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Bulletin 2011/10 - European Patent Office

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(C07D) I.1(1)<br />

(87) WO 2009/142522 2009/48 26.11.2009<br />

(30) 23.05.2008 PL 38526508<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

SOLIFENACIN UND/ODER DEN PHARMA-<br />

ZEUTISCH UNBEDENKLICHEN SALZEN<br />

DAVON IN HOHER PHARMAZEUTISCHER<br />

REINHEIT<br />

• PROCESS FOR PREPARATION OF SOLI-<br />

FENACIN AND/OR THE PHARMACEUTI-<br />

CALLY ACCEPTABLE SALTS THEREOF OF<br />

HIGH PHARMACEUTICAL PURITY<br />

• PROCEDE DE PREPARATION DE SOLIFE-<br />

NACINE ET/OU DE SES SELS PHARMA-<br />

CEUTIQUEMENT ACCEPTABLES DE<br />

HAUTE PURETE PHARMACEUTIQUE<br />

(71) Zaklady Farmaceutyczne "Polpharma" S.A.,<br />

Ul. Pelplinska 19, 83-200 Starogard Gdanski,<br />

PL<br />

(72) ZEGROCKA-STENDEL, Oliwia, PL-05-092<br />

Warszawa, PL<br />

ZAGRODZKA, Joanna, PL-01-772 Warszawa,<br />

PL<br />

LASZCZ, Marta, PL-02-904 Warszawa, PL<br />

(51) C07D 471/04 (11) 2 291 375 A1*<br />

A61K 31/437 A61P 35/00<br />

(25) De (26) De<br />

(21) 09772064.3 (22) 04.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) EP 2009/004013 04.06.2009<br />

(87) WO 20<strong>10</strong>/000364 20<strong>10</strong>/01 07.01.20<strong>10</strong><br />

(30) 03.07.2008 DE <strong>10</strong>2008031517<br />

(54) • PYRROLOPYRIDINYL-PYRIMIDIN-2-YL-<br />

AMIN-DERIVATE<br />

• PYRROLOPYRIDINYLPYRIMIDIN-2-YLA-<br />

MINE DERIVATIVES<br />

• DÉRIVÉ DE PYRROLOPYRIDINYLPYRIMI-<br />

DIN-2-YLAMINE<br />

(71) Merck <strong>Patent</strong> GmbH, Frankfurter Strasse<br />

250, 64293 Darmstadt, DE<br />

(72) WUCHERER-PLIETKER, Margarita, 64291<br />

Darmstadt, DE<br />

BRUGE, David, 60329 Frankfurt, DE<br />

FINSINGER, Dirk, 64291 Darmstadt, DE<br />

GRAEDLER, Ulrich, 69115 Heidelberg, DE<br />

DORSCH, Dieter, 64372 Ober-Ramstadt, DE<br />

ESDAR, Christina, 55128 Mainz, DE<br />

(51) C07D 471/04 (11) 2 291 376 A2*<br />

A61K 31/436 A61P 35/00<br />

(25) En (26) En<br />

(21) 09774230.8 (22) 29.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/049035 29.06.2009<br />

(87) WO 20<strong>10</strong>/002779 20<strong>10</strong>/01 07.01.20<strong>10</strong><br />

(30) 03.07.2008 US 134018<br />

(54) • NAPHTHYRIDININONE ALS AURORAKI-<br />

NASEHEMMER<br />

• NAPHTHYRIDININONES AS AURORA<br />

KINASE INHIBITORS<br />

• NAPHTYRIDININONES EN TANT QU INHI-<br />

BITEURS D AURORA KINASE<br />

(71) Merck <strong>Patent</strong> GmbH, Frankfurter Strasse<br />

250, 64293 Darmstadt, DE<br />

(72) XIAO, Yufang, Marshfield Massachusetts<br />

02050, US<br />

CHEN, Xiaoling, Newton Massachusetts<br />

02466, US<br />

KARRA, Srinivasa R., Pembroke Massachusetts<br />

02359, US<br />

HUCK, Bayard R., Sudbury Massachusetts<br />

01776, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

SUTTON, Amanda E., Hingham Massachusetts<br />

02043, US<br />

GOUTOPOULOS, Andreas, Boston Massachusetts<br />

02116, US<br />

(51) C07D 487/04 (11) 2 291 377 A1*<br />

A61K 31/519 A61P 31/18<br />

(25) En (26) En<br />

(21) 09771848.0 (22) 02.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) AU 2009/000857 02.07.2009<br />

(87) WO 20<strong>10</strong>/000031 20<strong>10</strong>/01 07.01.20<strong>10</strong><br />

(30) 02.07.2008 AU 2008903406<br />

20.03.2009 US 161931<br />

(54) • IMIDAZOPYRIMIDINONE UND IHRE VER-<br />

WENDUNGEN<br />

• IMIDAZOPYRIMIDINONES AND USES<br />

THEREOF<br />

• IMIDAZOPYRIMIDINONES ET LEURS UTI-<br />

LISATIONS<br />

(71) Avexa Limited, 576 Swan Street, Richmond,<br />

VIC 3121, AU<br />

(72) DEADMAN, John, Joseph, Carlton Victoria<br />

3053, AU<br />

JONES, Eric, Dale, Bentleigh East Victoria<br />

3165, AU<br />

LE, Giang, Thanh, Lower Templestowe<br />

Victoria 3<strong>10</strong>7, AU<br />

RHODES, David, Ian, Heidelberg Heights<br />

Victoria 3081, AU<br />

THIENTHONG, Neeranat, Malvern Victoria<br />

3144, AU<br />

VAN DE GRAFF, Nicholas, Andrew, Prahran<br />

Victoria 3181, AU<br />

WINFIELD, Lisa, Jane, Wymondham Norfolk<br />

NR18 0JJ, GB<br />

(74) Harrison Goddard Foote, Belgrave Hall Belgrave<br />

Street, Leeds LS2 8DD, GB<br />

(51) C07D 487/04 (11) 2 291 378 A2*<br />

(25) En (26) En<br />

(21) 09703852.5 (22) 22.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/031666 22.01.2009<br />

(87) WO 2009/094428 2009/31 30.07.2009<br />

(88) 01.<strong>10</strong>.2009<br />

(30) 22.01.2008 US 18172<br />

(54) • N- UND O-SUBSTITIERTE 4-[2-(DIPHE-<br />

NYLMETHOXY)-ETHYL]-1-[(PHENYL)<br />

METHYL]PIPERIDINANALOGA UND VER-<br />

FAHREN ZUR BEHANDLUNG VON ZNS-<br />

ERKRANKUNGEN DAMIT<br />

• N- AND O-SUBSTITUTED 4-Ý2-(DIPHE-<br />

NYLMETHOXY)-ETHYL¨-1-Ý(PHENYL)<br />

METHYL¨PIPERIDINE ANALOGS AND<br />

METHODS OF TREATING CNS DISORDERS<br />

THEREWITH<br />

• ANALOGUES DE LA 4-Ý2-(DIPHÉNYLMÉ-<br />

THOXY)-ÉTHYL¨-1-Ý(PHÉNYL)MÉTHYL¨-<br />

PIPÉRIDINE SUBSTITUÉS SUR N ET O ET<br />

PROCÉDÉS DE TRAITEMENT PAR CEUX-CI<br />

DE TROUBLES DU SYSTÈME NERVEUX<br />

CENTRAL<br />

(71) WAYNE STATE UNIVERSITY, 4043 Faculty/<br />

Administration Building, Detroit, MI 48202,<br />

US<br />

(72) DUTTA, Aloke, K., Novi, MI 48375, US<br />

(74) GPI & Associés, 1330, rue Guillibert de la<br />

Lauzière EuroParc de Pichaury, Bât B2,<br />

13856 Aix en Provence Cedex 3, FR<br />

60<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(51) C07D 487/04 (11) 2 291 379 A1*<br />

A61K 31/519 A61P 7/00<br />

(25) En (26) En<br />

(21) 09746112.3 (22) 13.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) GB 2009/050515 13.05.2009<br />

(87) WO 2009/138795 2009/47 19.11.2009<br />

(30) 16.05.2008 GB 0808953<br />

(54) • SUBSTITUIERTE CHINAZOLINE<br />

• SUBSTITUTED QUINAZOLINES<br />

• QUINAZOLINES SUBSTITUÉES<br />

(71) Shire LLC, 9200 Brookfield Court, Florence,<br />

KY 4<strong>10</strong>42, US<br />

(72) GOLDING, Bernard, Newcastle upon Tyne<br />

Tyne and Wear NE27 0EZ, GB<br />

FRANKLIN, Richard, Fleet hampshire GU51<br />

4NQ, GB<br />

(74) Harrison Goddard Foote, Belgrave Hall Belgrave<br />

Street, Leeds LS2 8DD, GB<br />

(51) C07D 489/08 (11) 2 291 380 A1*<br />

A61K 31/485 A61P 25/30<br />

(25) En (26) En<br />

(21) 09733923.8 (22) 23.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) EP 2009/054882 23.04.2009<br />

(87) WO 2009/130272 2009/44 29.<strong>10</strong>.2009<br />

(30) 24.04.2008 EP 08155094<br />

(54) • NALMEFEN-PRODRUGS<br />

• NALMEFENE PRODRUGS<br />

• PROMÉDICAMENTS DE NALMÉFÈNE<br />

(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) GUILLAUME, Michel, Joseph, Maurice,<br />

André, B-2340 Beerse, BE<br />

GAEKENS, Tim, B-2340 Beerse, BE<br />

(74) Verberckmoes, Filip Gerard, Janssen Pharmaceutica<br />

N.V., J&J <strong>Patent</strong> Law Department,<br />

Turnhoutseweg 30, 2340 Beerse, BE<br />

(51) C07D 491/04 (11) 2 291 381 A1*<br />

C07D 215/12 C07D 215/14<br />

C07D 215/20 A61K 31/47<br />

A61K 31/4725<br />

(25) Fr (26) Fr<br />

(21) 09761869.8 (22) 15.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) FR 2009/000573 15.05.2009<br />

(87) WO 2009/150318 2009/51 17.12.2009<br />

(30) 20.05.2008 FR 0802745<br />

(54) • NEUE 2-SUBSTITUIERTE CHINOLINDER-<br />

IVATE UND VERFAHREN ZU DEREN HER-<br />

STELLUNG<br />

• NOVEL 2-SUBSTITUTED QUINOLINE<br />

DERIVATIVES, AND METHOD FOR PRE-<br />

PARING SAME<br />

• NOUVEAUX DERIVES DE QUINOLEINES 2-<br />

SUBSTITUEES ET UN PROCEDE POUR<br />

LEUR PREPARATION<br />

(71) Institut De Recherche Pour Le Developpement,<br />

Le Sextant 44 bd de Dunkerque CS<br />

90009, 13572 Marseille Cedex 02, FR<br />

Alpha Chimica, Faculté de Pharmacie Paris-<br />

Sud 11 5 rue J.B. Clément, 92290 Châtenay-<br />

Malabry, FR<br />

(72) FOURNET, Alain, F-40290 Ossages, FR<br />

AKAGAH, Bernardin, F-92290 Chatenay-<br />

Malabry, FR

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