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PCT/2000/51 - World Intellectual Property Organization

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<strong>51</strong>/<strong>2000</strong><br />

19010 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 21 Dec/déc <strong>2000</strong><br />

MX MZ NO NZ PL RO SG SI SK SL TR TT<br />

TZ UA US UZ VN YU ZA.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 A61K 31/44<br />

(11) WO 00/76509 (13) A1<br />

(21) <strong>PCT</strong>/US00/04268<br />

(22) 18 Feb/fév <strong>2000</strong> (18.02.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/334,304 16 Jun/juin 1999 US<br />

(16.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) NASAL DELIVERY OF APOMOR-<br />

PHINE<br />

ADMINISTRATION D’APOMOR-<br />

PHINE PAR VOIE NASALE<br />

(71) NASTECH PHARMACEUTICAL COM-<br />

PANY, INC. [US/US]; 45 Davids Drive,<br />

Hauppauge, NY 11788 (US).<br />

(72) ACHARI, Raja, G.; 52 Indian Run, Millington,<br />

NJ 07946 (US). AHMED, Shamim; 64<br />

Coventry Lane, Central Islip, NY 11722 (US).<br />

BEHL, Charanjit, R.; Apartment 1-A, 658<br />

Veterans Memorial HIghway, Hauppauge,<br />

NY 11788 (US). DEMEIRELES, Jorge, C.;<br />

33 Renee Road, Syosset, NY 11791 (US).<br />

LIU, Tianquing; 35 Coventry Lane, Central<br />

Islip, NY 11722 (US). ROMEO, Vincent,<br />

D.; 104 Harbor Lane, Massapequa Park,<br />

NY 11762 (US). SILENO, Anthony, P.; 10<br />

Highview Boulevard, Brookhaven Hamlet,<br />

NY 11719 (US).<br />

(74) BODNER, Gerald, T.; Hoffmann & Baron,<br />

LLP, 6900 Jericho Turnpike, Syosset, NY<br />

11791 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW SD SL SZ TZ UG<br />

ZW); EA (AM AZ BY KG KZ MD RU TJ<br />

TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF<br />

BJ CF CG CI CM GA GN GW ML MR NE<br />

SN TD TG).<br />

(<strong>51</strong>) 7 A61K 31/445, C07D 211/40<br />

(11) WO 00/76<strong>51</strong>0<br />

(21) <strong>PCT</strong>/US00/15490<br />

(13) A1<br />

(22) 6 Jun/juin <strong>2000</strong> (06.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,353 10 Jun/juin 1999<br />

(10.06.1999)<br />

US<br />

(30) 60/179,267 31 Jan/jan <strong>2000</strong><br />

(31.01.<strong>2000</strong>)<br />

US<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) DERMAL ANESTHETIC AGENTS<br />

AGENTS<br />

MIQUES<br />

ANESTHESIQUES DER-<br />

(71) BRIDGE PHARMA, INC. [US/US]; 902<br />

Contento Street, Sarasota, FL 34242 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) ABERG, A., K., Gunnar [SE/US];<br />

902 Contento Street, Sarasota, FL 34242<br />

(US). WRIGHT, George, L. [US/US]; 298<br />

Highland Street, Worcester, MA 01602 (US).<br />

CHEN, Jan, L. [CN/US]; 216B East Mountain<br />

Street, Worcester, MA 01608 (US).<br />

(74) LEMACK, Kevin, S. et al. / etc.; Nields,<br />

Lemack & Dingman, Suite 8, 176 E. Main<br />

Street, Westboro, MA 01581 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 A61K 31/445, C07D 211/06, 401/08,<br />

409/08<br />

(11) WO 00/76<strong>51</strong>1 (13) A1<br />

(21) <strong>PCT</strong>/US00/15657<br />

(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,763 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) CYCLOPENTYL MODULATORS OF<br />

CHEMOKINE RECEPTOR ACTIVITY<br />

MODULATEURS CYCLOPENTYLE DE<br />

L’ACTIVITE DES RECEPTEURS DE LA<br />

CHIMIOKINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FINKE, Paul, E. [US/US]; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

MACCOSS, Malcolm [GB/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). MILLS, Sander, G. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). OATES, Bryan [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(74) MERCK & CO., INC.; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KR KZ LC LK LR LS LT<br />

LU LV MA MD MG MK MN MW MX MZ<br />

NO NZ PL PT RO RU SD SE SG SI SK SL<br />

TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 A61K 31/445, 31/4453, 31/454, C07D<br />

211/56, 211/92<br />

(11) WO 00/76<strong>51</strong>2 (13) A1<br />

(21) <strong>PCT</strong>/US00/15755<br />

(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/139,067 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) CYCLOPENTYL MODULATORS OF<br />

CHEMOKINE RECEPTOR ACTIVITY<br />

MODULATEURS CYCLOPENTY-<br />

LIQUES DE L’ACTIVITE DU RECEP-<br />

TEUR DE LA CHIMIOKINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). CHAPMAN, Kevin, T. [US/US];<br />

126 East Lincoln Avenue, Rahway, NJ<br />

07065-0907 (US). MACCOSS, Malcolm<br />

[GB/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). MILLS, Sander, G.<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US). OATES, Bryan<br />

[US/US]; 126 East Lincoln Avenue, Rahway,<br />

NJ 07065-0907 (US).<br />

(74) MERCK & CO., INC.; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065-0907 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KR KZ LC LK LR LS LT<br />

LU LV MA MD MG MK MN MW MX MZ<br />

NO NZ PL PT RO RU SD SE SG SI SK SL<br />

TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />

ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 A61K 31/445, 31/4453, 31/4465, C07D<br />

211/56, 211/92<br />

(11) WO 00/76<strong>51</strong>3 (13) A1<br />

(21) <strong>PCT</strong>/US00/15765<br />

(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/138,872 11 Jun/juin 1999 US<br />

(11.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) CYCLOPENTYL MODULATORS OF<br />

CHEMOKINE RECEPTOR ACTIVITY<br />

MODULATEURS CYCLOPENTY-<br />

LIQUES DE L’ACTIVITE DU RECEP-<br />

TEUR DE LA CHIMIOKINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907<br />

(US). LOEBACH, Jennifer, L. [US/US];

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