PCT/1998/43 - World Intellectual Property Organization

43/1998
29 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 15003
•
ARYL BICYCLIQUE OU NOYAU HETERO-
CYCLIQUE BICYCLIQUE CONTENANT
DES COMPOSES PRESENTANT UNE ACTI-
VITE ANTAGONISTE COMBINEE CONTRE
LES RECEPTEURS 5HT1A, 5HT1B ET
5HT1D
(71) SMITHKLINE BEECHAM PLC [GB/GB]; New
Horizons Court, Brentford, Middlesex TW8 9EP
(GB).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) GASTER, Laramie, Mary [GB/GB]; SmithKline
Beecham Pharmaceuticals, New Frontiers
Science Park South, Third Avenue, Harlow, Essex
CM19 5AW (GB). WYMAN, Paul, Adrian
[GB/GB]; SmithKline Beecham Pharmaceuticals,
New Frontiers Science Park South, Third Avenue,
Harlow, Essex CM19 5AW (GB).
(74) WATERS, David, Martin; SmithKline Beecham,
Corporate Intellectual Property, New Horizons
Court, Brentford, Middlesex TW8 9EP (GB).
(81) CA JP US; EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE).
(11) WO 98/47886 (13) A1
(21) PCT/EP98/01942
(22) 2 Apr/avr 1998 (02.04.1998)
(25) de (26) de
(31) 197 16 237.1 (32) 18 Apr/avr 1997 (33) DE
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 303/36, 203/12, C07C 251/60, 271/28,
251/42, A01N 43/04, 43/34, 47/20, 37/18, 37/10
(54) • SUBSTITUTED BENZYL OXIMINO
COMPOUNDS
• COMPOSES DU TYPE BENZYLO–
OXYMINO SUBSTITUES
(71) BASF AKTIENGESELLSCHAFT [DE/DE];
D–67056 Ludwigshafen (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) GRAMMENOS, Wassilios [DE/DE]; Borsigstrasse
5, D–67063 Ludwigshafen (DE). SAUTER,
Hubert [DE/DE]; Neckarpromenade 20, D–68167
Mannheim (DE). BAYER, Herbert [DE/DE];
D 3.4, D–68159 Mannheim (DE). GROTE,
Thomas [DE/DE]; Breslauer Strasse 6, D–67105
Schifferstadt (DE). GYPSER, Andreas [DE/DE];
B 4.4, D–68159 Mannheim (DE). KIRSTGEN,
Reinhard [DE/DE]; Karolinenstrasse 51, D–67434
Neustadt (DE). MÜLLER, Bernd [DE/DE];
Jean–Ganss–Strasse 21, D–67227 Frankenthal
(DE). PTOCK, Arne [DE/DE]; Eichenstrasse
23, D–67067 Ludwigshafen (DE). RÖHL, Franz
[DE/DE]; Sebastian–Kneipp–Strasse 17, D–67105
Schifferstadt (DE). GÖTZ, Roland [DE/DE];
Schumannstrasse 4, D–91541 Rothenburg (DE).
LORENZ, Gisela [DE/DE]; Erlenweg 13,
D–67434 Neustadt (DE). AMMERMANN, Eberhard
[DE/DE]; Von–Gagern–Strasse 2, D–64646
Heppenheim (DE). STRATHMANN, Siegfried
[DE/DE]; Donnersbergstrasse 9, D–67117 Limburgerhof
(DE). HARRIES, Volker [DE/DE];
Immengärtenweg 29e, D–67227 Frankenthal (DE).
(74) BASF AKTIENGESELLSCHAFT; D–67056
Ludwigshafen (DE).
(81) AL AU BG BR BY CA CN CZ GE HU ID IL JP
KR KZ LT LV MX NO NZ PL RO RU SG SI SK
TR UA US; EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH CY DE DK ES FI FR GB
GR IE IT LU MC NL PT SE).
Published / Publiée : (c)
(11) WO 98/47887 (13) A1
(21) PCT/JP98/01778
(22) 17 Apr/avr 1998 (17.04.1998)
(25) ja (26) ja
(31) 9/102151 (32) 18 Apr/avr 1997 (33) JP
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 303/48, A61K 31/335
(54) • NOVEL EPOXYSUCCINAMIDE DERIVA-
TIVES OR SALTS THEREOF
• NOUVEAUX DERIVES
D’EPOXYSUCCINAMIDE ET
SELS ASSOCIES
(71) TAIHO PHARMACEUTICAL CO., LTD.
[JP/JP]; 27, Kanda Nishikicho 1–chome,
Chiyoda–ku, Tokyo 101–0054 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ASAO, Tetsuji [JP/JP]; 48–2–504, 5063–1,
Yamaguchi, Tokorozawa–shi, Saitama 359–1145
(JP). YAMASHITA, Tomohiro [JP/JP]; 8–5, Musashidai
7–chome, Hidaka–shi, Saitama 350–1255
(JP). SUDA, Yoshimitsu [JP/JP]; 18–3–301,
Kotesashicho 4–chome, Tokorozawa–shi, Saitama
359–1141 (JP). OKAJIMA, Shigeo [JP/JP];
B101, 621–2, Iwasawa, Hanno–shi, Saitama
357–0023 (JP). TADA, Yukio [JP/JP]; 4–7,
Matsuyamacho 2–chome, Higashimatsuyama–shi,
Saitama 355–0018 (JP). KATSUNUMA, Nobuhiko
[JP/JP]; 246–2, Myodocho 3–chome,
Tokushima–shi, Tokushima 770–0047 (JP).
YAMADA, Shozo [JP/JP]; 75–3–101, Aoki,
Hanno–shi, Saitama 357–0003 (JP). SHIGENO,
Kazuhiko [JP/JP]; 5–26–203, Takakura 4–chome,
Iruma–shi, Saitama 358–0021 (JP). UEMURA,
Atsuhiko [JP/JP]; 13–3–406, Sayamadai 4–chome,
Sayama–shi, Saitama 350–1304 (JP).
(74) ARUGA, Mitsuyuki et al. / etc.; Kyodo Building,
3–6, Nihonbashiningyocho 1–chome, Chuo–ku,
Tokyo 103–0013 (JP).
(81) AU CA JP KR US; EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE).
(11) WO 98/47888
(21) PCT/EP98/02247
(13) A1
(22) 17 Apr/avr 1998 (17.04.1998)
(25) en (26) en
(31) 97106453.0
(34) DE et al. / etc.
(32) 18 Apr/avr 1997
(18.04.1997)
(33) EP
(31) 97109900.7 (32) 18 Jun/juin 1997 (33) EP
(34) DE et al. / etc.
(18.06.1997)
(31) 97120536.4
(34) DE et al. / etc.
(32) 24 Nov/nov 1997
(24.11.1997)
(33) EP
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 307/60, A61K 31/00, C12N 1/02, C12P
7/00 // (C12P 7/00, C12R 1:66)
(54) • KODAISTATINS A, B, C AND D, A PROCESS
FOR THEIR PRODUCTION AND THEIR USE
• CODAISTATINES A, B, C ET D, LEUR PRO-
CEDE DE PREPARATION ET LEUR UTILI-
SATION
(71) HOECHST MARION ROUSSEL DEUT-
SCHLAND GMBH [DE/DE]; Brüningstrasse 50,
D–65929 Frankfurt am Main (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) RAMAKRISHNA, Nirogi, Venkata, Satya
[IN/IN]; E–4/Flat, 303, Highland Park, Mulund
(W), Mumbai – 400 082 (IN). SWAMY, Keshavapura,
Hosamane, Sreedhara [IN/IN]; B–402,
Lok Rachana Amar Nagar, Mulund (W), Mumbai
– 400 082 (IN). VIJAYAKUMAR, Erra, Koteswara,
Satya [IN/IN]; K–3, Hoechst Qtrs., Amar
Nagar, Mulund (W), Mumbai – 400 082 (IN).
NADKARNI, Suresh, Rudra [IN/IN]; 5, Yagneshwar,
Kasturba Marg, Mulund (W), Mumbai
– 400 080 (IN). JAYVANTI, Kenia [IN/IN];
11, Dev Aashish, Ganesh Gwade Road, Mulund
(W), Mumbai – 400 080 (IN). HERLING, Andreas,
W. [DE/DE]; Am Walberstück 5, D–65520
Bad Camberg (DE). KOGLER, Herbert [DE/DE];
Dattenbachstrasse 12, D–61479 Schloßhorn (DE).
VERTESY, Laszlo [DE/DE]; Eppenhainer Weg
6, D–65817 Eppstein (DE). PANSHIKAR, Rajan,
Mukund [IN/IN]; Everest Builing No. 31,
Block No. 11, Pandit Dindayal Cross Lane, Dombivali
(W), Maharashtra 421202 (IN). SRIDEVI,
Kota [IN/IN]; K.S.R. Murthy, 503, Veena Vihar,
17/A, Flank Road Sion, Mumbai – 400 022 (IN).
RAMAN, Mythili [IN/IN]; G–34, Hoechst Qtrs.,
Amar Nagar, Muland (W), Mumbai – 400 082 (IN).
DALAL, Roda, Maneck [IN/IN]; G–21, Cusrow
Baug, S. Bhagat Singh Road, Colaba, Mumbai –
400 001 (IN).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47889 (13) A1
(21) PCT/EP98/02344
(22) 21 Apr/avr 1998 (21.04.1998)
(25) en (26) en
(31) 9708235.8 (32) 23 Apr/avr 1997 (33) GB
(23.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 311/58, A61K 31/35
(54) • CHROMAN DERIVATIVES
• DERIVES DE CHROMANE
(71) NOVARTIS AG [CH/CH]; Schwarzwaldallee 215,
CH–4058 Basel (CH).
(for all designated States except / pour tous les États
désignés sauf AT US)
(71) NOVARTIS–ERFINDUNGEN VERWAL-
TUNGSGESELLSCHAFT M.B.H. [AT/AT];
Brunner Strasse 59, A–1235 Vienna (AT).
(only for / seulement pour AT)
(72, 75) SWOBODA, Robert [AT/CH]; Moesliweg 30,
CH–3098 Koeniz (CH). POMBO VILLAR, Esteban
[CO/CH]; St.Johanns–Parkweg 5, CH–4056
Basel (CH).
(74) BECKER, Konrad; Novartis AG, Patent– und
Markenabteilung, Lichtstrasse 35, CH–4002 Basel
(CH).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
Published / Publiée : (c)
(11) WO 98/47890 (13) A1
(21) PCT/US98/07677
(22) 18 Apr/avr 1998 (18.04.1998)
(25) en (26) en