Bulletin 2011/35 - European Patent Office

(C07C) I.1(1)
C07C 319/18 → (51) C07C 45/52
C07C 319/20 → (51) C07C 45/52
C07C 323/22 → (51) C07C 45/52
C07C 323/52 → (51) C07C 45/52
C07C 323/58 → (51) C07C 45/52
(51) C07D 207/12 (11) 2 361 244 A1*
(25) En (26) En
(21) 09801288.3 (22) 24.11.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) IN 2009/000680 24.11.2009
(87) WO 2010/058429 2010/21 27.05.2010
(30) 24.11.2008 IN DE26482008
(54) • VERFAHREN ZUR HERSTELLUNG
OPTISCH AKTIVER N-BENZYL-3-HYDRO-
XYPYRROLIDINE
• A PROCESS FOR THE PREPARATION OF
OPTICALLY ACTIVE N-BENZYL-3 HYDRO-
XYPYRROLIDINES
• PROCÉDÉ DE PRÉPARATION DE N-BEN-
ZYL-3-HYDROXYPYRROLIDINES OPTI-
QUEMENT ACTIVES
(71) Council of Scientific & Industrial Research,
Anusandhan Bhawan, 2 Rafi Marg, New
Delhi 110 001, IN
(72) TANEJA, Subhash, Chandra, Jammu Tawi
180 001, IN
AGA, Mushtaq, Ahmad, Jammu Tawi 180
001, IN
KUMAR, Brijesh, Jammu Tawi 180 001, IN
SETHI, Vijay, Kumar, Jammu Tawi 180 001,
IN
ANDOTRA, Samar, Singh, Jammu Tawi 180
001, IN
QAZI, Gulham, Nabi, Jammu Tawi 180 001,
IN
(74) Jakobsson, Jeanette Helene, Awapatent AB
Bellevuevägen 46 P.O. Box 5117, 200 71
Malmö, SE
(51) C07D 209/12 (11) 2 361 245 A1*
A61K 31/12 A61K 31/335
A61K 31/381 A61K 31/403
A61K 31/404 A61K 31/415
A61K 31/47 A61P 35/00
C07C 49/237 C07C 49/255
C07D 209/86 C07D 215/14
C07D 231/06 C07D 333/56
(25) En (26) En
(21) 09828505.9 (22) 25.11.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) CA 2009/001719 25.11.2009
(87) WO 2010/060214 2010/22 03.06.2010
(30) 26.11.2008 US 118037 P
(54) • HYBRID-IONON- UND CURCUMINMOLE-
KÜLE ALS ANTIKREBSWIRKSTOFFE
• HYBRID -IONONE AND CURCUMIN
MOLECULES AS ANTICANCER AGENTS
• MOLÉCULES HYBRIDES D IONONE ET DE
CURCUMINE EN TANT QU AGENTS ANTI-
CANCÉREUX
(71) TRT Pharma Inc ., 2015 Peel Street, 5th
Floor, Montreal, QC H3A 1T8, CA
(72) WU, Jian Hui, Montreal, Quebec H4P 1P4,
CA
BATIST, Gerald, Montreal, Quebec H3W 2L8,
CA
ZHOU, Jinming, 100050 Beijing, CN
GENG, Guoyan, Montreal, Quebec H4E 1H3,
CA
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
LIN, Rongtuan, Dollard-Des -Ormeaux, Quebec
H9A 3G7, CA
(74) Rihm, Sven, Savic Patentanwälte Bayerstraße
83, DE-80355 München, DE
C07D 209/86 → (51) C07D 209/12
C07D 211/36 → (51) C07D 213/75
(51) C07D 211/76 (11) 2 361 246 A1*
C07D 405/10 C07D 409/10
C07D 309/14 A61K 31/351
A61K 31/381 A61K 31/4433
A61K 31/451 A61P 25/00
(25) En (26) En
(21) 09787251.9 (22) 18.09.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) IB 2009/054109 18.09.2009
(87) WO 2010/038167 2010/14 08.04.2010
(30) 02.10.2008 US 102095 P
(54) • OXOPIPERIDINYL- UND PYRANYLSULFO-
NAMIDE ALS AMPA-VERSTÄRKER
• OXOPIPERIDINYL AND PYRANYL SULFO-
NAMIDES AS AMPA POTENTIATORS
• OXOPIPÉRIDINYLSULFAMIDES ET PYRA-
NYLSULFAMIDES UTILISABLES EN TANT
QUE POTENTIALISATEURS DES RÉCEP-
TEURS AMPA
(71) Pfizer Inc., 235 East 42nd Street, New York,
NY 10017, US
(72) ESTEP, Kimberly Gail, Groton, Connecticut
06340, US
FLIRI, Anton F. J., Stonington, Connecticut
06378, US
GALLASCHUN, Randall James, Lebanon,
Connecticut 06249, US
O'DONNELL, Christopher John, Groton,
Connecticut 06340, US
PATEL, Nandini Chaturbhai, Groton, Connecticut
06340, US
SCHWARZ, Jacob Bradley, Waterford, Connecticut
06385, US
XIE, Longfei, Groton, Connecticut 06340, US
(74) Summers, Victoria Clare, Pfizer Limited
European Patent Department Ramsgate
Road, Sandwich, Kent CT13 9NJ, GB
(51) C07D 213/75 (11) 2 361 247 A2*
A61K 31/44 A61P 25/04
A61P 25/00 C07D 211/36
(25) En (26) En
(21) 09805531.2 (22) 06.08.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2009/052925 06.08.2009
(87) WO 2010/017343 2010/06 11.02.2010
(88) 14.05.2010
(30) 06.08.2008 US 86644 P
(54) • FLUPIRTINHYDROCHLORID-MALEIN-
SÄURE-COKRISTALL
• FLUPIRTINE HYDROCHLORIDE MALEIC
ACID COCRYSTAL
• COCRISTAL D HYDROCHLORURE DE
FLUPIRTINE ET D ACIDE MALÉIQUE
(71) Bionevia Pharmaceuticals Inc., 1 Nichols
Place, Cambridge, MA 02138, US
(72) KALOFONOS, Isabel, Cambridge MA 02138,
US
STAHLY, G., Patrick, West Lafayette IN
47906, US
MARTIN-DOYLE, William, Cambridge MA
02141, US
KALOFONOS, Dimitris, Cambridge MA
02138, US
STULTS, Jeffrey, S., West Lafayette IN
47906, US
48
Anmeldungen
Applications
Demandes (35/2011) 31.08.2011
HANKO, Jason, A., West Lafayette IN 47906,
US
SHIPPLETT, Rex, A., Wolcott IN 47995, US
(74) Cottrill, Emily Elizabeth Helen, A.A. Thornton
& Co. 235 High Holborn, London WC1V 7LE,
GB
C07D 215/14 → (51) C07D 209/12
C07D 231/06 → (51) C07D 209/12
C07D 233/76 → (51) C07C 45/52
C07D 235/26 → (51) A61K 31/41
(51) C07D 239/47 (11) 2 361 248 A1*
C07D 239/48 C07D 401/14
C07D 403/12 C07D 407/12
C07D 413/12 C07D 413/14
C07D 471/04 C07D 487/04
C07D 487/18 A61K 31/505
A61K 31/506 A61P 29/00
A61P 35/00 A61P 37/00
(25) En (26) En
(21) 09771102.2 (22) 26.06.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) US 2009/048784 26.06.2009
(87) WO 2009/158571 2009/53 30.12.2009
(30) 20.04.2009 US 170874 P
29.01.2009 US 148388 P
27.06.2008 US 76450 P
(54) • HETEROARYLVERBINDUNGEN UND IHRE
VERWENDUNGEN
• HETEROARYL COMPOUNDS AND USES
THEREOF
• COMPOSÉS HÉTÉRO-ARYLES ET LEURS
UTILISATIONS
(71) Avila Therapeutics, Inc., 100 Beaver Street,
First Floor, Waltham, MA 02453-8425, US
(72) KLUGE, Arthur, F., Lincoln MA 01773, US
PETTER, Russell, C., Stow MA 01775, US
TESTER, Richland, Wayne, Marlborough MA
01752, US
QIAO, Lixin, Tewksbury MA 01876, US
NIU, Deqiang, Lexington MA 02141, US
WESTLIN, William, Frederick, Boxborough
MA 01719, US
SINGH, Juswinder, Ashland MA 01721, US
MAZDIYASNI, Hormoz, Marlborough MA
01752, US
(74) Tostmann, Holger Carl, et al, Wallinger
Ricker Schlotter Foerstl Patent- und
Rechtsanwälte Zweibrückenstrasse 5-7,
80331 München, DE
C07D 239/48 → (51) C07D 239/47
C07D 295/192→ (51) C07C 229/10
C07D 307/02 → (51) C07D 307/58
(51) C07D 307/58 (11) 2 361 249 A2*
C07D 307/02 A61P 31/04
(25) En (26) En
(21) 09826824.6 (22) 13.11.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2009/064366 13.11.2009
(87) WO 2010/056978 2010/20 20.05.2010
(88) 22.07.2010
(30) 13.11.2008 US 114265 P