PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
PCT/2000/51 - World Intellectual Property Organization
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<strong>51</strong>/<strong>2000</strong><br />
21 Dec/déc <strong>2000</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 19097<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
Published / Publiée :(c)<br />
(<strong>51</strong>) 7 C07D 213/82, 239/42, 239/47, 239/48,<br />
403/12, 405/12, 409/12, 401/12, A61K<br />
31/455, 31/505, 31/506, 31/5377, A61P<br />
43/00, 9/10, 29/00, 35/00, 13/12<br />
(11) WO 00/76980 (13) A1<br />
(21) <strong>PCT</strong>/JP00/03768<br />
(22) 9 Jun/juin <strong>2000</strong> (09.06.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/163344 10 Jun/juin 1999<br />
(10.06.1999)<br />
(30) 11/165217 11 Jun/juin 1999<br />
(11.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) NOVEL NITROGEN-CONTAIING HET-<br />
EROCYCLIC DERIVATIVES OR SALTS<br />
THEREOF<br />
NOUVEAUX DERIVES HETEROCY-<br />
CLIQUES AZOTES OU LEURS SELS<br />
(71) YAMANOUCHI PHARMACEUTICAL<br />
CO., LTD. [JP/JP]; 3-11, Nihonbashi-honcho<br />
2-chome, Chuo-ku, Tokyo 103-8411 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) SUZUKI, Takayuki [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21,<br />
Miyukigaoka, Tsukuba-shi, Ibaraki 305-8585<br />
(JP). ONDA, Kenichi [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21, Miyukigaoka,<br />
Tsukuba-shi, Ibaraki 305-8585 (JP). MU-<br />
RAKAMI, Takeshi [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21, Miyukigaoka,<br />
Tsukuba-shi, Ibaraki 305-8585 (JP).<br />
NEGORO, Kenji [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21, Miyukigaoka,<br />
Tsukuba-shi, Ibaraki 305-8585 (JP).<br />
YAHIRO, Kiyoshi [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21, Miyukigaoka,<br />
Tsukuba-shi, Ibaraki 305-8585<br />
(JP). MARUYAMA, Tatsuya [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21,<br />
Miyukigaoka, Tsukuba-shi, Ibaraki 305-8585<br />
(JP). SHIMAYA, Akiyoshi [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21,<br />
Miyukigaoka, Tsukuba-shi, Ibaraki 305-8585<br />
(JP). OHTA, Mitsuaki [JP/JP]; Yamanouchi<br />
Pharmaceutical Co., Ltd., 21, Miyukigaoka,<br />
Tsukuba-shi, Ibaraki 305-8585 (JP).<br />
(74) NAGAI, Shozo et al. / etc.; Yamanouchi<br />
Pharmaceutical Co., Ltd., Patent Department,<br />
17-1, Hasune 3-chome, Itabashi-ku, Tokyo<br />
174-8612 (JP).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG US UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
JP<br />
JP<br />
(<strong>51</strong>) 7 C07D 215/38, 215/22, 223/16, 209/40,<br />
209/34, 401/04, A61K 31/404, 31/4704,<br />
31/55, A61P 25/00<br />
(11) WO 00/76981 (13) A1<br />
(21) <strong>PCT</strong>/US00/16784<br />
(22) 15 Jun/juin <strong>2000</strong> (15.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,187 15 Jun/juin 1999 US<br />
(15.06.1999)<br />
(30) 09/333,368 15 Jun/juin 1999 US<br />
(15.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) PIPERIDINYL AND PIPERAZINYL<br />
SUBSTITUTED BENZOFUSED LAC-<br />
TAMS<br />
LACTAMES BENZOFUSES A SUBSTI-<br />
TUTION PIPERIDINYLE ET PIPERAZI-<br />
NYLE<br />
(71) NEUROGEN CORPORATION [US/US];<br />
35 Northeast Industrial Road, Branford, CT<br />
06405 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) ZHAO, He [CN/US]; 4 Stoneridge Lane,<br />
Branford, CT 06405 (US). THURKAUF, Andrew<br />
[US/US]; 16 Fox Den Road, Danbury,<br />
CT 06811 (US).<br />
(74) SARUSSI, Steven, J.; McDonnell Boehnen<br />
Hulbert & Berghoff, Suite 3200, 300 South<br />
Wacker Drive, Chicago, IL 60606-6606 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM DZ EE<br />
ES FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
Published / Publiée :(c)<br />
(<strong>51</strong>) 7 C07D 215/44, 219/12, A61K 31/47, A61P<br />
37/06<br />
(11) WO 00/76982<br />
(21) <strong>PCT</strong>/US00/16723<br />
(13) A1<br />
(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,544 16 Jun/juin 1999<br />
(16.06.1999)<br />
US<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) ANTAGONISM OF IMMUNOSTIMU-<br />
LATORY CPG-OLIGONUCLEOTIDES<br />
BY 4-AMINOQUINOLINES AND<br />
OTHER WEAK BASES<br />
ANTAGONISME DES OLIGONUCLEO-<br />
TIDES CPG IMMUNOSTIMULATEURS<br />
PAR DES 4-AMINOQUINOLINES ET<br />
AUTRES BASES FAIBLES<br />
(71) UNIVERSITY OF IOWA RESEARCH<br />
FOUNDATION [US/US]; 100 Oakdale<br />
Campus #214-TIC, Iowa City, IA 52242-5000<br />
(US).<br />
(72) MACFARLANE, Donald, E.; 620 S.<br />
Summit Street, Iowa City, IA 52240 (US).<br />
STREKOWSKI, Lucjan; 6091 Windsong<br />
Way, Stone Mountain, GA 30087 (US).<br />
MANZEL, Lori; 3316 Timber Valley Ct.<br />
NE, Cedar Rapids, IA 52402 (US). ISMAIL,<br />
Fyaz; Department of Physical Sciences,<br />
University of Hertfordshire, Hartfield AL10<br />
9AB, Hertfordshire (GB). BARLIN, Gordon,<br />
B.; John Curtin School of Medical<br />
Research, Room D3044A, The Australian<br />
National University, Canberra, ACT 0200<br />
(AU).<br />
(74) SHISHIMA, Gina, N.; Fulbright & Jaworski,<br />
L.L.P., Suite 2400, 600 Congress<br />
Avenue, Austin, TX 78701 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG UZ VN YU ZA<br />
ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
Published / Publiée :(c)<br />
(<strong>51</strong>) 7 C07D 231/06, A61K 31/415<br />
(11) WO 00/76983 (13) A1<br />
(21) <strong>PCT</strong>/US00/16727<br />
(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/139,414 16 Jun/juin 1999 US<br />
(16.06.1999)<br />
(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />
(54) 1-(4-ARYLSULFONYL)-3-SUBSTI-<br />
TUTED-5-ARYL-2-PYRAZOLINES<br />
AS INHIBITORS OF CYCLOOXYGE-<br />
NASE-2<br />
1-(4-ARYLESULFONYLE)-3-SUB-<br />
STITUE-5-ARYLE-2-PYRAZOLINES<br />
COMME INHIBITEURS DE LA CY-<br />
CLO-OXYGENASE-2<br />
(71) TEMPLE UNIVERSITY - OF THE COM-<br />
MONWEALTH SYSTEM OF HIGHER<br />
EDUCATION [US/US]; Broad Street and<br />
Montgomery Avenue, Philadelphia, PA<br />
19122 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) REDDY, E., Premkumar [US/US];<br />
547 Atterbury Road, Villanova, PA 19085<br />
(US). REDDY, M., V., Ramana [IN/US];<br />
347B Beverly Boulevard, Upper Darby, PA<br />
19082-4504 (US).<br />
(74) MONACO, Daniel, A.; Seidel, Gonda, Lavorgna<br />
& Monaco, P.C., Suite 1800, Two<br />
Penn Center Plaza, Philadelphia, PA 19102<br />
(US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID IL<br />
IN IS JP KE KG KP KR KZ LC LK LR LS<br />
LT LU LV MA MD MG MK MN MW MX<br />
MZ NO NZ PL PT RO RU SD SE SG SI SK<br />
SL TJ TM TR TT TZ UA UG US UZ VN YU<br />
ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU
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