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European Patent Bulletin 2012/36 - European Patent Office

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(C07D) II.1(1)<br />

TOBE, Takahiko, Tokyo 103-8411, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München,<br />

DE<br />

C07D 211/34 → (51) C07D 213/56<br />

(51) C07D 211/46 (11) 2 286 811 B1<br />

C07D 491/04 A61K 31/4353<br />

(25) En (26) En<br />

(21) 10012138.3 (22) 13.11.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

AL LT LV MK RO SI<br />

(43) 23.02.2011<br />

(30) 21.11.2001 US 989086<br />

(54) Chemokine Rezeptor Antagonisten und<br />

Methoden zu deren Anwendung<br />

Chemokine receptor antagonists and<br />

methods of use thereof<br />

Antagonistes de récepteur de chemokine<br />

et leurs procédés d'utilisation<br />

(73) Millennium Pharmaceuticals, Inc., 40 Landsdowne<br />

Street, Cambridge, MA 02139, US<br />

Kyowa Hakko Kirin Co., Ltd., 1-6-1,<br />

Ohtemachi, Chiyoda-ku, Tokyo 100-8185, JP<br />

(72) Luly, Jay, R., Wellesley, MA 02481, US<br />

Nakasato, Yoshisuke, Susono-shi Shizuoka,<br />

JP<br />

Oshima, Etsuo, Nagareyama-shi Chiba, JP<br />

Harriman, Geraldine, C.B., Charlestown, RI<br />

02813, US<br />

Carson, Kenneth, G., Princenton New Jersey<br />

02445, US<br />

Ghosh, Shomir, Brookline, MA 02446, US<br />

Elder, Amy, M., Arlington, MA 02474, US<br />

Mattia, Karen, M., Marlborough MA 01752,<br />

US<br />

(74) Raynor, Stuart Andrew, J A Kemp 14 South<br />

Square Gray's Inn, London WC1R 5JJ, GB<br />

(62) 06004401.3 / 1 688 418<br />

02789725.5 / 1 448 566<br />

C07D 213/<strong>36</strong> → (51) C07C 311/18<br />

(51) C07D 213/40 (11) 1 951 673 B1<br />

C07D 213/61 C07D 277/28<br />

C07D 401/04 C07D 401/06<br />

C07D 401/12 C07D 405/06<br />

C07D 405/12 C07D 417/06<br />

C07D 417/12 A61K 31/345<br />

A61P 3/00 A61P 9/00<br />

(25) En (26) En<br />

(21) 06839919.5 (22) 16.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

HR MK RS<br />

(43) 06.08.2008<br />

(86) US 2006/060978 16.11.2006<br />

(87) WO 2007/062314 2007/22 31.05.2007<br />

(30) 23.11.2005 US 739322 P<br />

15.11.2006 US 559930<br />

(54) HETEROCYCLISCHE CETP-HEMMER<br />

HETEROCYCLIC CETP INHIBITORS<br />

INHIBITEURS DE CETP HETEROCYCLI-<br />

QUES<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton, NJ<br />

08543-4000, US<br />

(72) SALVATI, Mark E., Pennington, New Jersey<br />

08534, US<br />

FINLAY, Heather, Pennington, NJ 08534, US<br />

HARIKRISHNAN, Lalgudi S., Princeton, New<br />

Jersey 08543, US<br />

JIANG, Ji, Pennington, NJ 08543, US<br />

JOHNSON, James A., Pennington, NJ 08543,<br />

US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

KAMAU, Muthoni G., Princeton, NJ 08543,<br />

US<br />

LAWRENCE, R. Michael, Pennington, NJ<br />

08534, US<br />

MILLER, Michael M., Pennington, NJ 08534,<br />

US<br />

QIAO, Jennifer X., Pennington, NJ 08534,<br />

US<br />

WANG, Tammy C., Pennington, NJ 08534,<br />

US<br />

WANG, Yufeng, Pennington, NJ 08534, US<br />

YANG, Wu, Pennington, NJ 08534, US<br />

(74) Reitstötter - Kinzebach, <strong>Patent</strong>anwälte Sternwartstrasse<br />

4, 81679 München, DE<br />

C07D 213/55 → (51) C07C 311/18<br />

(51) C07D 213/56 (11) 1 495 002 B1<br />

C07D 215/12 C07D 237/08<br />

C07D 307/54 C07D 277/30<br />

C07D 239/26 C07D 239/42<br />

C07D 495/04 A61K 31/435<br />

A61K 31/495 A61P 35/00<br />

C07D 277/24 C07D 409/04<br />

C07D 213/74 C07D 487/04<br />

C07D 241/20 C07D 251/18<br />

C07D 211/34 C07D 401/04<br />

C07D 403/12<br />

(25) En (26) En<br />

(21) 03712442.7 (22) 02.04.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV<br />

(43) 12.01.2005<br />

(86) GB 2003/001442 02.04.2003<br />

(87) WO 2003/087057 2003/43 23.10.2003<br />

(30) 05.04.2002 GB 0207863<br />

21.12.2002 GB 0229930<br />

(54) BENZAMID-DERIVATE VERWENDBAR<br />

ALS HISTON-DEACETYLASE-INHIBITO-<br />

REN<br />

BENZAMIDE DERIVATIVES USEFUL AS<br />

HISTONE DEACETYLASE INHIBITORS<br />

DÉRIVÉS DE BENZAMIDE UTILES EN<br />

TANT QU'INHIBITEURS D'HISTONE<br />

DEACETYLASE<br />

(73) AstraZeneca AB, 151 85 Södertälje, SE<br />

(72) STOKES, Elaine S.E., AstraZeneca R & D<br />

Alderley, Macclesfield, Cheshire SK10 4TG,<br />

GB<br />

ROBERTS, C.A., AstraZeneca R & D Alderley,<br />

Macclesfield, Cheshire SK10 4TG, GB<br />

WARING, Michael J., AstraZeneca R & D<br />

Alderley, Macclesfield, Cheshire SK10 4TG,<br />

GB<br />

C07D 213/61 → (51) C07D 213/40<br />

(51) C07D 213/64 (11) 2 350 008 B1<br />

C07D 213/65 C07D 213/68<br />

A61K 31/44<br />

(25) En (26) En<br />

(21) 09778756.8 (22) 29.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(43) 03.08.2011<br />

(86) EP 2009/006986 29.09.2009<br />

(87) WO 2010/040461 2010/15 15.04.2010<br />

(30) 09.10.2008 EP 08166247<br />

(54) VERFAHREN ZUR HERSTELLUNG FUNK-<br />

TIONALISIERTER TRIHALOGENMETHOX-<br />

YSUBSTITUIERTER PYRIDINE<br />

METHOD FOR THE PREPARATION OF<br />

FUNCTIONALIZED TRIHALOMETHOXY<br />

SUBSTITUTED PYRIDINES<br />

PROCÉDÉ DE PRÉPARATION DE PYRI-<br />

DINES SUBSTITUÉES PAR UN RÉSIDU<br />

631<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

TRIHALOGÉNOMÉTHOXY FONCTIONNA-<br />

LISÉES<br />

(73) Bayer CropScience AG, Alfred-Nobel-Straße<br />

50, 40789 Monheim, DE<br />

Centre National de la Recherche Scientifique,<br />

3 Rue Michel Ange, 75795 Paris, FR<br />

Université de Strasbourg, 4, rue Blaise<br />

Pascal, 67000 Strasbourg, FR<br />

(72) PAZENOK, Sergii, 42699 Solingen, DE<br />

VORS, Jean-Pierre, 69110 Sainte Foy Les<br />

Lyon, FR<br />

LEROUX, Fréderic, R., 67850 Herrlisheim,<br />

FR<br />

MANTEAU, Baptiste, 17420 Saint Palais-sur-<br />

Mer, FR<br />

(74) Hildebrand, Steven, Bayer CropScience AG<br />

BPA-LP-<strong>Patent</strong>s & Licensing Alfred-Nobel-<br />

Straße 50 Building 6100, DE-40789 Monheim,<br />

DE<br />

C07D 213/65 → (51) C07D 213/64<br />

C07D 213/68 → (51) C07D 213/64<br />

C07D 213/74 → (51) C07D 213/56<br />

C07D 213/83 → (51) C07C 311/18<br />

C07D 215/12 → (51) C07D 213/56<br />

(51) C07D 215/14 (11) 2 085 388 B1<br />

A61K 31/47 A61K 31/4709<br />

A61P 1/04 A61P 3/04<br />

A61P 3/06 A61P 3/10<br />

A61P 3/14 A61P 5/00<br />

A61P 9/00 A61P 9/12<br />

A61P 11/00 A61P 11/02<br />

A61P 11/06 A61P 17/00<br />

A61P 25/00 A61P 25/18<br />

A61P 25/28 A61P 27/06<br />

A61P 37/00 C07D 215/20<br />

C07D 405/12 C07D 409/12<br />

(25) Ja (26) En<br />

(21) 07831812.8 (22) 14.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

(43) 05.08.2009<br />

(86) JP 2007/072082 14.11.2007<br />

(87) WO 2008/059866 2008/21 22.05.2008<br />

(30) 14.11.2006 JP 2006307651<br />

(54) NEUES 1,2-DIHYDROCHINOLINDERIVAT<br />

MIT SUBSTITUIERTER PHENYLAMINO-<br />

NIEDERALKYLGRUPPE UND ÜBER EINEN<br />

ESTER EINGEFÜHRTER PHENYLGRUPPE<br />

ALS SUBSTITUENTEN<br />

NOVEL 1,2-DIHYDROQUINOLINE DERI-<br />

VATIVE HAVING SUBSTITUTED PHENY-<br />

LAMINO LOWER ALKYL GROUP AND<br />

ESTER-INTRODUCED PHENYL GROUP AS<br />

SUBSTITUENTS<br />

NOUVEAU DÉRIVÉ 1,2-DIHYDROQUINO-<br />

LINE COMPRENANT UN GROUPE ALKYLE<br />

INFÉRIEUR À SUBSTITUTION PHÉNYLA-<br />

MINO ET UN GROUPE PHÉNYLE DANS<br />

LEQUEL EST INTRODUIT UN ESTER EN<br />

TANT QUE SUBSTITUANTS<br />

(73) Santen Pharmaceutical Co., Ltd, 9-19,<br />

Shimoshinjo 3-chome Higashiyodogawa-ku,<br />

Osaka-shi Osaka 533-8651, JP<br />

(72) MATSUDA, Mamoru, Ikoma-shi Nara 630-<br />

0101, JP<br />

NAGATSUKA, Masato, Ikoma-shi Nara 630-<br />

0101, JP<br />

MORI, Toshiyuki, Ikoma-shi Nara 630-0101,<br />

JP<br />

KOBAYASHI, Sachiko, Ikoma-shi Nara 630-<br />

0101, JP<br />

KATO, Masatomo, Ikoma-shi Nara 630-0101,<br />

JP

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