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European Patent Bulletin 2012/36 - European Patent Office

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(C07D) I.1(2)<br />

C07D 487/22 → (51) A61K 31/439<br />

C07D 493/08 → (51) A61K 31/352<br />

C07D 495/04 → (51) C08G 61/12<br />

C07D 519/00 → (51) C08G 61/12<br />

(51) C07F 9/6574 (11) 2 495 247 A1<br />

(25) Ja (26) En<br />

(21) 10820406.6 (22) 21.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/066322 21.09.2010<br />

(87) WO 2011/040287 2011/14 07.04.2011<br />

(30) 01.10.2009 JP 2009229622<br />

(54) VERFAHREN ZUR HERSTELLUNG VON<br />

ZYKLISCHEM ALKYLENPHOSPHOHALI-<br />

DAT UND EINES ZYKLISCHEN PHOS-<br />

PHORSÄUREESTERS<br />

PROCESSES FOR PRODUCTION OF<br />

CYCLIC ALKYLENE PHOSPHOHALIDATE<br />

AND CYCLIC PHOSPHORIC ACID ESTER<br />

PROCÉDÉS DE PRODUCTION DE PHOS-<br />

PHOHALIDATE D'ALKYLÈNE CYCLIQUE<br />

ET D'ESTER D'ACIDE PHOSPHORIQUE<br />

CYCLIQUE<br />

(71) Daihachi Chemical Industry Co., Ltd., 8-13,<br />

Hiranomachi 1-chome Chuo-ku Osaka-shi,<br />

Osaka 541-0046, JP<br />

(72) HAMADA, Toshiya, Osaka 577-0056, JP<br />

HAMADA, Sakiko, Osaka 577-0056, JP<br />

(74) Zanoli, Enrico, et al, Zanoli & Giavarini S.r.l.<br />

Via Melchiorre Gioia, 64, <strong>2012</strong>5 Milano, IT<br />

(51) C07H 19/06 (11) 2 495 248 A1<br />

A61K 31/712 C07H 19/16<br />

C07H 21/00<br />

(25) Ja (26) En<br />

(21) 10826568.7 (22) 19.10.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

(86) JP 2010/068409 19.10.2010<br />

(87) WO 2011/0524<strong>36</strong> 2011/18 05.05.2011<br />

(30) 29.10.2009 JP 2009248979<br />

04.02.2010 JP 2010023209<br />

(54) GEBRÜCKTES KÜNSTLICHES NUKLEOSID<br />

UND NUKLEOTID<br />

BRIDGED ARTIFICIAL NUCLEOSIDE AND<br />

NUCLEOTIDE<br />

NUCLÉOSIDE ET NUCLÉOTIDE ARTIFI-<br />

CIELS PONTÉS<br />

(71) Osaka University, 1-1, Yamadaoka, Suita-shi<br />

Osaka 565-0871, JP<br />

(72) OBIKA, Satoshi, Suita-shi Osaka 565-0871,<br />

JP<br />

HARI, Yoshiyuki, Suita-shi Osaka 565-0871,<br />

JP<br />

KODAMA, Tetsuya, Suita-shi Osaka 565-<br />

0871, JP<br />

YAHARA, Aiko, Suita-shi Osaka 565-0871,<br />

JP<br />

NISHIDA, Masaru, Suita-shi Osaka 565-<br />

0871, JP<br />

(74) Clements, Andrew Russell Niel, et al, Schlich<br />

LLP 34 New Road, Littlehampton, West<br />

Sussex BN17 5AT, GB<br />

C07H 19/16 → (51) C07H 19/06<br />

C07H 21/00 → (51) C07H 19/06<br />

C07H 21/02 → (51) C12N 15/113<br />

C07H 21/04 → (51) C12N 15/113<br />

C07H 21/04 → (51) C12Q 1/68<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

C07K 1/14 → (51) C07K 19/00<br />

C07K 1/22 → (51) C07K 14/31<br />

(51) C07K 5/06 (11) 2 495 249 A1<br />

C07K 5/08 A61K 38/06<br />

(25) En (26) En<br />

(21) 12164823.2 (22) 26.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(30) 26.02.2007 US 891634 P<br />

(54) Tertiäraminsubstituierte Peptide als HCV-<br />

Replikationshemmer<br />

Tertiary amine substituted peptides useful<br />

as inhibitors of HCV replication<br />

Peptides à amine tertiaire substituée utiles<br />

en tant qu'inhibiteurs de la réplication du<br />

VHC<br />

(71) Achillion Pharmaceuticals, Inc., 300 George<br />

Street, New Haven, CT 06511, US<br />

(72) Agarwal, Atul, Hamden, CT 06518, US<br />

Wang, Xiangzhu, Branford, CT 06405, US<br />

Chen, Dawei, Middletown, CT 06457, US<br />

Zhang, Suoming, Madison, CT 06443, US<br />

Phadke, Avinash, Branford, CT 06405, US<br />

(74) Smaggasgale, Gillian Helen, WP Thompson<br />

55 Drury Lane, London WC2B 5SQ, GB<br />

(62) 08726107.9 / 2 125 113<br />

C07K 5/08 → (51) C07K 5/06<br />

C07K 5/08 → (51) C07K 5/097<br />

(51) C07K 5/097 (11) 2 495 250 A2<br />

C07K 14/47 C12P 21/06<br />

A23J 3/10 A61K 38/06<br />

A61K 38/17 A61K 38/57<br />

A61P 9/12 A61P 17/18<br />

A61P 31/04 C07K 5/08<br />

(25) Es (26) En<br />

(21) 12158198.7 (22) 08.06.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

(30) 08.06.2005 ES 200501373<br />

(54) Biologisch aktive Peptide, die in enzymatischen<br />

Hydrolyzaten aus Milchcaseinen<br />

identifiziert wurden und Verfahren zu deren<br />

Erhalt<br />

Bioactive peptides identified in enzymatic<br />

hydrolyzates of milk caseins and method<br />

of obtaining same<br />

Peptides bioactifs identifiés dans des<br />

hydrolysats enzymatiques de caséine du<br />

lait et procédé d'obtention<br />

(71) Consejo Superior de Investigaciones Cientificas,<br />

Serrano, 117, 28006 Madrid, ES<br />

(72) Recio Sanchez, Isidra, 28006 Madrid, ES<br />

Contreras Gómez, Mar, 28006 Madrid, ES<br />

Quiros del Bosque, Ana, 28006 Madrid, ES<br />

Hernandez Ledesma, Blanca, 28006 Madrid,<br />

ES<br />

Gomez Ruiz, José Angel, 28006 Madrid, ES<br />

Miguel Castro, Marta, 28006 Madrid, ES<br />

Amigo Garrido, Maria Lourdes, 28006<br />

Madrid, ES<br />

Lopez Exposito, Ivan, 28006 Madrid, ES<br />

Ramos Gonzalez, Maria Mercedes, 28006<br />

Madrid, ES<br />

Aleixandre de Artiñano, Amaya, 28040<br />

Madrid, ES<br />

(74) Ungria Lopez, Javier, Avda. Ramón y Cajal,<br />

78, 28043 Madrid, ES<br />

(62) 06764378.3 / 1 905 779<br />

(51) C07K 9/00 (11) 2 495 251 A1<br />

(25) En (26) En<br />

(21) 12169694.2 (22) 21.10.2004<br />

277<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

LT LV<br />

(30) 22.10.2003 US 513359 P<br />

(54) Hydrochloridsalze eines Glycopeptidphosphonatderivats<br />

Hydrochloride salts of a glycopeptide<br />

phosphonate derivative<br />

Chlorhydrates d'un derivé de glycopeptide<br />

phosphonate<br />

(71) Theravance Inc, 901 Gateway Boulevard,<br />

South San Francisco, CA 94080, US<br />

(72) Liu, Jyanwei, Sunnyvale, CA 94087, US<br />

Lee, Junning, El Granada, CA 94018, US<br />

(74) Scott, Susan Margaret, et al, Abel & Imray<br />

20 Red Lion Street, London WC1R 4PQ, GB<br />

(62) 04796022.4 / 1 678 201<br />

C07K 14/11 → (51) C12N 15/44<br />

(51) C07K 14/115 (11) 2 495 252 A2<br />

A61K 39/155 C12N 15/62<br />

(25) En (26) En<br />

(21) 12157071.7 (22) 07.07.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

(30) 09.07.2004 US 586843 P<br />

(54) Lösliche Formen von Hendra- und Nipah-<br />

Virus-G-Glycoprotein<br />

Soluble forms of hendra and nipah virus G<br />

glycoprotein<br />

Formes solubles de glycoproteine G des<br />

virus hendra et nipah<br />

(71) The Henry M. Jackson Foundation for the<br />

Advancement of Military Medicine, Inc.,<br />

1401 Rockville Pike Suite 600, Rockville, MD<br />

20852, US<br />

(72) Broder, Christopher, C, Silver Spring, MD<br />

Maryland 20905, US<br />

Bossart, Katharine, N, San Francisco, CA<br />

California 94118, US<br />

(74) Harrison Goddard Foote, Belgrave Hall<br />

Belgrave Street, Leeds LS2 8DD, GB<br />

(62) 05857509.3 / 1 789 593<br />

(51) C07K 14/31 (11) 2 495 253 A1<br />

C07K 1/22<br />

(25) En (26) En<br />

(21) 1216<strong>36</strong>14.6 (22) 11.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(30) 11.08.2008 US 188549 P<br />

16.04.2009 US 212812 P<br />

(54) Neuartige immunoglobulinbindende Proteine<br />

mit verbesserter Spezifizität<br />

Novel immunoglobulin-binding proteins<br />

with improved specificity<br />

Nouvelles protéines se liant à des immunoglobulines<br />

dont la spécificité est<br />

améliorée<br />

(71) EMD Millipore Corporation, 290 Concord<br />

Road, Billerica, MA 01821, US<br />

(72) Spector, Shari, Billerica, MA 01821, US<br />

(74) Kirkham, Nicholas Andrew, et al, Graham<br />

Watt & Co. LLP St. Botolph's House 7-9 St.<br />

Botolph's Road, Sevenoaks, Kent TN13 3AJ,<br />

GB<br />

(62) 09167670.0 / 2 157 099<br />

(51) C07K 14/31 (11) 2 495 254 A1<br />

C07K 1/22<br />

(25) En (26) En<br />

(21) 1216<strong>36</strong>15.3 (22) 11.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR

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