PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
PCT/1998/43 - World Intellectual Property Organization
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<strong>43</strong>/<strong>1998</strong><br />
14944 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 29 Oct/oct <strong>1998</strong><br />
(54) •<br />
•<br />
METHOD FOR THE TREATMENT OF<br />
STROKE USING N–HETEROCYCLIC<br />
GLYOXYLAMIDE COMPOUNDS<br />
PROCEDE DE TRAITEMENT D’ACCIDENT<br />
CEREBROVASCULAIRE A L’AIDE DE<br />
COMPOSES DE GLYOXYLAMIDE N–<br />
HETEROCYCLIQUES<br />
(71) SHIONOGI & CO., LTD. [JP/JP]; 1–8, Doshomachi<br />
3–chome, Chuo–ku, Osaka–shi, Osaka<br />
541–0045 (JP).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) GEMBA, Takefumi [JP/JP]; 2–11–7, Obe, Kawanishi–shi,<br />
Hyogo 666–0014 (JP). HORI, Yozo<br />
[JP/JP]; 7–4–29, Nagaomotomachi, Hirakata–shi,<br />
Osaka 573–0163 (JP).<br />
(74) YAMAUCHI, Hideaki; 12–4, Sagisu 5–chome,<br />
Fukushima–ku, Osaka–shi, Osaka 553–0002 (JP).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/47509 (13) A1<br />
(21) <strong>PCT</strong>/US98/07318<br />
(22) 16 Apr/avr <strong>1998</strong> (16.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 60/044,626 (32) 18 Apr/avr 1997<br />
(18.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(33) US<br />
(51) 6 A61K 31/415, 31/635, 31/10, 31/18, 31/425,<br />
31/44, 31/42, 31/38, 31/35, 31/535, 31/54, 31/00,<br />
31/<strong>43</strong>5<br />
(54) • METHOD OF USING CYCLOOXYGENASE–<br />
2 INHIBITORS IN THE PREVENTION OF<br />
CARDIOVASCULAR DISORDERS<br />
• PROCEDE RELATIF A L’UTILISATION<br />
D’INHIBITEURS DE CYCLOOXYGENASE–2<br />
DANS LA PREVENTION DES MALADIES<br />
CARDIOVASCULAIRES<br />
(71) G.D. SEARLE & CO. [US/US]; P.O. Box 5110,<br />
Chicago, IL 60680 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) RONIKER, Barbara [US/US]; 1530 N.<br />
Dearborn Parkway, Chicago, IL 60610 (US). La-<br />
CHAPELLE, Richard, J. [US/US]; 1618 Central<br />
Avenue, Wilmette, IL 60091 (US). CONNOLLY,<br />
Daniel, T. [US/US]; 878 Mallard Woods Drive,<br />
Ballwin, MO 63021 (US). SEIBERT, Karen<br />
[US/US]; 11930 Greenwalk Drive, St. Louis, MO<br />
63146 (US). NEEDLEMAN, Philip [US/US]; 326<br />
New Salem Drive, Creve Coeur, MO 63146 (US).<br />
(74) BULOCK, Joseph, W. et al. / etc.; G.D. Searle<br />
& Co., Corporate Patent Dept., P.O. Box 5110,<br />
Chicago, IL 60680–5110 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/47510 (13) A1<br />
(21) <strong>PCT</strong>/JP98/01918<br />
(22) 24 Apr/avr <strong>1998</strong> (24.04.<strong>1998</strong>)<br />
(25) ja (26) ja<br />
(31) 9/107850 (32) 24 Apr/avr 1997 (33) JP<br />
(24.04.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 A61K 31/445, 45/00, 9/08<br />
(54) • EYE DROPS<br />
• COLLYRE<br />
(71) TAISHO PHARMACEUTICAL CO., LTD.<br />
[JP/JP]; 24–1, Takata 3–chome, Toshima–ku,<br />
Tokyo 170–8633 (JP).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) OKUDAIRA, Ichiro [JP/JP]; Taisho Pharmaceutical<br />
Co., Ltd., 24–1, Takata 3–chome,<br />
Toshima–ku, Tokyo 170–8633 (JP). TSUNODA,<br />
Kenji [JP/JP]; Taisho Pharmaceutical Co., Ltd.,<br />
24–1, Takata 3–chome, Toshima–ku, Tokyo<br />
170–8633 (JP).<br />
(74) KITAGAWA, Tomizo; Taisho Pharmaceutical Co.,<br />
Ltd., Patent Division, 24–1, Takata 3–chome, Toshima–ku,<br />
Tokyo 170–8633 (JP).<br />
(81) AU CA CN KR US; EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE).<br />
(11) WO 98/47511 (13) A1<br />
(21) <strong>PCT</strong>/FR98/00765<br />
(22) 16 Apr/avr <strong>1998</strong> (16.04.<strong>1998</strong>)<br />
(25) fr (26) fr<br />
(31) 97/04801 (32) 17 Apr/avr 1997<br />
(17.04.1997)<br />
(33) FR<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 A61K 31/505<br />
(54) • USE OF MIZOLASTINE FOR PREPARING<br />
A MEDICINE FOR TREATING INFLAMMA-<br />
TION<br />
• UTILISATION DE LA MIZOLASTINE<br />
POUR LA PREPARATION D’UN MEDICA-<br />
MENT DESTINE AU TRAITEMENT DE<br />
L’INFLAMMATION<br />
(71) SYNTHELABO [FR/FR]; 22, avenue Galilée,<br />
F–92350 Le Plessis Robinson (FR).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) ANGEL, Itzchak [IL/IL]; Lotus Street 22,<br />
Nes–Ziyyona (IL). ARBILLA, Sonia [FR/FR]; 16,<br />
rue J.M. de Hérédia, F–75007 Paris (FR). EVEN,<br />
Luc [FR/FR]; 77, rue Lecourbe, F–75015 Paris<br />
(FR). GOLDHILL, Jon [FR/FR]; 24, rue Champ<br />
de Mars, F–75007 Paris (FR). PICHAT, Philippe<br />
[FR/FR]; 28, rue de Chartres, F–91400 Orsay (FR).<br />
(74) THOURET–LEMAITRE, Elisabeth; Synthélabo,<br />
22, avenue Galilée, F–92350 Le Plessis Robinson<br />
(FR).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/47512<br />
(21) <strong>PCT</strong>/US98/07391<br />
(13) A1<br />
(22) 14 Apr/avr <strong>1998</strong> (14.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 08/837,637 (32) 21 Apr/avr 1997<br />
(21.04.1997)<br />
(33) US<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 A61K 31/53<br />
(54) • 1,2,4–BENZOTRIAZINE OXIDES FORMU-<br />
LATIONS<br />
• FORMULATIONS OXYDES DE 1,2,4–<br />
BENZOTRIAZINE<br />
(71) SANOFI<br />
[US/US];<br />
PHARMACEUTICALS, INC.<br />
90 Park Avenue, New York, NY<br />
10016 (US).<br />
(72) BROWN, Stephen; 17 The Croft, Ulgham, Morpeth,<br />
Northumberland NE61 3BB (GB). BAKER,<br />
Edward; 3 Bradshawgate, North Farm, Swinhoe,<br />
Chathill, Northumberland NE67 5AA (GB).<br />
(74) ALEXANDER, Michael, D.; Sanofi Pharmaceuticals,<br />
Inc., Patent Dept., 9 Great Valley Parkway,<br />
P.O. Box 3026, Malvern, PA 19355 (US).<br />
(81) AL AU BA BB BG BR CA CN CU CZ EE GE<br />
GW HU ID IL IS JP KP KR LC LK LR LT LV<br />
MG MK MN MX NO NZ PL RO SG SI SK SL<br />
TR TT UA UZ VN YU; AP (GH GM KE LS MW<br />
SD SZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF BJ CF<br />
CG CI CM GA GN ML MR NE SN TD TG).<br />
(11) WO 98/47513 (13) A1<br />
(21) <strong>PCT</strong>/GB98/01161<br />
(22) 22 Apr/avr <strong>1998</strong> (22.04.<strong>1998</strong>)<br />
(25) en (26) en<br />
(31) 9708289.5 (32) 24 Apr/avr 1997 (33) GB<br />
(24.04.1997)<br />
(31) 9721265.8 (32) 7 Oct/oct 1997 (33) GB<br />
(07.10.1997)<br />
(<strong>43</strong>) 29 Oct/oct <strong>1998</strong> (29.10.<strong>1998</strong>)<br />
(51) 6 A61K 31/535, 31/675, 31/<strong>43</strong>5, 31/445, 31/40,<br />
31/47<br />
(54) • USE OF NK–1 RECEPTOR ANTAGONISTS<br />
FOR TREATING EATING DISORDERS<br />
• UTILISATION DES ANTAGONISTES DU RE-<br />
CEPTEUR DE NK–1 DANS LE TRAITEMENT<br />
DES TROUBLES ALIMENTAIRES<br />
(71) MERCK SHARP & DOHME LIMITED<br />
[GB/GB]; Hertford Road, Hoddesdon, Hertfordshire<br />
EN11 9BU (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) HEFTI, Franz, F. [US/GB]; Terlings Park,<br />
Eastwick Road, Harlow, Essex CM20 2QR (GB).<br />
(74) HISCOCK, Ian; Merck & Co., Inc., European Patent<br />
Dept., Terlings Park, Eastwick Road, Harlow,<br />
Essex CM20 2QR (GB).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)