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European Patent Bulletin 2012/36 - European Patent Office

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(C07C) II.1(1)<br />

(72) Buyuktimkin, Servet, Lawrence, KS 66049,<br />

US<br />

Buyuktimkin, Nadir, Lawrence, KS 66049,<br />

US<br />

(74) Schnappauf, Georg, et al, Dr. Volker Vossius<br />

<strong>Patent</strong>- und Rechtsanwaltskanzlei Geibelstrasse<br />

6, 81679 München, DE<br />

(62) 00932524.2 / 1 097 126<br />

(51) C07C 227/32 (11) 2 213 653 B1<br />

C07C 229/<strong>36</strong> C07B 53/00<br />

C07C 67/31 C07C 69/732<br />

C07C 247/12 C07C 271/34<br />

C07D 203/06 C07K 1/04<br />

C07D 203/02<br />

(25) Es (26) En<br />

(21) 08852208.1 (22) 19.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 04.08.2010<br />

(86) ES 2008/000724 19.11.2008<br />

(87) WO 2009/065987 2009/22 28.05.2009<br />

(30) 19.11.2007 ES 200703112<br />

(54) VERFAHREN ZUR STEREOSELEKTIVEN<br />

HERSTELLUNG VON AMINOSÄUREDERI-<br />

VATEN<br />

METHOD FOR THE STEREOSELECTIVE<br />

PREPARATION OF AMINO ACID DERI-<br />

VATIVES<br />

PROCEDE DE PREPARATION STEREOSE-<br />

LECTIVE DE DERIVES D'ACIDES AMINES<br />

(73) BCN Peptides, S.A., Polígono Industrial Els<br />

Vinyets Els Fogars 2, Carretera Comarcal C-<br />

244 Km 22, 08777 Sant Quinti de Mediona-<br />

Barcelona, ES<br />

(72) RAFECAS JANE, Llorenç, Tarragona, ES<br />

RIERA ESCALE, Antoni, 08005 Barcelona,<br />

ES<br />

RAMON ALBALATE, Rosario, Barcelona, ES<br />

ALONSO XALMA, Monica, 08024 Barcelona,<br />

ES<br />

(74) Carvajal y Urquijo, Isabel, et al, Clarke,<br />

Modet & Co. c/ Goya, 11, 28001 Madrid, ES<br />

(51) C07C 227/42 (11) 1 300 392 B1<br />

C07C 229/<strong>36</strong> C07C 229/08<br />

C07C 231/24 C07C 237/06<br />

C07C 237/20 C12P 41/00<br />

C12P 13/04<br />

(25) Ja (26) En<br />

(21) 01930218.1 (22) 18.05.2001<br />

(84) CH DE FR GB LI<br />

(43) 09.04.2003<br />

(86) JP 2001/004191 18.05.2001<br />

(87) WO 2001/087819 2001/47 22.11.2001<br />

(30) 18.05.2000 JP 2000146663<br />

22.05.2000 JP 2000150285<br />

(54) VERFAHREN ZUR PRODUKTION EINER<br />

OPTISCH AKTIVEN ALPHA-AMINOSÄURE<br />

UND EINES OPTISCH AKTIVEN ALPHA-<br />

AMINOSÄUREAMIDS<br />

PROCESS FOR PRODUCING OPTICALLY<br />

ACTIVE ALPHA-AMINO ACID AND<br />

OPTICALLY ACTIVE ALPHA-AMINO ACID<br />

AMIDE<br />

PROCEDE DE PRODUCTION D'UN<br />

ALPHA-AMINO ACIDE OPTIQUEMENT<br />

ACTIF ET D'UN AMIDE D'ALPHA-AMINO<br />

ACIDE OPTIQUEMENT ACTIF<br />

(73) MITSUBISHI RAYON CO., LTD., 6-41, Konan<br />

1-chome, Minato-ku, Tokyo 108-8506, JP<br />

(72) KATOH, Osamu, Yokohama-shi, Kanagawa<br />

230-0053, JP<br />

URAGAKI, Toshitaka, Yokohama-shi,<br />

Kanagawa 230-0053, JP<br />

NAKAMURA, Tetsuji, Yokohama-shi,<br />

Kanagawa 230, JP<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München,<br />

DE<br />

C07C 227/42 → (51) C07C 227/18<br />

(51) C07C 229/00 (11) 1 546 085 B1<br />

C07C 249/00 C07C 381/00<br />

C07C 205/00 C07C 291/00<br />

C07C 233/00 C07C 211/00<br />

C07C 335/00 A61K 31/225<br />

A61P 35/00 A61P 35/04<br />

(25) En (26) En<br />

(21) 03710190.4 (22) 16.03.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 29.06.2005<br />

(86) IL 2003/000225 16.03.2003<br />

(87) WO 2004/028443 2004/15 08.04.2004<br />

(30) 25.09.2002 IL 15192102<br />

(54) LIPOPHILE DIESTER EINES CHELAT-<br />

BILDNERS ZUR HEMMUNG VON ENZYM-<br />

AKTIVITÄT<br />

LIPOPHILIC DIESTERS OF CHELATING<br />

AGENT FOR INHIBITION OF ENZYME<br />

ACTIVITY<br />

DIESTERS LIPOPHILES D'UN AGENT<br />

CHÉLATEUR POUR L`INHIBITION DE<br />

L'ACTIVITÉ ENZYMATIQUE<br />

(73) D-Pharm Ltd., Kiryat Weizmann Science<br />

Park, 76326 Rehovot, IL<br />

(72) STRIEM, Sarina, Rehovot 76469, IL<br />

FRIEDMAN, Jonathan, Eduard, Rehovot<br />

76529, IL<br />

REZNITSKY-COHEN, Dalia, Nes-Ziona<br />

74042, IL<br />

KOZAK, Alexander, Rehovot 76555, IL<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

C07C 229/08 → (51) C07C 227/42<br />

C07C 229/08 → (51) C07D 413/12<br />

C07C 229/<strong>36</strong> → (51) C07C 227/32<br />

C07C 229/<strong>36</strong> → (51) C07C 227/42<br />

(51) C07C 231/12 (11) 2 044 003 B1<br />

C07C 233/47<br />

(25) En (26) En<br />

(21) 07730270.1 (22) 20.06.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

(43) 08.04.2009<br />

(86) EP 2007/056140 20.06.2007<br />

(87) WO 2008/000671 2008/01 03.01.2008<br />

(30) 27.06.2006 US 475824<br />

(54) VERFAHREN ZUR UMWANDLUNG PRI-<br />

MÄRER AMIDOALKOHOLE IN AMIDO-<br />

CARBONSÄUREN IN HOHER AUSBEUTE<br />

UNTER VERWENDUNG VON WASSER<br />

ALS LÖSUNGSMITTEL<br />

PROCESS FOR CONVERTING PRIMARY<br />

AMIDOALCOHOLS TO AMIDOCAR-<br />

BOXYLIC ACIDS IN HIGH YIELD USING<br />

WATER AS SOLVENT<br />

PROCÉDÉ DE CONVERSION À RENDE-<br />

MENT ÉLEVÉ D'AMIDOALCOOLS<br />

PRIMAIRES EN ACIDES AMIDOCARBO-<br />

XYLIQUES EN EMPLOYANT L'EAU<br />

COMME SOLVANT<br />

(73) Unilever PLC, Unilever House 100 Victoria<br />

Embankment, London EC4Y 0DY, GB<br />

(84) CY GB IE MT<br />

(73) Unilever N.V., Weena 455, 3013 AL Rotterdam,<br />

NL<br />

629<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(84) AT BE BG CH CZ DE DK EE ES FI FR GR HU<br />

IS IT LI LT LU LV MC NL PL PT RO SE SI SK<br />

TR<br />

(72) HARICHIAN, Bijan, Trumbull, Connecticut<br />

06611, US<br />

CHEN, Hang, Trumbull, Connecticut 06611,<br />

US<br />

ROSA, Jose, Guillemo, Trumbull,<br />

Connecticut 06611, US<br />

(74) Baker, Colin John, et al, Potter Clarkson LLP<br />

Park View House 58 The Ropewalk,<br />

Nottingham NG1 5DD, GB<br />

C07C 231/24 → (51) C07C 227/42<br />

C07C 233/00 → (51) C07C 229/00<br />

C07C 233/47 → (51) C07C 231/12<br />

C07C 237/06 → (51) C07C 227/42<br />

C07C 237/20 → (51) C07C 227/42<br />

(51) C07C 237/<strong>36</strong> (11) 1 539 678 B1<br />

C07C 237/44 C07C 311/39<br />

C07D 207/323 C07D 217/24<br />

C07D 307/52 C07D 307/68<br />

C07D 307/81 C07D 307/82<br />

C07D 307/83 C07D 317/46<br />

C07D 319/18 C07D 333/20<br />

C07D 405/12 C07D 409/12<br />

C07D 409/14 C07D 413/12<br />

C07D 413/14 A61K 31/341<br />

A61K 31/<strong>36</strong> A61K 31/381<br />

(25) En (26) En<br />

(21) 03772075.2 (22) 30.07.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV MK<br />

(43) 15.06.2005<br />

(86) US 2003/023785 30.07.2003<br />

(87) WO 2004/011418 2004/06 05.02.2004<br />

(30) 30.07.2002 US 208412<br />

11.09.2002 US 241326<br />

(54) 3,4-DISUBSTITUIERTE CYCLOBUTEN-<br />

1,2-DIONE ALS LIGANDEN F R DEN CXC-<br />

CHEMOKINREZEPTOR<br />

3,4-DI-SUBSTITUTED CYCLOBUTENE-1,<br />

2-DIONES AS CXC-CHEMOKINE<br />

RECEPTOR LIGANDS<br />

CYCLOBUTENE-1, 2-DIONES 3,4-DI-<br />

SUBSTITUES UTILISES COMME LIGANDS<br />

DU RECEPTEUR DE CHIMIOKINE CXC<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

Pharmacopeia, LLC, 10275 Science Center<br />

Drive, San Diego, CA 92121, US<br />

(72) TAVERAS, Arthur, G., Southborough, MA<br />

01772, US<br />

AKI, Cynthia, J., Livingston, NJ 07039, US<br />

CHAO, Jianping, Summit, NJ 07901, US<br />

DWYER, Michael, Scotch Plains, NJ 07076,<br />

US<br />

CHAO, Jianhua, Pompton Lakes, NJ 07442,<br />

US<br />

YU, Younong, East Brunswick, NJ 08816,<br />

US<br />

MERRITT, J., Robert, Ewing, NJ 08618, US<br />

BIJU, Purakkattle, Scotch Plains, NJ 07076,<br />

US<br />

JAKWAY, James, Bridgewater, NJ 08807, US<br />

LAI, Gaifa, Edison, NJ 08837, US<br />

WU, Minglang, Monmouth Junction, NJ<br />

08852, US<br />

HECKER, Evan, A., East Windsor, NJ 08520,<br />

US<br />

LUNDELL, Daniel, Flemington, NJ 08822, US

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