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Bulletin 2011/10 - European Patent Office

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(A61K) I.1(2)<br />

(30) 12.02.2007 US 889336 P<br />

06.11.2007 US 985735 P<br />

(54) • Pyrazolderivate als 11-beta-HSD1-Hemmer<br />

• Pyrazole derivatives as 11-beta-HSD1<br />

inhibitors<br />

• Dérivés du pyrazole comme inhibiteurs de<br />

11-bêta-HSD1<br />

(71) AstraZeneca AB (Publ), 151 85 Södertälje,<br />

SE<br />

(72) Packer, Martin, Macclesfield, Cheshire SK<strong>10</strong><br />

4TG, GB<br />

Scott, James Stewart, Macclesfield, Cheshire<br />

SK<strong>10</strong> 4TG, GB<br />

Stocker, Andrew, Macclesfield, Cheshire<br />

SK<strong>10</strong> 4TG, GB<br />

Whittamore, Paul Robert Owen, Macclesfield,<br />

Cheshire SK<strong>10</strong> 4TG, GB<br />

(62) 08702088.9 / 2 124 937<br />

A61K 31/4155 → (51) A61K 31/415<br />

A61K 31/4188 → (51) C07D 471/04<br />

A61K 31/4192 → (51) C07D 249/04<br />

A61K 31/423 → (51) A61K 31/00<br />

A61K 31/435 → (51) A61K 31/198<br />

A61K 31/436 → (51) A61K 31/704<br />

A61K 31/4375 → (51) C07D 487/04<br />

A61K 31/438 → (51) C07D 498/<strong>10</strong><br />

A61K 31/439 → (51) A61K 45/00<br />

A61K 31/439 → (51) C07G 5/00<br />

A61K 31/44 → (51) C07C 311/18<br />

A61K 31/44 → (51) C07C 311/21<br />

A61K 31/4427 → (51) C07D 313/00<br />

A61K 31/4436 → (51) C07C 311/18<br />

A61K 31/4436 → (51) C07D 333/36<br />

A61K 31/4439 → (51) C07D 333/36<br />

A61K 31/4439 → (51) C07D 401/12<br />

A61K 31/444 → (51) C07D 333/36<br />

A61K 31/4523 → (51) C07D 313/00<br />

A61K 31/4525 → (51) A61K 31/00<br />

A61K 31/455 → (51) C07D 313/00<br />

A61K 31/47 → (51) C07D 487/04<br />

(51) A61K 31/485 (11) 2 292 229 A1<br />

A61K 9/22 A61K 9/32<br />

(25) En (26) En<br />

(21) <strong>10</strong>192641.8 (22) 24.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 25.08.2006 US 840244 P<br />

(54) • Manipulationssichere orale pharmazeutische<br />

Dosierformen enthaltend ein Opiatanalgetikum<br />

• Tamper resistant oral pharmaceutical<br />

dosage forms comprising an opioid<br />

analgesic<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• Formes de dosage pharmaceutiques orales<br />

anti-manipulation contenant un analgésique<br />

opioide<br />

(71) Purdue Pharma LP, One Stamford Forum<br />

201 Tresser Boulevard, Stamford, CT 06901,<br />

US<br />

(72) Mannion, Richard Owen, Furlong, PA 18925,<br />

US<br />

Huang, Haiyong Hugh, Princeton, NJ 08540,<br />

US<br />

McKenna, William Henry, Yonkers, NY<br />

<strong>10</strong>704, US<br />

O'Donnell, Edward, P., Basking Ridge, NJ<br />

07920, US<br />

(74) Ehlich, Eva Susanne, Maiwald <strong>Patent</strong>anwalts<br />

GmbH Elisenhof Elisenstraße 3, 80335<br />

München, DE<br />

(62) 09156832.9 / 2 070 538<br />

07114982.7 / 1 897 545<br />

(51) A61K 31/485 (11) 2 292 230 A1<br />

A61K 9/22 A61K 9/32<br />

(25) En (26) En<br />

(21) <strong>10</strong>192644.2 (22) 24.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 25.08.2006 US 840244 P<br />

(54) • Manipulationssichere orale pharmazeutische<br />

Dosierformen enthaltend ein Opiatanalgetikum<br />

• Tamper resistant oral pharmaceutical<br />

dosage forms comprising an opioid<br />

analgesic<br />

• Formes de dosage pharmaceutiques orales<br />

anti-manipulation contenant un analgésique<br />

opioide<br />

(71) Purdue Pharma LP, One Stamford Forum<br />

201 Tresser Boulevard, Stamford, CT 06901,<br />

US<br />

(72) Mannion, Richard Owen, Furlong, PA 18925,<br />

US<br />

Huang, Haiyong Hugh, Princeton, NJ 08540,<br />

US<br />

McKenna, William Henry, Yonkers, NY<br />

<strong>10</strong>704, US<br />

O'Donnell, Edward Patrick, Basking Ridge,<br />

NJ 07920, US<br />

(74) Ehlich, Eva Susanne, Maiwald <strong>Patent</strong>anwalts<br />

GmbH Elisenhof Elisenstraße 3, 80335<br />

München, DE<br />

(62) 09156832.9 / 2 070 538<br />

07114982.7 / 1 897 545<br />

A61K 31/485 → (51) A61K 31/00<br />

A61K 31/495 → (51) C07D 487/04<br />

A61K 31/496 → (51) C07D 333/36<br />

(51) A61K 31/4965 (11) 2 292 231 A1<br />

A61P 25/00 C07D 241/20<br />

(25) Ja (26) En<br />

(21) 09770<strong>10</strong>6.4 (22) 22.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) JP 2009/061285 22.06.2009<br />

(87) WO 2009/157396 2009/53 30.12.2009<br />

(30) 23.06.2008 JP 2008162638<br />

(54) • HEILMITTEL ZUR BEHANDLUNG VON<br />

SPINALER STENOSE<br />

• THERAPEUTIC AGENT FOR SPINAL CANAL<br />

STENOSIS<br />

• AGENT THÉRAPEUTIQUE POUR LA STÉ-<br />

NOSE DU CANAL SPINAL<br />

174<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(71) Nippon Shinyaku Co., Ltd., 14, Kisshoin<br />

Nishinosho Monguchicho Minami-ku, Kyotoshi<br />

Kyoto 601-8550, JP<br />

(72) KUWANO, Keiichi, Osaka-shi Osaka 547-<br />

0045, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

A61K 31/4965 → (51) C07C 237/20<br />

(51) A61K 31/4985 (11) 2 292 232 A1<br />

A61P 3/<strong>10</strong><br />

(25) En (26) En<br />

(21) <strong>10</strong>182449.8 (22) 05.07.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

AL LT LV MK<br />

(30) 06.07.2001 US 303474 P<br />

(54) • Beta-Amino-Tetrahydroimidazo(1,2-A)<br />

Pyrazine und Tetrahydrotriazolo(4,3-A)<br />

Ayrazine zur Verwendung zur Behandlung<br />

von Typ-II Diabetes<br />

• Beta-amino tetrahydroimidazo(1,2-A)pyrazines<br />

and tetrahydrotriazolo(4,3-A)pyrazines<br />

for use in the treatment of diabetes<br />

type II<br />

• Beta-amino tetrahydroimidazo(1,2-A)pyrazines<br />

et tetrahydrotriazolo(4,3-A)pyrazines<br />

pour une utilisation de traitement du<br />

diabete de type II<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) Edmondson, Scott, D., Rahway, NJ 07065-<br />

0907, US<br />

Fisher, Michael, H., Rahway, NJ 07065-0907,<br />

US<br />

Kim, Dooseop, Rahway, NJ 07065-0907, US<br />

Maccoss, Malcolm, Rahway, NJ 07065-<br />

0907, US<br />

Parmee, Emma, R., Rahway, NJ 07065-<br />

0907, US<br />

(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Hertford Road,<br />

Hoddesdon, Hertfordshire EN11 9BU, GB<br />

(62) <strong>10</strong>005997.1 / 2 226 324<br />

05077584.0 / 1 625 847<br />

02749813.8 / 1 412 357<br />

(51) A61K 31/505 (11) 2 292 233 A2<br />

(25) En (26) En<br />

(21) <strong>10</strong>185615.1 (22) 09.11.2000<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

AL LT LV MK RO SI<br />

(30) 11.11.1999 US 164907 P<br />

30.03.2000 US 193191 P<br />

23.05.2000 US 206420 P<br />

(54) • Pharmazeutische Verwendungen von N-(3-<br />

Ethynylphenyl)-6,7-bis(2-methoxyethoxy)-<br />

4-chinazolinamin<br />

• Pharmaceutical uses of N-(3-Ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine<br />

• Utilisations pharmaceutiques de N-(3ethynylphenyl)-6,7-bis(2-methoxyethoxy)-<br />

4-quinazolinamine<br />

(71) OSI Pharmaceuticals, Inc., 420 Saw Mill<br />

River Road, Ardsley, New York <strong>10</strong>502, US<br />

(72) Connell, Richard, D., East Lyme, CT 06333,<br />

US<br />

Moyer, James, D, East Lyme, CT 06333, US<br />

Morin, Michael, J, Waterford, CT 06385, US<br />

Kajiji, Shama, M, Mystic, CT 06355, US<br />

Foster, Barbara, A, Mystic, CT 06355, US<br />

Ferrante, Karen, J., East Greenwich, RI<br />

02818, US<br />

Norris, Timothy, Gales Ferry, CT 06335, US

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