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PCT/2002/18 - World Intellectual Property Organization

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<strong>18</strong>/<strong>2002</strong><br />

8550 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 2 May/mai <strong>2002</strong><br />

27, 06108 Halle/Saale (DE). FRIEDRICH,<br />

Daniel [DE/DE]; Glauchaer Str. 73, 06110<br />

Halle/Saale (DE).<br />

(74) FORSTMEYER, Dietmar et al. / etc.;<br />

Boeters & Bauer, Bereiteranger 15, 81541<br />

München (DE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GQ GW ML<br />

MR NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 02/34243 (13) A2<br />

(21) <strong>PCT</strong>/EP01/12479<br />

(22) 29 Oct/oct 2001 (29.10.2001)<br />

(25) en (26) en<br />

(30) 60/244,036 27 Oct/oct 2000 US<br />

(27.10.2000)<br />

(43) 2 May/mai <strong>2002</strong> (02.05.<strong>2002</strong>)<br />

(54) METHOD FOR THE TREATMENT OF<br />

NEUROLOGICAL AND NEUROPSY-<br />

CHOLOGICAL DISORDERS<br />

PROCEDE POUR LE TRAITEMENT<br />

DE TROUBLES NEUROLOGIQUES ET<br />

NEUROPSYCHOLOGIQUES<br />

(71) PROBIODRUG AG [DE/DE]; Weinbergweg<br />

22 / Biozentrum, 06120 Halle/Saale<br />

(DE).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) VON HÖRSTEN, Stephan [DE/DE];<br />

Birkenkamp 1, 30900 Wedemark (DE).<br />

KASK, Ants [EE/EE]; Kadaka pst. 12, EE<br />

10912 Tallinn (EE). DEMUTH, Hans-Ulrich<br />

[DE/DE]; Hegelstrasse 14, 06114<br />

Halle/Saale (DE). HOFFMANN, Matthias<br />

[DE/DE]; Frobelstrasse 1d, 06688 Wengelsdorf<br />

(DE). KRUBER, Susanne [DE/DE];<br />

Blumenauweg 29, 06120 Halle/Saale (DE).<br />

NGUYEN, Huu, Phuc [DE/DE]; Timmendorffstrasse<br />

6, 30625 Hannover (DE).<br />

(74) FORSTMEYER, DIETMAR et al. / etc.;<br />

Boeters & Bauer, Bereiteranger 15, 81541<br />

München (DE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GQ GW ML<br />

MR NE SN TD TG).<br />

Published / Publiée :(q1)<br />

(51) 7 A61K 31/00<br />

(11) WO 02/34244 (13) A2<br />

(21) <strong>PCT</strong>/EP01/12985<br />

(22) 25 Oct/oct 2001 (25.10.2001)<br />

(25) en (26) en<br />

(30) 60/243,431 27 Oct/oct 2000 US<br />

(27.10.2000)<br />

(30) 60/245,582 6 Nov/nov 2000 US<br />

(06.11.2000)<br />

(30) 60/250,138 1 Dec/déc 2000 US<br />

(01.12.2000)<br />

(43) 2 May/mai <strong>2002</strong> (02.05.<strong>2002</strong>)<br />

(54) A COMBINATION COMPRISING<br />

CAMPTOTHECIN AND A STILBENE<br />

DERIVATIVE FOR THE TREATMENT<br />

OF CANCER<br />

COMBINAISON DE CAMPTOTHE-<br />

CINE ET D’UN DERIVE DE STILBENE<br />

POUR LE TRAITEMENT DU CANCER<br />

(71) AVENTIS PHARMA S.A. [FR/FR]; 20, avenue<br />

Raymond Aron, F-92160 Antony (FR).<br />

(72) BISSERY, Marie-Christine; 5, rue Henri-<br />

Poincaré, F-94400 Vitry-sur-Seine (FR).<br />

(74) LE PENNEC, Magali; Aventis Pharma<br />

S.A., Patent Department, 20, avenue Raymond<br />

Aron, F-92165 Antony Cedex (FR).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS JP KE KG KP KR KZ<br />

LC LK LR LS LT LU LV MA MD MG MK<br />

MN MW MX MZ NO NZ PH PL PT RO RU<br />

SD SE SG SI SK SL TJ TM TR TT TZ UA<br />

UG UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GQ GW ML<br />

MR NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 02/34245<br />

(21) <strong>PCT</strong>/US01/27779<br />

(13) A2<br />

(22) 23 Oct/oct 2001 (23.10.2001)<br />

(25) en (26) en<br />

(30) 60/242,899 24 Oct/oct 2000<br />

(24.10.2000)<br />

US<br />

(30) 60/283,120 11 Apr/avr 2001<br />

(11.04.2001)<br />

US<br />

(30) 60/314,2<strong>18</strong> 22 Aug/août 2001<br />

(22.08.2001)<br />

US<br />

(43) 2 May/mai <strong>2002</strong> (02.05.<strong>2002</strong>)<br />

(54) USE OF TOLTERODINE TO TREAT<br />

ASTHMA<br />

UTILISATION DE TOLTERO-<br />

DINE DANS LE<br />

L’ASTHME<br />

TRAITEMENT DE<br />

(71) PHARMACIA & UPJOHN COMPANY<br />

[US/US]; 301 Henrietta Street, Kalamazoo,<br />

MI 49001 (US). PHARMACIA AB [SE/SE];<br />

Lindhagensgatan 133, S-0112 87 Stockholm<br />

(SE).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) GILLBERG, Per-Goran [SE/SE];<br />

Tallbacksvagen 44A, S-756 45 Uppsala<br />

(SE). SUNDQUIST, Staffan [SE/SE]; Sturgatan<br />

25, S-561 45 Huskvarna (SE). CAM-<br />

MARATA, Sue, K. [US/US]; 10147 Point<br />

O’Woods Drive, Portage, MI 49002 (US).<br />

(74) STEIN, Bruce; Global <strong>Intellectual</strong> <strong>Property</strong>,<br />

Pharmacia & Upjohn Company, 301 Henrietta<br />

Street, Kalamazoo, MI 49001 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EC EE ES FI GB GD GE GH GM<br />

HR HU ID IL IN IS JP KE KG KP KR KZ<br />

LC LK LR LS LT LU LV MA MD MG MK<br />

MN MW MX MZ NO NZ PH PL PT RO RU<br />

SD SE SG SI SK SL TJ TM TR TT TZ UA<br />

UG US UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GQ GW ML<br />

MR NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 02/34246<br />

(21) <strong>PCT</strong>/US01/30201<br />

(13) A2<br />

(22) 27 Sep/sep 2001 (27.09.2001)<br />

(25) en (26) en<br />

(30) 60/242,642 23 Oct/oct 2000<br />

(23.10.2000)<br />

US<br />

(43) 2 May/mai <strong>2002</strong> (02.05.<strong>2002</strong>)<br />

(54) USE OF HYDROPEROXYEICOSATE-<br />

TRAENOIC ACID DERIVATIVES FOL-<br />

LOWING REFRACTIVE SURGERY<br />

UTILISATION DE DERIVES D’ACIDE<br />

HYDROXYEICOSATETRANOIQUE<br />

(HETE) APRES UNE CHIRURGIE RE-<br />

FRACTIVE<br />

(71) ALCON UNIVERSAL LTD. [CH/CH];<br />

Bosch 69, P. O. Box 62, CH-6331 Hunenberg<br />

(CH).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) YANNI, John, M. [US/US]; 2821 Donnybrook<br />

Drive, Burleson, TX 76028 (US).<br />

GAMACHE, Daniel, A. [US/US]; 5610<br />

Hunterwood Lane, Arlington, TX 76017<br />

(US). MILLER, Steven, T. [US/US]; 5902<br />

Canberra Lane, Arlington, TX 76017 (US).<br />

(74) RYAN, Patrick, M. et al. / etc.; R & D Counsel<br />

Q-148, 6201 South Freeway, Fort Worth,<br />

TX 76134-2099 (US).<br />

(81) AU BR CA CN JP KR MX PH PL US ZA.<br />

(84) EP (AT BE CH CY DE DK ES FI FR GB GR<br />

IE IT LU MC NL PT SE TR).<br />

(51) 7 A61K 31/00<br />

(11) WO 02/34247<br />

(21) <strong>PCT</strong>/US01/326<strong>18</strong><br />

(13) A2<br />

(22) 23 Oct/oct 2001 (23.10.2001)<br />

(25) en (26) en<br />

(30) 60/241,955 23 Oct/oct 2000<br />

(23.10.2000)<br />

US<br />

(43) 2 May/mai <strong>2002</strong> (02.05.<strong>2002</strong>)<br />

(54) ANTICANCER AGENTS BASED ON<br />

REGULATION OF PROTEIN PRENY-<br />

LATION

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