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Bulletin 2011/10 - European Patent Office

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(C07D) II.1(1)<br />

• SUBSTITUTED PYRANO [2, 3 - B]PYRI-<br />

DINE DERIVATIVES AS CANNABINOID-1<br />

RECEPTOR MODULATORS<br />

• DÉRIVÉS DE PYRANO [2, 3 - B]PYRIDINE<br />

SUBSTITUÉE EN TANT QUE MODULA-<br />

TEURS DU RÉCEPTEUR DU CANNABI-<br />

NOÏDE-1<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) DEBENHAM, John, S., Rahway, New Jersey<br />

07065-0907, US<br />

HALE, Jeffrey, J., Rahway, New Jersey<br />

07065-0907, US<br />

HUO, Pei, Rahway, New Jersey 07065-0907,<br />

US<br />

MADSEN-DUGGAN, Christina, B., Rahway,<br />

New Jersey 07065-0907, US<br />

WALSH, Thomas, F., Rahway, New Jersey<br />

07065-0907, US<br />

YAN, Lin, Rahway, New Jersey 07065-0907,<br />

US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 491/16 → (51) C07D 491/052<br />

(51) C07D 495/02 (11) 2 176 269 B1<br />

(25) En (26) En<br />

(21) 08773248.3 (22) 08.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 21.04.20<strong>10</strong><br />

(86) CZ 2008/000079 08.07.2008<br />

(87) WO 2009/006859 2009/03 15.01.2009<br />

(30) 09.07.2007 CZ 20070456<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ESSIGSÄURE-5-[2-CYCLOPROPYL-1-(2-<br />

FLUORPHENYL)-2-OXOETHYL]-4,5,6,7-<br />

TETRAHYDROTHIENO[3,2-C]PYRIDIN-2-<br />

YL-ESTER (PRASUGREL)<br />

• A METHOD OF MANUFACTURING 5-[2-<br />

CYCLOPROPYL-1-(2-FLUOROPHENYL)-2-<br />

OXOETHYL]-4,5,6,7- TETRAHY-<br />

DROTHIENO[3,2-C]PYRIDIN-2-YL ACET-<br />

ATE (PRASUGREL)<br />

• PROCÉDÉ DE FABRICATION D'ACÉTATE<br />

DE 5-[2-CYCLOPROPYL-1-(2-FLUORO-<br />

PHÉNYL)-2-OXOÉTHYL]-4,5,6,7-TÉTRA-<br />

HYDROTHIÉNO[3,2-C]PYRIDIN-2-YLE<br />

(PRASUGREL)<br />

(73) Zentiva, k.s., U kabelovny 130, Dolni<br />

Mecholupy <strong>10</strong>2 37 Praha <strong>10</strong>, CZ<br />

(72) STEPANKOVA, Hana, 282 01 Cesky Brod, CZ<br />

HAJICEK, Josef, 128 00 Praha 2, CZ<br />

(74) Jirotkova, Ivana, et al, Rott, Ruzicka &<br />

Guttmann <strong>Patent</strong>, Trademark and Law <strong>Office</strong><br />

Vinohradskà 37, 120 00 Praha 2, CZ<br />

(51) C07D 495/04 (11) 1 656 381 B1<br />

(25) En (26) En<br />

(21) 04763994.3 (22) 11.08.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

AL HR LT LV MK<br />

(43) 17.05.2006<br />

(86) EP 2004/008989 11.08.2004<br />

(87) WO 2005/016931 2005/08 24.02.2005<br />

(30) 13.08.2003 DE <strong>10</strong>337773<br />

(54) • KRISTALLISATION VON FESTEN FORMEN<br />

VON CLOPIDOGRELADDITIONSSALZEN<br />

• CRYSTALLISATION OF SOLID FORMS OF<br />

CLOPIDOGREL ADDITION SALTS<br />

• CRISTALLISATION DE FORMES SOLIDES<br />

DE SELS D'ADDITION DU CLOPIDOGREL<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(73) Krka, Torvarna Zdravil, D.D., Novo Mesto,<br />

Smarjeska cesta 6, 8501 Novo mesto, SI<br />

(72) KOTAR-JORDAN, Berta, 8311 Kostanjevica<br />

na Krki, SI<br />

SIMONIC, Igor, 8351 Straza, SI<br />

ZUPET, Rok, 1211 Ljubljana, SI<br />

RUZIC, Milos, 3000 Celje, SI<br />

GRCMAN, Marija, 8212 Velika, SI<br />

PECAVAR, Anica, 8000 Novo mesto, SI<br />

(74) UEXKÜLL & STOLBERG, <strong>Patent</strong>anwälte<br />

Beselerstrasse 4, 22607 Hamburg, DE<br />

C07D 495/16 → (51) C07D 491/052<br />

(51) C07D 501/00 (11) 1 554 289 B1<br />

A61K 31/546<br />

(25) En (26) En<br />

(21) 03787771.9 (22) 12.08.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 20.07.2005<br />

(86) EP 2003/008944 12.08.2003<br />

(87) WO 2004/016623 2004/09 26.02.2004<br />

(30) 13.08.2002 AT 12232002<br />

18.<strong>10</strong>.2002 AT 15882002<br />

(54) • EIN CEFDINIR-ZWISCHENPRODUKT<br />

• A CEFDINIR INTERMEDIATE<br />

• INTERMEDIAIRE DE CEFDINIR<br />

(73) SANDOZ AG, Lichtstrasse 35, 4056 Basel,<br />

CH<br />

(72) KREMMINGER, Peter, 6330 Kufstein, AT<br />

WOLF, Siegfried, 6230 Brixlegg, AT<br />

LUDESCHER, Johannes, A-6252 Breitenbach,<br />

AT<br />

(60) 07111390.6 / 1 842 852<br />

(51) C07D 513/04 (11) 1 840 129 B1<br />

C07B 61/00 A61K 31/429<br />

A61P 31/04<br />

(25) Ja (26) En<br />

(21) 06711975.0 (22) 19.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 03.<strong>10</strong>.2007<br />

(86) JP 2006/300729 19.01.2006<br />

(87) WO 2006/077919 2006/30 27.07.2006<br />

(30) 19.01.2005 JP 2005011923<br />

(54) • IMIDAZOTHIAZOL-DERIVAT UND HER-<br />

STELLUNGSVERFAHREN DAFÜR<br />

• IMIDAZOTHIAZOLE DERIVATIVE AND<br />

METHOD FOR PRODUCING SAME<br />

• DÉRIVÉ D'IMIDAZOTHIAZOLE ET<br />

MÉTHODE DE SYNTHÈSE DUDIT DÉRIVÉ<br />

(73) Meiji Seika Kaisha Ltd., 4-16, Kyobashi 2chome,<br />

Chuo-ku, Tokyo <strong>10</strong>4-8002, JP<br />

SAGAMI CHEMICAL RESEARCH CENTER,<br />

2743-1, Hayakawa, Ayase-shi, Kanagawa<br />

252-1193, JP<br />

(72) SHITARA, Eiki, uhoku-ku, Yokohama-shi,<br />

Kanagawa, 222856, JP<br />

ATSUMI, Kunio, uhoku-ku, Yokohama-shi,<br />

Kanagawa, 222856, JP<br />

AJITO, Keiichi, me, Chuo-ku, Tokyo,<br />

<strong>10</strong>48002, JP<br />

IKEDA, Shinya, -shi, Kanagawa, 2500852, JP<br />

KATOH, Tadashi, i, Miyagi, 9800801, JP<br />

INOUE, Munenori, 30403, JP<br />

NAKATANI, Mari, Shizuoka-ken, JP<br />

(74) Warcoin, Jacques, et al, Cabinet Régimbeau<br />

20, rue de Chazelles, 75847 Paris Cedex 17,<br />

FR<br />

(51) C07D 519/00 (11) 2 024 375 B1<br />

A61P 31/12 A61K 31/55<br />

(25) En (26) En<br />

(21) 07761873.4 (22) 04.05.2007<br />

590<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

HR<br />

(43) 18.02.2009<br />

(86) US 2007/068209 04.05.2007<br />

(87) WO 2007/136982 2007/48 29.11.2007<br />

(30) 17.05.2006 US 801125 P<br />

19.05.2006 US 802005 P<br />

16.<strong>10</strong>.2006 US 852084 P<br />

14.03.2007 US 894757 P<br />

(54) • CYCLOPROPYL-ANNELIERTE INDOLO-<br />

BENZAZEPINE ALS HCV-NS5B-INHIBITO-<br />

REN<br />

• CYCLOPROPYL FUSED INDOLOBENZAZE-<br />

PINE HCV NS5B INHIBITORS<br />

• INHIBITEURS DE VHC NS5B DE TYPE<br />

INDOLOBENZAZÉPINE FUSIONNÉE À UN<br />

CYCLOPROPYLE<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton, NJ<br />

08543-4000, US<br />

(72) BENDER, John A., Wallingford, Connecticut<br />

06492, US<br />

DING, Min, Wallingford, Connecticut 06492,<br />

US<br />

GENTLES, Robert G., Wallingford, Connecticut<br />

06492, US<br />

HEWAWASAM, Piyasena, Wallingford, Connecticut<br />

06492, US<br />

(74) Reitstötter - Kinzebach, <strong>Patent</strong>anwälte<br />

Sternwartstrasse 4, 81679 München, DE<br />

(51) C07F 5/02 (11) 1 355 9<strong>10</strong> B1<br />

C07F 5/04 C07K 5/078<br />

A61K 38/05 A61K 31/69<br />

A61P 35/00 A61P 29/00<br />

(25) En (26) En<br />

(21) 02709145.3 (22) 25.01.2002<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 29.<strong>10</strong>.2003<br />

(86) US 2002/001907 25.01.2002<br />

(87) WO 2002/059130 2002/31 01.08.2002<br />

(30) 25.01.2001 US 264160 P<br />

(54) • FORMULIERUNGEN VON BORSÄURE-<br />

VERBINDUNGEN<br />

• FORMULATION OF BORONIC ACID COM-<br />

POUNDS<br />

• FORMULATION DE COMPOSES D'ACIDE<br />

BORONIQUE<br />

(73) The United States of America, represented by<br />

the Secretary, Department of Health and<br />

Human Services, National Institutes of<br />

Health, <strong>Office</strong> of Technology Transfer, Suite<br />

325, 6011 Executive Boulevard, Rockville,<br />

MD 20852, US<br />

(72) GUPTA, Shanker, Rockville, MD 20850, US<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

(60) <strong>10</strong>006835.2 / 2 251 344<br />

C07F 5/04 → (51) C07F 5/02<br />

C07F 5/06 → (51) B01J 31/14<br />

C07F 7/08 → (51) C07B 63/02<br />

C07F 7/12 → (51) C07B 63/02<br />

C07F 7/18 → (51) C07B 63/02<br />

C07F 7/18 → (51) C07D 239/42<br />

C07F 7/18 → (51) C09J 183/04<br />

C07F 7/22 → (51) C07B 63/02

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