PCT/1998/43 - World Intellectual Property Organization

43/1998
15006 PCT Gazette - Section I - Gazette du PCT 29 Oct/oct 1998
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM
GW HU ID IL IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MD MG MK MN MW MX NO
NZ PL PT RO RU SD SE SG SI SK SL TJ TM
TR TT UA UG UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47901 (13) A1
(21) PCT/JP98/01752
(22) 16 Apr/avr 1998 (16.04.1998)
(25) en (26) en
(31) 9/101254 (32) 18 Apr/avr 1997 (33) JP
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 471/16, 211/96, 207/48 // (C07D 471/16,
235:00, 235:00, 221:00) (C07D 471/16, 241:00,
235:00, 221:00)
(54) • PROCESS FOR PRODUCING TRICYCLIC
COMPOUNDS AND THEIR INTERME-
DIATES
• PROCEDE DE PRODUCTION DE
COMPOSES TRICYCLIQUES ET DE LEURS
INTERMEDIAIRES
(71) TAKEDA CHEMICAL INDUSTRIES, LTD.
[JP/JP]; 1–1, Doshomachi 4–chome, Chuo–ku,
Osaka–shi, Osaka 541–0045 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) IKEMOTO, Tomomi [JP/JP]; 11–5, Yamamotomarubashi
2–chome, Takarazuka–shi,
Hyogo 665–0815 (JP). WAKIMASU, Mitsuhiro
[JP/JP]; 1–37, Suimeidai 3–chome, Kawanishi–shi,
Hyogo 666–0116 (JP).
(74) ASAHINA, Tadao et al. / etc.; Osaka Plant of
Takeda Chemical Industries, Ltd., 17–85, Jusohonmachi
2–chome, Yodogawa–ku, Osaka–shi, Osaka
532–0024 (JP).
(81) AL AM AU AZ BA BB BG BR BY CA CN CU
CZ EE GE GW HU ID IL IS KG KR KZ LC LK
LR LT LV MD MG MK MN MX NO NZ PL RO
RU SG SI SK SL TJ TM TR TT UA US UZ VN
YU; AP (GH GM KE LS MW SD SZ UG ZW);
EA (AM AZ BY KG KZ MD RU TJ TM); EP (AT
BE CH CY DE DK ES FI FR GB GR IE IT LU
MC NL PT SE); OA (BF BJ CF CG CI CM GA
GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/47902
(21) PCT/EP98/02252
(13) A1
(22) 17 Apr/avr 1998 (17.04.1998)
(25) en (26) en
(31) MI97A000938 (32) 22 Apr/avr 1997
(22.04.1997)
(33) IT
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 487/18, 471/18, A61K 31/495 // (C07D
487/18, 241:00, 209:00, 209:00) (C07D 471/18,
241:00, 221:00, 221:00)
(54) • 9,10–DIAZATRICYCLO[4.2.1.12,5]DECANE
AND 9,10–
DIAZATRICYCLO[3.3.1.12,6]DECANE DERIVATIVES HAVING ANALGESIC
ACTIVITY
• DERIVES DE 9,10–
DIAZATRICYCLO[4.2.1.12,5]DECANE ET
9,10–DIAZATRICYCLO[3.3.1.12,6]DECANE PRESENTANT UNE ACTIVITE
ANALGESIQUE
(71) NEUROSCIENZE S.C.A.R.L. [IT/IT]; Via Palabanda,
9, I–09125 Cagliari (IT).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) CIGNARELLA, Giorgio [IT/IT]; Universita’
Degli Studi di Milano, Istituto di Chimica Farmaceutica
e Tossicologica, Viale Abruzzi, 42, I–20131
Milano (IT). VIANELLO, Paola [IT/IT]; Universita’
Degli Studi di Milano, Istituto di Chimica
Farmaceutica e Tossicologica, Viale Abruzzi, 42,
I–20131 Milano (IT).
(74) MINOJA, Fabrizio; Bianchetti Bracco Minoja
S.r.l., Via Rossini, 8, I–20122 Milano (IT).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47903 (13) A1
(21) PCT/EP98/02268
(22) 15 Apr/avr 1998 (15.04.1998)
(25) en (26) en
(31) 60/044,524 (32) 22 Apr/avr 1997 (33) US
(22.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 495/04, A61K 31/44, 31/38 // (C07D
495/04, 333:00, 221:00)
(54) • CRF ANTAGONISTIC THIOPHENOPYRI-
DINES
• THIOPHENOPYRIDINES ANTAGONISTES
DU CRF
(71) JANSSEN PHARMACEUTICA N.V. [BE/BE];
Turnhoutseweg 30, B–2340 Beerse (BE). NEURO-
CRINE BIOSCIENCES INC. [US/US]; 3050
Science Park Road, San Diego, CA 92121–1102
(US).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) WEBB, Thomas, R. [US/US]; 2250 Colony
Terrace, Olivenhain, CA 92024 (US). McCAR-
THY, James, R. [US/US]; Neurocrine Biosciences
Inc., 3050 Science Park Road, San Diego, CA
92121–1102 (US).
(74) WANTE, Dirk; Janssen Pharmaceutica N.V., Patent
Dept., Turnhoutseweg 30, B–2340 Beerse
(BE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
Published / Publiée : (c)
(11) WO 98/47904 (13) A1
(21) PCT/US98/08002
(22) 20 Apr/avr 1998 (20.04.1998)
(25) en (26) en
(31) 60/044,145 (32) 22 Apr/avr 1997
(22.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(33) US
(51) 6 C07D 513/04, 249/12, 239/54, 257/04, 211/88,
231/16, 231/14, A01N 43/836
(54) • HERBICIDAL SULFONAMIDES
• SULFONAMIDES HERBICIDES
(71) E.I. DU PONT DE NEMOURS AND COM-
PANY [US/US]; 1007 Market Street, Wilmington,
DE 19898 (US). DEGUSSA AKTIENGE-
SELLSCHAFT [DE/DE]; Weissfrauenstrasse 9,
D–60311 Frankfurt am Main (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) DRAUZ, Karlheinz [DE/DE]; Zur Marienrhe
13, D–63579 Freigericht (DE). HONG, Wonpyo
[KR/US]; 8506 Marburg Manor Drive, Lutherville,
MD 21093 (US). KAMIREDDY, Balreddy
[IN/US]; 204 Golding Court, Hockessin, DE
19707 (US). VOGT, Anne [DE/DE]; Am Markt
19, D–63450 Hanau (DE). WECKBECKER,
Christoph, Helmut [DE/DE]; Grunau Strasse
5, D–63457 Hanau (DE). KLEMENT, Ingo
[DE/DE]; Busring 3, D–35043 Marburg (DE).
(74) KING, Karen, K.; E.I. du Pont de Nemours
and Company, Legal Patent Records Center, 1007
Market Street, Wilmington, DE 19898 (US).
(81) AL AM AU AZ BA BB BG BR BY CA CN CU
CZ EE GE GW HU ID IL IS JP KG KP KR KZ
LC LK LR LT LV MD MG MK MN MX NO NZ
PL RO RU SG SI SK SL TJ TM TR TT UA US
UZ VN YU; AP (GH GM KE LS MW SD SZ UG
ZW); EA (AM AZ BY KG KZ MD RU TJ TM);
EP (AT BE CH CY DE DK ES FI FR GB GR IE
IT LU MC NL PT SE); OA (BF BJ CF CG CI CM
GA GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/47905 (13) A1
(21) PCT/EP98/02414
(22) 23 Apr/avr 1998 (23.04.1998)
(25) de (26) de
(31) 197 17 130.3 (32) 23 Apr/avr 1997 (33) DE
(23.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07F 9/38
(54) • METHOD FOR PRODUCING AMINO ME-
THANE PHOSPHONIC ACID
• PROCEDE DE FABRICATION D’ACIDE
AMINOMETHANEPHOSPHONIQUE
(71) SKW TROSTBERG AKTIENGESELL-
SCHAFT [DE/DE]; Dr.–Albert–Frank–Strasse
32, D–83308 Trostberg (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) NEUMANN, Thomas [DE/DE]; Heinrich–Braun–Strasse
7, D–83308 Trostberg (DE).
FLEISCHER, Frank [DE/DE]; Harter Strasse
19, D–83349 Palling (DE). GRAEFE, Jürgen
[DE/DE]; Bergleite 15, D–83308 Trostberg (DE).
HAMMER, Benedikt [DE/DE]; Am Anger 24,
D–83342 Tacherting (DE).
(74) WEICKMANN, H. et al. / etc.; Kopernikusstrasse
9, D–81679 München (DE).
(81) AU CA NZ US; EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE).
Published / Publiée : (c)
(11) WO 98/47906
(21) PCT/US98/07522
(13) A1
(22) 13 Apr/avr 1998 (13.04.1998)
(25) en (26) en
(31) 08/842,360 (32) 24 Apr/avr 1997
(24.04.1997)
(33) US