PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
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<strong>51</strong>/<strong>2000</strong><br />
19010 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 21 Dec/déc <strong>2000</strong><br />
MX MZ NO NZ PL RO SG SI SK SL TR TT<br />
TZ UA US UZ VN YU ZA.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/44<br />
(11) WO 00/76509 (13) A1<br />
(21) <strong>PCT</strong>/US00/04268<br />
(22) 18 Feb/fév <strong>2000</strong> (18.02.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 09/334,304 16 Jun/juin 1999 US<br />
(16.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) NASAL DELIVERY OF APOMOR-<br />
PHINE<br />
ADMINISTRATION D’APOMOR-<br />
PHINE PAR VOIE NASALE<br />
(71) NASTECH PHARMACEUTICAL COM-<br />
PANY, INC. [US/US]; 45 Davids Drive,<br />
Hauppauge, NY 11788 (US).<br />
(72) ACHARI, Raja, G.; 52 Indian Run, Millington,<br />
NJ 07946 (US). AHMED, Shamim; 64<br />
Coventry Lane, Central Islip, NY 11722 (US).<br />
BEHL, Charanjit, R.; Apartment 1-A, 658<br />
Veterans Memorial HIghway, Hauppauge,<br />
NY 11788 (US). DEMEIRELES, Jorge, C.;<br />
33 Renee Road, Syosset, NY 11791 (US).<br />
LIU, Tianquing; 35 Coventry Lane, Central<br />
Islip, NY 11722 (US). ROMEO, Vincent,<br />
D.; 104 Harbor Lane, Massapequa Park,<br />
NY 11762 (US). SILENO, Anthony, P.; 10<br />
Highview Boulevard, Brookhaven Hamlet,<br />
NY 11719 (US).<br />
(74) BODNER, Gerald, T.; Hoffmann & Baron,<br />
LLP, 6900 Jericho Turnpike, Syosset, NY<br />
11791 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES FI<br />
GB GD GE GH GM HR HU ID IL IN IS JP<br />
KE KG KP KR KZ LC LK LR LS LT LU LV<br />
MA MD MG MK MN MW MX NO NZ PL<br />
PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT TZ UA UG UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(<strong>51</strong>) 7 A61K 31/445, C07D 211/40<br />
(11) WO 00/76<strong>51</strong>0<br />
(21) <strong>PCT</strong>/US00/15490<br />
(13) A1<br />
(22) 6 Jun/juin <strong>2000</strong> (06.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,353 10 Jun/juin 1999<br />
(10.06.1999)<br />
US<br />
(30) 60/179,267 31 Jan/jan <strong>2000</strong><br />
(31.01.<strong>2000</strong>)<br />
US<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) DERMAL ANESTHETIC AGENTS<br />
AGENTS<br />
MIQUES<br />
ANESTHESIQUES DER-<br />
(71) BRIDGE PHARMA, INC. [US/US]; 902<br />
Contento Street, Sarasota, FL 34242 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) ABERG, A., K., Gunnar [SE/US];<br />
902 Contento Street, Sarasota, FL 34242<br />
(US). WRIGHT, George, L. [US/US]; 298<br />
Highland Street, Worcester, MA 01602 (US).<br />
CHEN, Jan, L. [CN/US]; 216B East Mountain<br />
Street, Worcester, MA 01608 (US).<br />
(74) LEMACK, Kevin, S. et al. / etc.; Nields,<br />
Lemack & Dingman, Suite 8, 176 E. Main<br />
Street, Westboro, MA 01581 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES FI<br />
GB GD GE GH GM HR HU ID IL IN IS JP<br />
KE KG KP KR KZ LC LK LR LS LT LU LV<br />
MA MD MG MK MN MW MX NO NZ PL<br />
PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT TZ UA UG US UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/445, C07D 211/06, 401/08,<br />
409/08<br />
(11) WO 00/76<strong>51</strong>1 (13) A1<br />
(21) <strong>PCT</strong>/US00/15657<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,763 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS CYCLOPENTYLE DE<br />
L’ACTIVITE DES RECEPTEURS DE LA<br />
CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
MACCOSS, Malcolm [GB/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). MILLS, Sander, G. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). OATES, Bryan [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/445, 31/4453, 31/454, C07D<br />
211/56, 211/92<br />
(11) WO 00/76<strong>51</strong>2 (13) A1<br />
(21) <strong>PCT</strong>/US00/15755<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,067 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS CYCLOPENTY-<br />
LIQUES DE L’ACTIVITE DU RECEP-<br />
TEUR DE LA CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). CHAPMAN, Kevin, T. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065-0907 (US). MACCOSS, Malcolm<br />
[GB/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). MILLS, Sander, G.<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US). OATES, Bryan<br />
[US/US]; 126 East Lincoln Avenue, Rahway,<br />
NJ 07065-0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065-0907 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX MZ<br />
NO NZ PL PT RO RU SD SE SG SI SK SL<br />
TJ TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(<strong>51</strong>) 7 A61K 31/445, 31/4453, 31/4465, C07D<br />
211/56, 211/92<br />
(11) WO 00/76<strong>51</strong>3 (13) A1<br />
(21) <strong>PCT</strong>/US00/15765<br />
(22) 8 Jun/juin <strong>2000</strong> (08.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/138,872 11 Jun/juin 1999 US<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) CYCLOPENTYL MODULATORS OF<br />
CHEMOKINE RECEPTOR ACTIVITY<br />
MODULATEURS CYCLOPENTY-<br />
LIQUES DE L’ACTIVITE DU RECEP-<br />
TEUR DE LA CHIMIOKINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) FINKE, Paul, E. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065-0907<br />
(US). LOEBACH, Jennifer, L. [US/US];