Bulletin 2009/06 - European Patent Office
Bulletin 2009/06 - European Patent Office
Bulletin 2009/06 - European Patent Office
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(C07C) II.1(1)<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
<strong>Patent</strong>e<br />
<strong>Patent</strong>s<br />
Brevets (<strong>06</strong>/<strong>2009</strong>) 04.02.<strong>2009</strong><br />
(51) C07C 45/50 (11) 1 279 658 B1<br />
C07C 29/156<br />
(25) De (26) De<br />
(21) 02012800.5 (22) 10.<strong>06</strong>.2002<br />
(84) BE DE FR GB NL<br />
(43) 29.01.2003<br />
(30) 24.07.2001 DE 101359<strong>06</strong><br />
(54) • Verfahren zur Hydroformylierung von<br />
höheren Olefinen mit Kobaltverbindungen<br />
als Katalysator<br />
• Process for the hydroformylation of higher<br />
olefins in presence of cobalt compounds as<br />
catalyst<br />
• Procédé pour l'hydroformylation d'oléfines<br />
supérieures en présence de composés de<br />
cobalt comme catalyseur<br />
(73) Evonik Oxeno GmbH, Paul-Baumann-Strasse<br />
1, 45772 Marl, DE<br />
(72) Scholz, Bernhard, Dr., 45768 Marl, DE<br />
Tötsch, Walter, Dr., 45770 Marl, DE<br />
Drees, Stefan, 48249 Dülmen, DE<br />
Kaizik, Alfred, Dr., 45772 Marl, DE<br />
Trocha, Martin, Dr., 45136 Essen, DE<br />
Büschken, Wilfried, Dr., 45721 Haltern, DE<br />
(74) Hirsch, Hans-Ludwig, et al, Evonik Degussa<br />
GmbH DG-IPM-PAT Bau 1042 / PB 15 Paul-<br />
Baumann-Strasse 1, 45764 Marl, DE<br />
C07C 49/647 → (51) C07C 35/18<br />
C07C 49/683 → (51) C07C 35/18<br />
(51) C07C 59/68 (11) 1 538 140 B1<br />
C11D 1/74<br />
(25) De (26) De<br />
(21) 04026130.7 (22) 04.11.2004<br />
(84) BE DE ES FR GB IT<br />
(43) 08.<strong>06</strong>.2005<br />
(30) 17.11.2003 DE 10353603<br />
(54) • Ethercarbonsäuren auf Basis alkoxylierter<br />
Styrylphenole<br />
• Ether carboxylic acids based on alkoxylated<br />
styrylphenol<br />
• Acides carboxyliques d'éther à base de<br />
styrylphenol alcoxylé<br />
(73) Clariant Produkte (Deutschland) GmbH,<br />
Brüningstrasse 50, 65929 Frankfurt am<br />
Main, DE<br />
(72) Dahlmann, Uwe, Dr., 69126 Heidelberg, DE<br />
Kupfer, Rainer, Dr., 65795 Hattersheim, DE<br />
(51) C07C 59/90 (11) 1 565 422 B1<br />
C07C 62/24 C07C 69/78<br />
C07C 235/34 C07C 311/50<br />
C07C 317/28 C07D 257/<strong>06</strong><br />
C07D 277/34 A61K 31/12<br />
A61K 31/165 A61K 31/18<br />
A61K 31/19 A61K 31/192<br />
A61K 31/235 A61K 31/41<br />
A61K 31/426<br />
(25) En (26) En<br />
(21) 03781741.8 (22) 20.11.2003<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PT RO SE SI SK<br />
TR<br />
AL LT LV MK<br />
(43) 24.08.2005<br />
(86) US 2003/035055 20.11.2003<br />
(87) WO 2004/048309 2004/24 10.<strong>06</strong>.2004<br />
(30) 22.11.2002 US 429041 P<br />
(54) • MODULATOREN VON VITAMIN D<br />
REZEPTOREN<br />
• VITAMIN D RECEPTOR MODULATORS<br />
• MODULATEURS DE RECEPTEUR DE<br />
VITAMINE D<br />
(73) ELI LILLY AND COMPANY, Lilly Corporate<br />
Center, Indianapolis IN 46285, US<br />
(72) BUNEL, Emilio, Enrique, Thousand Oaks,<br />
California 91362, US<br />
GAJEWSKI, Robert, Peter, Indianapolis, IN<br />
46217, US<br />
JONES, Charles, David, Indianapolis, IN<br />
46227, US<br />
LU, Jianliang, Fishers, IN 46038, US<br />
MA, Tianwei, Carmel, IN 46033, US<br />
NAGPAL, Sunil, Carmel, IN 46033, US<br />
YEE, Ying, Kwong, Carmel, IN 46033, US<br />
(74) Hiscock, Ian James, <strong>European</strong> <strong>Patent</strong><br />
Operations, Eli Lilly and Company Limited,<br />
Lilly Research Centre, Erl Wood Manor,<br />
Sunninghill Road Windlesham GU20 6PH,<br />
GB<br />
C07C 62/24 → (51) C07C 59/90<br />
C07C 69/78 → (51) C07C 59/90<br />
C07C 235/34 → (51) C07C 59/90<br />
C07C 255/23 → (51) A61L 24/<strong>06</strong><br />
C07C 311/50 → (51) C07C 59/90<br />
(51) C07C 317/14 (11) 1 824 817 B1<br />
C07D 213/71 C07D 215/36<br />
C07D 471/02 C07D 241/12<br />
A61K 31/10 A61K 31/275<br />
A61K 31/4409 A61K 31/47<br />
A61P 25/00<br />
(25) En (26) En<br />
(21) 05813608.6 (22) 28.11.2005<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
(43) 29.08.2007<br />
(86) GB 2005/050215 28.11.2005<br />
(87) WO 20<strong>06</strong>/059149 20<strong>06</strong>/23 08.<strong>06</strong>.20<strong>06</strong><br />
(30) 01.12.2004 GB 0426313<br />
(54) • ARYLSULFONYLNAPHTHALINDERIVATE<br />
ALS 5HT2A-ANTAGONISTEN<br />
• ARYLSULFONYLNAPHTHALENE DERIVA-<br />
TIVES AS 5HT2A ANTAGONISTS<br />
• DERIVES DE L'ARYLSULFONYLNAPHTA-<br />
LENE UTILISES EN TANT QU'ANTAGO-<br />
NISTES DE 5HT2A<br />
(73) MERCK SHARP & DOHME LTD., Hertford<br />
Road, Hoddesdon, Hertfordshire EN11 9BU,<br />
GB<br />
(72) CHAMBERS, Mark, Stuart, Harlow, Essex<br />
CM20 2QR, GB<br />
CURTIS, Neil, Roy, Eastwick Road, Harlow,<br />
Essex CM20 2QR, GB<br />
GANCIA, Emanuela, Harlow, Essex CM20<br />
2QR, GB<br />
GILLIGAN, Myra, Harlow, Essex CM20 2QR,<br />
GB<br />
HUMPHRIES, Alexander, Charles, Harlow,<br />
Essex CM20 2QR, GB<br />
LADDUWAHETTY, Tamara, Harlow, Essex<br />
CM20 2QR, GB<br />
MAXEY, Robert, James, Harlow, Essex CM20<br />
2QR, GB<br />
MERCHANT, Kevin, John, Harlow, Essex<br />
CM20 2QR, GB<br />
(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />
<strong>European</strong> <strong>Patent</strong> Department Hertford Road,<br />
Hoddesdon, Hertfordshire EN11 9BU, GB<br />
C07C 317/28 → (51) C07C 59/90<br />
(51) C07D 211/22 (11) 1 002 794 B1<br />
A61K 31/4465<br />
(25) Es (26) En<br />
(21) 99500208.6 (22) 10.11.1999<br />
(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />
LU MC NL PT SE<br />
(43) 24.05.2000<br />
(30) 18.11.1998 ES 9802420<br />
(54) • 4-¬(Aryl)(aryloxy)methyl piperidinderivate<br />
und ihre Verwendung als Serotonin und/<br />
oder Noradrenalin Reuptake Inhibitoren<br />
• 4-¬(Aryl)(aryloxy)methyl piperidine derivatives<br />
and their use as serotonin and/or<br />
noradrenaline reuptake inhibitors<br />
• Dérivés de 4-¬(aryl)(aryloxy)methyl pipéridine<br />
et leur usage comme inhibiteurs de la<br />
réabsorption de sérotonine et/ou de noradrénaline<br />
(73) FAES, Fabrica Espanola de Productos Quimicos<br />
y Farmaceuticos, S.A., Maximo<br />
Aguirre, 14, 48940 Lejona, Vizcaya, ES<br />
(72) Orjales Venero, Aurelio, 48990 Neguri (Vizcaya),<br />
ES<br />
Toledo Avello, Antonio, 48990 Algorta (Vizcaya),<br />
ES<br />
Pumar Duran, Carmen, 48110 Gatika (Vizcaya),<br />
ES<br />
(74) ABG <strong>Patent</strong>es, S.L., Avenida de Burgos 16D<br />
Edificio Euromor, 28036 Madrid, ES<br />
C07D 213/71 → (51) C07C 317/14<br />
(51) C07D 213/79 (11) 1 601 653 B1<br />
C07D 213/80 C07D 405/12<br />
C07D 409/12 C07D 401/12<br />
C07D 413/12 C07D 417/12<br />
C07D 401/<strong>06</strong> C07D 401/08<br />
C07D 417/<strong>06</strong> C07D 417/08<br />
C07D 413/<strong>06</strong> C07D 413/08<br />
(25) En (26) En<br />
(21) 04717574.0 (22) 05.03.2004<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />
TR<br />
(43) 07.12.2005<br />
(86) EP 2004/002291 05.03.2004<br />
(87) WO 2004/078729 2004/38 16.09.2004<br />
(30) 07.03.2003 CH 373032003<br />
(54) • VERFAHREN ZUR HERSTELLUNG SUB-<br />
STITUIERTER NIKOTINSÄUREESTER<br />
• PROCESS FOR THE PRODUCTION OF<br />
SUBSTITUTED NICOTINIC ACID ESTERS<br />
• PROCEDE DE PRODUCTION D'ESTERS<br />
D'ACIDES NICOTINIQUES SUBSTITUES<br />
(73) Syngenta Participations AG, Schwarzwaldallee<br />
215, 4058 Basel, CH<br />
(72) JACKSON, David Anthony, Syngenta Huddersfield,<br />
West Yorkshire, HD2 1FF, GB<br />
BOWDEN, Martin Charles, Huddersfield,<br />
West Yorkshire, HD2 1FF, GB<br />
(74) Hölscher, Ingo, et al, Syngenta Participations<br />
AG Intellectual Property P.O. Box, 4002<br />
Basel, CH<br />
C07D 213/80 → (51) C07D 213/79<br />
C07D 215/36 → (51) C07C 317/14<br />
(51) C07D 231/12 (11) 1 492 773 B1<br />
C07D 401/04 C07D 307/46<br />
C07D 263/38 C07D 277/34<br />
C07D 261/08 A61K 31/34<br />
A61K 31/415 A61K 31/42<br />
A61K 31/425 A61K 31/44<br />
A61P 29/00<br />
(25) En (26) En<br />
(21) 03733003.2 (22) 01.04.2003<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PT RO SE SI SK<br />
TR<br />
(43) 05.01.2005<br />
(86) IN 2003/000133 01.04.2003<br />
229