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PCT/2000/51 - World Intellectual Property Organization

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<strong>51</strong>/<strong>2000</strong><br />

19108 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 21 Dec/déc <strong>2000</strong><br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07K 5/02, A61K 38/05<br />

(11) WO 00/77030 (13) A1<br />

(21) <strong>PCT</strong>/US00/16643<br />

(22) 15 Jun/juin <strong>2000</strong> (15.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/139,173 15 Jun/juin 1999 US<br />

(15.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) STATINE-DERIVED TETRAPEPTIDE<br />

INHIBITORS OF BETA-SECRETASE<br />

INHIBITEURS TETRAPEPTIDES DE-<br />

RIVES DE LA STATINE DE β-SECRE-<br />

TASE<br />

(71) ELAN PHARMACEUTICALS, INC.<br />

[US/US]; 800 Gateway Boulevard, South San<br />

Francisco, CA 94080 (US).<br />

(72) JOHN, Varghese; 1722 18th Street, San<br />

Francisco, CA 94122 (US). TUNG, Jay;<br />

2224 Semeria Avenue, Belmont, CA 94002<br />

(US). FANG, Lawrence; 1193 Beach Park<br />

Boulevard, Foster City, CA 94404 (US).<br />

MAMO, Shumeye, S.; 564 Oakland Avenue<br />

#14, Oakland, CA 95611 (US).<br />

(74) HOCH, J., Mark; Elan Pharmaceuticals,<br />

Inc., 800 Gateway Boulevard, South San<br />

Francisco, CA 94080 (US).<br />

(81) AE AG AL AM AT AT (Utility model / modèle<br />

d’utilité) AUAZBABBBGBRBYCA<br />

CH CN CR CU CZ CZ (Utility model / modèle<br />

d’utilité) DE DE (Utility model / modèle<br />

d’utilité) DK DK (Utility model / modèle<br />

d’utilité) DM DZ EE EE (Utility model / modèle<br />

d’utilité) ES FI FI (Utility model / modèle<br />

d’utilité) GBGDGEGHGMHRHUIDIL<br />

IN IS JP KE KG KP KR KR (Utility model<br />

/ modèle d’utilité) KZLCLKLRLSLTLU<br />

LV MA MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SK (Utility<br />

model / modèle d’utilité) SLTJTMTRTT<br />

TZ UA UG UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

Published / Publiée :(c)<br />

(<strong>51</strong>) 7 C07K 7/00<br />

(11) WO 00/77031 (13) A2<br />

(21) <strong>PCT</strong>/CA00/00711<br />

(22) 15 Jun/juin <strong>2000</strong> (15.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/139,263 15 Jun/juin 1999<br />

(15.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) MUC1 LIGANDS<br />

US<br />

LIGANDS MUC1<br />

(71) UNIVERSITY HEALTH NETWORK<br />

[CA/CA]; Room 7-504, 610 University Avenue,<br />

Toronto, Ontario M5G 2M9 (CA).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) GARIEPY, Jean [CA/CA]; 29 Elmsthorpe<br />

Avenue, Toronto, Ontario M5P 2L5<br />

(CA). YANG, Shaoxian [CA/CA]; 309-36<br />

Thorncliffe Park Drive, Toronto, Ontario<br />

M4H 1J8 (CA).<br />

(74) BERESKIN & PARR; 40th floor, 40 King<br />

Street West, Toronto, Ontario M5H 3Y2<br />

(CA).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES FI<br />

GB GD GE GH GM HR HU ID IL IN IS JP<br />

KE KG KP KR KZ LC LK LR LS LT LU LV<br />

MA MD MG MK MN MW MX NO NZ PL<br />

PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT TZ UA UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07K 7/00<br />

(11) WO 00/77032 (13) A2<br />

(21) <strong>PCT</strong>/GB00/02364<br />

(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 9914045.1 16 Jun/juin 1999 GB<br />

(16.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) NOVEL COMPOUNDS<br />

NOUVEAUX COMPOSES<br />

(71) SMITHKLINE BEECHAM P.L.C.<br />

[GB/GB]; New Horizons Court, Brentford,<br />

Middlesex TW8 9EP (GB). CAMBRIDGE<br />

UNIVERSITY TECHNICAL SERVICES<br />

LTD. [GB/GB]; The Old Schools, Cambridge<br />

University, Cambridge, Cambridgeshire CB2<br />

1TS (GB).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) CAMILLERI, Patrick [MT/GB];<br />

SmithKline Beecham Pharmaceuticals, New<br />

Frontiers Science Park South, Third Avenue,<br />

Harlow, Essex CM19 5AW (GB).<br />

GUÉDAT, Philippe [FR/FR]; University<br />

of Cambridge, Department of Chemistry,<br />

University Chemical Laboratory, Lensfield<br />

Road, Cambridge CB2 1EW (GB). KIRBY,<br />

Anthony, John [GB/GB]; University of<br />

Cambridge, Department of Chemistry, University<br />

Chemical Laboratory, Lensfield Road,<br />

Cambridge, Cambridgeshire CB2 1EW (GB).<br />

KREMER, Andreas [DE/GB]; SmithKline<br />

Beecham Pharmaceuticals, New Frontiers<br />

Science Park South, Third Avenue, Harlow,<br />

Essex CM19 5AW (GB).<br />

(74) GIDDINGS, Peter, John; SmithKline<br />

Beecham, Two New Horizons Court, Brentford,<br />

Middlesex TW8 9EP (GB).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

(<strong>51</strong>) 7 C07K 7/00, 14/47, 14/52, A61K 38/16,<br />

38/19, 38/20<br />

(11) WO 00/77033 (13) A1<br />

(21) <strong>PCT</strong>/US00/40227<br />

(22) 16 Jun/juin <strong>2000</strong> (16.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/139,687 16 Jun/juin 1999 US<br />

(16.06.1999)<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) RETRO-INVERSO PEPTIDES DE-<br />

RIVED FROM INTERLEUKIN-6<br />

PEPTIDES RÉTRO-INVERSES DÉRI-<br />

VÉS DEL’INTERLEUKINE 6<br />

(71) MYELOS CORPORATION [US/US];<br />

Suite M, 4940 Carroll Canyon Road, San<br />

Diego, CA 92121 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) WRIGHT, David, E. [US/US]; 17140<br />

Woodson View Lane, Ramona, CA 92065<br />

(US). PARKS, D., Elliot [US/US]; 709 Kalamath<br />

Drive, Del Mar, CA 92014 (US).<br />

(74) HUNT, Dale, C.; Knobbe, Martens, Olson<br />

& Bear, LLP, 16th floor, 620 Newport Center<br />

Drive, Newport Beach, CA 92660 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID IL<br />

IN IS JP KE KG KP KR KZ LC LK LR LS<br />

LT LU LV MA MD MG MK MN MW MX<br />

MZ NO NZ PL PT RO RU SD SE SG SI SK<br />

SL TJ TM TR TT TZ UA UG US UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

Published / Publiée :(c)<br />

(<strong>51</strong>) 7 C07K 14/00<br />

(11) WO 00/77034<br />

(21) <strong>PCT</strong>/CA00/00714<br />

(13) A2<br />

(22) 12 Jun/juin <strong>2000</strong> (12.06.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 2,274,414 11 Jun/juin 1999<br />

(11.06.1999)<br />

CA<br />

(43) 21 Dec/déc <strong>2000</strong> (21.12.<strong>2000</strong>)<br />

(54) AMINO ACIDS FROM FISH AND SOY<br />

PROTEINS IMPROVE INSULIN SENSI-<br />

TIVITY<br />

ACIDES AMINES PROVENANT DE<br />

PROTEINES DE POISSON ET DE SOJA<br />

AMELIORANT<br />

L’INSULINE<br />

LA SENSIBILITE A<br />

(71) UNIVERSITE LAVAL [CA/CA]; Cité Universitaire,<br />

Quebec, Quebec G1K 7P4 (CA).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)

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