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European Patent Bulletin 2012/36 - European Patent Office

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(A61K) I.1(1)<br />

A61K 31/517 → (51) C07D 239/94<br />

(51) A61K 31/519 (11) 2 493 473 A1*<br />

A61P 25/18<br />

(25) En (26) En<br />

(21) 10773821.3 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

BA ME<br />

(86) US 2010/054807 29.10.2010<br />

(87) WO 2011/053829 2011/18 05.05.2011<br />

(30) 30.10.2009 US 256696 P<br />

(54) DOSIERPLAN IM ZUSAMMENHANG MIT<br />

LANGWIRKENDEN INJIZIERBAREN PALI-<br />

PERIDONESTERN<br />

DOSING REGIMEN ASSOCIATED WITH<br />

LONG-ACTING INJECTABLE PALI-<br />

PERIDONE ESTERS<br />

POSOLOGIE ASSOCIÉE À DES ESTERS<br />

DE PALIPÉRIDONE INJECTABLES À<br />

ACTION PROLONGÉE<br />

(71) Janssen Pharmaceutica NV, Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) LEWYN-BRISCOE, Peter, H., Newtown PA<br />

18940, US<br />

GASSMANN-MAYER, Cristiana, Pennington<br />

NJ 08534, US<br />

GOPAL, Srihari, Belle Mead NJ 08502, US<br />

HOUGH, David, W., Wallingford PA 19086,<br />

US<br />

REMMERIE, Bart, M. M., B-9000 Gent, BE<br />

SAMTANI, Mahesh, N., Flemington NJ<br />

08822, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

A61K 31/519 → (51) A01N 43/90<br />

A61K 31/519 → (51) A61K 31/52<br />

A61K 31/519 → (51) C07D 239/94<br />

(51) A61K 31/52 (11) 2 493 474 A2*<br />

A61K 31/522 A61K 31/519<br />

A61K 9/06 A61K 9/70<br />

A61P 9/12 A61P 9/00<br />

A61P 25/34<br />

(25) En (26) En<br />

(21) 10827530.6 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/0547<strong>36</strong> 29.10.2010<br />

(87) WO 2011/053792 2011/18 05.05.2011<br />

(88) 22.09.2011<br />

(30) 30.10.2009 US 256614 P<br />

23.12.2009 US 289471 P<br />

(54) VERFAHREN UND ZUSAMMENSETZUN-<br />

GEN FÜR VERZÖGERTE WIRKSTOFFFREI-<br />

SETZUNG<br />

METHODS AND COMPOSITIONS FOR<br />

SUSTAINED DELIVERY OF DRUGS<br />

MÉTHODES ET COMPOSITIONS POUR<br />

UNE LIBÉRATION PROLONGÉE DE MÉDI-<br />

CAMENTS<br />

(71) Intratus, Inc., 9834 Genesee Avenue Suite<br />

406, La Jolla, California 92037, US<br />

(72) NANDURI, Padma, La Jolla California 92037,<br />

US<br />

DYER, T. Aaron, La Jolla California 92037,<br />

US<br />

(74) Müller-Boré & Partner <strong>Patent</strong>anwälte, Grafinger<br />

Straße 2, 81671 München, DE<br />

(51) A61K 31/52 (11) 2 493 475 A2*<br />

A61K 31/522 A61K 31/519<br />

A61P 27/02 A61P 27/00<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(25) En (26) En<br />

(21) 10827537.1 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054752 29.10.2010<br />

(87) WO 2011/053801 2011/18 05.05.2011<br />

(88) 29.09.2011<br />

(30) 30.10.2009 US 256614 P<br />

23.12.2009 US 289471 P<br />

(54) VERFAHREN UND KOSMETIKPRÄPARATE<br />

ZUR VERZÖGERTEN FREISETZUNG THE-<br />

RAPEUTISCHER WIRKSTOFFE IM AUGE<br />

METHODS AND COSMETIC<br />

PREPARATIONS FOR THE SUSTAINED<br />

DELIVERY OF THERAPEUTIC AGENTS TO<br />

THE EYE<br />

MÉTHODES ET PRÉPARATIONS COSMÉ-<br />

TIQUES POUR LA LIBÉRATION<br />

PROLONGÉE D'AGENTS THÉRAPEUTI-<br />

QUES DANS L'OEIL<br />

(71) Intratus, Inc., 9834 Genesee Avenue Suite<br />

406, La Jolla, California 92037, US<br />

(72) NANDURI, Padma, La Jolla CA 92037, US<br />

DYER, T., Aaron, La Jolla CA 92037, US<br />

(74) Müller-Boré & Partner <strong>Patent</strong>anwälte, Grafinger<br />

Straße 2, 81671 München, DE<br />

A61K 31/52 → (51) C07D 519/04<br />

A61K 31/522 → (51) A61K 31/52<br />

A61K 31/522 → (51) C07D 519/04<br />

A61K 31/535 → (51) A61K 31/00<br />

A61K 31/5<strong>36</strong>5 → (51) C07D 471/04<br />

A61K 31/5377 → (51) C07D 231/14<br />

A61K 31/5377 → (51) C07D 311/22<br />

(51) A61K 31/54 (11) 2 493 476 A1*<br />

(25) En (26) En<br />

(21) 10828886.1 (22) 27.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054276 27.10.2010<br />

(87) WO 2011/056647 2011/19 12.05.2011<br />

(30) 28.10.2009 US 255728 P<br />

(54) DEUTERIERTE 5,6-DIHYDRO-1H-PYRI-<br />

DIN-2-ON-VERBINDUNGEN<br />

DEUTERATED 5,6-DIHYDRO-1H-<br />

PYRIDIN-2-ONE COMPOUNDS<br />

COMPOSÉS 5,6-DIHYDRO-1H-PYRIDINE-<br />

2-UN DEUTÉRÉS<br />

(71) Anadys Pharmaceuticals, Inc., 5871 Oberlin<br />

Drive Suite 200, San Diego, California<br />

92121, US<br />

(72) WEBBER, Stephen, E., San Diego CA 92122,<br />

US<br />

(74) Schiweck, Weinzierl & Koch, <strong>European</strong> <strong>Patent</strong><br />

Attorneys Landsberger Straße 98,<br />

80339 München, DE<br />

A61K 31/5415 → (51) A61K 31/135<br />

(51) A61K 31/55 (11) 2 493 477 A2*<br />

A61K 9/16 A61K 9/20<br />

A61K 9/28 A61K 31/404<br />

(25) En (26) En<br />

(21) 10776863.2 (22) 26.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054022 26.10.2010<br />

(87) WO 2011/056532 2011/19 12.05.2011<br />

(88) 15.12.2011<br />

43<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(30) 27.10.2009 US 255216 P<br />

(54) BAZEDOXIFENFORMULIERUNGEN MIT<br />

ANTIOXIDATIONSMITTELN<br />

BAZEDOXIFENE FORMULATIONS WITH<br />

ANTIOXIDANTS<br />

PREPARATIONS DE BAZEDOXIFENE<br />

AVEC ANTIOXYDANTS<br />

(71) Wyeth LLC, <strong>Patent</strong> Law Department Five<br />

Giralda Farms, Madison, NJ 07940, US<br />

(72) AGRAWAL, Anjali, Nyack New York 10960,<br />

US<br />

CHATLAPALLI, Ramarao S., Hopewell<br />

Junction New York 12533, US<br />

NAGI, Arwinder S., Thiells New York 10984,<br />

US<br />

VAN PELT, Lawrence, Garnerville New York<br />

10923, US<br />

CHIRRA, Srinivas, North Brunswick New<br />

Jersey 08902, US<br />

(74) Pfizer, <strong>European</strong> <strong>Patent</strong> Department 23-25<br />

avenue du Docteur Lannelongue, 75668<br />

Paris Cedex 14, FR<br />

A61K 31/55 → (51) A61K 31/00<br />

A61K 31/55 → (51) C07D 471/04<br />

A61K 31/55 → (51) C07D 498/20<br />

A61K 31/551 → (51) C07D 471/04<br />

A61K 31/553 → (51) C07D 471/04<br />

A61K 31/554 → (51) A61K 31/135<br />

A61K 31/558 → (51) C07D 311/22<br />

A61K 31/56 → (51) A61K 31/164<br />

A61K 31/565 → (51) A61K 47/10<br />

A61K 31/568 → (51) A61K 47/10<br />

A61K 31/57 → (51) A61K 47/10<br />

A61K 31/60 → (51) A61K 31/135<br />

A61K 31/66 → (51) C07F 9/6574<br />

A61K 31/675 → (51) A61K 31/70<br />

(51) A61K 31/683 (11) 2 493 478 A1*<br />

A61P 3/00 A61P 9/00<br />

(25) En (26) En<br />

(21) 10825905.2 (22) 29.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) CA 2010/001720 29.10.2010<br />

(87) WO 2011/050474 2011/18 05.05.2011<br />

(30) 29.10.2009 US 256106 P<br />

(54) KONZENTRIERTE THERAPEUTISCHE<br />

PHOSPHOLIPID-ZUSAMMENSETZUNGEN<br />

CONCENTRATED THERAPEUTIC PHOS-<br />

PHOLIPID COMPOSITIONS<br />

COMPOSITIONS DE PHOSPHOLIPIDES<br />

THÉRAPEUTIQUES CONCENTRÉES<br />

(71) Acasti Pharma, Inc., 225 Promenade Du<br />

Centropolis Suite 200, Laval, Quebec H7T<br />

0B3, CA<br />

(72) SAMPALIS, Fotini, Laval Quebec H7W 3J8,<br />

CA<br />

HARLAND, Henri, Rosemere Quebec J7A<br />

4H8, CA<br />

(74) Wills, Andrew Jonathan, et al, Mewburn Ellis<br />

LLP 33 Gutter Lane, London EC2V 8AS, GB<br />

(51) A61K 31/70 (11) 2 493 479 A1*<br />

A61K 31/675<br />

(25) En (26) En

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