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European Patent Bulletin 2012/36 - European Patent Office

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(A61K) I.1(1)<br />

RAUCHENBERGER, Robert, 82152 Martinsried/Planegg,<br />

DE<br />

RUTZ, Mark, 82152 Martinsried/Planegg, DE<br />

ALMAGRO, Juan, Carlos, Radnor, PA 19087,<br />

US<br />

TAUDTE, Susann, Radnor, PA 19087, US<br />

WU, Bingyuan, Radnor, PA 19087, US<br />

OBMOLOVA, Galina, Radnor, PA 19087, US<br />

MALIA, Thomas, Radnor, PA 19087, US<br />

(74) Carpmaels & Ransford, One Southampton<br />

Row, London WC1B 5HA, GB<br />

(51) A61K 39/395 (11) 2 493 507 A2*<br />

C07K 16/00<br />

(25) En (26) En<br />

(21) 10827525.6 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054714 29.10.2010<br />

(87) WO 2011/053783 2011/18 05.05.2011<br />

(88) 28.07.2011<br />

(30) 30.10.2009 US 256732 P<br />

12.04.2010 US 323148 P<br />

(54) AX213- UND AX132-PCSK9-ANTAGONIS-<br />

TEN UND VARIANTEN DAVON<br />

AX213 AND AX132 PCSK9 ANTAGONISTS<br />

AND VARIANTS<br />

ANTAGONISTES ET VARIANTS AX213 ET<br />

AX132 PCSK9<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) LUO, Peter Peizhi, Lansdale Pennsylvania<br />

19446, US<br />

NI, Yan, Rahway New Jersey 07065-0907,<br />

US<br />

WANG, Kevin Caili, West Point Pennsylvania<br />

19486, US<br />

HSIEH, Mark, West Point Pennsylvania<br />

19486, US<br />

WANG, Xinwei, West Point Pennsylvania<br />

19486, US<br />

DONG, Feng, West Point Pennsylvania<br />

19486, US<br />

GOLOSOV, Andrei, West Point Pennsylvania<br />

19486, US<br />

WANG, Weirong, West Point Pennsylvania<br />

19486, US<br />

LI, Yan, West Point Pennsylvania 19486, US<br />

ZHONG, Pingyu, Blue Bell Pennsylvania<br />

19422, US<br />

PETERSON, Laurence, B., Westfield New<br />

Jersey 07090, US<br />

CUBBON, Rose, Fanwood New Jersey<br />

07023, US<br />

SHARMA, Sujata, West Point Pennsylvania<br />

19486, US<br />

CONDRA, Jon, West Point Pennsylvania<br />

19486, US<br />

LU, Jun, West Point Pennsylvania 19486, US<br />

PARTHASARATHY, Gopalakrishnan, West<br />

Point Pennsylvania 19486, US<br />

SOISSON, Stephen, West Point Pennsylvania<br />

19486, US<br />

BYRNE, Noel, West Point Pennsylvania<br />

19486, US<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

& Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

A61K 39/395 → (51) A61K 35/14<br />

A61K 39/395 → (51) C07K 16/00<br />

A61K 39/395 → (51) C07K 16/24<br />

A61K 39/395 → (51) C07K 16/28<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

A61K 41/00 → (51) A61L 2/00<br />

A61K 41/00 → (51) A61P 17/02<br />

A61K 45/06 → (51) A61K 31/135<br />

A61K 45/06 → (51) A61K 31/164<br />

(51) A61K 47/10 (11) 2 493 508 A2*<br />

A61K 47/12 A61K 47/14<br />

A61K 9/06 A61K 9/08<br />

A61K 31/565 A61K 31/568<br />

A61K 31/57<br />

(25) En (26) En<br />

(21) 10768983.8 (22) 27.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) EP 2010/066283 27.10.2010<br />

(87) WO 2011/051354 2011/18 05.05.2011<br />

(88) 01.03.<strong>2012</strong><br />

(30) 10.12.2009 EP 09178762<br />

27.10.2009 US 255241 P<br />

(54) TRANSDERMALE PHARMAZEUTISCHE<br />

ZUSAMMENSETZUNGEN MIT WIRKSTOF-<br />

FEN<br />

TRANSDERMAL PHARMACEUTICAL<br />

COMPOSITIONS COMPRISING ACTIVE<br />

AGENTS<br />

COMPOSITIONS PHARMACEUTIQUES<br />

TRANSDERMIQUES CONTENANT DES<br />

AGENTS ACTIFS<br />

(71) Besins Healthcare Luxembourg SARL, 67<br />

boulevard Grande-Duchesse Charlotte, 1331<br />

Luxembourg, LU<br />

(72) MASINI-ETEVE, Valérie, F-92340 Bourg La<br />

Reine, FR<br />

CANET, Denis, B-1050 Bruxelles, BE<br />

(74) Cabinet Plasseraud, 52, rue de la Victoire,<br />

75440 Paris Cedex 09, FR<br />

(51) A61K 47/12 (11) 2 493 509 A2*<br />

A61K 47/14 A61K 9/00<br />

A61K 31/00<br />

(25) En (26) En<br />

(21) 10796168.2 (22) 27.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) NL 2010/050720 27.10.2010<br />

(87) WO 2011/053139 2011/18 05.05.2011<br />

(88) 23.06.2011<br />

(30) 27.10.2009 NL 2003711<br />

(54) WÄSSRIGE ZUSAMMENSETZUNG FÜR<br />

TOPISCHE ANWENDUNG, ZUBEREI-<br />

TUNGSVERFAHREN, VERWENDUNG UND<br />

VORRICHTUNG<br />

AQUEOUS COMPOSITION FOR TOPICAL<br />

APPLICATION, METHOD OF<br />

PREPARATION, USES AND DEVICE<br />

COMPOSITION AQUEUSE POUR APPLI-<br />

CATION TOPIQUE, PROCÉDÉ DE PRÉPA-<br />

RATION, UTILISATIONS ET DISPOSITIF<br />

(71) Medner B.V., Professor Tulpstraat 18, 1018<br />

HA Amsterdam, NL<br />

(72) CLAPPOSEN, Miriam, NL-1070 AR Amsterdam,<br />

NL<br />

(74) Jansen, Bart Antonius Johannes, Zacco<br />

Netherlands B.V. Nachtwachtlaan 20, 1058<br />

EA Amsterdam, NL<br />

A61K 47/12 → (51) A61K 47/10<br />

A61K 47/14 → (51) A61K 47/10<br />

A61K 47/14 → (51) A61K 47/12<br />

A61K 47/30 → (51) A23L 1/05<br />

48<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(51) A61K 47/48 (11) 2 493 510 A1*<br />

(25) En (26) En<br />

(21) 10779848.0 (22) 30.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) IB 2010/002565 30.09.2010<br />

(87) WO 2011/1386<strong>36</strong> 2011/45 10.11.2011<br />

(30) 30.09.2009 US 247518 P<br />

(54) KONJUGATION VON KAPSELFÖRMIGEN<br />

POLYSACCHARIDEN TYP 5 UND TYP 8<br />

AUS STAPHYLOCOCCUS AUREUS<br />

CONJUGATION OF STAPHYLOCOCCUS<br />

AUREUS TYPE 5 AND TYPE 8 CAPSULAR<br />

POLYSACCHARIDES<br />

CONJUGAISON DE POLYSACCHARIDES<br />

CAPSULAIRES DE STAPHYLOCOCCUS<br />

AUREUS DE TYPE 5 ET DE TYPE 8<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) BERTI, Francesco, I-53100 Siena, IT<br />

COSTANTINO, Paolo, I-53100 Siena, IT<br />

ROMANO, Maria, Rosaria, I-53100 Siena, IT<br />

(74) Marshall, Cameron John, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

A61K 47/48 → (51) A61K 9/16<br />

A61K 47/48 → (51) A61L 2/00<br />

A61K 47/48 → (51) C07K 14/<strong>36</strong><br />

A61K 48/00 → (51) C12N 15/86<br />

(51) A61K 49/04 (11) 2 493 511 A1*<br />

(25) En (26) En<br />

(21) 10771120.2 (22) 28.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) EP 2010/066351 28.10.2010<br />

(87) WO 2011/051387 2011/18 05.05.2011<br />

(30) 29.10.2009 EP 09174413<br />

(54) DIAGNOSTISCHE ZUSAMMENSETZUNG<br />

MIT PLASMAKATIONEN MIT VERBES-<br />

SERTEM SICHERHEITSPROFIL<br />

DIAGNOSTIC COMPOSITION<br />

COMPRISING PLASMA CATIONS HAVING<br />

SUPERIOR SAFETY PROFILE<br />

COMPOSITION DE DIAGNOSTIC<br />

COMPORTANT DES CATIONS PLASMATI-<br />

QUES AYANT UN PROFIL D'INNOCUITÉ<br />

SUPÉRIEUR<br />

(71) GE Healthcare AS, Nycoveien 1-2 P.O. Box<br />

4220 Nydalen, 0401 Oslo, NO<br />

(72) WISTRAND, Lars-Göran, N-0401 Oslo, NO<br />

THANING, Mikkel, N-0401 Oslo, NO<br />

NEWTON, Ben, Amersham Buckinghamshire<br />

HP7 9LL, GB<br />

(74) Wulff, Marianne Weiby, et al, GE Healthcare<br />

AS P.O. Box 4220 Nydalen Nycoveien 1-2,<br />

0401 Oslo, NO<br />

(51) A61K 49/18 (11) 2 493 512 A2*<br />

(25) En (26) En<br />

(21) 10771742.3 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) EP 2010/066429 29.10.2010<br />

(87) WO 2011/051422 2011/18 05.05.2011<br />

(88) 21.07.2011<br />

(30) 30.10.2009 US 609799<br />

(54) BEHANDLUNG WASSERUNLÖSLICHER<br />

NANOPARTIKEL MIT HYDROPHILEN AL-<br />

PHA-HYDROXYPHOSPHONSÄUREKON-<br />

JUGATEN, IN DIESEM VERFAHREN MO-<br />

DIFIZIERTE NANOPARTIKEL UND IHRE<br />

VERWENDUNG ALS KONTRASTMITTEL

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