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PCT/1998/43 - World Intellectual Property Organization

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<strong>43</strong>/<strong>1998</strong><br />

14998 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 29 Oct/oct <strong>1998</strong><br />

(74) CAVATTONI, Fabio et al. / etc.; Cavattoni<br />

Raimondi, Viale dei Parioli, 160, I–00197 Roma<br />

(IT).<br />

(81) AL AU BA BB BG BR CA CN CU CZ EE GE<br />

GW HU ID IL IS JP KP KR LC LK LR LS LT LV<br />

MG MK MN MW MX NO NZ PL RO SG SI SK<br />

SL TR TT UA US UZ VN YU; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/47858 (13) A1<br />

(21) <strong>PCT</strong>/US98/08311<br />

(22) 21 Apr/avr <strong>1998</strong> (21.04.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 08/845,247 (32) 21 Apr/avr 1997 (33) US<br />

(21.04.1997)<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 229/22, 235/12, A61K 31/495, 31/225,<br />

31/19<br />

(54) • CHELATE DERIVATIVES AS PROTECTORS<br />

AGAINST TISSUE INJURY<br />

• DERIVES DE CHELATES, UTILISES<br />

COMME PROTECTEURS CONTRE LES<br />

LESIONS TISSULAIRES<br />

(63) US 08/845,247 (CON)<br />

21 Apr/avr 1997 (21.04.1997)<br />

(71) EASTERN VIRGINIA MEDICAL SCHOOL<br />

[US/US]; 700 Olney Road, P.O. Box 1980,<br />

Norfolk, VA 23501–1980 (US).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) SCHELLENBERG, Karl, A. [US/US]; 1332<br />

Lakeview Drive, Virginia Beach, VA 23455 (US).<br />

SHAEFFER, James [US/US]; 325 Jule Drive,<br />

Chesapeake, VA 23322 (US). LATTANZIO,<br />

Frank, A., Jr. [US/US]; 3209 Mistletoe Way,<br />

Chesapeake, VA 23323 (US).<br />

(74) WOLFFE, Susan, A. et al. / etc.; Banner &<br />

Witcoff, Ltd., 11th floor, 1001 G Street, N.W.,<br />

Washington, DC 20001–4597 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/47859<br />

(21) <strong>PCT</strong>/US98/07980<br />

(13) A1<br />

(22) 20 Apr/avr <strong>1998</strong> (20.04.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 08/847,951 (32) 22 Apr/avr 1997<br />

(22.04.1997)<br />

(33) US<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 229/26, 227/08, C07D 295/14, C11D 1/10,<br />

1/28, 1/90, B01F 17/00, A61K 7/50<br />

(54) • AMPHOTERIC SURFACTANTS HAVING<br />

MULTIPLE HYDROPHOBIC AND HYDRO-<br />

PHILIC GROUPS<br />

• TENSIO–ACTIFS AMPHOTERES PORTANT<br />

PLUSIEURS GROUPES HYDROPHOBES ET<br />

HYDROPHILES<br />

(71) RHODIA INC. [US/US]; 259 Prospect Plains<br />

Road, Cranbury, NJ 08512–7500 (US).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) TRACY, David, James [US/US]; 37–03<br />

Ravens Crest Drive, Plainsboro, NJ 08536 (US).<br />

LI, Ruoxin [US/US]; 1415 Ravens Crest Drive,<br />

Plainsboro, NJ 08536 (US). YANG, Jiang<br />

[CN/US]; 616 Quil Ridge Drive, Plainsboro, NJ<br />

08536 (US).<br />

(74) SHEDDEN, John, A. et al. / etc.; Rhodia Inc., 259<br />

Prospect Plains Road, Cranbury, NJ 08512–7500<br />

(US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/47860 (13) A1<br />

(21) <strong>PCT</strong>/EP98/01781<br />

(22) 19 Mar/mar <strong>1998</strong> (19.03.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 08/837,844 (32) 22 Apr/avr 1997<br />

(22.04.1997)<br />

(33) US<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 231/02<br />

(54) • PROCESS FOR MAKING CARBOXYLIC<br />

AMIDES<br />

• PROCEDE DE PREPARATION D’AMIDES<br />

CARBOXYLIQUES<br />

(71) AKZO NOBEL N.V. [NL/NL]; Velperweg 76,<br />

NL–6824 BM Arnhem (NL).<br />

(72) MAISONNEUVE, Bernard; 307 Fulle Drive, Valley<br />

Cottage, NY 10989 (US). STEICHEN, Dale,<br />

Stanley; 2 Birch Crest Drive, Danbury, CT 06811<br />

(US). FRANKLIN, Ralph; 25 Tammany Trail,<br />

Danbury, CT 06811 (US). OVERKEMPE, Kornelis;<br />

Erve Lukensveld 27, NL–7451 WH Holten<br />

(NL).<br />

(74) SCHALKWIJK, Pieter, Cornelis; Akzo Nobel<br />

N.V., Patent Dept. (Dept. APTA), P.O. Box 9300,<br />

NL–6800 SB Arnhem (NL).<br />

(81) CA JP; EP (AT BE CH DE DK ES FI FR GB GR<br />

IE IT LU MC NL PT SE).<br />

Published / Publiée : (c)<br />

(11) WO 98/47861<br />

(21) <strong>PCT</strong>/US98/06214<br />

(13) A1<br />

(22) 30 Mar/mar <strong>1998</strong> (30.03.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 60/044,186 (32) 24 Apr/avr 1997<br />

(24.04.1997)<br />

(33) US<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 235/00, 237/00, 239/00<br />

(54) • RETINOID–LIKE COMPOUNDS<br />

• COMPOSES DE TYPE RETINOIDE<br />

(71) BRISTOL–MYERS SQUIBB COMPANY<br />

[US/US]; 5 Research Parkway, Wallingford, CT<br />

06492 (US).<br />

(72) ZUSI, Fred, C.; 20 Nolan Road, Hamden, CT<br />

06514 (US). RECZEK, Peter, R.; 22 Towhee<br />

Court, E. Amherst, NY 14051 (US). OS-<br />

TROWSKI, Jacek; 111 Bywater Drive, Getzville,<br />

NY 14068 (US).<br />

(74) MORSE, David, M.; Bristol–Myers Squibb Company,<br />

5 Research Parkway, Wallingford, CT 06492<br />

(US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG UZ VN YU ZW; AP (GH GM KE LS<br />

MW SD SZ UG ZW); EA (AM AZ BY KG KZ<br />

MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN ML MR NE SN TD TG).<br />

(11) WO 98/47862 (13) A1<br />

(21) <strong>PCT</strong>/EP98/02175<br />

(22) 14 Apr/avr <strong>1998</strong> (14.04.<strong>1998</strong>)<br />

(25) de (26) de<br />

(31) 197 17 231.8 (32) 24 Apr/avr 1997<br />

(24.04.1997)<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 255/57, 251/48, 65/30, 25/13<br />

(33) DE<br />

(54) • 3–CYANO–2,4,5–TRIFLUORO–BENZOYL<br />

FLUORIDE AND INTERMEDIATE PRO-<br />

DUCTS FOR THE PRODUCTION THEREOF<br />

• FLUORURE DE 3–CYANO–2,4,5–<br />

TRIFLUORO–BENZOYLE ET PRODUITS<br />

INTERMEDIAIRES POUR SA FABRICATION<br />

(71) BAYER AKTIENGESELLSCHAFT [DE/DE];<br />

D–51368 Leverkusen (DE).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) MARHOLD, Albrecht [DE/DE];<br />

Carl–Duisberg–Strasse 329, D–51373 Leverkusen<br />

(DE). WOLFRUM, Peter [DE/DE]; Landecker<br />

Weg 18, D–40789 Monheim (DE).<br />

(74) BAYER AKTIENGESELLSCHAFT; D–51368<br />

Leverkusen (DE).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/47863<br />

(21) <strong>PCT</strong>/FR98/00801<br />

(13) A1<br />

(22) 21 Apr/avr <strong>1998</strong> (21.04.<strong>1998</strong>)<br />

(25) fr (26) fr<br />

(31) 97/04971 (32) 22 Apr/avr 1997<br />

(22.04.1997)<br />

(33) FR<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 C07C 259/06, 323/41, C07D 209/26, A61K<br />

31/16, 31/40<br />

(54) • AMINO ACID DERIVATIVES INHIBITING<br />

EXTRACELLULAR MATRIX METALLO-<br />

PROTEINASE AND TNF ALPHA RELEASE<br />

• DERIVES D’AMINO–ACIDES INHIBITEURS<br />

DES METALLOPROTEASES DE LA MA-<br />

TRICE EXTRACELLULAIRE ET DE LA<br />

LIBERATION DU TNF

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