PCT/1998/43 - World Intellectual Property Organization

43/1998
15002 PCT Gazette - Section I - Gazette du PCT 29 Oct/oct 1998
(25) en (26) en
(31) 9/118871 (32) 21 Apr/avr 1997 (33) JP
(21.04.1997)
(31) 9/367154 (32) 24 Dec/déc 1997 (33) JP
(24.12.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 261/14, 261/08, 413/12, 417/12, 413/14,
A61K 31/42
(54) • ISOXAZOLE DERIVATIVES
• DERIVES D’ISOXAZOLE
(71) SUMITOMO PHARMACEUTICALS COM-
PANY, LIMITED [JP/JP]; 2–8, Doshomachi
2–chome, Chuo–ku, Osaka–shi, Osaka 541–8510
(JP).
(72) NAKATSUKA, Masashi; 3–2–4–807, Yamazaki,
Shimamotocho, Mishima–gun, Osaka 618–0001
(JP). UENO, Yoshihide; 2–3–37–112, Matsuzakicho,
Abeno–ku, Osaka–shi, Osaka 545–0053
(JP). OKADA, Shin–ichiro; 2–17–18, Okutenjincho,
Takatsuki–shi, Osaka 569–1118 (JP). NI-
SHIKAKU, Fumio; 1–21, Sakuragaoka 5–chome,
Itami–shi, Hyogo 664–0897 (JP).
(74) ASAMURA, Kiyoshi et al. / etc.; Room 331, New
Ohtemachi Building, 2–1, Ohtemachi 2–chome,
Chiyoda–ku, Tokyo 100–0004 (JP).
(81) CN ID KR MX; EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE).
(11) WO 98/47881 (13) A1
(21) PCT/EP98/02182
(22) 14 Apr/avr 1998 (14.04.1998)
(25) de (26) de
(31) 197 17 228.8 (32) 24 Apr/avr 1997 (33) DE
(24.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 263/14, A01N 43/76
(54) • SUBSTITUTED DIPHENYL OXAZOLIN DE-
RIVATIVES WITH INSECTICIDAL EFFECT
• DERIVES DE DIPHENYL–OXAZOLINE
SUBSTITUES A ACTION INSECTICIDE
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];
D–51368 Leverkusen (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) KRÄMER, Wolfgang [DE/DE]; Rosenkranz
25, D–51399 Burscheid (DE). KRAATZ, Udo
[DE/DE]; Andreasstrasse 22a, D–51375 Leverkusen
(DE). LANTZSCH, Reinhard [DE/DE];
Am Buschhäuschen 51, D–42115 Wuppertal
(DE). MARHOLD, Albrecht [DE/DE];
Carl–Duisberg–Strasse 329, D–51373 Leverkusen
(DE). ERDELEN, Christoph [DE/DE];
Unterbüscherhof 15, D–42799 Leichlingen
(DE). WACHENDORFF–NEUMANN, Ulrike
[DE/DE]; Oberer Markenweg 85, D–56566 Neuwied
(DE). TURBERG, Andreas [DE/DE];
Naheweg 19, D–40699 Erkrath (DE). MENCKE,
Norbert [DE/DE]; Grundermühle 2, D–51381
Leverkusen (DE).
(74) BAYER AKTIENGESELLSCHAFT; D–51368
Leverkusen (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
Published / Publiée : (c)
(11) WO 98/47882 (13) A1
(21) PCT/JP98/01797
(22) 20 Apr/avr 1998 (20.04.1998)
(25) en (26) en
(31) 9/103138 (32) 21 Apr/avr 1997 (33) JP
(21.04.1997)
(31) 9/319545 (32) 20 Nov/nov 1997 (33) JP
(20.11.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 267/14, 243/24, 281/10, 413/04, 413/06,
417/06, 417/12, A61K 31/55
(54) • 4,1–BENZOXAZEPINES, THEIR
ANALOGUES, AND THEIR USE AS SO-
MATOSTATIN AGONISTS
• 4,1 BENZOXAZEPINES, LEURS
ANALOGUES ET LEUR UTILISATION
COMME AGONISTES DE LA SOMATOSTA-
TINE
(71) TAKEDA CHEMICAL INDUSTRIES, LTD.
[JP/JP]; 1–1, Doshomachi 4–chome, Chuo–ku,
Osaka–shi, Osaka 541–0045 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) MABUCHI, Hiroshi [JP/JP]; 555–33, Ayameikeminami
7–chome, Nara–shi, Nara 631–0033
(JP). SUZUKI, Nobuhiro [JP/JP]; 1077–50,
Oaza–yatabe, Tsukuba–shi, Ibaraki 305–0861 (JP).
MIKI, Takashi [JP/JP]; 1–7–502, Hannancho
2–chome, Abeno–ku, Osaka–shi, Osaka 545–0021
(JP).
(74) ASAHINA, Tadao et al. / etc.; Osaka Plant of
Takeda Chemical Industries, Ltd., 17–85, Jusohonmachi
2–chome, Yodogawa–ku, Osaka–shi, Osaka
532–0024 (JP).
(81) AL AM AU AZ BA BB BG BR BY CA CN CU
CZ EE GE GW HU ID IL IS KG KR KZ LC LK
LR LT LV MD MG MK MN MX NO NZ PL RO
RU SG SI SK SL TJ TM TR TT UA US UZ VN
YU; AP (GH GM KE LS MW SD SZ UG ZW);
EA (AM AZ BY KG KZ MD RU TJ TM); EP (AT
BE CH CY DE DK ES FI FR GB GR IE IT LU
MC NL PT SE); OA (BF BJ CF CG CI CM GA
GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/47883 (13) A1
(21) PCT/EP98/01990
(22) 6 Apr/avr 1998 (06.04.1998)
(25) de (26) de
(31) 197 16 260.6 (32) 18 Apr/avr 1997
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 271/07, A01N 43/82
(54) • SULFONYLOXADIAZOLONES
• SULFONYLOXADIAZOLONES
(33) DE
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];
D–51368 Leverkusen (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ASSMANN, Lutz [DE/DE]; Eichblatt 2,
D–23701 Eutin (DE). GERDES, Peter [DE/DE];
Waldstrasse 75, D–52080 Aachen (DE). STEN-
ZEL, Klaus [DE/DE]; Seesener Strasse 17,
D–40595 Düsseldorf (DE). DENG, Chuan–
Zheng [CN/CN]; Building 5, Flat 401, Lane 715,
Mao–Tai Road, Shanghai 200335 (CN). YUAN,
Li–Ping [CN/CN]; Building 10, Flat 406, Lane 65,
Tian–Lin Road, Shanghai 200233 (CN). ZHAO,
Jian–Mei [CN/CN]; Building 142, Room 402,
Mei Long Yi Cun, Shanghai 200237 (CN).
(74) BAYER AKTIENGESELLSCHAFT; D–51368
Leverkusen (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
Published / Publiée : (c)
(11) WO 98/47884 (13) A1
(21) PCT/GB98/01034
(22) 8 Apr/avr 1998 (08.04.1998)
(25) en (26) en
(31) 9708280.4 (32) 24 Apr/avr 1997 (33) GB
(24.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 277/36, 277/32
(54) • PROCESS FOR THE PRODUCTION OF
5–CHLORO–2– (4,4–DIFLUOROBUT–3–
ENYLSULPHONYL) THIAZOLE AND
INTERMEDIATES THEREFOR
• PROCEDE SERVANT A PREPARER 5–
CHLORO–2– (4,4–DIFLUOROBUT–3–
ENYLSULFONYL) THIAZOLE ET IN-
TERMEDIAIRES
(71) ZENECA LIMITED [GB/GB]; 15 Stanhope Gate,
London W1Y 6LN (GB).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) BOWDEN, Martin, Charles [GB/GB]; Zeneca
Huddersfield Works, Leeds Road, P.O. Box
A38, Huddersfield, West Yorkshire HD2 1FF (GB).
BROWN, Stephen, Martin [GB/GB]; Zeneca
Huddersfield Works, Leeds Road, P.O. Box A 38,
Huddersfield, West Yorkshire HD2 1FF (GB).
(74) BISHOP, Nigel, Douglas et al. / etc.; Zeneca
Agrochemicals, Intellectual Property Dept.,
Jealott’s Hill Research Station, P.O. Box 3538, Bracknell,
Berkshire RG42 6YA (GB).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47885
(21) PCT/EP98/02265
(13) A1
(22) 14 Apr/avr 1998 (14.04.1998)
(25) en (26) en
(31) 9707876.0 (32) 18 Apr/avr 1997
(18.04.1997)
(33) GB
(31) 9801635.5 (32) 26 Jan/jan 1998
(26.01.1998)
(33) GB
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 295/12, A61K 31/495, 31/445, C07D
213/56, 213/40, 215/50, 215/38, 217/02, 209/08,
277/62, 285/14, 307/79, 317/60, 401/12, 401/10
(54) • A BICYCLIC ARYL OR A BICYCLIC
HETEROCYCLIC RING CONTAINING
COMPOUNDS HAVING A COMBINED
5HT1A, 5HT1B AND 5HT1D RECEPTOR
ANTAGONISTIC ACTIVITY