PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
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<strong>51</strong>/<strong>2000</strong><br />
21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19095<br />
Road, Heaton Moor, Stockport SK4 4LD<br />
(GB). CAMP, Nicholas, Paul [GB/GB]; Flat<br />
2, Sliver Court, Fosseway, Nailsea, Avon<br />
BS48 2BX (GB). JONES, Stuart, Donald<br />
[GB/GB]; 17 Oakwood Drive, Prestbury,<br />
Cheshire SK10 4HG (GB). MORGAN,<br />
Phillip, John [GB/GB]; 11 Woodland Avenue,<br />
Congleton, Cheshire CW12 1LN (GB).<br />
RICHARDS, Simon, James [GB/GB];<br />
39 Vicarage Road, Blackrod, Bolton BL6<br />
5DA (GB). WYLIE, William, Alexander<br />
[GB/GB]; Flat 4, 39 Station Road, Reddish,<br />
Stockport SK5 6LT (GB). MASTERS, John,<br />
Joseph [US/US]; 12047 Flint Stone Court,<br />
Fishers, IN 46038 (US). WILEY, Michael,<br />
Robert [US/US]; 7725 Langwood Drive,<br />
Indianapolis, IN 46268 (US).<br />
(74) HAY, Martin, A.; Martin A. Hay & Co., 13<br />
Queen Victoria Street, Macclesfield, Cheshire<br />
SK11 6LP (GB).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG US UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07D 211/14, 271/12, 239/42, 231/12,<br />
277/30, 263/32, A61K 31/4409, A61P 37/00,<br />
31/18<br />
(11) WO 00/76972 (13) A1<br />
(21) <strong>PCT</strong>/US00/15736<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,886 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(30) 09/330,810 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) N-CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS N-CYCLOPENTY-<br />
LIQUES DE L’ACTIVITE DU RECEP-<br />
TEUR DE LA CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). HILFIKER, Kerry, A. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065-0907 (US). MACCOSS, Malcolm<br />
[GB/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). CHAPMAN, Kevin, T.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). LOEBACH, Jennifer,<br />
L. [US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MILLS, Sander,<br />
G. [US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). GUTHIKONDA,<br />
Ravi, N. [US/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065-0907 (US). SHAH,<br />
Shrenik, K. [US/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065-0907 (US). KIM,<br />
Dooseop [KR/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065-0907 (US). SHEN,<br />
Dong-Ming [US/US]; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
OATES, Bryan [US/US]; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
Published / Publiée :(c)<br />
(<strong>51</strong>) 7 C07D 211/54, 211/56, 401/06, 403/06,<br />
409/06, 413/06, A61K 31/4453, C07F<br />
31/4453<br />
(11) WO 00/76973 (13) A1<br />
(21) <strong>PCT</strong>/US00/15724<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,078 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) N-CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS N-CYCLOPENTY-<br />
LIQUES DE L’ACTIVITE DU RECEP-<br />
TEUR DE LA CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). CHAPMAN, Kevin, T. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065-0907 (US). LOEBACH, Jennifer, L.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MACCOSS, Malcolm<br />
[GB/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MILLS, Sander, G.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). OATES, Bryan<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07D 211/60, 207/16, 241/24, A61K<br />
31/40, 31/4523, 31/496, A61P 43/00<br />
(11) WO 00/76974 (13) A2<br />
(21) <strong>PCT</strong>/US00/16188<br />
(22) 13 Jun/juin <strong>2000</strong> (13.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,972 14 Jun/juin 1999 US<br />
(14.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) OLIGOMERS AND POLYMERS OF<br />
CYCLIC IMINO CARBOXYLIC ACIDS<br />
OLIGOMERES ET POLYMERES<br />
D’ACIDES IMINO CARBOXYLIQUES<br />
CYCLIQUES<br />
(71) WISCONSIN ALUMNI RESEARCH<br />
FOUNDATION [US/US]; 614 Walnut<br />
Street, Madison, WI 53707-7365 (US).<br />
(72) GELLMAN, Samuel, H.; 222 Glacier<br />
Drive, Madison, WI 53705 (US). HUCK,<br />
Bayard, R.; 304 Princeton Avenue, #6,<br />
Madison, WI 53705 (US). RICHARDS,<br />
Michele, R.; 155 Lakewood Gardens Lane,<br />
Madison, WI 53704 (US).<br />
(74) LEONE, Joseph, T. et al. / etc.; DeWitt Ross<br />
& Stevens S.C., 8000 Excelsior Drive, Madison,<br />
WI 53717-1914 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 C07D 213/22 // 213/84, 401/04<br />
(11) WO 00/76975<br />
(21) <strong>PCT</strong>/JP00/03831<br />
(13) A1<br />
(22) 13 Jun/juin <strong>2000</strong> (13.06.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/167308 14 Jun/juin 1999<br />
(14.06.1999)<br />
JP<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) PROCESS FOR THE PRODUCTION OF<br />
2-PYRIDYLPYRIDINE DERIVATIVES<br />
PROCEDE DE PRODUCTION DE DE-<br />
RIVES DE 2-PYRIDYLPYRIDINE<br />
(71) SANKIO CHEMICAL CO., LTD. [JP/JP];<br />
1-1, Kyobashi 1-chome, Chuo-ku, Tokyo 104-<br />
0031 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) IKEUCHI, Fumiaki [JP/JP]; Sankio<br />
Chemical Co., Ltd., Synthetic Chemistry<br />
Research Laboratory, 2-3, Higashiyawata<br />
5-chome, Hiratsuka-shi, Kanagawa 254-0016<br />
(JP). SHINTOU, Taichi [JP/JP]; Sankio<br />
Chemical Co., Ltd., Synthetic Chemistry<br />
Research Laboratory, 2-3, Higashiyawata