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Bulletin 2011/10 - European Patent Office

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(C07D) II.1(1)<br />

JANETKA, James, AstraZeneca R & D<br />

Boston, Waltham, Massachusetts 02451, US<br />

LYNE, Paul, AstraZeneca R & D Boston,<br />

Waltham, Massachusetts 02451, US<br />

SU, Mei, AstraZeneca R & D Boston,<br />

Waltham, Massachusetts 02451, US<br />

TOADER, Dorin, AstraZeneca R & D Boston,<br />

Waltham, Massachusetts 02451, US<br />

YU, Dingwei, AstraZeneca R & D Boston,<br />

Waltham, Massachusetts 02451, US<br />

YU, Yan, AstraZeneca R & D Boston,<br />

Waltham, Massachusetts 02451, US<br />

(60) <strong>10</strong>184816.6<br />

C07D 409/12 → (51) C07D 231/44<br />

C07D 409/14 → (51) C07D 409/04<br />

C07D 409/14 → (51) C07D 409/12<br />

C07D 411/04 → (51) C07D 409/04<br />

C07D 413/06 → (51) C07D 417/04<br />

(51) C07D 413/12 (11) 2 144 904 B1<br />

A61K 31/42 A61P 31/12<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 08749348.2 (22) 06.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 20.01.20<strong>10</strong><br />

(86) EP 2008/003626 06.05.2008<br />

(87) WO 2008/138516 2008/47 20.11.2008<br />

(30) 09.05.2007 US 924321 P<br />

(54) • (S,R)-3-PHENYL-4,5 DIHYDRO-5-ISOXA-<br />

ZOLESSIGSÄURE-STICKOXID UND VER-<br />

WENDUNG ALS KREBSMITTEL UND<br />

VIRUZID<br />

• (S,R)-3-PHENYL-4,5 DIHYDRO-5-ISOXA-<br />

ZOLE ACETIC ACID-NITRIC OXIDE AND<br />

USE THEREOF AS ANTI-CANCER AND<br />

ANTIVIRAL AGENT<br />

• OXYDE NITRIQUE DE L'ACIDE (S,R)-3-<br />

PHÉNYL-4,5-DIHYDRO-5-ISOXAZOLE-<br />

ACÉTIQUE ET SON UTILISATION EN TANT<br />

QU'AGENT ANTICANCÉREUX ET ANTIVI-<br />

RAL<br />

(73) Ganial Immunotherapeutics Inc., The Corporation<br />

Trust Center 1209 Orange Street,<br />

Wilmington, DE 19801, US<br />

(72) NICOLETTI, Ferninando, 95021 Cannizzaro,<br />

IT<br />

AL-ABED, Yousef, Locust Valley, NY 11560,<br />

US<br />

GAROTTA, Gianni, 74380 Lucinges, FR<br />

(74) Minoja, Fabrizio, Bianchetti Bracco Minoja S.<br />

r.l. Via Plinio 63, 20129 Milano, IT<br />

(51) C07D 413/12 (11) 2 201 006 B1<br />

C07D 417/12 A61K 31/427<br />

A61K 31/422 A61P 37/00<br />

(25) En (26) En<br />

(21) 08840589.9 (22) 17.<strong>10</strong>.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 30.06.20<strong>10</strong><br />

(86) EP 2008/064023 17.<strong>10</strong>.2008<br />

(87) WO 2009/050258 2009/17 23.04.2009<br />

(30) 18.<strong>10</strong>.2007 EP 07020396<br />

(54) • (R)-4-(HETEROARYL)PHENYLETHYLDER-<br />

IVATE UND PHARMAZEUTISCHE ZUSAM-<br />

MENSETZUNGEN DAMIT<br />

• (R)-4-(HETEROARYL) PHENYLETHYL<br />

DERIVATIVES AND PHARMACEUTICAL<br />

COMPOSITIONS CONTAINING THEM<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• DÉRIVÉS DE (R)-4-(HÉTÉROARYL)PHÉ-<br />

NYLÉTHYLE ET COMPOSITIONS PHAR-<br />

MACEUTIQUES LES CONTENANT<br />

(73) Dompé S.p.a., Via Campo di Pile snc, 67<strong>10</strong>0<br />

L'aquila, IT<br />

(72) MORICONI, Alessio, I-67<strong>10</strong>0 L'aquila, IT<br />

ARAMINI, Andrea, I-67<strong>10</strong>0 L'aquila, IT<br />

(74) Perani, Aurelio, et al, Perani & Partners<br />

Piazza San Babila, 5, 20122 Milano, IT<br />

C07D 413/12 → (51) C07D 209/30<br />

C07D 413/12 → (51) C07D 237/30<br />

C07D 413/12 → (51) C07D 249/06<br />

C07D 413/12 → (51) C07D 409/12<br />

C07D 413/14 → (51) C07D 409/12<br />

(51) C07D 417/04 (11) 1 620 434 B1<br />

C07D 417/06 C07D 417/14<br />

C07D 403/06 C07D 413/06<br />

A61P 25/00 A61K 31/425<br />

A61K 31/404 A61K 31/423<br />

(25) En (26) En<br />

(21) 04751135.7 (22) 03.05.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(43) 01.02.2006<br />

(86) US 2004/013606 03.05.2004<br />

(87) WO 2004/<strong>10</strong>1559 2004/48 25.11.2004<br />

(30) 07.05.2003 US 431152<br />

25.09.2003 US 670629<br />

(54) • KONDENSIERTE BIZYKLISCH SUBSTITU-<br />

IERTE AMINE ALS HISTAMIN 3 REZEPTOR<br />

LIGANDEN<br />

• FUSED BICYCLIC-SUBSTITUTED AMINES<br />

AS HISTAMINE-3 RECEPTOR LIGANDS<br />

• AMINES SUBSTITUEES BICYCLIQUES<br />

HYBRIDES SERVANT DE LIGANDS AU<br />

RECEPTEUR D'HISTAMINE 3<br />

(73) ABBOTT LABORATORIES, Dept. 377, Bldg<br />

AP6A-1A <strong>10</strong>0 Abbott Park Road, Abbott<br />

Park, IL 60064-6008, US<br />

(72) COWART, Marlon, D., Round Lake Beach, IL<br />

60073, US<br />

KU, Yin-Yin, Buffalo Grove, IL 60089, US<br />

CHANG, Sou-Jen, Prairie View, IL 60069, US<br />

FERNANDO, Dilinie, P., Gurnee, IL 60031,<br />

US<br />

GRIEME, Timothy, A., Chicago, IL 60640, US<br />

ALTENBACH, Robert, A., Chicago, IL 60631,<br />

US<br />

(74) Modiano, Micaela Nadia, et al, Modiano Josif<br />

Pisanty & Staub Ltd Thierschstrasse 11,<br />

80538 München, DE<br />

(60) <strong>10</strong>180403.7<br />

C07D 417/06 → (51) C07D 417/04<br />

C07D 417/<strong>10</strong> → (51) C07D 237/30<br />

C07D 417/12 → (51) C07D 209/30<br />

C07D 417/12 → (51) C07D 401/06<br />

C07D 417/12 → (51) C07D 413/12<br />

C07D 417/14 → (51) C07D 401/14<br />

C07D 417/14 → (51) C07D 409/12<br />

C07D 417/14 → (51) C07D 417/04<br />

C07D 453/02 → (51) C07D 409/12<br />

588<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(51) C07D 471/04 (11) 1 874 770 B1<br />

C07D 235/04 A61K 31/4184<br />

A61K 31/4188 A61P 35/00<br />

A61P 35/02<br />

(25) En (26) En<br />

(21) 06724286.7 (22) 12.04.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 09.01.2008<br />

(86) EP 2006/003380 12.04.2006<br />

(87) WO 2006/<strong>10</strong>8640 2006/42 19.<strong>10</strong>.2006<br />

(30) 14.04.2005 GB 0507575<br />

(54) • ALS PROTEINKINASEINHIBITOREN<br />

GEEIGNETE PHENYLACETAMIDE<br />

• PHENYLACETAMIDES SUITABLE AS PRO-<br />

TEIN KINASE INHIBITORS<br />

• PHENYLACETAMIDES APPROPRIES EN<br />

TANT QU'INHIBITEURS DE PROTEINES<br />

KINASES<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) BOLD, Guido, CH-5073 Gipf-Oberfrick, CH<br />

FURET, Pascal, F-68800 Thann, FR<br />

GUAGNANO, Vito, CH-4054 Basel, CH<br />

MCCARTHY, Clive, Novartis AG, CH-4056<br />

Basel, CH<br />

VAUPEL, Andrea, CH-4125 Riehen, CH<br />

(74) Roth, Peter Richard, et al, Novartis AG<br />

Corporate Intellectual Property, 4002 Basel,<br />

CH<br />

C07D 471/04 → (51) C07D 237/30<br />

C07D 471/04 → (51) C07D 401/06<br />

C07D 471/04 → (51) C07D 405/14<br />

(51) C07D 471/08 (11) 1 996 194 B1<br />

A61K 31/437 A61P 25/00<br />

(25) En (26) En<br />

(21) 07752887.5 (22) 12.03.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 03.12.2008<br />

(86) US 2007/006219 12.03.2007<br />

(87) WO 2007/<strong>10</strong>6439 2007/38 20.09.2007<br />

(30) <strong>10</strong>.03.2006 US 781245 P<br />

(54) • HOMOTROPANE MIT ZNS-AKTIVITÄT<br />

• HOMOTROPANES WITH CENTRAL NER-<br />

VOUS SYSTEM ACTIVITY<br />

• HOMOTROPANES AGISSANT SUR LE<br />

SYSTÈME NERVEUX CENTRAL<br />

(73) THE RESEARCH FOUNDATION OF STATE<br />

UNIVERSITY OF NEW YORK, STOR Intellectual<br />

Property Division, UB Technology Incubator,<br />

Suite 111, Amherst, NY 14228-2567,<br />

US<br />

(72) DAVIES, Huw, M.l., E. Amherst, NY 14051,<br />

US<br />

(74) Pidgeon, Robert John, Appleyard Lees 15<br />

Clare Road, GB-Halifax, West Yorkshire HX1<br />

2HY, GB<br />

(51) C07D 471/14 (11) 1 641 795 B1<br />

C07D 487/04 A61K 31/519<br />

A61P 9/00<br />

(25) En (26) En<br />

(21) 04726960.0 (22) 13.04.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(43) 05.04.2006<br />

(86) EP 2004/003851 13.04.2004<br />

(87) WO 2004/094425 2004/45 04.11.2004<br />

(30) 24.04.2003 EP 03009286

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