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2.1 ReferencesPart-IIIAim of the Present Work1. Saponara, S.; Kawase, M.; Shah, A.; Motohashi, N.; Molnar, J.; Ugocsai, K.;Sgaragli, G.; Fusi, F. Br. J. Pharmacol. 2004, 141, 415.2. Fusi, F.; Saponara, S.; Valoti, M.; Dragoni, S.; D’Elia, P.; Sgaragli, T.; Alderighi,D.; Kawase, M.; Shah, A.; Motohashi, N.; Sgaragli, G. Curr. Drug Targets 2006,7, 949; 7, 1729.3. Saponara, S.; Ferrara, A.; Gorelli, B.; Shah, A.; Kawase, M.; Motohashi, N.;Molnar, J.; Sgaragli, G.; Fusi, F. Eur. J. Pharmacol. 2007, 563, 160.4. Mayer, T. U.; Kapoor, T. M.; Haggarty, S. J.; King, R. W.; Schreiber, S. I.;Mitchison, T. J. Science 1999, 268, 971.5. Maliga, Z.; Kapoor, T. M.; Mitchison, T. J. Chem. Biol. 2000, 9, 989.6. Biginelli, P.; P. Gazz. Chim. Ital. 1893, 23, 360.7. Kappe, C. O. Tetrahedron 1993, 49, 6937.8. Kappe, C. O. QSAR Comb. Sci. 2003, 22, 630.9. Lou, S.; Taoka, B. M.; Ting, A.; Schaus, S. E. J. Am. Chem. Soc. 2005, 127,11256.10. Munoz-Muniz, O.; Juaristi, E. Arkivoc 2003, 11, 16.11. Dondoni, A.; Massi, A.; Sabbatini, S.; Bertolasi, V. J. Org. Chem. 2002, 67, 6974.12. Dondoni, A.; Massi, A.; Minghini, E.; Sabbatini, S.; Bertolasi, V. J. Org. Chem.2003, 68, 6172.13. Huang, Y.; Yang, F.; Zhu, C. J. Am. Chem. Soc. 2005, 127, 16386.14. Hu, E. H.; Sidler, D. R.; Dolling, U.-H. J. Org. Chem. 1998, 63, 3454.15. Ranu, B. C.; Hajra, A.; Jana, U. J. Org. Chem. 2000, 65, 6270.16. Lu, J.; Bai, Y. Synthesis 2002, 466.17. Chen, R.-F.; Quian, C.-T. Chin. J. Chem. 2002, 20, 427.18. Bose, D. S.; Fatima, L.; Mereyala, H. B. J. Org. Chem. 2003, 68, 587.19. Narsaiah, A. V.; Basak, A. K.; Nagaiah, K. Synthesis 2004, 1253.20. Salehi, H.; Guo, Q.-X. Chin. J. Chem. 2005, 23, 91.21. Russowsky, D.; Lopes, F. A.; daSilva, V. S. S.; Canto, K. F. S.; D’Oca, M. G. M.Godoi, M. N. J. Br. Chem. Soc. 2004, 15, 165.22. D’Oca, M. G. M.; Godoi, M. N.; Kramer, E.; Costenaro, H. S.; Russowsky, D.Quı´mica Nova 2005, 12, 738.453

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