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European Patent Bulletin 2012/36 - European Patent Office

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(A01N) I.1(1)<br />

ALLEVIATING OXIDATIVE STRESS<br />

DISORDERS WITH PUFA DERIVATIVES<br />

SOULAGEMENT DE TROUBLES LIÉS AU<br />

STRESS OXYDATIF PAR DES DÉRIVÉS<br />

DE PUFA<br />

(71) Retrotope, Inc., 12133 Foothill Lane, Los<br />

Altos Hills, CA 94022-3319, US<br />

(72) SHCHEPINOV, Mikhail, S., Oxford<br />

Oxfordshire OX3 0PN, GB<br />

(74) Carpintero Lopez, Francisco, et al, Herrero &<br />

Asociados, S.L. Alcalá 35, 28014 Madrid, ES<br />

A01N 37/06 → (51) C07C 69/67<br />

(51) A01N 37/12 (11) 2 493 297 A1*<br />

A01N 37/18 A61K 31/16<br />

(25) En (26) En<br />

(21) 10827<strong>36</strong>1.6 (22) 25.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/053908 25.10.2010<br />

(87) WO 2011/053542 2011/18 05.05.2011<br />

(30) 30.10.2009 US 256740 P<br />

(54) HETEROCYCLISCHE AMID-CALCIUM-<br />

KANALANTAGONISTEN VOM TYP T<br />

HETEROCYCLE AMIDE T-TYPE CALCIUM<br />

CHANNEL ANTAGONISTS<br />

ANTAGONISTES DES CANAUX CALCI-<br />

QUES DE TYPE T AMIDES HÉTÉROCY-<br />

CLIQUES<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) SCHLEGEL, Kelly-Ann, West Point, Pennsylvania<br />

19486, US<br />

SHU, Yoheng, West Point, Pennsylvania<br />

19486, US<br />

YANG, Zhi-Qiang, West Point, Pennsylvania<br />

19486, US<br />

BARROW, James, Arnold, Maryland 21012,<br />

US<br />

(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Hertford Road,<br />

Hoddesdon, Hertfordshire EN11 9BU, GB<br />

(51) A01N 37/12 (11) 2 493 298 A1*<br />

A61K 31/195<br />

(25) En (26) En<br />

(21) 10827583.5 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054872 29.10.2010<br />

(87) WO 2011/053876 2011/18 05.05.2011<br />

(30) 01.12.2009 US 265468 P<br />

30.10.2009 US 256927 P<br />

(54) VERWENDUNG VON CI-994 UND DINA-<br />

LIN ZUR BEHANDLUNG VON GEDÄCHT-<br />

NIS-/KOGNITIVEN UND ANGSTSTÖRUN-<br />

GEN<br />

THE USE OF CI-994 AND DINALINE FOR<br />

THE TREATMENT OF MEMORY/<br />

COGNITION AND ANXIETY DISORDERS<br />

UTILISATION DE CI-994 ET DE DINALINE<br />

POUR LE TRAITEMENT DE TROUBLES DE<br />

LA MÉMOIRE/COGNITION ET DE L'AN-<br />

XIÉTÉ<br />

(71) Massachusetts Institute of Technology, 77<br />

Massachusetts Avenue, Cambridge, MA<br />

02139, US<br />

The General Hospital Corporation d/b/a<br />

Massachusetts General Hospital, 55 Fruit<br />

Street, Boston, MA 02114, US<br />

The Broad Institute, Inc., 7 Cambridge<br />

Center, Cambridge, MA02142, US<br />

(72) TSAI, Li-Huei, Cambridge MA 02138, US<br />

GUAN, Ji-Song, Medford MA 02155, US<br />

HAGGARTY, Stephen, J., Dorchester MA<br />

02125, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

HOLSON, Edward, Newton Highlands MA<br />

02461, US<br />

WAGNER, Florence, Ashland MA 01721, US<br />

GRAEFF, Johannes, Waban MA 02468, US<br />

(74) Korn, Richard Mervyn, Potter Clarkson LLP<br />

Park View House 58 The Ropewalk,<br />

Nottingham NG1 5DD, GB<br />

(51) A01N 37/18 (11) 2 493 299 A1*<br />

A61K 31/16<br />

(25) En (26) En<br />

(21) 10827347.5 (22) 22.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/05<strong>36</strong>87 22.10.2010<br />

(87) WO 2011/053522 2011/18 05.05.2011<br />

(30) 29.10.2009 US 255916 P<br />

(54) TERTIÄRE AMIDOREXINREZEPTORANTA-<br />

GONISTEN<br />

TERTIARY AMIDE OREXIN RECEPTOR<br />

ANTAGONISTS<br />

ANTAGONISTES DE RÉCEPTEURS<br />

D'OREXINES AMIDES TERTIAIRES<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) COLEMAN, Paul, J., West Point, Pennsylvania<br />

19486, US<br />

MERCER, Swati, P., West Point, Pennsylvania<br />

19486, US<br />

ROECKER, Anthony, J., West Point, Pennsylvania<br />

19486, US<br />

(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Hertford Road,<br />

Hoddesdon, Hertfordshire EN11 9BU, GB<br />

A01N 37/18 → (51) A01N 37/12<br />

(51) A01N 37/34 (11) 2 493 300 A1*<br />

(25) En (26) En<br />

(21) 10826219.7 (22) 18.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) IL 2010/000848 18.10.2010<br />

(87) WO 2011/051932 2011/18 05.05.2011<br />

(30) 29.10.2009 US 255889 P<br />

(54) BREITBAND-BIOZIDZUSAMMENSETZUN-<br />

GEN UND VERFAHREN ZU IHRER HER-<br />

STELLUNG<br />

BROAD-SPECTRUM BIOCIDE COMPO-<br />

SITIONS AND A METHOD FOR THEIR<br />

PREPARATION<br />

COMPOSITIONS BIOCIDES À SPECTRE<br />

LARGE ET PROCÉDÉ POUR LEUR<br />

PRÉPARATION<br />

(71) Bromine Compounds Ltd., Makleff House<br />

P.O.B. 180, 84894 Beer-Sheva, IL<br />

(72) SHAPIRO, Evgeny, 32922 Haifa, IL<br />

ZOLKOV, Chen, <strong>36</strong>081 Kiryat Tivon, IL<br />

KHODAKOVSKAYA, Rimma, 33061 Haifa, IL<br />

EFFENBERGER, Reinhard, 34<strong>36</strong>7 Haifa, IL<br />

(74) Bottero, Carlo, et al, Barzanò & Zanardo<br />

Milano S.p.A. Via Borgonuovo, 10, <strong>2012</strong>1<br />

Milano, IT<br />

A01N 39/02 → (51) A01N 43/40<br />

(51) A01N 41/10 (11) 2 493 301 A1*<br />

(25) En (26) En<br />

(21) 10830412.2 (22) 22.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/053701 22.10.2010<br />

(87) WO 2011/059661 2011/20 19.05.2011<br />

(30) 29.10.2009 US 256201 P<br />

19<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(54) QUECKSILBERENTFERNUNG MITHILFE<br />

VON AMINSORPTIONSMITTELN<br />

MERCURY REMOVAL WITH AMINE<br />

SORBENTS<br />

ELIMINATION DE MERCURE AVEC DES<br />

SORBANTS AMINÉS<br />

(71) Conocophillips Company, IP Services Group<br />

Attn: Docketing 600 N. Dairy Ashford MA-<br />

1135, Houston, Texas 77079, US<br />

(72) HAYS, John, Michael, Bartlesville Oklahoma<br />

74006, US<br />

CROSS, Joe B., Bartlesville Oklahoma<br />

74006, US<br />

(74) Hyden, Martin Douglas, FINNEGAN LLP<br />

Avenue Louise, 326 PO Box 37, 1050<br />

Brussels, BE<br />

A01N 43/18 → (51) A01N 43/40<br />

(51) A01N 43/38 (11) 2 493 302 A1*<br />

A61K 31/40<br />

(25) En (26) En<br />

(21) 10827377.2 (22) 26.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054035 26.10.2010<br />

(87) WO 2011/053567 2011/18 05.05.2011<br />

(30) 30.10.2009 US 256631 P<br />

09.03.2010 US 311954 P<br />

(54) HEXAHYDROCYCLOPENTYL-[F-]INDA-<br />

ZOL-PYRIDYLETHANOLE UND DERIVATE<br />

DAVON ALS SELEKTIVE GLUCOCORTI-<br />

COID-REZEPTOR-MODULATOREN<br />

HEXAHYDROCYCLOPENTYL[F]INDAZOLE<br />

PYRIDYL ETHANOLS AND DERIVATIVES<br />

THEREOF AS SELECTIVE GLUCOCOR-<br />

TICOID RECEPTOR MODULATORS<br />

HEXAHYDROCYCLOPENTYL[F]INDAZO-<br />

LEPYRIDYL ÉTHANOLS ET LEUR<br />

DÉRIVÉS COMME MODULATEURS<br />

SÉLECTIFS DES RÉCEPTEURS AUX<br />

GLUCOCORTICOÏDES<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) MITCHELL, Helen, J., West Point, Pennsylvania<br />

19486, US<br />

DANKULICH, William, P., West Point, New<br />

Jersey 19486, US<br />

KAUFMAN, Mildred, L., West Point, Pennsylvania<br />

19486, US<br />

MEISSNER, Robert, S., West Point, Pennsylvania<br />

19486, US<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

& Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon EN11 9BU, GB<br />

(51) A01N 43/38 (11) 2 493 303 A1*<br />

A61K 31/40<br />

(25) En (26) En<br />

(21) 10827382.2 (22) 26.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054052 26.10.2010<br />

(87) WO 2011/053574 2011/18 05.05.2011<br />

(30) 30.10.2009 US 256676 P<br />

(54) 2- [1-PHENYL-5-HYDROXY-4A-SUBSTI-<br />

TUTIERTE-HEXAHYDROCYCLOPENTA<br />

[F]INDAZOL-5-YL]ETHYLPHENYLDERI-<br />

VATE ALS GLUCOCORTICOIDREZEPT-<br />

ORLIGANDEN<br />

2- [1-PHENYL-5-HYDROXY-4a-<br />

SUBSTITUTED-HEXAHYDROCY-<br />

CLOPENTA [F]INDAZOL-5-YL]ETHYL<br />

PHENYL DERIVATIVES AS GLUCOCOR-<br />

TICOID RECEPTOR LIGANDS<br />

DÉRIVÉS 2-[1-PHÉNYL-5-HYDROXY-4A-<br />

SUBSTITUÉS-HEXAHYDROCYCLOPEN-<br />

TA[F]INDAZOL-5-YL]ÉTHYL PHÉNYLÉS

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