PCT/1998/43 - World Intellectual Property Organization

43/1998
29 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 15005
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 409/14, A61K 31/44, C07D 417/14,
401/14, 413/14
(54) • 2–OXO–1–AZETIDINE SULFONIC ACID DE-
RIVATIVES AS POTENT –LACTAMASE IN-
HIBITORS
• DERIVES D’ACIDE 2–OXO–1–AZETIDINE
SULFONIQUE AGISSANT COMME INHIBI-
TEURS PUISSANTS DE –LACTAMASE
(71) SYNPHAR LABORATORIES, INC. [CA/CA];
Taiho Alberta Center #2, 4290–91A Street,
Edmonton, Alberta T6E 5V2 (CA). TAIHO
PHARMACEUTICAL CO., LTD. [JP/JP]; 1–27,
Misugidal, Hanno, Saitama 357 (JP).
(72) MAITI, Samarendra, N.; 6756–39 Avenue,
Edmonton, Alberta T6K 1T8 (CA). SETTI,
Eduardo, L.; 202 High Street, Nutley, NJ 07110
(US). PHILLIPS, Oludotun, A.; 4733–35
Avenue, Edmonton, Alberta T6L 3P8 (CA).
REDDY, Andhe, V., Narender; 1503–104 Street,
Edmonton, Alberta T6J 5T2 (CA). MICETICH,
Ronald, G.; 12 Braeside Terrace, Sherwood Park,
Alberta T8A 3V6 (CA). SINGH, Rajeshwar;
7927–22 Avenue, Edmonton, Alberta T6K 1Z2
(CA). HIGASHITANI, Fusahiro; 3–22–9,
Kamiyoshino–cho, Tokushima 770 (JP). KUNU-
GITA, Chieko; 45–11, Myoujinshita, Nakamura,
Kitajima–cho, Itano–gun, Tokushima 771–02 (JP).
NISHIDA, Koichi; 47–5, Kouzima, Syouzui,
Atzumi–cho, Itano–gun, Tokushima 771–12 (JP).
UJI, Tatsuya; 2–31–1–208, Kitayaso–cho, Tokushima
770 (JP).
(81) AU CA HU JP KP KR NO; EP (AT BE CH CY
DE DK ES FI FR GB GR IE IT LU MC NL PT
SE).
(11) WO 98/47896 (13) A1
(21) PCT/JP98/01819
(22) 21 Apr/avr 1998 (21.04.1998)
(25) ja (26) ja
(31) 9/139088 (32) 22 Apr/avr 1997 (33) JP
(22.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 413/04, A61K 31/41, 31/445
(54) • SYDONONIMINE DERIVATIVES
• DERIVES DE SYDONONIMINE
(71) CHUGAI SEIYAKU KABUSHIKI KAISHA
[JP/JP]; 5–1, Ukima 5–chome, Kita–ku, Tokyo
115–8543 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) KOGA, Hiroshi [JP/JP]; Chugai Seiyaku Kabushiki
Kaisha, 1–9, Kyobashi 2–chome, Chuo–ku,
Tokyo 104–8301 (JP). SATO, Haruhiko [JP/JP];
Chugai Seiyaku Kabushiki Kaisha, 135, Komakado
1–chome, Gotenba–shi, Shizuoka 412–8513
(JP). TAKAHASHI, Tadakatsu [JP/JP]; Chugai
Seiyaku Kabushiki Kaisha, 135, Komakado
1–chome, Gotenba–shi, Shizuoka 412–8513 (JP).
IMAOKA, Ikuhiro [JP/JP]; Chugai Seiyaku
Kabushiki Kaisha, 135, Komakado 1–chome,
Gotenba–shi, Shizuoka 412–8513 (JP).
(74) SHAMOTO, Ichio et al. / etc.; Yuasa and Hara,
Section 206, New Ohtemachi Building, 2–1, Ohtemachi
2–chome, Chiyoda–ku, Tokyo 100–0004
(JP).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM
GW HU ID IL IS KE KG KR KZ LC LK LR LS
LT LU LV MD MG MK MN MW MX NO NZ PL
PT RO RU SD SE SG SI SK SL TJ TM TR TT
UA UG US UZ VN YU ZW; AP (GH GM KE LS
MW SD SZ UG ZW); EA (AM AZ BY KG KZ
MD RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE); OA (BF
BJ CF CG CI CM GA GN ML MR NE SN TD
TG).
(11) WO 98/47897 (13) A1
(21) PCT/EP98/01989
(22) 6 Apr/avr 1998 (06.04.1998)
(25) de (26) de
(31) 197 16 258.4 (32) 18 Apr/avr 1997
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(33) DE
(51) 6 C07D 413/12, 271/07, A01N 43/836
(54) • SULFONYLOXADIAZOLONES AND THEIR
USE AS MICROBICIDES
• SULFONYLOXADIAZOLONES ET LEUR
UTILISATION COMME MICROBICIDES
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];
D–51368 Leverkusen (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ASSMANN, Lutz [DE/DE]; Eichblatt 2,
D–23701 Eutin (DE). GERDES, Peter [DE/DE];
Waldstrasse 75, D–52080 Aachen (DE). STEN-
ZEL, Klaus [DE/DE]; Seesener Strasse 17,
D–40595 Düsseldorf (DE).
(74) BAYER AKTIENGESELLSCHAFT; D–51368
Leverkusen (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47898 (13) A1
(21) PCT/FR98/00754
(22) 15 Apr/avr 1998 (15.04.1998)
(25) fr (26) fr
(31) 97/04802 (32) 18 Apr/avr 1997
(18.04.1997)
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 451/04, A61K 31/46
(33) FR
(54) • 5–ARYL–3–(8–AZABICYCLO(3.2.2)OCT–3–
YL)–1,3,4–OXADIAZOL–2(3H)–ONE DERI-
VATIVES AS 5–HT4 RECEPTOR LIGANDS
• DERIVES DE 5–ARYL–3–(8–
AZABICYCLO(3.2.2)OCT–3–YL)–1,3,4–
OXADIAZOL–2(3H)–ONE EN TANT QUE
LIGANDS DES RECEPTEURS 5–HT4
(71) SYNTHELABO [FR/FR]; 22, avenue Galilée,
F–92350 Le Plessis Robinson (FR).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) JEGHAM, Samir [TN/FR]; 65, rue du Lieutenant
Colonel Prudhon, F–95100 Argenteuil (FR).
LOCHEAD, Alistair [GB/FR]; 95, rue de Paris,
F–94220 Charenton (FR). GALLI, Frédéric
[FR/FR]; 3, résidence de l’Orangerie, F–78170
La Celle Saint Cloud (FR). NEDELEC, Alain
[FR/FR]; 97, rue Victor Hugo, F–92700 Colombes
(FR). SAMSON, Axelle [FR/FR]; 6, rue du Renard,
F–75004 Paris (FR). GALLET, Thierry
[FR/FR]; 105, boulevard de Palaiseau, F–91120 Palaiseau
(FR).
(74) LUDWIG, Jacques; Synthelabo, 22, avenue Galilée,
F–92350 Le Plessis Robinson (FR).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR
TT UA UG US UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/47899
(21) PCT/US98/07831
(13) A1
(22) 17 Apr/avr 1998 (17.04.1998)
(25) en (26) en
(31) 60/044,244 (32) 24 Apr/avr 1997
(24.04.1997)
(33) US
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 471/04, A61K 31/44, C07F 7/18 // (C07D
471/04, 221:00, 209:00)
(54) • SUBSTITUTED PYRROLOPYRIDINES USE-
FUL IN THE TREATMENT OF INFLAM-
MATORY DISEASES
• PYRROLOPYRIDINES SUBSTITUEES UTI-
LISEES DANS LE TRAITEMENT DES MA-
LADIES INFLAMMATOIRES
(71) ORTHO–MCNEIL CORPORATION, INC.
[US/US]; U.S. Route #202, P.O. Box 300, Raritan,
NJ 08869–0606 (US).
(72) DODD, John, H.; 15 Alexandria Drive, Pittstown,
NJ 08867 (US). HENRY, James, R.; 260 Turkey
Hill Road, Bloomsbury, NJ 08804 (US). RUPERT,
Kenneth; 426 Centre Street, South Orange, NJ
08079 (US).
(74) CIAMPORCERO, Audley, A., Jr. et al. / etc.;
Johnson & Johnson, One Johnson & Johnson Plaza,
New Brunswick, NJ 08933 (US).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU IL
IS JP KE KG KP KR KZ LC LK LR LS LT LU
LV MD MG MK MN MW MX NO NZ PL PT RO
RU SD SE SG SI SK SL TJ TM TR TT UA UG
UZ VN YU ZW; AP (GH GM KE LS MW SD
SZ UG ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH CY DE DK ES FI FR GB
GR IE IT LU MC NL PT SE); OA (BF BJ CF CG
CI CM GA GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/47900
(21) PCT/DK98/00156
(13) A1
(22) 15 Apr/avr 1998 (15.04.1998)
(25) en (26) en
(31) 0455/97 (32) 22 Apr/avr 1997
(22.04.1997)
(33) DK
(31) 1114/97 (32) 29 Sep/sep 1997
(29.09.1997)
(33) DK
(43) 29 Oct/oct 1998 (29.10.1998)
(51) 6 C07D 471/08, 453/02, 487/08, A61K 31/41
(54) • HETEROCYCLIC COMPOUNDS AND THEIR
PREPARATION AND USE
• COMPOSES HETEROCYCLIQUES, LEUR
PREPARATION ET LEUR UTILISATION
(71) NOVO NORDISK A/S [DK/DK]; Novo Allé,
DK–2880 Bagsværd (DK).
(72) JEPPESEN, Lone; Malmmosevej 121, DK–2830
Virum (DK). SAUERBERG, Per; Syrenvaenget
27, DK–3520 Farum (DK).