PCT/2002/18 - World Intellectual Property Organization

18/2002
8638 PCT Gazette - Section I - Gazette du PCT 2 May/mai 2002
(51) 7 C07C 209/48, 211/29, 29/09, 33/46, 67/14,
69/743
(11) WO 02/34707 (13) A1
(21) PCT/GB01/04692
(22) 18 Oct/oct 2001 (18.10.2001)
(25) en (26) en
(30) 0026348.3 27 Oct/oct 2000 GB
(27.10.2000)
(43) 2 May/mai 2002 (02.05.2002)
(54) PREPARATION OF 4-METHYL-2,3,5,6-
TETRAFLUOROBENZYL ALCOHOL
PREPARATION D’ALCOOL DE 4-ME-
THYL-2,3,5,6-TETRAFLUOROBEN-
ZYLE
(71) SYNGENTA LIMITED [GB/GB]; Fernhurst,
Haslemere, Surrey GU27 3JE (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) JONES, Raymond, Vincent, Heavon
[GB/GB]; Grangemouth Manufacturing Centre,
Earls Road, Grangemouth, Stirlingshire
FK3 8XG (GB). BROWN, Stephen, Martin
[GB/GB]; Process Technology DepART-
MENT, Leeds Road, Huddersfield, West
Yorkshire HD2 1FF (GB).
(74) WATERMAN, John, Richard et al. / etc.;
Intellectual Property Department, Syngenta
Limited, Jealott’s Hill Research Centre, PO
Box 3538, Bracknell RG42 6YA (GB).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC
LK LR LS LT LU LV MA MD MG MK MN
MW MX MZ NO NZ PH PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT TZ UA UG
US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
(51) 7 C07C 225/32, A61K 31/35, C07D 213/38,
A61P 35/00
(11) WO 02/34708 (13) A2
(21) PCT/IB01/01993
(22) 24 Oct/oct 2001 (24.10.2001)
(25) en (26) en
(30) 00 1 30048.2 25 Oct/oct 2000 CN
(25.10.2000)
(43) 2 May/mai 2002 (02.05.2002)
(54) ALIPHATIC AMINO-SUBSTITUTED
DEMETHOXYLATED HYPOCRE-
LLINS AND THEIR SYNTHESIS
HYPOCRELLINES DEMETHOXYLEES
AMINO-SUBSTITUEES ALIPHA-
TIQUES ET SYNTHESE DE CELLES-CI
(71) ALTACHEM PHARMA, LTD. [CA/CA];
17215 - 108 Avenue, Edmonton, Alberta
T5S 1G2 (CA). INSTITUTE OF PHOTO-
GRAPHIC CHEMISTRY ACADEMIA
SINICA [CN/CN]; Beijing 100101 (CN).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ZHANG, Manhua [CN/CN]; Suite 301,
Building 313, 311 Kexue Yuan Nanli, Beijing
(CN). XU, Shangjie [CN/CN]; Room
413, Building 3, 3A Datun Road, Beijing
(CN). WU, Tao [CN/CN]; Room 413, Building
3, 3A Datun Road (CN). CHEN, Shen
[CN/CN]; Suite 421, Building 1, 3A Datun
Road, Beijing (CN). SHEN, Tao [CN/CN];
Suite 306, Building 510, 311 Kexue Yuan
Nanli, Beijing (CN).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EE ES FI GB GD GE GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC
LK LR LS LT LU LV MA MD MG MK MN
MW MX MZ NO NZ PL PT RO RU SD SE
SG SI SK SL TJ TM TR TT TZ UA UG US
UZ VN YU ZA ZW.
Declaration / Déclaration :
(u) for / pour US only / seulement
(51) 7 C07C 227/40, 227/42, 229/28
(11) WO 02/34709 (13) A1
(21) PCT/EP01/11867
(22) 15 Oct/oct 2001 (15.10.2001)
(25) en (26) en
(30) MI2000A002285 23 Oct/oct 2000 IT
(23.10.2000)
(43) 2 May/mai 2002 (02.05.2002)
(54) PROCESS FOR THE PREPARATION OF
GABAPENTIN
PROCEDE DE PREPARATION DE GA-
BAPENTINE
(71) ZAMBON GROUP S.P.A. [IT/IT]; via della
Chimica, 9, I-36100 Vicenza (IT).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) CANNATA, Vincenzo [IT/IT]; via Annibale
Clò, 12, I-40037 Sasso Marconi (IT).
NICOLI, Andrea [IT/IT]; via Monzambano,
50, I-36100 Vicenza (IT). CORCELLA,
Francesco [IT/IT]; via Europa, 25, Quinto
Stampi, I-20089 Rozzano (IT).
(74) ZAMBON GROUP S.P.A.; I.P. & Intelligence,
via Lillo del Duca, 10, I-20091 Bresso
(IT).
(81) AL AT CA CH DE DK ES FI GB HU IL IN
JP LT LU LV MK PT RO SE SI US.
Published / Publiée :(c)
Declaration / Déclaration :
(u) for / pour US only / seulement
(51) 7 C07C 229/30, 227/16, 67/313, 403/16
(11) WO 02/34710
(21) PCT/FR01/03331
(13) A2
(22) 26 Oct/oct 2001 (26.10.2001)
(25) fr (26) fr
(30) 00/13726 26 Oct/oct 2000
(26.10.2000)
FR
(43) 2 May/mai 2002 (02.05.2002)
(54) NOVEL INTERMEDIATES FOR USE IN
RETINOID SYNTHESIS
NOUVEAUX INTERMEDIAIRES
UTILES POUR LA SYNTHESE DE
RETINOIDES
(71) CENTRE NATIONAL DE LA
RECHERCHE SCIENTIFIQUE (CNRS)
[FR/FR]; 3, rue Michel Ange, F-75794 Paris
Cedex 16 (FR).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) VALLA, Alain [FR/FR]; Impasse
Ty Guen, Ezer, F-29750 Loctudy (FR).
CARTIER, Dominique [FR/FR]; 16,
rue M. Curie, F-29000 Quimper (FR).
LABIA, Roger [FR/FR]; Trogour-Huella,
F-29180 Plougonnec (FR). POTIER, Pierre,
Jean-Paul [FR/FR]; 14, avenue de Breteuil,
F-75007 Paris (FR).
(74) MARTIN, Jean-Jacques et al. / etc.; Cabinet
Regimbeau, 20, rue de Chazelles, F-75847
Paris Cedex 17 (FR).
(81) CA JP US.
Declaration / Déclaration :
(u) for / pour US only / seulement
(51) 7 C07C 229/38, 317/22, 63/04, 257/00, C07D
333/22, 307/02, 277/30, 207/30, 207/08,
211/70, 311/78, 239/02, 265/30, 277/62,
211/70, 317/44, 231/56, A61K 31/24, 31/69,
31/38, 31/34, 31/38, 31/34, 31/255, 31/425,
31/40, 31/55, 31/495, 31/505, 31/535,
31/425, 31/415, 31/44, 31/27, 31/155
(11) WO 02/34711 (13) A1
(21) PCT/US01/32582
(22) 22 Oct/oct 2001 (22.10.2001)
(25) en (26) en
(30) 60/241,848 20 Oct/oct 2000 US
(20.10.2000)
(30) 60/281,735 6 Apr/avr 2001 US
(06.04.2001)
(43) 2 May/mai 2002 (02.05.2002)
(54) BIARYL COMPOUNDS AS SERINE
PROTEASE INHIBITORS
COMPOSES BIARYLE UTILISES
COMME INHIBITEURS DE SERINE
PROTEASE
(71) BIOCRYST PHARMACEUTICALS,
INC. [US/US]; 2910 Parkway Lake Drive,
Birmingham, AL 35244 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BABU, Yarlagadda, S. [IN/US]; 3441
Strollway Drive, Birmingham, AL 35226
(US). ROWLAND, Scott, R. [US/US]; 3436
Tamasee Lane, Hoover, AL 35226 (US).
CHAND, Pooran [US/US]; 509 Creekwood
Place, Birmingham, AL 35226 (US). KO-
TIAN, Pravin, L. [IN/US]; 1313 Atkins
Trimm Blvd., Birmingham, AL 35226 (US).
EL-KATTAN, Yahya [LB/US]; 5023 Rime
Village, Hoover, AL 35216 (US). NIWAS,
Shri [US/US]; 3348 Castle Crest Drive,
Birmingham, AL 35244 (US).
(74) AMERNICK, Burton, A. et al. / etc.; Connolly
Bove Lodge & Hutz LLP, P.O. Box
19088, Washington, DC 20036 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PH PL PT RO RU
SD SE SG SI SK SL TJ TM TR TT TZ UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
Published / Publiée :(c)