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Bulletin 2011/10 - European Patent Office

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(C07F) II.1(1)<br />

C07F 9/02 → (51) C07F 9/50<br />

C07F 9/09 → (51) C07D 213/64<br />

C07F 9/40 → (51) C09K 11/77<br />

(51) C07F 9/50 (11) 1 975 170 B1<br />

C07F 9/02<br />

(25) En (26) En<br />

(21) 08153127.9 (22) 20.03.2008<br />

(84) DE FR GB<br />

(43) 01.<strong>10</strong>.2008<br />

(30) 26.03.2007 JP 2007078384<br />

(54) • Bisphosphin-Liganden für asymmetrische<br />

Synthesen<br />

• Bisphosphine ligands for asymmetric<br />

syntheses<br />

• Ligands de bisphosphine pour synthèses<br />

asymmétriques<br />

(73) Daiichi Fine Chemical Co., Ltd., 530, Chokeiji,<br />

Takaoka-shi, Toyama 933-8511, JP<br />

(72) Watanabe, Michimasa, Toyama Toyama 933-<br />

8511, JP<br />

Takeuchi, Yuhki, Toyama Toyama 933-8511,<br />

JP<br />

Isobe, Takahiro, Toyama Toyama 933-8511,<br />

JP<br />

Takeuchi, Tadashi, Toyama Toyama 933-<br />

8511, JP<br />

(74) Polypatent, Postfach 40 02 43, 514<strong>10</strong><br />

Bergisch Gladbach, DE<br />

C07F 9/535 → (51) C07D 239/42<br />

C07H 15/26 → (51) A61K 47/48<br />

(51) C07H 17/08 (11) 1 000 952 B1<br />

A61K 31/70 A61P 31/04<br />

(25) Fr (26) Fr<br />

(21) 99402523.7 (22) 14.<strong>10</strong>.1999<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE<br />

(43) 17.05.2000<br />

(30) 15.<strong>10</strong>.1998 FR 9812937<br />

(54) • Neue 2-Halogen-Derivate von 5-O-Desosaminylerythronolid<br />

A, Verfahren zu deren<br />

Herstellung sowie deren Verwendung als<br />

Arzneimittel<br />

• New 2-halogenated derivatives of 5-Odeosaminylerythronolide<br />

A, process for<br />

making them as well as their use as<br />

medicines<br />

• Nouveaux dérivés 2-halogénés de 5-0désosaminylérythronolide<br />

A, leur procédé<br />

de préparation et leur application comme<br />

médicaments<br />

(73) Aventis Pharma S.A., 20, avenue Raymond<br />

Aron, 92160 Antony, FR<br />

(72) Agouridas, Constantin, 94130 Nogent sur<br />

Marne, FR<br />

Denis, Alexis, 75011 Paris, FR<br />

Bretin, Francois, 77330 Ozoir la Ferriere, FR<br />

Fromentin, Claude, 75019 Paris, FR<br />

(74) Le Coupanec, Pascale A.M.P., et al, Nony &<br />

Associés 3, rue de Penthièvre, 75008 Paris,<br />

FR<br />

(51) C07H 19/04 (11) 2 049 557 B1<br />

A61K 31/706<br />

(25) En (26) En<br />

(21) 07791887.8 (22) 27.07.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 22.04.2009<br />

(86) JP 2007/065213 27.07.2007<br />

(87) WO 2008/013322 2008/05 31.01.2008<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(30) 27.07.2006 US 820604 P<br />

23.01.2007 US 886178 P<br />

(54) • 1-(D-GLYKOPYRANOSYL)-3-(4-CYCLO-<br />

PROPYLPHENYLMETHYL)-4-HALOGENIN-<br />

DOLDERIVATE UND DEREN<br />

VERWENDUNG ALS SGLT-INHIBITOREN<br />

• 1- (-D-GLYCOPYRANOSYL) - 3 - (4-<br />

CYCLOPROPYLPHENYLMETHYL) - 4 -<br />

HALOGENO INDOLE DERIVATIVES AND<br />

USE THEREOF AS SGLT INHIBITORS.<br />

• DÉRIVÉS 1-(D-GLYCOPYRANOSYL)-3-(4-<br />

CYCLOPROPYLPHÉNYLMÉTHYL)-4-HALO-<br />

GÉNÉS D'INDOLE ET LEUR EMPLOI EN<br />

TANT QU'INHIBITEURS DE SGLT<br />

(73) Mitsubishi Tanabe Pharma Corporation, 2-6-<br />

18, Kitahama Chuo-ku Osaka-shi, Osaka<br />

541-8505, JP<br />

(72) NOMURA, Sumihiro, Osaka 541-8505, JP<br />

SAKAMAKI, Shigeki, Osaka 541-8505, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) C07H 21/00 (11) 2 081 948 B1<br />

C12Q 1/68 G01N 21/64<br />

(25) Fr (26) Fr<br />

(21) 07823852.4 (22) 26.09.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 29.07.2009<br />

(86) FR 2007/052007 26.09.2007<br />

(87) WO 2008/037924 2008/14 03.04.2008<br />

(30) 28.09.2006 FR 0653982<br />

(54) • NEUES MARKIERTES OLIGONUKLEOTID<br />

• NOVEL LABELLED OLIGONUCLEOTIDE<br />

• NOUVEL OLIGONUCLEOTIDE MARQUE<br />

(73) bioMérieux S.A., Chemin de l'Orme, 69280<br />

Marcy l'Etoile, FR<br />

(72) BERNAL-MENDEZ, Eloy, 38070 Saint-Quentin-Fallavier,<br />

FR<br />

LAAYOUN, Ali, 38690 Colombe, FR<br />

LAURENT, Alain, 38<strong>10</strong>0 Grenoble, FR<br />

(51) C07H 21/04 (11) 1 355 918 B1<br />

C12N 15/63 C07K 14/00<br />

G01N 33/68 C07K 14/315<br />

G01N 33/569<br />

(25) En (26) En<br />

(21) 01996301.6 (22) 28.12.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 29.<strong>10</strong>.2003<br />

(86) US 2001/049650 28.12.2001<br />

(87) WO 2002/053761 2002/28 11.07.2002<br />

(30) 28.12.2000 US 258841 P<br />

(54) • REKOMBINANTES SCHUTZPROTEIN AUS<br />

STREPTOCOCCUS PNEUMONIAE<br />

• RECOMBINANT PROTECTIVE PROTEIN<br />

FROM $I(STREPTOCOCCUS PNEUMO-<br />

NIAE)<br />

• PROTEINE PROTECTRICE RECOMBINEE<br />

ISSUE DE $I(STREPTOCOCCUS PNEUMO-<br />

NIAE)<br />

(73) Wyeth LLC, Five Giralda Farms, Madison, NJ<br />

07940, US<br />

(72) GREEN, Bruce, A., Pittsford, NY 14534, US<br />

MASI, Amy, W., Caledonia, NY 14423, US<br />

(74) Ricol, David Gerard, et al, Pfizer Limited<br />

<strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich, Kent CT13 9NJ, GB<br />

(60) <strong>10</strong>184194.8<br />

C07H 21/04 → (51) C12N 15/861<br />

(51) C07J 1/00 (11) 1 622 925 B1<br />

C07J 43/00 C07J 75/00<br />

A61K 31/566<br />

A61P 19/<strong>10</strong><br />

A61K 31/58<br />

591<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(25) Fr (26) Fr<br />

(21) 04742577.2 (22) 27.04.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(43) 08.02.2006<br />

(86) FR 2004/00<strong>10</strong><strong>10</strong> 27.04.2004<br />

(87) WO 2004/096828 2004/46 11.11.2004<br />

(30) 29.04.2003 FR 0305221<br />

(54) • NEUES VERFAHREN UND ZWISCHEN-<br />

PRODUKTE ZUR HERSTELLUNG VON 19-<br />

NOR-STEROIDEN<br />

• NOVEL METHOD AND INTERMEDIATES<br />

FOR THE PREPARATION OF 19-NOR-<br />

STEROID COMPOUNDS<br />

• NOUVEAU PROCEDE ET INTERMEDIAIRES<br />

DE PREPARATION DE COMPOSES 19-<br />

NOR-STEROÏDES<br />

(73) Aventis Pharma S.A., 20, avenue Raymond<br />

Aron, 92160 Antony, FR<br />

(72) PRAT, Denis, F-93500 Pantin, FR<br />

MORATILLE, Christian, F-94360 Bry sur<br />

Marne, FR<br />

BENEDETTI, Françoise, F-931<strong>10</strong> Rosny sous<br />

Bois, FR<br />

NAIT-BOUDA, Lahlou, F- 94320 Thiais, FR<br />

(74) Ulmann, Catherine Claire, et al, Santarelli 14,<br />

avenue de la Grande Armée B.P. 237, 75822<br />

Paris Cedex 17, FR<br />

(51) C07J 17/00 (11) 1 756 140 B1<br />

A61K 31/70 A61P 3/04<br />

(25) En (26) En<br />

(21) 05744278.2 (22) 20.05.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 28.02.2007<br />

(86) GB 2005/001995 20.05.2005<br />

(87) WO 2005/116049 2005/49 08.12.2005<br />

(30) 25.05.2004 GB 0411703<br />

(54) • SELEKTIVE ABTRENNUNG ODER<br />

EXTRAKTION VON STEROIDALEN GLYCO-<br />

SIDEN DURCH EXTRAKTION MIT SUPER-<br />

KRITISCHER FLÜSSIGKEIT UNTER<br />

EINSATZ VON KOHLENDIOXID<br />

• SELECTIVE SEPARATION OR EXTRACTION<br />

OF STEROIDAL GLYCOSIDES BY SUPER-<br />

CRITICAL FLUID EXTRACTION USING<br />

CARBON DIOXIDE<br />

• SEPARATION OU EXTRACTION SELECTIVE<br />

DE GLYCOSIDES STEROIDIQUES PAR<br />

EXTRACTION DE FLUIDE SUPER CRI-<br />

TIQUE UTILISANT DU DIOXYDE DE CAR-<br />

BONE<br />

(73) Unilever N.V., Weena 455, 3013 AL Rotterdam,<br />

NL<br />

(72) GUNNING, Philip James, c/o Phytopharm<br />

plc, Godmanchester, Cambridgeshire PE29<br />

2HY, GB<br />

ROSE, Paul Martin, c/oBotanix Limited,<br />

Paddock Wood, Kent TN12 6DQ, GB<br />

MARRIOT, Raymond,John, c/oBotanix Limited,<br />

Paddock Wood, Kent TN12 6DQ, GB<br />

(74) Brown, David Leslie, Haseltine Lake LLP<br />

Redcliff Quay 120 Redcliff Street, Bristol BS1<br />

6HU, GB<br />

C07J 43/00 → (51) C07J 1/00<br />

C07J 75/00 → (51) C07J 1/00<br />

C07K 1/02 → (51) A61K 38/02<br />

(51) C07K 1/04 (11) 1 644 401 B1<br />

(25) En (26) En<br />

(21) 04739972.0 (22) 17.06.2004

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