Bulletin 2009/06 - European Patent Office
Bulletin 2009/06 - European Patent Office
Bulletin 2009/06 - European Patent Office
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(C07D) I.1(1)<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
Anmeldungen<br />
Applications<br />
Demandes (<strong>06</strong>/<strong>2009</strong>) 04.02.<strong>2009</strong><br />
ALONSO CASCÓN, Mercedes, 28036 Madrid,<br />
ES<br />
FUERTES HUERTA, Ana, 28003 Madrid, ES<br />
NAVARRO RICO, María Luisa, 28014 Madrid,<br />
ES<br />
PÉREZ PUERTO, María José, 28008 Madrid,<br />
ES<br />
DEL MONTE MILLÁN, María, 28032 Madrid,<br />
ES<br />
(74) ABG <strong>Patent</strong>es, S.L., Avenida de Burgos 16D<br />
Edificio Euromor, 28036 Madrid, ES<br />
(51) C07D 417/12 (11) 2 019 829 A1*<br />
A61K 31/426 A61K 31/427<br />
A61P 25/28<br />
(25) En (26) En<br />
(21) 07728642.5 (22) 27.04.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) EP 2007/054188 27.04.2007<br />
(87) WO 2007/125110 2007/45 08.11.2007<br />
(30) 28.04.20<strong>06</strong> EP <strong>06</strong>380099<br />
04.01.2007 US 878386 P<br />
(54) • N-(2-THIAZOLYL)AMIDDERIVATE ALS<br />
GSK-3-INHIBITOREN<br />
• N- ( 2-THIAZOLYL) -AMIDE DERIVATIVES<br />
AS GSK-3 INHIBITORS<br />
• UTILISATION DE DÉRIVÉS DE N-(2-THIA-<br />
ZOLYL)-AMIDES EN TANT QU'INHIBI-<br />
TEURS DE LA GSK-3<br />
(71) Noscira, S.A., Avenida de la Industria, 52,<br />
28760 Tres Cantos, ES<br />
(72) MARTÍNEZ GIL, Ana, E-28004 Madrid, ES<br />
CASTRO MORERA, Ana, E-28028 Madrid, ES<br />
MEDINA PADILLA, Miguel, E-28035 Madrid,<br />
ES<br />
MARTÍN APARICIO, Ester, E-28411 Moralzarzal<br />
- Madrid, ES<br />
ALONSO CASCÓN, Mercedes, E-28036<br />
Madrid, ES<br />
FUERTES HUERTA, Ana, E-28003 Madrid, ES<br />
NAVARRO RICO, María Luisa, E-28014<br />
Madrid, ES<br />
PÉREZ PUERTO, María José, E-28008<br />
Madrid, ES<br />
DEL MONTE MILLÁN, María, E-28032<br />
Madrid, ES<br />
(74) ABG <strong>Patent</strong>es, S.L., Avenida de Burgos 16D<br />
Edificio Euromor, 28036 Madrid, ES<br />
C07D 417/12 → (51) C07D 207/10<br />
C07D 417/12 → (51) C07D 277/46<br />
C07D 417/14 → (51) C07D 409/14<br />
(51) C07D 487/04 (11) 2 019 830 A2*<br />
A61K 31/519 A61K 31/662<br />
C07F 9/32 A61P 31/22<br />
(25) En (26) En<br />
(21) 07761888.2 (22) 04.05.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 2007/<strong>06</strong>8241 04.05.2007<br />
(87) WO 2007/131168 2007/46 15.11.2007<br />
(88) 20.11.2008<br />
(30) 04.05.20<strong>06</strong> US 797581 P<br />
(54) • HEMMER DER SEKRETION VON HEPATI-<br />
TIS-B-VIRUS-ANTIGENEN ZUR BEHAND-<br />
LUNG EINES CHRONISCHEN HEPATITIS-<br />
VIRUS<br />
• INHIBITORS OF SECRETION OF HEPATITIS<br />
B VIRUS ANTIGENS FOR TREATMENT OF<br />
A CHRONIC HEPATITIS VIRUS<br />
• INHIBITEURS DE LA SÉCRÉTION D'ANTI-<br />
GÈNES DU VIRUS DE L'HÉPATITE B<br />
DESTINÉS AU TRAITEMENT D'UN VIRUS<br />
DE L'HÉPATITE CHRONIQUE<br />
(71) Institute For Hepatitis And Virus Research,<br />
3805 Old Easton Road, Doylestown, PA<br />
18902, US<br />
Drexel University, 3225 Arch Street, Ground<br />
Floor, Philadelphia, PA 19104, US<br />
(72) CUCONATI, Andrea, Oreland, PA 19075, US<br />
BLOCK, Timothy M., Doylestown, PA 18901,<br />
US<br />
XU, Xiaodong, Doylestown, PA 18902, US<br />
(74) Leissler-Gerstl, Gabriele, et al, Hoefer &<br />
Partner <strong>Patent</strong>anwälte Pilgersheimer Strasse<br />
20, 81543 München, DE<br />
(51) C07D 491/22 (11) 2 019 831 A1*<br />
A61K 31/439 A61P 25/00<br />
A61P 25/18 A61P 25/22<br />
A61P 25/34<br />
(25) En (26) En<br />
(21) 07748149.7 (22) 16.05.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) SE 2007/000485 16.05.2007<br />
(87) WO 2007/133155 2007/47 22.11.2007<br />
(30) 17.05.20<strong>06</strong> US 747476 P<br />
08.09.20<strong>06</strong> US 824975 P<br />
(54) • LIGANDEN DES NIKOTINISCHEN ACETYL-<br />
CHOLINREZEPTORS 101<br />
• NICOTINIC ACETYLCHOLINE RECEPTOR<br />
LIGANDS 101<br />
• LIGAND 101 DU RÉCEPTEUR D'ACÉTYL-<br />
CHOLINE NICOTINIQUE<br />
(71) Astra Zeneca AB, S-151 85 Södertalje, SE<br />
(72) CHANG, Hui-Fang, Wilmington, Delaware<br />
19850-5437, US<br />
HOLMQUIST, Christopher, Wilmington,<br />
Delaware 19850-5437, US<br />
PHILLIPS, Eifion, Boothwyn, Pennsylvania<br />
19<strong>06</strong>1, US<br />
PISER, Timothy, Wilmington, Delaware<br />
19850-5437, US<br />
SIMPSON, Thomas, Wilmington, Delaware<br />
19850-5437, US<br />
URBANEK, Rebecca, Wilmington, Delaware<br />
19850-5437, US<br />
WOODS, James, Wilmington, Delaware<br />
19850-5437, US<br />
XIONG, Hui, Wilmington, Delaware 19850-<br />
5437, US<br />
(74) Larsson, Birgitta, et al, AstraZeneca AB,<br />
Intellectual Property, <strong>Patent</strong>s, 151 85<br />
Södertälje, SE<br />
(51) C07F 9/02 (11) 2 019 832 A1*<br />
(25) En (26) En<br />
(21) 07732773.2 (22) 14.05.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) GB 2007/001748 14.05.2007<br />
(87) WO 2007/132210 2007/47 22.11.2007<br />
(30) 16.05.20<strong>06</strong> GB <strong>06</strong>09617<br />
(54) • VERFAHREN ZUR HERSTELLUNG VON<br />
PYRAZOLYLAMINOCHINAZOLINDERIVA-<br />
TEN MIT EINER PHOSPHATGRUPPE<br />
• PROCESS FOR THE PREPARATION OF<br />
PYRAZOLYLAMINOQUINAZOLINE DERI-<br />
VATIVES COMPRISING A PHOSPHATE<br />
GROUP<br />
• PROCÉDÉ DE PRÉPARATION DE DÉRIVÉS<br />
PYRAZOLYLAMINOQUINAZOLINE COM-<br />
PRENANT UN GROUPE PHOSPHATE<br />
(71) AstraZeneca AB, 151 85 Södertälje, SE<br />
(72) PITTAM, John, David, Macclesfield Cheshire<br />
SK10 2NA, GB<br />
SEPENDA, George, Joseph, Macclesfield<br />
Cheshire SK10 2NA, GB<br />
C07F 9/32 → (51) C07D 487/04<br />
(51) C07H 13/<strong>06</strong> (11) 2 019 833 A1*<br />
C07C 67/03<br />
(25) En (26) En<br />
(21) 07732566.0 (22) 26.04.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) GB 2007/001529 26.04.2007<br />
(87) WO 2007/125328 2007/45 08.11.2007<br />
(30) 28.04.20<strong>06</strong> GB <strong>06</strong>08512<br />
(54) • VERFAHREN ZUR HERSTELLUNG VON<br />
ESTERN VON ZUCKERN UND ZUCKER-<br />
DERIVATEN<br />
• PROCESS FOR THE PRODUCTION OF<br />
ESTERS OF SUGARS AND SUGAR DERI-<br />
VATIVES<br />
• PROCEDE DE PRODUCTION D'ESTERS DE<br />
SUCRES ET DE DERIVES DE SUCRE<br />
(71) Sebus Ltd, Oswald House, 24-26 Queens<br />
Road Reading RG1 4AU, GB<br />
(72) JAMES, Kenneth, Reading RG1 4AU, GB<br />
SMITH, James, Frederick, Reading RG1 4AU,<br />
GB<br />
(74) Beresford, Keith Denis Lewis, et al, Beresford<br />
& Co 16 High Holborn, London WC1V 6BX,<br />
GB<br />
(51) C07H 19/<strong>06</strong> (11) 2 019 834 A1*<br />
C07H 19/16 A61P 29/00<br />
A61P 27/02 A61P 25/00<br />
A61P 11/00 A61K 31/7052<br />
(25) En (26) En<br />
(21) 07729500.4 (22) 24.05.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) EP 2007/055071 24.05.2007<br />
(87) WO 2007/135195 2007/48 29.11.2007<br />
(30) 24.05.20<strong>06</strong> EP <strong>06</strong>114534<br />
(54) • ECTONUKLEOTDASEINHIBITOREN<br />
• ECTONUCLEOTIDASE INHIBITORS<br />
• INHIBITEURS D'ECTONUCLÉOTIDASES<br />
(71) Rheinische Friedrich-Wilhelms-Universität<br />
Bonn, Regina-Pacis-Weg 3, 53113 Bonn, DE<br />
(72) MÜLLER, Christa E., 53113 Bonn, DE<br />
BRUNSCHWEIGER, Andreas, 53225 Bonn-<br />
Beuel, DE<br />
IQBAL, Jamshed, 53115 Bonn, DE<br />
(74) Helbing, Jörg, et al, <strong>Patent</strong>anwälte von<br />
Kreisler Selting Werner Bahnhofsvorplatz 1<br />
Deichmannhaus am Dom, 5<strong>06</strong>67 Köln, DE<br />
C07H 19/16 → (51) C07H 19/<strong>06</strong><br />
(51) C07H 21/00 (11) 2 019 835 A1*<br />
A61K 31/7088 A61P 11/00<br />
A61P 29/00<br />
(25) En (26) En<br />
(21) 07719824.0 (22) 18.05.2007<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) CA 2007/000902 18.05.2007<br />
(87) WO 2007/134451 2007/48 29.11.2007<br />
(30) 19.05.20<strong>06</strong> US 801384 P<br />
50