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European Patent Bulletin 2012/36 - European Patent Office

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(C07D) II.1(1)<br />

SAKATA, Masahiro, Osaka 569-1125, JP<br />

KONDO, Wataru, Tokyo 105-8422, JP<br />

HORI, Yoshikazu, Osaka 569-1125, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) C07D 413/12 (11) 1 851 214 B1<br />

C07D 413/14 C07C 229/08<br />

A61K 31/422 A61P 29/00<br />

(25) En (26) En<br />

(21) 06716026.7 (22) 21.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

(43) 07.11.2007<br />

(86) KR 2006/000576 21.02.2006<br />

(87) WO 2006/090997 2006/35 31.08.2006<br />

(30) 26.02.2005 KR 20050016203<br />

(54) ISOXAZOLINDERIVAT UND NEUES VER-<br />

FAHREN ZU DESSEN HERSTELLUNG<br />

ISOXAZOLINE DERIVATIVE AND NOVEL<br />

PROCESS FOR ITS PREPARATION<br />

DERIVES D'ISOXAZOLINE ET SON<br />

NOUVEAU PROCEDE DE PRODUCTION<br />

(73) LG Life Sciences Ltd., LG Twin Tower, East<br />

Tower, 20, Yoido-dong, Youngdungpo-gu,<br />

Seoul 150-010, KR<br />

(72) SHIN, Hyun Ik R & D Park, LG Life Sciences<br />

Ltd., Daejeon 305-380, KR<br />

CHOI, Hyeong Wook R & D Park, LG Life<br />

Sciences Ltd, Daejeon 305-380, KR<br />

HEO, Tae Ho R & D Park, LG Life Sciences<br />

Ltd., Daejeon 305-380, KR<br />

LEE, Kyu Woong R & D Park, LG Life<br />

Sciences Ltd., Daekepm 305-380, KR<br />

LEE, Jae Hoon R & D Park, LG Life Sciences<br />

Ltd., Daejeon 305-380, KR<br />

PARK, Ki Sook R & D Park, LG Life Sciences<br />

Ltd., 104-1, Moongi-dong, Yuseong-gu<br />

Daejeon 3, KR<br />

(74) Gillard, Richard Edward, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

C07D 413/12 → (51) C07C 237/<strong>36</strong><br />

C07D 413/14 → (51) C07C 237/<strong>36</strong><br />

C07D 413/14 → (51) C07D 413/04<br />

C07D 413/14 → (51) C07D 413/12<br />

C07D 417/06 → (51) C07D 213/40<br />

C07D 417/12 → (51) C07D 213/40<br />

C07D 417/12 → (51) C07D 277/34<br />

C07D 417/14 → (51) C07D 401/04<br />

(51) C07D 471/04 (11) 1 912 986 B1<br />

A61K 31/435 A61P 3/00<br />

(25) En (26) En<br />

(21) 06772525.9 (22) 08.06.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT<br />

RO SE SI SK TR<br />

HR MK RS<br />

(43) 23.04.2008<br />

(86) US 2006/022260 08.06.2006<br />

(87) WO 2006/135667 2006/51 21.12.2006<br />

(30) 09.06.2005 US 688993 P<br />

07.06.2006 US 448946<br />

(54) IMIDAZO- UND TRIAZOLOPYRIDINE ALS<br />

INHIBITOREN VON 11-BETA-HYDROXYS-<br />

TEROIDDEHYDROGENASE VOM TYP I<br />

IMIDIAZO -AND TRIAZOLOPYRIDINES AS<br />

INHIBITORS OF 11-BETA HYDROXYS-<br />

TEROID DEHYDROGENASE TYPE I<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

IMIDIAZO- ET TRIAZOLOPYRIDINES<br />

COMME INHIBITEURS DE LA 11-BÊTA<br />

HYDROXYSTÉROÏDE DÉSHYDROGÉNASE<br />

TYPE I<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton, NJ<br />

08543-4000, US<br />

(72) LI, James, J., Pennington, New Jersey<br />

08534, US<br />

HAMANN, Lawrence, G., North Grafton,<br />

Massachusetts 015<strong>36</strong>, US<br />

WANG, Haixia, Princeton, New Jersey<br />

08540, US<br />

(74) Beacham, Annabel Rose, Dehns St Bride's<br />

House 10 Salisbury Square, London EC4Y<br />

8JD, GB<br />

(51) C07D 471/04 (11) 2 046 789 B1<br />

C07D 219/06 A61K 31/165<br />

C07D 209/42 C07D 215/54<br />

C07D 217/26 C07D 235/24<br />

C07D 237/26 C07D 333/68<br />

C07D 233/62<br />

(25) En (26) En<br />

(21) 07805258.6 (22) 27.07.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL<br />

PT RO SE SI SK TR<br />

(43) 15.04.2009<br />

(86) IB 2007/052992 27.07.2007<br />

(87) WO 2008/012782 2008/05 31.01.2008<br />

(30) 27.07.2006 FR 0653138<br />

(54) MARKIERTE HALOBENZAMID-ANALOGA<br />

ALS RADIOPHARMAZEUTIKA<br />

LABELLED ANALOGUES OF HALOBEN-<br />

ZAMIDES AS RADIOPHARMACEUTICALS<br />

ANALOGUES MARQUES D'HALOBENZA-<br />

MIDES UTILISES COMME PRODUITS<br />

RADIOPHARMACEUTIQUES<br />

(73) INSTITUT NATIONAL DE LA SANTE ET DE<br />

LA RECHERCHE MEDICALE (INSERM), 101,<br />

rue de Tolbiac, 75013 Paris, FR<br />

Université d'Auvergne, Clermont-Ferrand 1,<br />

49, boulevard François-Mitterand, 63001<br />

Clermont-Ferrand Cedex 1, FR<br />

(72) MADELMONT, Jean-Claude, F-63540 Romagnat,<br />

FR<br />

CHEZAL, Jean-Michel, F-63400 Chamalieres,<br />

FR<br />

CHAVIGNON, Oliver, 63730 Les Martres De<br />

Veyre, FR<br />

TEULADE, Jean-Claude, 34430 Saint Jean<br />

De Vedas, FR<br />

MOINS, Nicole, 63000 Clemont-Ferrand, FR<br />

(74) Tanty, François, Cabinet Nony 3, rue de<br />

Penthièvre, 75008 Paris, FR<br />

(60) 11167370.3 / 2 <strong>36</strong>3 399<br />

(51) C07D 471/04 (11) 2 265 609 B1<br />

C07C 311/08 A61K 31/437<br />

A61P 35/00 A61P 13/12<br />

(25) En (26) En<br />

(21) 09716688.8 (22) 27.02.2009<br />

(84) CH DE ES FR GB IT LI TR<br />

AL BA RS<br />

(43) 29.12.2010<br />

(86) US 2009/035379 27.02.2009<br />

(87) WO 2009/111277 2009/37 11.09.2009<br />

(30) 29.02.2008 US 32801<br />

(54) ALS RAF-INHIBITOREN VERWENDETE<br />

IMIDAZO[4,5-B]PYRIDINDERIVATE<br />

IMDIZO [4. 5-B] PYRIDINE DERIVATIVES<br />

USED AS RAF INHIBITORS<br />

DÉRIVÉS D'IMIDAZO [4. 5-B] PYRIDINE<br />

UTILISÉS COMME INHIBITEURS DE RAF<br />

(73) Array Biopharma, Inc., 3200 Walnut Street,<br />

Boulder, CO 80301, US<br />

Genentech, Inc., 1 DNA Way, South San<br />

Francisco, CA 94080-4990, US<br />

634<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>36</strong>/<strong>2012</strong>) 05.09.<strong>2012</strong><br />

(72) AHRENDT, Kateri, A., Boulder Colorado<br />

80301, US<br />

BUCKMELTER, Alexandre, J., Boulder<br />

Colorado 80301, US<br />

GRINA, Jonas, Boulder Colorado 80301, US<br />

HANSEN, Joshua, D., Boulder Colorado<br />

80301, US<br />

LAIRD, Ellen, R., Boulder Colorado 80301,<br />

US<br />

NEWHOUSE, Brad, Boulder Colorado 80301,<br />

US<br />

REN, Li, Boulder Colorado 80301, US<br />

WENGLOWSKY, Steven, M., Boulder<br />

Colorado 80301, US<br />

FENG, Bainian, South San Francisco California<br />

94080-4900, US<br />

MALESKY, Kim, South San Francisco<br />

Colorado 94080-4900, US<br />

MATHIEU, Simon, South San Francisco California<br />

94080-4990, US<br />

RUDOLPH, Joachim, South San Francisco<br />

California 94080-4990, US<br />

WEN, Zhaoyang, South San Francisco California<br />

94080-4990, US<br />

YOUNG, Wendy, B., South San Francisco<br />

California 94080-4990, US<br />

MORENO, David, A., Boulder CO 80301, US<br />

(74) Bailey, Sam Rogerson, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

(51) C07D 471/04 (11) 2 303 879 B1<br />

A61K 31/437 A61P 3/10<br />

A61P 3/04<br />

(25) De (26) De<br />

(21) 09777108.3 (22) 10.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(43) 06.04.2011<br />

(86) EP 2009/005024 10.07.2009<br />

(87) WO 2010/020308 2010/08 25.02.2010<br />

(30) 18.08.2008 DE 102008038221<br />

(54) 7-AZAINDOLDERIVATE<br />

7-AZAINDOLE DERIVATIVES<br />

DÉRIVÉS DE 7-AZAINDOLE<br />

(73) Merck <strong>Patent</strong> GmbH, Frankfurter Strasse<br />

250, 64293 Darmstadt, DE<br />

(72) KLEIN, Markus, 64291 Darmstadt, DE<br />

C07D 471/04 → (51) C07D 401/06<br />

C07D 471/04 → (51) C07D 401/14<br />

(51) C07D 471/08 (11) 1 699 790 B1<br />

C07D 275/06 C07D 207/40<br />

(25) En (26) En<br />

(21) 04815907.3 (22) 29.12.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 13.09.2006<br />

(86) US 2004/043917 29.12.2004<br />

(87) WO 2005/065370 2005/29 21.07.2005<br />

(30) 30.12.2003 US 533169 P<br />

17.12.2004 US 15399<br />

(54) LÖSLICHE POLYMERE ALS AMIN-CAP-<br />

TURE-MITTEL UND METHODEN<br />

SOLUBLE POLYMERS AS AMINE<br />

CAPTURE AGENTS AND METHODS<br />

POLYMERES SOLUBLES EN TANT<br />

QU'AGENTS DE CAPTURE D'AMINES ET<br />

PROCEDES ASSOCIES<br />

(73) 3M Innovative Properties Company, 3M<br />

Center P.O.Box 33427, St. Paul, MN 55133-<br />

3427, US<br />

(72) BENSON, Karl, E., Saint Paul, MN 55133-<br />

3427, US<br />

BOMMARITO, G., Marco, Saint Paul, MN<br />

55133-3427, US

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