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PCT/1998/43 - World Intellectual Property Organization

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<strong>43</strong>/<strong>1998</strong><br />

14944 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 29 Oct/oct <strong>1998</strong><br />

(54) •<br />

•<br />

METHOD FOR THE TREATMENT OF<br />

STROKE USING N–HETEROCYCLIC<br />

GLYOXYLAMIDE COMPOUNDS<br />

PROCEDE DE TRAITEMENT D’ACCIDENT<br />

CEREBROVASCULAIRE A L’AIDE DE<br />

COMPOSES DE GLYOXYLAMIDE N–<br />

HETEROCYCLIQUES<br />

(71) SHIONOGI & CO., LTD. [JP/JP]; 1–8, Doshomachi<br />

3–chome, Chuo–ku, Osaka–shi, Osaka<br />

541–0045 (JP).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) GEMBA, Takefumi [JP/JP]; 2–11–7, Obe, Kawanishi–shi,<br />

Hyogo 666–0014 (JP). HORI, Yozo<br />

[JP/JP]; 7–4–29, Nagaomotomachi, Hirakata–shi,<br />

Osaka 573–0163 (JP).<br />

(74) YAMAUCHI, Hideaki; 12–4, Sagisu 5–chome,<br />

Fukushima–ku, Osaka–shi, Osaka 553–0002 (JP).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM<br />

GW HU ID IL IS JP KE KG KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/47509 (13) A1<br />

(21) <strong>PCT</strong>/US98/07318<br />

(22) 16 Apr/avr <strong>1998</strong> (16.04.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 60/044,626 (32) 18 Apr/avr 1997<br />

(18.04.1997)<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(33) US<br />

(51) 6 A61K 31/415, 31/635, 31/10, 31/18, 31/425,<br />

31/44, 31/42, 31/38, 31/35, 31/535, 31/54, 31/00,<br />

31/<strong>43</strong>5<br />

(54) • METHOD OF USING CYCLOOXYGENASE–<br />

2 INHIBITORS IN THE PREVENTION OF<br />

CARDIOVASCULAR DISORDERS<br />

• PROCEDE RELATIF A L’UTILISATION<br />

D’INHIBITEURS DE CYCLOOXYGENASE–2<br />

DANS LA PREVENTION DES MALADIES<br />

CARDIOVASCULAIRES<br />

(71) G.D. SEARLE & CO. [US/US]; P.O. Box 5110,<br />

Chicago, IL 60680 (US).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) RONIKER, Barbara [US/US]; 1530 N.<br />

Dearborn Parkway, Chicago, IL 60610 (US). La-<br />

CHAPELLE, Richard, J. [US/US]; 1618 Central<br />

Avenue, Wilmette, IL 60091 (US). CONNOLLY,<br />

Daniel, T. [US/US]; 878 Mallard Woods Drive,<br />

Ballwin, MO 63021 (US). SEIBERT, Karen<br />

[US/US]; 11930 Greenwalk Drive, St. Louis, MO<br />

63146 (US). NEEDLEMAN, Philip [US/US]; 326<br />

New Salem Drive, Creve Coeur, MO 63146 (US).<br />

(74) BULOCK, Joseph, W. et al. / etc.; G.D. Searle<br />

& Co., Corporate Patent Dept., P.O. Box 5110,<br />

Chicago, IL 60680–5110 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/47510 (13) A1<br />

(21) <strong>PCT</strong>/JP98/01918<br />

(22) 24 Apr/avr <strong>1998</strong> (24.04.<strong>1998</strong>)<br />

(25) ja (26) ja<br />

(31) 9/107850 (32) 24 Apr/avr 1997 (33) JP<br />

(24.04.1997)<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 A61K 31/445, 45/00, 9/08<br />

(54) • EYE DROPS<br />

• COLLYRE<br />

(71) TAISHO PHARMACEUTICAL CO., LTD.<br />

[JP/JP]; 24–1, Takata 3–chome, Toshima–ku,<br />

Tokyo 170–8633 (JP).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) OKUDAIRA, Ichiro [JP/JP]; Taisho Pharmaceutical<br />

Co., Ltd., 24–1, Takata 3–chome,<br />

Toshima–ku, Tokyo 170–8633 (JP). TSUNODA,<br />

Kenji [JP/JP]; Taisho Pharmaceutical Co., Ltd.,<br />

24–1, Takata 3–chome, Toshima–ku, Tokyo<br />

170–8633 (JP).<br />

(74) KITAGAWA, Tomizo; Taisho Pharmaceutical Co.,<br />

Ltd., Patent Division, 24–1, Takata 3–chome, Toshima–ku,<br />

Tokyo 170–8633 (JP).<br />

(81) AU CA CN KR US; EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE).<br />

(11) WO 98/47511 (13) A1<br />

(21) <strong>PCT</strong>/FR98/00765<br />

(22) 16 Apr/avr <strong>1998</strong> (16.04.<strong>1998</strong>)<br />

(25) fr (26) fr<br />

(31) 97/04801 (32) 17 Apr/avr 1997<br />

(17.04.1997)<br />

(33) FR<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 A61K 31/505<br />

(54) • USE OF MIZOLASTINE FOR PREPARING<br />

A MEDICINE FOR TREATING INFLAMMA-<br />

TION<br />

• UTILISATION DE LA MIZOLASTINE<br />

POUR LA PREPARATION D’UN MEDICA-<br />

MENT DESTINE AU TRAITEMENT DE<br />

L’INFLAMMATION<br />

(71) SYNTHELABO [FR/FR]; 22, avenue Galilée,<br />

F–92350 Le Plessis Robinson (FR).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) ANGEL, Itzchak [IL/IL]; Lotus Street 22,<br />

Nes–Ziyyona (IL). ARBILLA, Sonia [FR/FR]; 16,<br />

rue J.M. de Hérédia, F–75007 Paris (FR). EVEN,<br />

Luc [FR/FR]; 77, rue Lecourbe, F–75015 Paris<br />

(FR). GOLDHILL, Jon [FR/FR]; 24, rue Champ<br />

de Mars, F–75007 Paris (FR). PICHAT, Philippe<br />

[FR/FR]; 28, rue de Chartres, F–91400 Orsay (FR).<br />

(74) THOURET–LEMAITRE, Elisabeth; Synthélabo,<br />

22, avenue Galilée, F–92350 Le Plessis Robinson<br />

(FR).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/47512<br />

(21) <strong>PCT</strong>/US98/07391<br />

(13) A1<br />

(22) 14 Apr/avr <strong>1998</strong> (14.04.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 08/837,637 (32) 21 Apr/avr 1997<br />

(21.04.1997)<br />

(33) US<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 A61K 31/53<br />

(54) • 1,2,4–BENZOTRIAZINE OXIDES FORMU-<br />

LATIONS<br />

• FORMULATIONS OXYDES DE 1,2,4–<br />

BENZOTRIAZINE<br />

(71) SANOFI<br />

[US/US];<br />

PHARMACEUTICALS, INC.<br />

90 Park Avenue, New York, NY<br />

10016 (US).<br />

(72) BROWN, Stephen; 17 The Croft, Ulgham, Morpeth,<br />

Northumberland NE61 3BB (GB). BAKER,<br />

Edward; 3 Bradshawgate, North Farm, Swinhoe,<br />

Chathill, Northumberland NE67 5AA (GB).<br />

(74) ALEXANDER, Michael, D.; Sanofi Pharmaceuticals,<br />

Inc., Patent Dept., 9 Great Valley Parkway,<br />

P.O. Box 3026, Malvern, PA 19355 (US).<br />

(81) AL AU BA BB BG BR CA CN CU CZ EE GE<br />

GW HU ID IL IS JP KP KR LC LK LR LT LV<br />

MG MK MN MX NO NZ PL RO SG SI SK SL<br />

TR TT UA UZ VN YU; AP (GH GM KE LS MW<br />

SD SZ UG ZW); EA (AM AZ BY KG KZ MD<br />

RU TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF BJ CF<br />

CG CI CM GA GN ML MR NE SN TD TG).<br />

(11) WO 98/47513 (13) A1<br />

(21) <strong>PCT</strong>/GB98/01161<br />

(22) 22 Apr/avr <strong>1998</strong> (22.04.<strong>1998</strong>)<br />

(25) en (26) en<br />

(31) 9708289.5 (32) 24 Apr/avr 1997 (33) GB<br />

(24.04.1997)<br />

(31) 9721265.8 (32) 7 Oct/oct 1997 (33) GB<br />

(07.10.1997)<br />

(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />

(51) 6 A61K 31/535, 31/675, 31/<strong>43</strong>5, 31/445, 31/40,<br />

31/47<br />

(54) • USE OF NK–1 RECEPTOR ANTAGONISTS<br />

FOR TREATING EATING DISORDERS<br />

• UTILISATION DES ANTAGONISTES DU RE-<br />

CEPTEUR DE NK–1 DANS LE TRAITEMENT<br />

DES TROUBLES ALIMENTAIRES<br />

(71) MERCK SHARP & DOHME LIMITED<br />

[GB/GB]; Hertford Road, Hoddesdon, Hertfordshire<br />

EN11 9BU (GB).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) HEFTI, Franz, F. [US/GB]; Terlings Park,<br />

Eastwick Road, Harlow, Essex CM20 2QR (GB).<br />

(74) HISCOCK, Ian; Merck & Co., Inc., European Patent<br />

Dept., Terlings Park, Eastwick Road, Harlow,<br />

Essex CM20 2QR (GB).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)

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