(30) 11/167308 14 Jun/juin 1999<br />

(14.06.1999)<br />

JP<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) PROCESS FOR THE PRODUCTION OF<br />

2-PYRIDYLPYRIDINE DERIVATIVES<br />

PROCEDE DE PRODUCTION DE DE-<br />

RIVES DE 2-PYRIDYLPYRIDINE<br />

(71) SANKIO CHEMICAL CO., LTD. [JP/JP];<br />

1-1, Kyobashi 1-chome, Chuo-ku, Tokyo 104-<br />

0031 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) IKEUCHI, Fumiaki [JP/JP]; Sankio<br />

Chemical Co., Ltd., Synthetic Chemistry<br />

Research Laboratory, 2-3, Higashiyawata<br />

5-chome, Hiratsuka-shi, Kanagawa 254-0016<br />

(JP). SHINTOU, Taichi [JP/JP]; Sankio<br />

Chemical Co., Ltd., Synthetic Chemistry<br />

Research Laboratory, 2-3, Higashiyawata

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