PCT/2002/18 - World Intellectual Property Organization

18/2002
8648 PCT Gazette - Section I - Gazette du PCT 2 May/mai 2002
NJ 07065-0907 (US). ILLIG, Kathleen, J.
[US/US]; 126 East Lincoln Avenue, Rahway,
NJ 07065-0907 (US). KANIKE, Anand
[IN/US]; 126 East Lincoln Avenue, Rahway,
NJ 07065-0907 (US). PATEL, Hiren
[IN/US]; 126 East Lincoln Avenue, Rahway,
NJ 07065-0907 (US). REYNOLDS, Scott,
D. [US/US]; 126 East Lincoln Avenue, Rahway,
NJ 07065-0907 (US). TSINONTIDES,
Stelios, C. [US/US]; 126 East Lincoln Avenue,
Rahway, NJ 07065-0907 (US).
(74) MERCK & CO., INC.; 126 East Lincoln
Avenue, Rahway, NJ 07065-0907 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 487/04, A61P 29/00
(11) WO 02/34751 (13) A1
(21) PCT/EP01/12251
(22) 23 Oct/oct 2001 (23.10.2001)
(25) en (26) en
(30) 0026106.5 25 Oct/oct 2000 GB
(25.10.2000)
(43) 2 May/mai 2002 (02.05.2002)
(54) HEXAHYDRO-4-OXOAZEPINO[3,2,1-
HI]INDOLES
HEXAHYDRO-4-OXOAZE-
PINO[3,2,1-HI] INDOLES
(71) NOVARTIS AG [CH/CH]; Lichtstrasse 35,
Basel 4056 (CH).
(for all designated States except / pour tous
les États désignés sauf AT US)
(71) NOVARTIS-ERFINDUNGEN VER-
WALTUNGSGESELLSCHAFT M.B.H.
[AT/AT]; Brunner Strasse 59, A-1230 Vienna
(AT).
(only for / seulement pour AT)
(72, 75) ROGGO, Silvio [CH/CH]; Stettbrunnenweg
36, CH-4132 Muttenz (CH). HIN-
TERMANN, Samuel [CH/CH]; Klingelbergstrasse
93, CH-4056 Basel (CH).
RASETTI, Vittorio [CH/CH]; Mohrhaldenstrasse
196, CH-4125 Riehen (CH). VON
KROSIGK, Ulrike [DE/CH]; Wettsteinallee
83, CH-4058 Basel (CH).
(74) BECKER, Konrad; Novartis AG, Corporate
Intellectual Property, Patent & Trademark Department,
CH-4002 Basel (CH).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PH PL PT RO RU
SD SE SG SI SK SL TJ TM TR TT TZ UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
(51) 7 C07D 487/04, A61K 31/55, A61P 31/10
(11) WO 02/34752 (13) A1
(21) PCT/EP01/12287
(22) 17 Oct/oct 2001 (17.10.2001)
(25) en (26) en
(30) 00203726.5 23 Oct/oct 2000 EP
(23.10.2000)
(43) 2 May/mai 2002 (02.05.2002)
(54) ANTIFUNGAL 4-SUBSTITUTED
5,6-DIHYDRO-4H-PYRROLO[1,2-
A][1,4]BENZODIAZEPINES
BENZODIAZEPINES 5,6-DIHY-
DRO-4H-PYRROLO[1,2-A][1,4] SUB-
STITUEES EN 4, ANTIFONGIQUES
(71) JANSSEN PHARMACEUTICA N.V.
[BE/BE]; Turnhoutseweg 30, B-2340 Beerse
(BE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) GILKERSON, Terence [GB/GB];
Krown Synthesis, 11 The Ness, Canterbury,
Kent CT1 3NL (GB). NASH, Roger,
John [GB/GB]; Merlin Synthesis, University
of London, Wye College, WYE, Ashford,
Kent TN25 5AH (GB). VAN GESTEL,
Jozef, Frans, Elisabetha [BE/BE]; Renier
Sniederspad 9, B-2350 Vosselaar (BE).
MEERPOEL, Lieven [BE/BE]; Janssen
Pharmaceutica N.V., Turnhoutseweg 30,
B-2340 Beerse (BE).
(74) QUAGHEBEUR, Luc et al. / etc.; Janssen
Pharmaceutica N.V., Turnhoutseweg 30,
B-2340 Beerse (BE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PH PL PT RO RU
SD SE SG SI SK SL TJ TM TR TT TZ UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 487/10, A61K 31/527, A61P 29/00,
35/00, C07D 471/10 // (C07D 487/10,
239:00, 209:00) (C07D 471/10, 239:00,
221:00)
(11) WO 02/34753
(21) PCT/IB01/01986
(13) A2
(22) 23 Oct/oct 2001 (23.10.2001)
(25) en (26) en
(30) 60/243,389 26 Oct/oct 2000
(26.10.2000)
US
(43) 2 May/mai 2002 (02.05.2002)
(54) SPIRO-PYRIMIDINE-2,4,6-TRIONE
METALLOPROTEINASE INHIBITORS
INHIBITEURS DE METALLOPROTEI-
NASE
ONE
SPIRO-PYRIMIDINE-2,4,6-TRI-
(71) PFIZER PRODUCTS INC. [US/US]; Eastern
Point Road, Groton, CT 06340 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BRONK, Brian, Scott [US/US]; Pfizer
Global Research and Development, Eastern
Point Road, Groton, CT 06340 (US). NOE,
Mark, Carl [US/US]; Pfizer Global Research
and Development, Eastern Point Road,
Groton, CT 06340 (US). WYTHES, Martin,
James [GB/US]; Pfizer Global Research and
Development, Eastern Point Road, Groton,
CT 06340 (US).
(74) LUMB, J., Trevor et al. / etc.; c/o Simpson,
Alison, Urquhart-Dykes & Lord, 30 Welbeck
Street, London, W1G 8ER (GB).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PH PL PT RO RU
SD SE SG SI SK SL TJ TM TR TT TZ UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
(51) 7 C07D 498/00
(11) WO 02/34754
(21) PCT/EP01/12344
(13) A2
(22) 22 Oct/oct 2001 (22.10.2001)
(25) en (26) en
(30) 0026224.6 26 Oct/oct 2000
(26.10.2000)
GB
(30) 0111858.7 15 May/mai 2001
(15.05.2001)
GB
(43) 2 May/mai 2002 (02.05.2002)
(54) BENZOXAZINONE DERIVATIVES,
THEIR PREPARATION AND USE
DERIVES DE BENZOXAZINONE,
LEUR PREPARATION ET
TION
UTILISA-
(71) SMITHKLINE BEECHAM P.L.C.
[GB/GB]; New Horizons Court, Brentford,
Middlesex TW8 9EP (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) JOHNSON, Christopher, Norbert
[GB/GB]; GlaxoSmithKline Pharmaceuticals,
New Frontiers Science Park South,
Third Avenue, Harlow, Essex CM19 5AW
(GB). RAMI, Harshad, Kantilal [GB/GB];
SmithKline Beecham Pharmaceuticals, New
Frontiers Science Park South, Third Avenue,
Harlow, Essex CM19 5AW (GB). STEMP,
Geoffrey [GB/GB]; GlaxoSmithKline Pharmaceuticals,
New Frontiers Science Park
South, Third Avenue, Harlow, Essex CM19
5AW (GB). THEWLIS, Kevin [GB/GB];
GlaxoSmithKline Pharmaceuticals, New
Frontiers Science Park South, Third Avenue,
Harlow, Essex CM19 5AW (GB). THOMP-
SON, Mervyn [GB/GB]; GlaxoSmithKline
Pharmaceuticals, New Frontiers Science Park
South, Third Avenue, Harlow, Essex CM19
5AW (GB). VONG, Antonio, Kuok, Keong
[GB/GB]; SmithKline Beecham Pharmaceuticals,
New Frontiers Science Park South,