PCT/2002/18 - World Intellectual Property Organization

18/2002
2 May/mai 2002 PCT Gazette - Section I - Gazette du PCT 8641
(51) 7 C07D 231/54, 401/12, 409/12, A61K
31/416, A61P 35/00
(11) WO 02/34721
(21) PCT/US00/28952
(13) A1
(22) 20 Oct/oct 2000 (20.10.2000)
(25) en (26) en
(43) 2 May/mai 2002 (02.05.2002)
(54) ACYLSEMICARBAZIDES AND THEIR
USE AS CYCLIN DEPENDENT KI-
NASE (CDK) INHIBITORS
SEMI-CARBAZIDES ACYLE ET UTI-
LISATIONS DE CELLES-CI COMME
INHIBITEURS DE KINASE DEPEN-
DANTE DES CYCLINES (CDK)
(71) DU PONT PHARMACEUTICALS COM-
PANY [US/US]; Chestnut Run Plaza, 974
Centre Road, Wilmington, DE 19805 (US).
(72) NUGIEL, David, A.; 8 Vanessa Court,
Cherry Hill, NJ 08003 (US). CARINI,
David, J.; 1921 Julian Road, Wilmington,
DE 19803 (US). DI MEO, Susan, V.; 406
Clayton Avenue, Wilmington, DE 19809
(US). VIDWANS, Anup; 3120 Naamans
Road, Apartment F-8, Wilmington, DE
19810 (US). YUE, Eddy, W.; 9 Altemus
Drive, Landenberg, PA 19350 (US).
(74) DOLAN, Peter, L.; Du Pont Pharmaceuticals
Company, Legal Patent Records Center,
1007 Market Street, Wilmington, DE 19898
(US).
(81) AU BR CA CN CZ EE HU IL IN JP KR LT
LV MX NO NZ PL RO SG SI SK TR UA VN
ZA.
(84) EA (AM AZ BY KG KZ MD RU TJ TM); EP
(ATBECHCYDEDKESFIFRGBGRIE
IT LU MC NL PT SE).
(51) 7 C07D 233/54, C07F 5/02, C07C 307/02,
C08F 4/00, 36/04
(11) WO 02/34722
(21) PCT/IB01/02003
(13) A1
(22) 25 Oct/oct 2001 (25.10.2001)
(25) en (26) en
(30) 00403008.6 27 Oct/oct 2000
(27.10.2000)
EP
(43) 2 May/mai 2002 (02.05.2002)
(54) IMIDAZOLIUM SALTS AND THEIR
USE OF THESE IONIC LIQUIDS AS A
SOLVENT
SELS D’IMIDAZOLIUM ET UTILISA-
TION DE CES LIQUIDES IONIQUES
COMME SOLVANT
(71) CENTRE NATIONAL DE LA
RECHERCHE SCIENTIFIQUE
(C.N.R.S.) [FR/FR]; 3, rue Michel Ange,
F-75016 Paris (FR).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) CHAUVIN, Yves [FR/FR]; 10, Place
François Sicard, F-37000 Tours (FR).
MAGNA, Lionel [FR/FR]; Le Fenouillet,
Les Jonquilles C1, F-83400 Hyeres (FR).
NICCOLAI, Gerald, Peter [FR/FR]; 1, rue
du Professeur Calmette, F-69100 Villeurbanne
(FR). BASSET, Jean-Marie [FR/FR];
18, Chemin J.B. Gilliard, F-69300 Caluire
(FR).
(74) JACOBSON, Claude; Cabinet Lavoix, 2,
place d’Estienne-d’Orves, F-75441 Paris
Cedex 09 (FR).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CO CR CU CZ DE DK
DM DZ EC EE ES FI GB GD GE GH GM
HR HU ID IL IN IS JP KE KG KP KR KZ
LC LK LR LS LT LU LV MA MD MG MK
MN MW MX MZ NO NZ PH PL PT RO RU
SD SE SG SI SK SL TJ TM TR TT TZ UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GQ GW ML
MR NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 235/06, C07F 15/00, C08G 61/08,
B01J 31/32
(11) WO 02/34723 (13) A1
(21) PCT/JP01/09206
(22) 19 Oct/oct 2001 (19.10.2001)
(25) ja (26) ja
(30) 2000-322554 23 Oct/oct 2000 JP
(23.10.2000)
(30) 2000-324452 24 Oct/oct 2000 JP
(24.10.2000)
(30) 2001-126970 25 Apr/avr 2001 JP
(25.04.2001)
(43) 2 May/mai 2002 (02.05.2002)
(54) PROCESS FOR PREPARATION OF
DIAMINOCARBENE-TRANSITION
METAL COMPLEXES, RUTHENIUM
COMPOUNDS AND THEIR USAGE
METHODE DE PREPARATION DE
COMPLEXES DE METAUX DE TRAN-
SITION A BASE DE DIAMINOCAR-
BENE
(71) ZEON CORPORATION [JP/JP]; 6-1,
Marunouchi 2-chome, Chiyoda-ku, Tokyo
100-8323 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) OKADA, Seiji [JP/JP]; c/o ZEON
CORPORATION, Research & Development
Center, 2-1, Yako 1-chome, Kawasaki-ku,
Kawasaki-shi, Kanagawa 210-9507 (JP).
TAGUCHI, Kazunori [JP/JP]; c/o ZEON
CORPORATION, Research & Development
Center, 2-1, Yako 1-chome, Kawasaki-ku,
Kawasaki-shi, Kanagawa 210-9507 (JP).
TSUNOGAE, Yasuo [JP/JP]; c/o ZEON
CORPORATION, Research & Development
Center, 2-1, Yako 1-chome, Kawasaki-ku,
Kawasaki-shi, Kanagawa 210-9507 (JP).
(74) WADA, Yasuro; c/o ZEON CORPORA-
TION, 6-1, Marunouchi 2-chome, Chiyoda-ku,
Tokyo 100-0005 (JP).
(81) US.
(84) EP (DE GB).
(51) 7 C07D 239/34, 401/12, 409/12, A01N 43/54
(11) WO 02/34724 (13) A1
(21) PCT/CN01/01395
(22) 13 Sep/sep 2001 (13.09.2001)
(25) zh (26) zh
(30) 00 1 30735.5 16 Oct/oct 2000 CN
(16.10.2000)
(30) 01 1 12689.2 20 Apr/avr 2001 CN
(20.04.2001)
(30) 01 1 13199.3 29 Jun/juin 2001 CN
(29.06.2001)
(43) 2 May/mai 2002 (02.05.2002)
(54) NEW 2-PYRIMIDINYLOXY-N-ARYL-
BENZYLAMINE DERIVATIVES,
THEIR PROCESSES AND USES
NOUVEAUX DERIVES DE 2-PYRI-
MIDINYLOXY-N-ARYL-BENZYLA-
MINE, LEUR PROCEDE DE PREPARA-
TION ET LEURS APPLICATIONS
(71) SHANGHAI INSTITUTE OF ORGANIC
CHEMISTRY, CHINESE ACADEMY
OF SCIENCES [CN/CN]; 354, Feng lin
Road, Shanghai 200032 (CN). ZHEJIANG
CHEMICAL INDUSTRY RESEARCH
INSTITUTE [CN/CN]; 47, Huan Cheng Bei
Road, Zhejiang Province, Hangzhou 310023
(CN).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) LU, Long [CN/CN]; 354, Feng Lin
Road, Shanghai 200032 (CN). CHEN,
Jie [CN/CN]; 387, Tian Mu Shan Road,
Hangzhou, Zhejiang 310023 (CN). WU,
Jun [CN/CN]; 387, Tian Mu Shan Road,
Hangzhou, Zhejiang 310023 (CN). LING,
Wen [CN/CN]; 354, Feng Lin Road, Shanghai
200032 (CN). MAO, Lisheng [CN/CN];
354, Feng Lin Road, Shanghai 200032
(CN). LI, Mingzhi [CN/CN]; 387, Tian Mu
Shan Road, Hangzhou, Zhejiang 310023
(CN). CAI, Xian [CN/CN]; 354, Feng
Lin Road, Shanghai 200032 (CN). PENG,
Weili [CN/CN]; 387, Tian Mu Shan Road,
Hangzhou, Zhejiang 310023 (CN). WU,
Yong [CN/CN]; 354, Feng Lin Road, Shanghai
200032 (CN). WU, Shenggan [CN/CN];
387, Tian Mu Shan Road, Hangzhou, Zhejiang
310023 (CN). WANG, Hongjun
[CN/CN]; 354, Feng Lin Road, Shanghai
200032 (CN). WANG, Guochao [CN/CN];
387, Tian Mu Shan Road, Hangzhou, Zhejiang
310023 (CN). CUI, Hu [CN/CN]; 354,
Feng Lin Road, Shanghai 200032 (CN).
HAN, Shidong [CN/CN]; 387, Tian Mu
Shan Road, Hangzhou, Zhejiang 310023
(CN). QIU, Weilian [CN/CN]; 354, Feng
Lin Road, Shanghai 200032 (CN). WANG,
Yonghua [CN/CN]; 387, Tian Mu Shan
Road, Hangzhou, Zhejiang 310023 (CN).
(74) SHANGHAI ZHI XIN PATENT AGENT
LTD.; 10/F, Italy Building, 446 Zhao Jia Bang
Road, Shanghai 200031 (CN).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CO CR CU CZ DE DK DM
DZ EC EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW MX
MZ NO NZ PL PT RO RU SD SE SG SI SK
SL TJ TM TR TT TZ UA UG US UZ VN YU
ZA ZW.
Declarations / Déclarations :
(s) for the following designations / pour les
désignations suivantes : AE AG AL AM AT AU AZ
BA BB BG BR BY BZ CA CH CO CR CU CZ DE
DK DM DZ EC EE ES FI GB GD GE GH GM HR
HU ID IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW MX MZ
NO NZ PL PT RO RU SD SE SG SI SK SL TJ TM
TR TT TZ UA UG UZ VN YU ZA ZW AP (GH GM