PCT/2000/51 - World Intellectual Property Organization

51/2000
19094 PCT Gazette - Section I - Gazette du PCT 21 Dec/déc 2000
(22) 26 May/mai 2000 (26.05.2000)
(25) en (26) en
(30) P 9901939 10 Jun/juin 1999 HU
(10.06.1999)
(43) 21 Dec/déc 2000 (21.12.2000)
(54) PROCESS FOR THE SYNTHESIS OF
A-NOR-SECO COMPOUNDS WITH
STERANE SKELETON
PROCEDE DE SYNTHESE DE COM-
POSES A-NOR-SECO A L’AIDE D’UN
SQUELETTE DE STERANE
(71) RICHTER GEDEON VEGYÉSZETI
GYÁR RT. [HU/HU]; Gyömrői út 19-21,
H-1103 Budapest (HU).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) SÁNTA, Csaba [HU/HU]; Sasvár u.
44, H-1165 Budapest (HU). TUBA, Zoltán
[HU/HU]; Bogár u. 20/b, H-1022 Budapest
(HU). MAHÓ, Sándor [HU/HU]; Rím
u. 20, H-1183 Budapest (HU). SZÉLES,
János [HU/HU]; Haller u. 82, H-1096 Budapest
(HU). BALOGH, Gábor [HU/HU];
Csontváry K.T. u. 18, H-1181 Budapest
(HU). BRLIK, János [HU/HU]; Klapka
György u. 29, H-1154 Budapest (HU).
TRISCHLER, Ferenc [HU/HU]; Úttörő u.
16, H-1171 Budapest (HU). SZILÁGYI,
Gabriella [HU/HU]; Tövishát u. 47, H-1186
Budapest (HU). BAKCSI, Erika [HU/HU];
Nóra u. 12, H-1028 Budapest (HU).
(74) RICHTER GEDEON VEGYÉSZETI
GYÁR RT.; Gyömrói út 19-21, H-1103
Budapest (HU).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID IL
IN IS JP KE KG KP KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
NO NZ PL PT RO RU SD SE SG SI SK SL
TJ TM TR TT TZ UA UG US UZ VN YU ZA
ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07D 209/44, A61K 31/4035, A61P 43/00,
C07D 403/12, 401/12
(11) WO 00/76969
(21) PCT/US00/15073
(13) A1
(22) 31 May/mai 2000 (31.05.2000)
(25) en (26) en
(30) 60/138,543 10 Jun/juin 1999
(10.06.1999)
US
(43) 21 Dec/déc 2000 (21.12.2000)
(54) METHOD OF INHIBITING AMYLOID
PROTEIN AGGREGATION AND IMAG-
ING AMYLOID DEPOSITS USING
ISOINDOLINE DERIVATIVES
PROCEDE D’INHIBITION D’AGRE-
GATION DE PROTEINES AMYLOIDES
ET D’IMAGERIE DE DEPOTS AMY-
LOIDES AU MOYEN DE DERIVES
D’ISOINDOLINE
(71) WARNER-LAMBERT COMPANY
[US/US]; 201 Tabor Road, Morris Plains,
NJ 07950 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) AUGELLI-SZAFRAN, Corinne, Elizabeth
[US/US]; 2812 Aspen Ridge Drive,
Ann Arbor, MI 48103 (US). LAI, Yingjie
[CA/US]; 27H Reading Road, Edison, NJ
08817 (US). SAKKAB, Annette, Theresa
[US/US]; 39790 Foxway Court, Northville,
MI 48167 (US). WALKER, Lary, Craswell
[US/US]; 4890 North Ridgeside Circle, Ann
Arbor, MI 48105 (US).
(74) RYAN, M., Andrea; Warner-Lambert Company,
201 Tabor Road, Morris Plains, NJ
07950 (US) et al. / etc.
(81) AE AG AL AU BA BB BG BR CA CN CR
CU CZ DM DZ EE GD GE HR HU ID IL IN
IS JP KP KR LC LK LR LT LV MA MG MK
MN MX MZ NO NZ PL RO SG SI SK SL TR
TT UA US UZ VN YU ZA.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07D 211/00
(11) WO 00/76970
(21) PCT/GB00/02296
(13) A2
(22) 13 Jun/juin 2000 (13.06.2000)
(25) en (26) en
(30) 9913823.2 14 Jun/juin 1999
(14.06.1999)
GB
(30) 60/142,064 2 Jul/juil 1999
(02.07.1999)
US
(30) 9918741.1 9 Aug/août 1999
(09.08.1999)
GB
(30) 9929552.9 14 Dec/déc 1999
(14.12.1999)
GB
(30) 9929553.7 14 Dec/déc 1999
(14.12.1999)
GB
(43) 21 Dec/déc 2000 (21.12.2000)
(54) COMPOUNDS
COMPOSES
(71) ELI LILLY AND COMPANY [US/US];
Lilly Corporate Center, Indianapolis, IN
46285 (US). PROTHERICS MOLECU-
LAR DESIGN LIMITED [GB/GB]; Beechfield
House, Lyme Green Business Park,
Macclesfield, Cheshire SK11 0JL (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) LIEBESCHUETZ, John, Walter
[GB/GB]; Laburnum Cottage, 42 Bollington
Road, Bollington, Cheshire SK10 5EJ (GB).
LYONS, Amanda, Jane [GB/GB]; 3 Thistleton
Close, Macclesfield, Cheshire SK11 8BE
(GB). MURRAY, Christopher, William
[GB/GB]; 1 Wheatfield Close, Tytherington,
Maeclesfield, Cheshire SK10 2TT (GB).
RIMMER, Andrew, David [GB/GB]; 9
Stamford Drive, Whittle-le-Woods, Chorley,
Lancashire PR6 7HP (GB). YOUNG,
Stephen, Clinton [GB/GB]; 8 Cranbourne
Road, Heaton Moor, Stockport SK4 4LD
(GB). CAMP, Nicholas, Paul [GB/GB]; Flat
2, Sliver Court, Fosseway, Nailsea, Avon
BS48 2BX (GB). JONES, Stuart, Donald
[GB/GB]; 17 Oakwood Drive, Prestbury,
Cheshire SK10 4HG (GB). MORGAN,
Phillip, John [GB/GB]; 11 Woodland Avenue,
Congleton, Cheshire CW12 1LN (GB).
RICHARDS, Simon, James [GB/GB];
39 Vicarage Road, Blackrod, Bolton BL6
5DA (GB). WYLIE, William Alexander
[GB/GB]; Flat 4, 39 Station Road, Reddish,
Stockport SK5 6LT (GB). LIVELY,
Sarah, Elizabeth [GB/GB]; Hillcrest, Reads
Lane, Congleton, Cheshire CW12 3PJ (GB).
HARRISON, Martin, James [GB/GB];
29 Grenfell Road, Didsbury, Manchester
M20 6TG (GB). WASZKOWYCZ, Bohdan
[GB/GB]; 46 Grange Park Avenue, Wilmslow,
Cheshire SK9 4AL (GB). MASTERS,
John, Joseph [US/US]; 12047 Flint Stone
Court, Fishers, IN 46038 (US). WILEY,
Michael, John [US/US]; 7725 Langwood
Drive, Indianapolis, IN 46268 (US).
(74) HAY, Martin, A.; Martin A. Hay & Co., 13
Queen Victoria Street, Macclesfield, Cheshire
SK11 6LP (GB).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID IL
IN IS JP KE KG KP KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
MZ NO NZ PL PT RO RU SD SE SG SI SK
SL TJ TM TR TT TZ UA UG US UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 211/00
(11) WO 00/76971
(21) PCT/GB00/02302
(13) A2
(22) 13 Jun/juin 2000 (13.06.2000)
(25) en (26) en
(30) 9913823.2 14 Jun/juin 1999
(14.06.1999)
GB
(30) 60/142,064 2 Jul/juil 1999
(02.07.1999)
US
(30) 9918741.1 9 Aug/août 1999
(09.08.1999)
GB
(30) 9929553.7 14 Dec/déc 1999
(14.12.1999)
GB
(43) 21 Dec/déc 2000 (21.12.2000)
(54) COMPOUNDS
COMPOSES
(71) ELI LILLY AND COMPANY [US/US];
Lilly Corporate Center, Indianapolis, IN
46285 (US). PROTHERICS MOLECU-
LAR DESIGN LIMITED [GB/GB]; Beechfield
House, Lyme Green Business Park,
Macclesfield, Cheshire SK11 0JL (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) LIEBESCHUETZ, John, Walter
[GB/GB]; Laburnum Cottage, 42 Bollington
Road, Bollington, Cheshire SK10 5EJ (GB).
LYONS, Amanda, Jane [GB/GB]; 3 Thistleton
Close, Macclesfield, Cheshire SK11 8BE
(GB). MURRAY, Christopher, William
[GB/GB]; 1 Wheatfield Close, Tytherington,
Macclesfield, Cheshire SK10 2TT (GB).
RIMMER, Andrew, David [GB/GB]; 9
Stamford Drive, Whittle-le-Woods, Chorley,
Lancashire PR6 7HP (GB). YOUNG,
Stephen, Clinton [GB/GB]; 8 Cranbourne