PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
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<strong>43</strong>/<strong>1998</strong><br />
14998 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 29 Oct/oct <strong>1998</strong><br />
(74) CAVATTONI, Fabio et al. / etc.; Cavattoni<br />
Raimondi, Viale dei Parioli, 160, I–00197 Roma<br />
(IT).<br />
(81) AL AU BA BB BG BR CA CN CU CZ EE GE<br />
GW HU ID IL IS JP KP KR LC LK LR LS LT LV<br />
MG MK MN MW MX NO NZ PL RO SG SI SK<br />
SL TR TT UA US UZ VN YU; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47858 (13) A1<br />
(21) <strong>PCT</strong>/US98/08311<br />
(22) 21 Apr/avr <strong>1998</strong> (21.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/845,247 (32) 21 Apr/avr 1997 (33) US<br />
(21.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 229/22, 235/12, A61K 31/495, 31/225,<br />
31/19<br />
(54) • CHELATE DERIVATIVES AS PROTECTORS<br />
AGAINST TISSUE INJURY<br />
• DERIVES DE CHELATES, UTILISES<br />
COMME PROTECTEURS CONTRE LES<br />
LESIONS TISSULAIRES<br />
(63) US 08/845,247 (CON)<br />
21 Apr/avr 1997 (21.04.1997)<br />
(71) EASTERN VIRGINIA MEDICAL SCHOOL<br />
[US/US]; 700 Olney Road, P.O. Box 1980,<br />
Norfolk, VA 23501–1980 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) SCHELLENBERG, Karl, A. [US/US]; 1332<br />
Lakeview Drive, Virginia Beach, VA 23455 (US).<br />
SHAEFFER, James [US/US]; 325 Jule Drive,<br />
Chesapeake, VA 23322 (US). LATTANZIO,<br />
Frank, A., Jr. [US/US]; 3209 Mistletoe Way,<br />
Chesapeake, VA 23323 (US).<br />
(74) WOLFFE, Susan, A. et al. / etc.; Banner &<br />
Witcoff, Ltd., 11th floor, 1001 G Street, N.W.,<br />
Washington, DC 20001–4597 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/47859<br />
(21) <strong>PCT</strong>/US98/07980<br />
(13) A1<br />
(22) 20 Apr/avr <strong>1998</strong> (20.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/847,951 (32) 22 Apr/avr 1997<br />
(22.04.1997)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 229/26, 227/08, C07D 295/14, C11D 1/10,<br />
1/28, 1/90, B01F 17/00, A61K 7/50<br />
(54) • AMPHOTERIC SURFACTANTS HAVING<br />
MULTIPLE HYDROPHOBIC AND HYDRO-<br />
PHILIC GROUPS<br />
• TENSIO–ACTIFS AMPHOTERES PORTANT<br />
PLUSIEURS GROUPES HYDROPHOBES ET<br />
HYDROPHILES<br />
(71) RHODIA INC. [US/US]; 259 Prospect Plains<br />
Road, Cranbury, NJ 08512–7500 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) TRACY, David, James [US/US]; 37–03<br />
Ravens Crest Drive, Plainsboro, NJ 08536 (US).<br />
LI, Ruoxin [US/US]; 1415 Ravens Crest Drive,<br />
Plainsboro, NJ 08536 (US). YANG, Jiang<br />
[CN/US]; 616 Quil Ridge Drive, Plainsboro, NJ<br />
08536 (US).<br />
(74) SHEDDEN, John, A. et al. / etc.; Rhodia Inc., 259<br />
Prospect Plains Road, Cranbury, NJ 08512–7500<br />
(US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47860 (13) A1<br />
(21) <strong>PCT</strong>/EP98/01781<br />
(22) 19 Mar/mar <strong>1998</strong> (19.03.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/837,844 (32) 22 Apr/avr 1997<br />
(22.04.1997)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 231/02<br />
(54) • PROCESS FOR MAKING CARBOXYLIC<br />
AMIDES<br />
• PROCEDE DE PREPARATION D’AMIDES<br />
CARBOXYLIQUES<br />
(71) AKZO NOBEL N.V. [NL/NL]; Velperweg 76,<br />
NL–6824 BM Arnhem (NL).<br />
(72) MAISONNEUVE, Bernard; 307 Fulle Drive, Valley<br />
Cottage, NY 10989 (US). STEICHEN, Dale,<br />
Stanley; 2 Birch Crest Drive, Danbury, CT 06811<br />
(US). FRANKLIN, Ralph; 25 Tammany Trail,<br />
Danbury, CT 06811 (US). OVERKEMPE, Kornelis;<br />
Erve Lukensveld 27, NL–7451 WH Holten<br />
(NL).<br />
(74) SCHALKWIJK, Pieter, Cornelis; Akzo Nobel<br />
N.V., Patent Dept. (Dept. APTA), P.O. Box 9300,<br />
NL–6800 SB Arnhem (NL).<br />
(81) CA JP; EP (AT BE CH DE DK ES FI FR GB GR<br />
IE IT LU MC NL PT SE).<br />
Published / Publiée : (c)<br />
(11) WO 98/47861<br />
(21) <strong>PCT</strong>/US98/06214<br />
(13) A1<br />
(22) 30 Mar/mar <strong>1998</strong> (30.03.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 60/044,186 (32) 24 Apr/avr 1997<br />
(24.04.1997)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 235/00, 237/00, 239/00<br />
(54) • RETINOID–LIKE COMPOUNDS<br />
• COMPOSES DE TYPE RETINOIDE<br />
(71) BRISTOL–MYERS SQUIBB COMPANY<br />
[US/US]; 5 Research Parkway, Wallingford, CT<br />
06492 (US).<br />
(72) ZUSI, Fred, C.; 20 Nolan Road, Hamden, CT<br />
06514 (US). RECZEK, Peter, R.; 22 Towhee<br />
Court, E. Amherst, NY 14051 (US). OS-<br />
TROWSKI, Jacek; 111 Bywater Drive, Getzville,<br />
NY 14068 (US).<br />
(74) MORSE, David, M.; Bristol–Myers Squibb Company,<br />
5 Research Parkway, Wallingford, CT 06492<br />
(US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG UZ VN YU ZW; AP (GH GM KE LS<br />
MW SD SZ UG ZW); EA (AM AZ BY KG KZ<br />
MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN ML MR NE SN TD TG).<br />
(11) WO 98/47862 (13) A1<br />
(21) <strong>PCT</strong>/EP98/02175<br />
(22) 14 Apr/avr <strong>1998</strong> (14.04.<strong>1998</strong>)<br />
(25) de (26) de<br />
(31) 197 17 231.8 (32) 24 Apr/avr 1997<br />
(24.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 255/57, 251/48, 65/30, 25/13<br />
(33) DE<br />
(54) • 3–CYANO–2,4,5–TRIFLUORO–BENZOYL<br />
FLUORIDE AND INTERMEDIATE PRO-<br />
DUCTS FOR THE PRODUCTION THEREOF<br />
• FLUORURE DE 3–CYANO–2,4,5–<br />
TRIFLUORO–BENZOYLE ET PRODUITS<br />
INTERMEDIAIRES POUR SA FABRICATION<br />
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];<br />
D–51368 Leverkusen (DE).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) MARHOLD, Albrecht [DE/DE];<br />
Carl–Duisberg–Strasse 329, D–51373 Leverkusen<br />
(DE). WOLFRUM, Peter [DE/DE]; Landecker<br />
Weg 18, D–40789 Monheim (DE).<br />
(74) BAYER AKTIENGESELLSCHAFT; D–51368<br />
Leverkusen (DE).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47863<br />
(21) <strong>PCT</strong>/FR98/00801<br />
(13) A1<br />
(22) 21 Apr/avr <strong>1998</strong> (21.04.<strong>1998</strong>)<br />
(25) fr (26) fr<br />
(31) 97/04971 (32) 22 Apr/avr 1997<br />
(22.04.1997)<br />
(33) FR<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 C07C 259/06, 323/41, C07D 209/26, A61K<br />
31/16, 31/40<br />
(54) • AMINO ACID DERIVATIVES INHIBITING<br />
EXTRACELLULAR MATRIX METALLO-<br />
PROTEINASE AND TNF ALPHA RELEASE<br />
• DERIVES D’AMINO–ACIDES INHIBITEURS<br />
DES METALLOPROTEASES DE LA MA-<br />
TRICE EXTRACELLULAIRE ET DE LA<br />
LIBERATION DU TNF