PCT/1998/43 - World Intellectual Property Organization

43/1998
29 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 14941
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 9/19, 47/18, 47/12
(54) • STABLE PHARMACEUTICAL ADMINIS-
TRATION FORMS OF PEPTIDES, PROTEINS
AND NUCLEIC ACIDS
• FORMES DE PREPARATIONS PHARMA-
CEUTIQUES STABLES POUR PEPTIDES,
PROTEINES ET ACIDES NUCLEIQUES
(71) BOEHRINGER MANNHEIM GMBH [DE/DE];
D–68298 Mannheim (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) RÖDEL, Wolfgang [DE/DE]; Johanniterstrasse
9, D–69123 Heidelberg (DE). MATTERN,
Markus [DE/DE]; Friedrichstrasse 17, D–64646
Heppenheim (DE). WINTER, Gerhard [DE/DE];
Jahnstrasse 20e, D–69221 Dossenheim (DE).
(74) BOEHRINGER MANNHEIM GMBH; Patentabteilung,
D–68298 Mannheim (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU IL
IS JP KE KG KP KR KZ LC LK LR LS LT LU
LV MD MG MK MN MW MX NO NZ PL PT RO
RU SD SE SG SI SK SL TJ TM TR TT UA UG
US UZ VN YU ZW; AP (GH GM KE LS MW SD
SZ UG ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH CY DE DK ES FI FR GB
GR IE IT LU MC NL PT SE); OA (BF BJ CF CG
CI CM GA GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/47491 (13) A2
(21) PCT/CA98/00274
(22) 3 Apr/avr 1998 (03.04.1998)
(25) en (26) en
(31) 60/036,551 (32) 21 Apr/avr 1997 (33) US
(21.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 9/22
(54) • CONTROLLED RELEASE FORMULATIONS
USING INTELLIGENT POLYMERS
• COMPOSITIONS A LIBERATION REGULEE
UTILISANT DES POLYMERES INTELLI-
GENTS
(71, 72) ODIDI, Isa [NG/CA]; 2136 Opal Court, Mississauga,
Ontario L5K 2S5 (CA). ODIDI, Amina
[NG/CA]; 2136 Opan Court, Mississauga, Ontario
L5K 2S5 (CA).
(74) BARTOSZEWICZ, Lola, A.; Sim & McBurney,
6th floor, 330 University Avenue, Toronto, Ontario
M5G 1R7 (CA).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47492 (13) A1
(21) PCT/US98/07845
(22) 14 Apr/avr 1998 (14.04.1998)
(25) en (26) en
(31) 08/844,015 (32) 18 Apr/avr 1997
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(33) US
(51) 6 A61K 9/51, 31/00, 9/14, 31/635
(54) • NANOSIZED ASPARTYL PROTEASE INHI-
BITORS
• INHIBITEURS D’ASPARTYLE PROTEASE
NANOMETRIQUES
(63) US 08/844,015 (CIP)
18 Apr/avr 1997 (18.04.1997)
(71) VERTEX PHARMACEUTICALS INCORPO-
RATED [US/US]; 130 Waverly Street, Cambridge,
MA 02139–4242 (US).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) CHATURVEDI, Pravin, Ramsewak [IN/US];
4 Turning Mill Lane, Quincy, MA 02169 (US).
TUNG, Roger, Dennis [US/US]; 54 Richfield
Road, Arlington, MA 01274 (US). BOGER, Joshua,
S. [US/US]; 243 Old Pickard Road, Concord,
MA 01742 (US).
(74) HALEY, James, F., Jr.; Fish & Neave, 1251
Avenue of the Americas, New York, NY 10020
(US) et al. / etc.
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
Published / Publiée : (c)
(11) WO 98/47493 (13) A1
(21) PCT/AU98/00296
(22) 23 Apr/avr 1998 (23.04.1998)
(25) en (26) en
(31) PO 6371 (32) 23 Apr/avr 1997 (33) AU
(23.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 9/52, 9/60
(54) • TASTE MASKED PHARMACEUTICAL
COMPOSITIONS
• COMPOSITIONS PHARMACEUTIQUES A
GOUT MASQUE
(71) F.H. FAULDING & CO. LIMITED [AU/AU];
115 Sherriff Street, Underdale, S.A. 5032 (AU).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) PITMAN, Ian, Hamilton [AU/AU]; 4/182
Gover Street, North Adelaide, S.A. 5006 (AU).
(74) PHILLIPS ORMONDE & FITZPATRICK; 367
Collins Street, Melbourne, VIC 3000 (AU).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47494 (13) A2
(21) PCT/GB98/01169
(22) 22 Apr/avr 1998 (22.04.1998)
(25) en (26) en
(31) 9708133.5 (32) 22 Apr/avr 1997
(22.04.1997)
(33) GB
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 31/00
(54) • NOVEL USE OF MATRIX METALLOPROTEI-
NASE INHIBITORS
• NOUVELLE UTILISATION D’INHIBITEURS
DE METALLOPROTEINASE MATRICIELLE
(71) BRITISH BIOTECH PHARMACEUTICALS
LIMITED [GB/GB]; Watlington Road, Cowley,
Oxford OX4 5LY (GB).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) DAVIDSON, Alan, Hornsby [GB/GB]; British
Biotech Pharmaceuticals Limited, Watlington
Road, Cowley, Oxford OX4 5LY (GB). BAKER,
Rodney, Cyril [GB/GB]; British Biotech Pharmaceuticals
Limited, Watlington Road, Cowley,
Oxford OX4 5LY (GB).
(74) WALLS, Alan, J.; British Biotech Pharmaceuticals
Limited, Watlington Road, Cowley, Oxford 0X4
5LY (GB).
(81) AU BR CA CN CZ DE GB HU IL JP KR MX NO
NZ PL RU SG TR US; EP (AT BE CH CY DE
DK ES FI FR GB GR IE IT LU MC NL PT SE).
(11) WO 98/47495 (13) A1
(21) PCT/SE98/00301
(22) 20 Feb/fév 1998 (20.02.1998)
(25) en (26) en
(31) 9700617–5 (32) 22 Apr/avr 1997 (33) SE
(22.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 31/00, 33/00, 33/02, 31/375
(54) • NEW COMPOSITION
• NOUVELLE COMPOSITION
(71) NITRICARE KB [SE/SE]; Alving Kjell,
Spetsvägen 40, S–757 57 Uppsala (SE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ALVING, Kjell [SE/SE]; Spetsvägen 40,
S–757 57 Uppsala (SE). LUNDBERG, Jan, M.
[SE/SE]; Helgevägen 10, S–182 64 Djursholm
(SE). LUNDBERG, Jon [SE/SE]; Tomtebogatan
40, S–113 35 Stockholm (SE). WEITZBERG, Eddie
[SE/SE]; Nybrogatan 24, S–114 39 Stockholm
(SE). WIKLUND, Peter [SE/SE]; Bergsätravägen
22A, S–181 61 Lidingö (SE).
(74) ONN, Thorsten et al. / etc.; AB Stockholms
Patentbyrå, Zacco & Bruhn (Publ), P.O. Box 23101,
S–104 35 Stockholm (SE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR TT
UA UG US UZ VN YU ZW; AP (GH GM KE LS
MW SD SZ UG ZW); EA (AM AZ BY KG KZ
MD RU TJ TM); EP (AT BE CH DE DK ES FI
FR GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN ML MR NE SN TD TG).
(11) WO 98/47496 (13) A2
(21) PCT/US98/07659
(22) 15 Apr/avr 1998 (15.04.1998)
(25) en (26) en
(31) 60/044,701 (32) 18 Apr/avr 1997
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 A61K 31/00
(33) US