PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
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<strong>43</strong>/<strong>1998</strong><br />
29 Oct/oct <strong>1998</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 15007<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07F 9/38, A61K 31/66, C07F 9/40, 9/24, 9/09<br />
(54) • PHOSPHONIC ACID DERIVATIVES<br />
• DERIVES D’ACIDE PHOSPHONIQUE<br />
(71) GUILFORD PHARMACEUTICALS INC.<br />
[US/US]; 6611 Tributary Street, Baltimore, MD<br />
21224 (US).<br />
(72) JACKSON, Paul, F.; 310 Huntsman Court, Bel<br />
Air, MD 21015 (US). TAYS, Kevin, L.; Apartment<br />
1415, 6847 Old Waterloo Road, Elkridge, MD<br />
21227 (US). MACLIN, Keith, M.; 5005 Remmell<br />
Avenue, Baltimore, MD 21206 (US). SLUSHER,<br />
Barbara, S.; 7424 Longfield Drive, Kingsville,<br />
MD 21087 (US).<br />
(74) NATH, Gary, M.; Nath & Associates, Suite 750,<br />
1835 K Street, N.W., Washington, DC 20006 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47907 (13) A1<br />
(21) <strong>PCT</strong>/EP98/01865<br />
(22) 31 Mar/mar <strong>1998</strong> (31.03.<strong>1998</strong>)<br />
(25) de (26) de<br />
(31) 197 17 178.8 (32) 24 Apr/avr 1997 (33) DE<br />
(24.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07F 13/00<br />
(54) • DIRECT SYNTHESIS OF ORGANO–<br />
RHENIUM OXIDES FROM COMPOUNDS<br />
CONTAINING RHENIUM<br />
• SYNTHESE DIRECTE D’OXYDES<br />
D’ORGANORHENIUM A PARTIR DE<br />
COMPOSES CONTENANT DU RHENIUM<br />
(71) HOECHST RESEARCH & TECHNOLOGY<br />
DEUTSCHLAND GMBH & CO. KGS [DE/DE];<br />
Brüningstrasse 50, D–65929 Frankfurt am Main<br />
(DE).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) FISCHER, Richard, Walter [DE/DE];<br />
Königsteiner Strasse 203, D–65812 Bad Soden<br />
(DE). HERRMANN, Wolfgang, Anton [DE/DE];<br />
Gartenstrasse 69c, D–85354 Freising (DE). KRAT-<br />
ZER, Roland [DE/DE]; Fasanenweg 8, D–85356<br />
Freising (DE).<br />
(81) AU CA CN IL JP MX NO SG US; EP (AT BE CH<br />
DE DK ES FI FR GB GR IE IT LU MC NL PT<br />
SE).<br />
Published / Publiée : (a)<br />
(11) WO 98/47908 (13) A1<br />
(21) <strong>PCT</strong>/EP98/02245<br />
(22) 17 Apr/avr <strong>1998</strong> (17.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) MI97A000889 (32) 17 Apr/avr 1997<br />
(17.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07H 3/04, C13K 13/00<br />
(33) IT<br />
(54) • PROCESS FOR THE PREPARATION OF A<br />
LACTULOSE SYRUP BY LACTOSE ISOME-<br />
RIZATION<br />
• PROCEDE DE PREPARATION D’UN SIROP<br />
DE LACTULOSE PAR ISOMERISATION DU<br />
LACTOSE<br />
(71) INALCO S.P.A. [IT/IT]; Via C. Goldoni, 11,<br />
I–20129 Milan (IT).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) CAROBBI, Renato [IT/IT]; Via Dalmazia,<br />
168, I–51100 Pistoia (IT). BIMBI, Giuseppe<br />
[IT/IT]; Via de Nicola, 99, I–56025 Pontedera<br />
(IT). CIPOLLETTI, Giovanni [IT/IT]; Via Tagliamento,<br />
21, I–20139 Milan (IT).<br />
(74) GERVASI, Gemma; Notarbartolo & Gervasi<br />
S.p.A., Corso di Porta Vittoria, 9, I–20122 Milan<br />
(IT).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/47909<br />
(21) <strong>PCT</strong>/US98/06708<br />
(13) A1<br />
(22) 3 Apr/avr <strong>1998</strong> (03.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/844,590 (32) 21 Apr/avr 1997<br />
(21.04.1997)<br />
(33) US<br />
(31) 08/914,7<strong>43</strong> (32) 19 Aug/août 1997<br />
(19.08.1997)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07H 13/06, A23D 9/013, A23L 1/308<br />
(54) • A FLOWABLE NONDIGESTIBLE OIL AND<br />
PROCESS FOR MAKING IT<br />
• HUILE FLUIDE NON ASSIMILABLE ET SON<br />
PROCEDE DE PRODUCTION<br />
(71) THE PROCTER & GAMBLE COMPANY<br />
[US/US]; One Procter & Gamble Plaza, Cincinnati,<br />
OH 45202 (US).<br />
(72) CERRETA, Michael, Kenneth; 44 Bennetts<br />
Bridge Road, Newtown, CT 06482 (US). LIN,<br />
Peter, Yau–Tak; 6753 Netherland Drive, Middletown,<br />
OH 45044 (US). EDWARDS, Penelope,<br />
Marie; 19 Robinson Drive, Greendale, IN 47025<br />
(US). AGERTON, Mark, Lewis; 4126 Ballard<br />
Avenue, Cincinnati, OH 45209 (US).<br />
(74) REED, T., David et al. / etc.; The Procter &<br />
Gamble Company, 5299 Spring Grove Avenue,<br />
Cincinnati, OH 45217 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47910 (13) A1<br />
(21) <strong>PCT</strong>/US98/08192<br />
(22) 20 Apr/avr <strong>1998</strong> (20.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/8<strong>43</strong>,820 (32) 21 Apr/avr 1997 (33) US<br />
(21.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07H 19/00, 21/00, 21/02, 21/04<br />
(54) • METHOD FOR SOLUTION PHASE SYNTHE-<br />
SIS OF OLIGONUCLEOTIDES<br />
• SYNTHESE D’OLIGONUCLEOTIDES EN<br />
SOLUTION<br />
(63) US 08/8<strong>43</strong>,820 (CIP)<br />
21 Apr/avr 1997 (21.04.1997)<br />
(71) NEXSTAR PHARMACEUTICALS, INC.<br />
[US/US]; Suite 200, 2860 Wilderness Place,<br />
Boulder, CO 80301 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) PIEKEN, Wolfgang [US/US]; 4190 South<br />
Hampton Circle, Boulder, CO 80301 (US). MC-<br />
GEE, Danny [CA/US]; 20 South Grant Street,<br />
San Mateo, CA 94401 (US). SETTLE, Alecia<br />
[US/US]; 1497 East Riverbend Street, Superior,<br />
CO 80027 (US). ZHAI, Yansheng [CN/US];<br />
1072 Colorado Place, Palo Alto, CA 9<strong>43</strong>03 (US).<br />
HUANG, JianPing [CN/US]; 1407 Orchard Court,<br />
Lafayette, CO 80026 (US). HILL, Ken [US/US];<br />
115 E. 5th Street, Nederland, CO 80466 (US).<br />
SMITH, Randall, S. [US/US]; 6175 Habitat Drive<br />
#1072, Boulder, CO 80301 (US).<br />
(74) SWANSON, Barry, J. et al. / etc.; Swanson &<br />
Bratschun, L.L.C., Suite 200, 8400 E. Prentice<br />
Avenue, Englewood, CO 80111 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/47911<br />
(21) <strong>PCT</strong>/US98/07397<br />
(13) A1<br />
(22) 13 Apr/avr <strong>1998</strong> (13.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 60/044,507 (32) 21 Apr/avr 1997<br />
(21.04.1997)<br />
(33) US<br />
(31) 09/018,125 (32) 3 Feb/fév <strong>1998</strong><br />
(03.02.<strong>1998</strong>)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07H 21/00, 21/02, C12Q 1/68, A61K 48/00<br />
(54) • RNASE L ACTIVATORS AND ANTISENSE<br />
OLIGONUCLEOTIDES EFFECTIVE TO<br />
TREAT TELOMERASE–EXPRESSING MA-<br />
LIGNANCIES<br />
• ACTIVATEURS DU RNASE L ET OLIGONU-<br />
CLEOTIDES ANTISENS POUVANT TRAI-<br />
TER EFFICACEMENT DES AFFECTIONS<br />
MALIGNES EXPRIMANT TELOMERASE<br />
(71) THE CLEVELAND CLINIC FOUNDATION<br />
[US/US]; 9500 Euclid Avenue, Cleveland, OH<br />
44195 (US). NATIONAL INSTITUTES OF<br />
HEALTH [US/US]; 6011 Executive Boulevard,<br />
Rockville, MD 20852 (US).<br />
(72) SILVERMAN, Robert, H.; 24607 Letchworth<br />
Road, Beachwood, OH 44122 (US). KONDO,<br />
Seiji; 20826 Fairmount Boulevard, Shaker Heights,<br />
OH 44118 (US). COWELL, John, K.; 14808<br />
Shaker Boulevard, Shaker Heights, OH 44120<br />
(US). LI, Guiying; 5011 South Alston Avenue,<br />
Durham, NC 21713 (US). TORRENCE, Paul, F.;<br />
14912 McIntosh Court, Silver Spring, MD 20905<br />
(US).