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European Patent Bulletin 2012/36 - European Patent Office

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(A61K) I.1(1)<br />

(54) PHARMAZEUTISCHE ZUSAMMENSET-<br />

ZUNG MIT EINER INDOLVERBINDUNG<br />

PHARMACEUTICAL COMPOSITION<br />

COMPRISING INDOLE COMPOUND<br />

COMPOSITION PHARMACEUTIQUE<br />

CONTENANT UN COMPOSÉ INDOLE<br />

(71) LG Life Sciences Ltd, LG Gwanghwamun<br />

Bldg. 92 Sinmunno 2-ga, Jongno-gu, Seoul<br />

110-062, KR<br />

(72) KIM, Soon Ha, Daejeon 305-380, KR<br />

KIM, Hyoung Jin, Daejeon 305-380, KR<br />

PARK, Heui Sul, Daejeon 305-380, KR<br />

GU, Seon Yeong, Daejeon 305-380, KR<br />

KWAK, Hyo Shin, Daejeon 305-380, KR<br />

PARK, Du Hee, Daejeon 305-380, KR<br />

KIM, Hyo Soo, Daejeon 305-380, KR<br />

CHO, Hyun Jai, Daejeon 305-380, KR<br />

KIM, Ji Hyun, Daejeon 305-380, KR<br />

KIM, Ju Young, Daejeon 305-380, KR<br />

PARK, Kwang Min, Daejeon 305-380, KR<br />

(74) Nicolle, Frederick Joseph, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

GB-London EC1N 2HA, GB<br />

A61K 31/404 → (51) A61K 31/55<br />

A61K 31/415 → (51) A01N 43/50<br />

A61K 31/415 → (51) C07D 231/38<br />

A61K 31/416 → (51) C07D 231/14<br />

A61K 31/416 → (51) C07D 401/04<br />

A61K 31/4164 → (51) C07D 233/64<br />

A61K 31/4178 → (51) C07D 233/64<br />

A61K 31/42 → (51) C07D 231/14<br />

A61K 31/42 → (51) C07D 261/20<br />

A61K 31/421 → (51) C07D 263/20<br />

A61K 31/4245 → (51) C07D 205/04<br />

A61K 31/425 → (51) A01N 43/78<br />

A61K 31/425 → (51) A61K 31/135<br />

A61K 31/435 → (51) A61K 31/135<br />

A61K 31/437 → (51) A61K 9/20<br />

A61K 31/437 → (51) A61K 31/10<br />

A61K 31/437 → (51) C07D 471/04<br />

A61K 31/4375 → (51) C07D 219/10<br />

A61K 31/4375 → (51) C07D 471/04<br />

A61K 31/438 → (51) C07D 231/14<br />

A61K 31/439 → (51) C07D 498/20<br />

A61K 31/44 → (51) A01N 43/42<br />

A61K 31/44 → (51) C07D 213/74<br />

A61K 31/44 → (51) C07D 231/14<br />

A61K 31/4402 → (51) A61K 31/135<br />

A61K 31/4427 → (51) C07D 213/74<br />

A61K 31/4439 → (51) C07D 403/12<br />

A61K 31/444 → (51) A61K 31/135<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

A61K 31/444 → (51) C07D 205/04<br />

A61K 31/445 → (51) C07D 211/28<br />

A61K 31/45 → (51) C07D 211/28<br />

A61K 31/4523 → (51) C07D 211/28<br />

A61K 31/4523 → (51) C07D 231/14<br />

A61K 31/46 → (51) C07D 401/12<br />

A61K 31/4706 → (51) A61P 33/06<br />

(51) A61K 31/4709 (11) 2 493 470 A1*<br />

A61K 31/7056 A61K 38/21<br />

A61P 31/14<br />

(25) En (26) En<br />

(21) 10773799.1 (22) 27.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/054194 27.10.2010<br />

(87) WO 2011/05<strong>36</strong>17 2011/18 05.05.2011<br />

(30) 30.10.2009 US 256516 P<br />

(54) DOSIERPLÄNE FÜR EINE HCV-KOMBINA-<br />

TIONSTHERAPIE AUS BI201335, INTER-<br />

FERON ALPHA UND RIBAVIRIN<br />

DOSAGE REGIMENS FOR HCV COMBI-<br />

NATION THERAPY COMPRISING<br />

BI201335, INTERFERON ALPHA AND<br />

RIBAVIRIN<br />

RÉGIMES POSOLOGIQUES POUR UNE<br />

THÉRAPIE EN COMBINAISON CONTRE LE<br />

VHC COMPRENANT BI201335, L'INTER-<br />

FÉRON ALPHA ET LA RIBAVIRINE<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim, DE<br />

(72) HAEFNER, Carla, 55216 Ingelheim am Rhein,<br />

DE<br />

STEINMANN, Gerhard, 55216 Ingelheim am<br />

Rhein, DE<br />

STERN, Jerry O., Ridgefield, Connecticut<br />

06877-0<strong>36</strong>8, US<br />

YONG, Chan-Loi, Ridgefield, Connecticut<br />

06877-0<strong>36</strong>8, US<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

Pharma GmbH & Co. KG Binger<br />

Strasse 173, 55216 Ingelheim am Rhein, DE<br />

A61K 31/473 → (51) C07D 311/68<br />

(51) A61K 31/485 (11) 2 493 471 A1*<br />

A61K 31/70<strong>36</strong> A61P 1/12<br />

A61K 31/165 A61K 31/7048<br />

A61P 25/16 A61K 31/166<br />

A61P 1/08 A61P 25/28<br />

A61K 31/496 A61P 1/10<br />

(25) En (26) En<br />

(21) 10825843.5 (22) 22.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) AU 2010/001410 22.10.2010<br />

(87) WO 2011/050397 2011/18 05.05.2011<br />

(30) 26.10.2009 AU 2009905229<br />

(54) NEUE ENTERALE KOMBINATIONSTHERA-<br />

PIE<br />

NOVEL ENTERIC COMBINATION<br />

THERAPY<br />

NOUVELLE POLYTHÉRAPIE GASTRO-<br />

RÉSISTANTE<br />

(71) Borody, Thomas Julius, Level 1, 229 Great<br />

North Road, Five Dock NSW 2046, AU<br />

(72) Borody, Thomas Julius, Five Dock NSW<br />

2046, AU<br />

(74) Zwicker, Jörk, et al, Dr. Volker Vossius <strong>Patent</strong>-<br />

und Rechtsanwaltskanzlei Geibelstrasse<br />

6, 81679 München, DE<br />

42<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

A61K 31/495 → (51) A61K 31/135<br />

A61K 31/496 → (51) A61K 31/485<br />

A61K 31/496 → (51) C07D 401/06<br />

(51) A61K 31/497 (11) 2 493 472 A1*<br />

(25) En (26) En<br />

(21) 10827343.4 (22) 22.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) US 2010/05<strong>36</strong>78 22.10.2010<br />

(87) WO 2011/053518 2011/18 05.05.2011<br />

(30) 27.04.2010 US 328480 P<br />

26.10.2009 US 254917 P<br />

(54) VERFAHREN ZUR SYNTHESE UND REI-<br />

NIGUNG VON HETEROARYLVERBINDUN-<br />

GEN<br />

METHODS OF SYNTHESIS AND PURIFI-<br />

CATION OF HETEROARYL COMPOUNDS<br />

PROCÉDÉS DE SYNTHÈSE ET DE PURIFI-<br />

CATION DE COMPOSÉS HÉTÉROARYLES<br />

(71) Signal Pharmaceuticals, LLC, 4550 Towne<br />

Centre Court, San Diego, CA 92121, US<br />

(72) HARRIS, Roy, L., San Diego, CA 92109, US<br />

SAPIENZA, John, Chula Vista, CA 91913, US<br />

SHEVLIN, Graziella, San Diego, CA 92129,<br />

US<br />

PAPA, Patrick, Carlsbad, CA 92008, US<br />

LEE, Branden, Gingsee, San Diego, CA<br />

92130, US<br />

PACKARD, Garrick, San Diego, CA 92121,<br />

US<br />

ZHAO, Jingjing, San Diego, CA 92129, US<br />

JOKIEL, Patrick, Anthony, Princeton, NJ<br />

08540, US<br />

MORTENSEN, Deborah, San Diego, CA<br />

92117, US<br />

RIGGS, Jennifer, Cardiff, CA 92007, US<br />

GAMBOA, Juan, Antonio, New York, NY<br />

10009, US<br />

BEAUCHAMPS, Marie, Georges, Flanders, NJ<br />

078<strong>36</strong>, US<br />

KREILEIN, Matthew, Michael, Watchung, NJ<br />

07069, US<br />

KOTHARE, Mohit, Atul, Bridgewater, NJ<br />

08807, US<br />

PERRIN-NINKOVIC, Sophie, La Jolla, CA<br />

92037, US<br />

PYE, Philip, Scotch Plains, NJ 07076, US<br />

LEONG, William, Wei-Hwa, Westfield, NJ<br />

07090, US<br />

ELSNER, Jan, San Diego, CA 92122, US<br />

CHOUDHURY, Anusuya, Churchville, PA<br />

18966, US<br />

(74) Jones Day, Rechtsanwälte, Attorneys-at-Law<br />

<strong>Patent</strong>anwälte Intellectual Property Prinzregentenstraße<br />

11, 80538 München, DE<br />

A61K 31/497 → (51) C07D 231/14<br />

A61K 31/497 → (51) C07D 401/14<br />

A61K 31/4985 → (51) C07D 471/04<br />

A61K 31/5025 → (51) C07D 487/04<br />

A61K 31/505 → (51) C07D 213/74<br />

A61K 31/506 → (51) C07D 213/74<br />

A61K 31/506 → (51) C07D 219/10<br />

A61K 31/506 → (51) C07D 239/28<br />

A61K 31/506 → (51) C07D 239/48<br />

A61K 31/506 → (51) C07D 401/14

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